G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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MCUF-651
CAS:2747162-85-0
MCUF-651 is a guanylyl cyclase A receptor positive allosteric modulators, EC50=0.45 μM.
Formula:
C17H22F2N4OS
Purity:
99.57%
Color and Shape:
Soild
Molecular weight:
368.44
Ref: TM-T67734
| 1mg | 170.00 € | ||
| 1ml | 413.00 € | ||
| 5mg | 395.00 € | ||
| 10mg | 587.00 € | ||
| 25mg | 925.00 € | ||
| 50mg | 1,236.00 € | ||
| 100mg | 1,662.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Dynorphin B (1-9)
CAS:126050-26-8
Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its …
Formula:
C54H78N16O12
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1143.3
Ref: TM-T80463
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
N-0500 HCl
CAS:100935-99-7
N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.
Formula:
C15H22ClNO2
Purity:
98.3% - 98.42%
Color and Shape:
Solid
Molecular weight:
283.79
Ref: TM-T60107
| 1ml | 55.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 54.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
UCM-1306
CAS:2258608-78-3
UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive …
Formula:
C14H14FNO2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
279.33
Ref: TM-T67729
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 464.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SDF-1α (human)
CAS:1268129-65-2
SDF-1α (human) serves as a chemotactic agent for mononuclear cells through its interaction with the …
Formula:
C356H578N106O93S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
7959.34
Ref: TM-T80130
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.
Formula:
C20H26ClF3N4O2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
446.89
Ref: TM-T60047L
| 1mg | 41.00 € | ||
| 1ml | 98.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 227.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 482.00 € | ||
| 200mg | 661.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Dodoviscin A
CAS:1372527-25-7
Dodoviscin A: a potential agent for altering pigmentation, inhibits melanin synthesis; also promotes fat cell …
Formula:
C27H32O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.544
Ref: TM-TN3882
| 1ml | 1,171.00 € | ||
| 5mg | 774.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Leumorphin, human
CAS:88846-98-4
Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and …
Formula:
C150H224N42O46
Purity:
98%
Color and Shape:
Solid
Molecular weight:
3351.64
Ref: TM-T81938
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
NOX-6-18
CAS:898211-21-7
NOX-6-18 (GPR132-B-160) is a GPR132 antagonist with insulin-promoting activity and reduced weight gain.
Formula:
C18H17NO5S
Purity:
99.29%
Color and Shape:
Soild
Molecular weight:
359.4
Ref: TM-T83972
| 1mg | 75.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 809.00 € | ||
| 100mg | 1,290.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Serazapine
CAS:115313-22-9
Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment …
Formula:
C22H23N3O2
Purity:
98% - 99%
Color and Shape:
Solid
Molecular weight:
361.44
Ref: TM-T68142
| 1mg | 197.00 € | ||
| 5mg | 505.00 € | ||
| 10mg | 723.00 € | ||
| 25mg | 1,103.00 € | ||
| 50mg | 1,504.00 € | ||
| 100mg | 2,023.00 € | ||
| 500mg | 4,057.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB2R/FAAH modulator-3
CAS:2876918-67-9
CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.
Formula:
C22H31NO2
Purity:
99.02%
Color and Shape:
Soild
Molecular weight:
341.49
Ref: TM-T67747
| 1mg | 45.00 € | ||
| 1ml | 95.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,328.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for …
Formula:
C31H44N6O9
Purity:
98%
Color and Shape:
Soild
Molecular weight:
644.72
Ref: TM-T32511L
| 1mg | 185.00 € | ||
| 5mg | 422.00 € | ||
| 10mg | 637.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,630.00 € | ||
| 100mg | 2,449.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GLP-1 (9-36) amide
CAS:161748-29-4
GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
Formula:
C140H214N36O43
Purity:
97%
Color and Shape:
Solid
Molecular weight:
3089.41
Ref: TM-TP2252
| 1mg | 88.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 353.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 823.00 € | ||
| 100mg | 1,109.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Adrenomedullin (AM) (22-52), human acetate
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the …
Formula:
C161H256N46O50
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
3636.09
Ref: TM-TP1257L
| 1mg | 206.00 € | ||
| 5mg | 807.00 € | ||
| 10mg | 1,204.00 € | ||
| 25mg | 2,180.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Uroguanylin (human)
CAS:154525-25-4
Uroguanylin (human) serves as a natural ligand for the Guanylyl Cyclase C (GCC) receptor in …
Formula:
C64H102N18O26S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1667.86
Ref: TM-T80067
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB1R/AMPK modulator 1
Compound 38-S is an orally active CB1R/AMPK modulator with a K i of 0.81 nM …
Formula:
C25H22Cl2N6O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
557.45
Ref: TM-T79649
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Licoarylcoumarin
CAS:125709-31-1
Licoarylcoumarin inhibits cAMP phosphodiesterase, fights VRE bacteria, has anti-HIV properties, and blocks xanthine oxidase.
Formula:
C21H20O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
368.38
Ref: TM-TN4433
| 1ml | 869.00 € | ||
| 5mg | 850.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Eledoisin
CAS:69-25-0
Eledoisin (Eledone peptide) is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide …
Formula:
C54H85N13O15S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1188.4
Ref: TM-TP1177
| 1mg | 204.00 € | ||
| 5mg | 797.00 € | ||
| 10mg | 1,394.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PAR-4 Agonist Peptide, amide
CAS:352017-71-1
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
Formula:
C34H48N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.79
Ref: TM-T7623
| 1mg | 51.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 230.00 € | ||
| 25mg | 391.00 € | ||
| 50mg | 563.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
ITIC-4F
CAS:2097998-59-7
ITIC-4F: a postfullerene IDTT electron acceptor for high-efficiency PSCs, relevant in binary, ternary, and tandem …
Formula:
C94H78F4N4O2S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1499.92
Ref: TM-T19385
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
