G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Avexitide acetate
CAS:2051593-46-3
Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the …
Formula:
C155H246N40O53S
Purity:
96.64%
Color and Shape:
Liquid
Molecular weight:
3549.91
Ref: TM-TP2100L
| 1mg | 162.00 € | ||
| 5mg | 457.00 € | ||
| 10mg | 641.00 € | ||
| 25mg | 991.00 € | ||
| 50mg | 1,342.00 € | ||
| 100mg | 1,805.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial …
Formula:
C102H163N31O26
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
2239.58
Ref: TM-TP2075L
| 1mg | 303.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 1,033.00 € | ||
| 25mg | 1,838.00 € | ||
| 50mg | 2,755.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Formula:
C38H39ClFN3O12
Purity:
95%
Color and Shape:
Liquid
Molecular weight:
784.18
Ref: TM-T9579L
| 1mg | 181.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,738.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
L 152804
CAS:6508-43-6
L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese …
Formula:
C23H26O4
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
366.45
Ref: TM-T15679
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 174.00 € | ||
| 100mg | 253.00 € | ||
| 200mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMS-193885
CAS:186185-03-5
BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a …
Formula:
C33H42N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.71
Ref: TM-T14671
| 1mg | 34.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GSK270822A
CAS:864082-23-5
GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, …
Formula:
C24H20N4O2
Purity:
98.13% - 98.77%
Color and Shape:
Liquid
Molecular weight:
396.44
Ref: TM-T27467
| 1mg | 222.00 € | ||
| 5mg | 542.00 € | ||
| 10mg | 721.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,461.00 € | ||
| 100mg | 1,964.00 € | ||
| 1mL*10mM (DMSO) | 564.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GV-150013X
CAS:151386-96-8
GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKi
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Soild
Molecular weight:
534.65
Ref: TM-T27503L
| 1mg | 183.00 € | ||
| 5mg | 444.00 € | ||
| 10mg | 608.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,235.00 € | ||
| 100mg | 1,625.00 € | ||
| 1mL*10mM (DMSO) | 638.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Seglitide acetate
CAS:99248-33-6
Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.
Formula:
C46H60N8O9
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
869.02
Ref: TM-T28743
| 1mg | 111.00 € | ||
| 2mg | 159.00 € | ||
| 5mg | 247.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 763.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,392.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Quipazine dimaleate
CAS:150323-78-7
Quipazine dimaleate is a selective 5-HT3 agonist.
Formula:
C21H23N3O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
445.42
Ref: TM-T23212
| 10mg | 35.00 € | ||
| 25mg | 52.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Deltorphin
CAS:119975-64-3
Deltorphin (Dermenkephalin) is Isolated from the skin of Phyllomedusa Sauvage. It also has an affinity …
Formula:
C44H62N10O10S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
955.15
Ref: TM-T20166
| 1mg | 167.00 € | ||
| 5mg | 291.00 € | ||
| 10mg | 556.00 € | ||
| 25mg | 888.00 € | ||
| 50mg | 1,198.00 € | ||
| 100mg | 1,606.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GRK2-IN-1 hydrochloride (2055990-90-2 free base)
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 …
Formula:
C24H26ClFN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
488.94
Ref: TM-T13714L
| 1mg | 106.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 294.00 € | ||
| 10mg | 459.00 € | ||
| 25mg | 824.00 € | ||
| 50mg | 1,372.00 € | ||
| 100mg | 1,870.00 € | ||
| 200mg | To inquire | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 316.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
W140 HBr
CAS:1246817-25-3
[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.
Formula:
C16H28BrN2O4P
Purity:
99.34%
Color and Shape:
Soild
Molecular weight:
423.28
Ref: TM-T60204
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
FSCPX
CAS:156547-56-7
FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting …
Formula:
C23H27FN4O6S
Purity:
98.00%
Color and Shape:
Liquid
Molecular weight:
506.55
Ref: TM-T39039
| 1mg | 176.00 € | ||
| 5mg | 446.00 € | ||
| 10mg | 668.00 € | ||
| 25mg | 1,135.00 € | ||
| 50mg | 1,516.00 € | ||
| 100mg | 2,037.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Litoxetine HCl
Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles …
Formula:
C16H20ClNO
Purity:
98.98% - 99.19%
Color and Shape:
Soild
Molecular weight:
277.79
Ref: TM-T67956L
| 1mg | 95.00 € | ||
| 5mg | 213.00 € | ||
| 10mg | 319.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,078.00 € | ||
| 1mL*10mM (DMSO) | 207.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Vibozilimod
CAS:1403232-33-6
Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .
Formula:
C29H36ClN3O5
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
542.07
Ref: TM-T38826
| 1mg | 74.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 223.00 € | ||
| 25mg | 387.00 € | ||
| 50mg | 559.00 € | ||
| 100mg | 765.00 € | ||
| 200mg | 1,012.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CB2R/FAAH modulator-1
CAS:928892-60-8
CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. …
Formula:
C24H27NO2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
361.48
Ref: TM-T67896
| 1mg | 113.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 552.00 € | ||
| 50mg | 772.00 € | ||
| 100mg | 1,053.00 € | ||
| 500mg | 2,106.00 € | ||
| 1mL*10mM (DMSO) | 262.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Balixafortide
CAS:1051366-32-5
Balixafortide (POL6326), a potent CXCR4 blocker with IC50 < 10 nM, mobilizes HSPCs and is anti-cancer, …
Formula:
C84H118N24O21S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1864.14
Ref: TM-TP2141L
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Orforglipron
CAS:2212020-52-3
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist …
Formula:
C48H48F2N10O5
Purity:
99.15% - 99.61%
Color and Shape:
Solid
Molecular weight:
882.96
Ref: TM-T11408
| 1mg | 239.00 € | ||
| 5mg | 587.00 € | ||
| 10mg | 922.00 € | ||
| 25mg | 1,848.00 € | ||
| 50mg | 2,499.00 € | ||
| 100mg | 3,378.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in …
Formula:
C52H77N15O14
Purity:
99.46%
Color and Shape:
Liquid
Molecular weight:
1136.26
Ref: TM-T36442L
| 1mg | 87.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 643.00 € | ||
| 100mg | 919.00 € | ||
| 500mg | 1,791.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Samelisant
CAS:1394808-82-2
Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.
Formula:
C21H31N3O3
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
373.49
Ref: TM-T9770
| 1mg | 111.00 € | ||
| 2mg | 163.00 € | ||
| 5mg | 275.00 € | ||
| 10mg | 440.00 € | ||
| 25mg | 724.00 € | ||
| 50mg | 1,015.00 € | ||
| 100mg | 1,357.00 € | ||
| 500mg | 2,683.00 € | ||
| 1mL*10mM (DMSO) | 282.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
