G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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EP4-IN-1
CAS:2455480-28-9
EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.
Formula:
C27H24N2O4
Purity:
100%
Color and Shape:
Soild
Molecular weight:
440.49
Ref: TM-T77699
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
(+)-OSU 6162
CAS:160777-43-5
(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant …
Formula:
C15H23NO2S
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
281.41
Ref: TM-T60027
| 1mg | 113.00 € | ||
| 5mg | 244.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,031.00 € | ||
| 500mg | 2,070.00 € | ||
| 1mL*10mM (DMSO) | 261.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
(1S,2R)-2-PCCA
(1S,2R)-2-PCCA is a novel and potent small molecule GPR88 receptor agonist with an EC50 value …
Formula:
C30H39Cl2N3O
Purity:
99.34%
Color and Shape:
Soild
Molecular weight:
528.56
Ref: TM-T13423L
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € | ||
| 100mg | 1,803.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to …
Formula:
C25H31F3N6O8
Purity:
98.40%
Color and Shape:
Soild
Molecular weight:
600.55
Ref: TM-T26641L
| 1mg | 735.00 € | ||
| 5mg | 1,834.00 € | ||
| 25mg | 3,167.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
DALDA TFA
DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant …
Formula:
C30H45N9O5·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
611.74 (free base)
Ref: TM-T80086
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Sonepcizumab
CAS:1031360-18-5
Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.
Purity:
SDS-PAGE:95% SEC-HPLC:98.90%
Color and Shape:
Liquid
Molecular weight:
146.43 kDa
Ref: TM-T76828
| 1mg | 269.00 € | ||
| 5mg | 616.00 € | ||
| 10mg | 829.00 € | ||
| 25mg | 1,255.00 € | ||
| 50mg | 1,691.00 € | ||
| 100mg | 2,277.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Galanin (1-13)-Neuropeptide Y (25-36) amide
CAS:147138-51-0
Galanin (1-13)-Neuropeptide Y (25-36) amide exhibits high-affinity binding to galanin receptors, similar to that of …
Formula:
C136H209N41O34
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2962.37
Ref: TM-T80143
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
![[(pF)Phe4]Nociceptin(1-13)NH2 acetate](https://static.cymitquimica.com/products/TM/thumb/TP1885L1.jpg)
[(pF)Phe4]Nociceptin(1-13)NH2 acetate
[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and …
Formula:
C63H103FN22O17
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
1459.63
Ref: TM-TP1885L1
| 1mg | 304.00 € | ||
| 2mg | 457.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 1,031.00 € | ||
| 25mg | 1,533.00 € | ||
| 50mg | 2,079.00 € | ||
| 100mg | 2,720.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
![[Orn8]-Urotensin II acetate](https://static.cymitquimica.com/products/TM/thumb/T37527L.jpg)
[Orn8]-Urotensin II acetate
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.
Formula:
C65H87N13O20S2
Purity:
98.63%
Color and Shape:
Liquid
Molecular weight:
1434.59
Ref: TM-T37527L
| 1mg | 185.00 € | ||
| 5mg | 415.00 € | ||
| 10mg | 613.00 € | ||
| 25mg | 937.00 € | ||
| 50mg | 1,309.00 € | ||
| 100mg | 1,764.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Neurokinin A(4-10)
CAS:97559-35-8
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
Formula:
C34H54N8O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
766.91
Ref: TM-T7559
| 1mg | 123.00 € | ||
| 5mg | 243.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 850.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
![[D-Ala2]leucine-enkephalin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1367L.jpg)
[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study …
Formula:
C31H43N5O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
629.65
Ref: TM-TP1367L
| 5mg | 55.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 349.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
![[DPro10] Dynorphin A (1-11)acetate,porcine](https://static.cymitquimica.com/products/TM/thumb/T76341L.jpg)
[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value …
Formula:
C65H107N21O15
Purity:
99.05%
Color and Shape:
Soild
Molecular weight:
1422.7
Ref: TM-T76341L
| 1mg | 60.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 646.00 € | ||
| 500mg | 1,364.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Mogamulizumab
CAS:1159266-37-1
Mogamulizumab is a monoclonal antibody targeting CC chemokine receptor 4 with anticancer effects, used in …
Purity:
SDS-PAGE:97.3%;SEC-HPLC:99.4%
Color and Shape:
Liquid
Molecular weight:
146.43 kDa
Ref: TM-T76782
| 1mg | 445.00 € | ||
| 5mg | 916.00 € | ||
| 10mg | 1,281.00 € | ||
| 25mg | 1,839.00 € | ||
| 50mg | 2,591.00 € | ||
| 100mg | 3,533.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
GB-6
CAS:2413262-74-3
GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), …
Formula:
C32H45N11O8
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
711.77
Ref: TM-T80266
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Samidorphan HCl
CAS:2328045-02-7
Samidorphan HCl is an orally active and highly potent modulator of the opioid system that …
Formula:
C21H27ClN2O4
Purity:
98.25% - 99.60%
Color and Shape:
Soild
Molecular weight:
406.9
Ref: TM-T67888L
| 1mg | 162.00 € | ||
| 5mg | 386.00 € | ||
| 10mg | 573.00 € | ||
| 25mg | 909.00 € | ||
| 50mg | 1,225.00 € | ||
| 100mg | 1,652.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist …
Formula:
C37H47Cl2N5O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
680.71
Ref: TM-T79547
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Galcanezumab
CAS:1578199-75-3
Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.
Purity:
> 95%
Color and Shape:
Liquid
Molecular weight:
144.08 kDa
Ref: TM-T76682
| 1mg | 125.00 € | ||
| 5mg | 370.00 € | ||
| 10mg | 594.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,233.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Drinabant
CAS:358970-97-5
Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.
Formula:
C23H20Cl2F2N2O2S
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
497.38
Ref: TM-T21861
| 1mg | 85.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 585.00 € | ||
| 100mg | 791.00 € | ||
| 500mg | 1,588.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Isobutyryl-L-carnitine
CAS:25518-49-4
Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a …
Formula:
C11H21NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
231.29
Ref: TM-T19381
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning …
Formula:
C24H29ClF3N5O5S
Purity:
96.67%
Color and Shape:
Soild
Molecular weight:
592.03
Ref: TM-T67972L
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
