G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CB2 receptor agonist 2
CAS:1314230-75-5
CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.
Formula:
C30H36N2O4
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
488.62
Ref: TM-T22009
| 1mg | 116.00 € | ||
| 2mg | 170.00 € | ||
| 5mg | 266.00 € | ||
| 10mg | 391.00 € | ||
| 25mg | 615.00 € | ||
| 50mg | 827.00 € | ||
| 100mg | 1,111.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
S1R agonist 2 hydrochloride
Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 …
Formula:
C21H28ClNO
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
345.91
Ref: TM-T78087
| 2mg | 96.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
SLB1122168 formic
SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of …
Formula:
C23H37N3O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
403.56
Ref: TM-T78160
| 2mg | 128.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
TUG-499
CAS:1206629-08-4
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 …
Formula:
C16H11Cl2NO2
Purity:
99.59%
Color and Shape:
Soild
Molecular weight:
320.17
Ref: TM-T60184
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 279.00 € | ||
| 200mg | 395.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used …
Formula:
C21H26NO10P
Purity:
95.50%
Color and Shape:
Soild
Molecular weight:
483.41
Ref: TM-T68132L
| 1mg | 185.00 € | ||
| 5mg | 409.00 € | ||
| 10mg | 605.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,293.00 € | ||
| 100mg | 1,738.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
JHU 75528
CAS:947696-17-5
JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can …
Formula:
C23H21Cl2N5O2
Purity:
99.97%
Color and Shape:
Liquid
Molecular weight:
470.35
Ref: TM-T77634
| 1mg | 185.00 € | ||
| 5mg | 409.00 € | ||
| 10mg | 605.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,293.00 € | ||
| 100mg | 1,738.00 € | ||
| 500mg | 3,496.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
AT-121 hydrochloride
CAS:2099681-71-5
AT-121 hydrochloride: dual nociception/mu-opioid agonist, Ki 3.67/16.49 nM, safe, non-addictive pain reliever with analgesic effects.
Formula:
C24H39ClN4O3S
Purity:
100% - 97.28%
Color and Shape:
Liquid
Molecular weight:
499.11
Ref: TM-T39529
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
2-PCCA hydrochloride
CAS:1609563-70-3
2-PCCA hydrochloride, a racemate, is a potent and selective GPR88 receptor agonist showing inhibition of …
Formula:
C30H39Cl2N3O
Purity:
99.65% - 99.96%
Color and Shape:
Soild
Molecular weight:
528.56
Ref: TM-T80666
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € | ||
| 500mg | 3,734.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Oxmetidine
CAS:72830-39-8
Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular …
Formula:
C19H21N5O3S
Purity:
99.67%
Color and Shape:
Liquid
Molecular weight:
399.47
Ref: TM-T68122
| 1mg | 378.00 € | ||
| 5mg | 895.00 € | ||
| 10mg | 1,216.00 € | ||
| 25mg | 1,786.00 € | ||
| 50mg | 2,442.00 € | ||
| 100mg | 3,287.00 € | ||
| 500mg | 6,603.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Retatrutide sodium salt
Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study …
Purity:
99.97%
Color and Shape:
Soild
Ref: TM-T76279L1
| 1mg | 235.00 € | ||
| 5mg | 590.00 € | ||
| 10mg | 948.00 € | ||
| 25mg | 1,396.00 € | ||
| 50mg | 1,890.00 € | ||
| 100mg | 2,555.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Delequamine
CAS:119905-05-4
Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability …
Formula:
C18H26N2O3S
Purity:
98.75%
Color and Shape:
Liquid
Molecular weight:
350.48
Ref: TM-T68051
| 1mg | 245.00 € | ||
| 5mg | 615.00 € | ||
| 10mg | 873.00 € | ||
| 25mg | 1,311.00 € | ||
| 50mg | 1,768.00 € | ||
| 100mg | 2,365.00 € | ||
| 500mg | 4,684.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
![[D-Trp34]-Neuropeptide Y Acetate](https://static.cymitquimica.com/products/TM/thumb/TP1984L.jpg)
[D-Trp34]-Neuropeptide Y Acetate
[D-Trp34]-Neuropeptide Y Acetate is a potent Y5 receptor agonist that increases rat food intake; less …
Formula:
C198H293N55O58
Purity:
99.73%
Color and Shape:
Soild
Molecular weight:
4371.78
Ref: TM-TP1984L
| 1mg | 185.00 € | ||
| 5mg | 427.00 € | ||
| 10mg | 642.00 € | ||
| 25mg | 1,096.00 € | ||
| 50mg | 1,644.00 € | ||
| 100mg | 2,465.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
GLP-1R Agonist DMB
CAS:281209-71-0
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 …
Formula:
C13H15Cl2N3O2S
Purity:
99.52%
Color and Shape:
Liquid
Molecular weight:
348.25
Ref: TM-T36579
| 1mg | 51.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 236.00 € | ||
| 25mg | 404.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
CGRP 8-37 (rat)
CAS:129121-73-9
CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects …
Formula:
C138H224N42O41
Purity:
99.28%
Color and Shape:
Solid
Molecular weight:
3127.51
Ref: TM-TP1323
| 1mg | 273.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
DF-1012 FA
DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study …
Formula:
C17H22N4O3
Purity:
99.13% - 99.61%
Color and Shape:
Liquid
Molecular weight:
330.382
Ref: TM-T27158L
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Neuropeptide AF (human) acetate
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, …
Purity:
99.89%
Color and Shape:
Soild
Ref: TM-TP1082L
| 1mg | 172.00 € | ||
| 5mg | 427.00 € | ||
| 10mg | 630.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,320.00 € | ||
| 100mg | 1,786.00 € | ||
| 500mg | 3,600.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
Des His1, Glu8 Exendin-4
Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose …
Formula:
C179H277N47O59S
Purity:
99.92%
Color and Shape:
Liquid
Molecular weight:
4063.46
Ref: TM-T76291
| 1mg | 235.00 € | ||
| 5mg | 515.00 € | ||
| 10mg | 772.00 € | ||
| 25mg | 1,311.00 € | ||
| 50mg | 1,967.00 € | ||
| 100mg | 2,650.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
CB2R/FAAH modulator-2
CAS:2876918-68-0
CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.
Formula:
C24H33NO2
Purity:
99.52%
Color and Shape:
Soild
Molecular weight:
367.52
Ref: TM-T67745
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 430.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
2'-Hydroxydaidzein
CAS:7678-85-5
2'-Hydroxydaidzein is an isoflavonoid phytonutrient found in plant species, when a natural compound. 2'-Hydroxydaidzein has …
Formula:
C15H10O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
270.24
Ref: TM-TN2766
| 1mg | To inquire |
Estimated delivery in United States, on Monday 31 Mar 2025
Nelivaptan
CAS:439687-69-1
Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective …
Formula:
C30H32ClN3O8S
Purity:
98% - 98.39%
Color and Shape:
Solid
Molecular weight:
630.11
Ref: TM-T28153
| 1mg | 78.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 210.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 517.00 € | ||
| 100mg | 745.00 € | ||
| 500mg | 1,549.00 € |
Estimated delivery in United States, on Monday 31 Mar 2025
