G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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BIMU 8
CAS:134296-40-5
BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, …
Formula:
C19H27ClN4O2
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
378.9
Ref: TM-T21946
| 1mg | 88.00 € | ||
| 1ml | 184.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 601.00 € | ||
| 100mg | 854.00 € | ||
| 500mg | 1,734.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Phoenixin-14
CAS:1415039-79-0
Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH …
Formula:
C75H110N18O20
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1583.78
Ref: TM-T80422
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Upidosin
CAS:152735-23-4
Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.
Formula:
C31H33N3O4
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
511.61
Ref: TM-T9762
| 1ml | 53.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 125.00 € | ||
| 100mg | 181.00 € | ||
| 200mg | 272.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Balixafortide TFA (1051366-32-5 free base)
Balixafortide TFA is a selective CXCR4 antagonist with IC50 < 10nM, over 1000x preference for CXCR4, …
Formula:
C82H113N22F3O23S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1896.05
Ref: TM-TP2141
| 5mg | 150.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 875.00 € | ||
| 100mg | To inquire | ||
| 200mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Panaxydol
CAS:72800-72-7
Panaxydol has anti-cancer activity, can inhibit the growth and apoptosis of cancer cells, the signaling …
Formula:
C17H24O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
260.37
Ref: TM-TN2039
| 1mg | 208.00 € | ||
| 5mg | 991.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Neurokinin A(4-10)
CAS:97559-35-8
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
Formula:
C34H54N8O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
766.91
Ref: TM-T7559
| 1mg | 123.00 € | ||
| 5mg | 243.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 850.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[D-Ala2]leucine-enkephalin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1367L.jpg)
[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study …
Formula:
C31H43N5O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
629.65
Ref: TM-TP1367L
| 5mg | 55.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 349.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Val9-Oxytocin
CAS:1021701-88-1
Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete …
Formula:
C46H72N12O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1049.27
Ref: TM-T80136
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Conopeptide rho-TIA
CAS:381725-58-2
Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at …
Formula:
C105H160N36O21S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2390.88
Ref: TM-T80175
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Catalpalactone
CAS:1585-68-8
Catalpalactone: antitermitic, cytotoxic, inhibits NO in cells (IC50 9.80µM), reduces dopamine synthesis, hinders TPA-induced EBV-EA …
Formula:
C15H14O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
258.27
Ref: TM-TN3607
| 1ml | To inquire | ||
| 5mg | 1,378.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
AB21 HCl
AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces …
Formula:
C23H29ClN2O
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
384.2
Ref: TM-T77340L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 593.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Drinabant
CAS:358970-97-5
Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.
Formula:
C23H20Cl2F2N2O2S
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
497.38
Ref: TM-T21861
| 1mg | 85.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 585.00 € | ||
| 100mg | 791.00 € | ||
| 500mg | 1,588.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PIT
CAS:56583-49-4
PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with …
Formula:
C20H16N2O5S
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
396.42
Ref: TM-T23164
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 310.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SB-408124
CAS:288150-92-5
SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x …
Formula:
C19H18F2N4O
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
356.37
Ref: TM-T6658
| 1ml | 65.00 € | ||
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 201.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Sigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic …
Formula:
C26H27N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
397.51
Ref: TM-T78734
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
WAY-298630
CAS:303134-93-2
Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.
Formula:
C17H15FN2O3S
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
346.38
Ref: TM-T77601
| 1mg | 181.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,710.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Bucindolol Formate
Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.
Formula:
C23H27N3O4
Purity:
99.11% - 99.61%
Color and Shape:
Solid
Molecular weight:
409.48
Ref: TM-T10631L
| 1mg | 181.00 € | ||
| 1ml | 462.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,282.00 € | ||
| 100mg | 1,733.00 € | ||
| 500mg | 3,452.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Latanoprost acid
CAS:41639-83-2
Latanoprost acid is a prostanoid receptor agonist that blocks RANKL and can be used to …
Formula:
C23H34O5
Purity:
96.97%
Color and Shape:
Pale Yellow Oil
Molecular weight:
390.51
Ref: TM-T15718
| 1mg | 94.00 € | ||
| 1ml | 257.00 € | ||
| 2mg | 132.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 374.00 € | ||
| 25mg | 750.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,504.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonist
Formula:
C7H13N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
171.2
Ref: TM-T23038L
| 1mg | 192.00 € | ||
| 5mg | 474.00 € | ||
| 10mg | 665.00 € | ||
| 25mg | 1,037.00 € | ||
| 50mg | 1,431.00 € | ||
| 100mg | 1,832.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Zalospirone
CAS:114298-18-9
Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and …
Formula:
C24H29N5O2
Purity:
100% - 99%
Color and Shape:
Solid
Molecular weight:
419.52
Ref: TM-T68172
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,336.00 € | ||
| 500mg | 4,564.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
