G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PF-06478939 TFA
PF-06478939 TFA is a peptide that acts as a non-brain-penetrating agonist at the oxytocin (OT) …
Formula:
C78H134N14O22S2·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Ref: TM-T79174
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[Deamino-Pen1,Val4,D-Arg8]-vasopressin](https://static.cymitquimica.com/products/TM/thumb/T83501.jpg)
[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:64158-84-5
[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).
Formula:
C48H69N13O11S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1068.27
Ref: TM-T83501
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Pro8-Oxytocin
CAS:24327-19-3
Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR …
Formula:
C42H62N12O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
991.14
Ref: TM-T80133
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(1S,2R)-2-PCCA
(1S,2R)-2-PCCA is a novel and potent small molecule GPR88 receptor agonist with an EC50 value …
Formula:
C30H39Cl2N3O
Purity:
99.34%
Color and Shape:
Soild
Molecular weight:
528.56
Ref: TM-T13423L
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € | ||
| 100mg | 1,803.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
DALDA TFA
DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant …
Formula:
C30H45N9O5·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
611.74 (free base)
Ref: TM-T80086
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Galanin (1-13)-Neuropeptide Y (25-36) amide
CAS:147138-51-0
Galanin (1-13)-Neuropeptide Y (25-36) amide exhibits high-affinity binding to galanin receptors, similar to that of …
Formula:
C136H209N41O34
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2962.37
Ref: TM-T80143
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Sergliflozin A
CAS:360775-96-8
Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It …
Formula:
C20H24O7
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
376.4
Ref: TM-T68174
| 1mg | 108.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 609.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,348.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Gevotroline
CAS:107266-06-8
Gevotroline, a chemical in palm wine that can be used to treat psychosis, is a …
Formula:
C19H20FN3
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
309.38
Ref: TM-T68080
| 1mg | 87.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,007.00 € | ||
| 500mg | 2,042.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formula:
C141H221N33O42S
Purity:
96.52%
Color and Shape:
Solid
Molecular weight:
3082.52
Ref: TM-T38193L
| 1mg | 111.00 € | ||
| 2mg | 157.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 355.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,016.00 € | ||
| 200mg | 1,354.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[Des-Arg9]-Bradykinin](https://static.cymitquimica.com/products/TM/thumb/T7645.jpg)
[Des-Arg9]-Bradykinin
CAS:15958-92-6
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
Formula:
C44H61N11O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
904.02
Ref: TM-T7645
| 5mg | 252.00 € | ||
| 10mg | 444.00 € | ||
| 25mg | 936.00 € | ||
| 50mg | 1,470.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GB-6
CAS:2413262-74-3
GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), …
Formula:
C32H45N11O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
711.77
Ref: TM-T80266
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
EP4-IN-1
CAS:2455480-28-9
EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.
Formula:
C27H24N2O4
Purity:
100%
Color and Shape:
Soild
Molecular weight:
440.49
Ref: TM-T77699
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist …
Formula:
C37H47Cl2N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.71
Ref: TM-T79547
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.
Formula:
C33H35F3N6O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
620.66
Ref: TM-T11671
| 1ml | 763.00 € | ||
| 2mg | 374.00 € | ||
| 5mg | 560.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[(pF)Phe4]Nociceptin(1-13)NH2 acetate](https://static.cymitquimica.com/products/TM/thumb/TP1885L1.jpg)
[(pF)Phe4]Nociceptin(1-13)NH2 acetate
[(pF)Phe4]Nociceptin(1-13)NH2 acetate is a selective agonist of NOP receptor with a pKi of 10.68 and …
Formula:
C63H103FN22O17
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
1459.63
Ref: TM-TP1885L1
| 1mg | 304.00 € | ||
| 2mg | 457.00 € | ||
| 5mg | 684.00 € | ||
| 10mg | 1,031.00 € | ||
| 25mg | 1,533.00 € | ||
| 50mg | 2,079.00 € | ||
| 100mg | 2,720.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[Orn8]-Urotensin II acetate](https://static.cymitquimica.com/products/TM/thumb/T37527L.jpg)
[Orn8]-Urotensin II acetate
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.
Formula:
C65H87N13O20S2
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
1434.59
Ref: TM-T37527L
| 1mg | 182.00 € | ||
| 1ml | 873.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,726.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MK-3207 Hydrochloride
CAS:957116-20-0
MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 …
Formula:
C31H29F2N5O3·HCl
Purity:
98%
Color and Shape:
Solid
Molecular weight:
594.05
Ref: TM-T6590
| 5mg | To inquire | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 1ml*10 (DMSO) | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning …
Formula:
C24H29ClF3N5O5S
Purity:
96.67%
Color and Shape:
Soild
Molecular weight:
592.03
Ref: TM-T67972L
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
FGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K …
Formula:
C33H36N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
520.66
Ref: TM-T79312
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is …
Formula:
C42H61N11O19
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1024.01
Ref: TM-TP1452L1
| 1mg | 251.00 € | ||
| 5mg | 513.00 € | ||
| 10mg | 777.00 € | ||
| 25mg | 1,398.00 € | ||
| 50mg | 2,095.00 € | ||
| 100mg | 3,143.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
