G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
Formula:
C23H27F3N2O3
Purity:
98.10%
Color and Shape:
Soild
Molecular weight:
436.47
Ref: TM-T68023L
| 1mg | 115.00 € | ||
| 5mg | 245.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 562.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
CB1R/AMPK modulator 1
Compound 38-S is an orally active CB1R/AMPK modulator with a K i of 0.81 nM …
Formula:
C25H22Cl2N6O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
557.45
Ref: TM-T79649
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Mar 2025
NOX-6-18
CAS:898211-21-7
NOX-6-18 (GPR132-B-160) is a GPR132 antagonist with insulin-promoting activity and reduced weight gain.
Formula:
C18H17NO5S
Purity:
99.29%
Color and Shape:
Soild
Molecular weight:
359.4
Ref: TM-T83972
| 1mg | 74.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 810.00 € | ||
| 100mg | 1,293.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Upidosin
CAS:152735-23-4
Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.
Formula:
C31H33N3O4
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
511.61
Ref: TM-T9762
| 5mg | 44.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 129.00 € | ||
| 100mg | 187.00 € | ||
| 200mg | 281.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in …
Formula:
C52H77N15O14
Purity:
99.46%
Color and Shape:
Liquid
Molecular weight:
1136.26
Ref: TM-T36442L
| 1mg | 87.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 439.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 919.00 € | ||
| 500mg | 1,833.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
PAR-4 Agonist Peptide, amide
CAS:352017-71-1
PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
Formula:
C34H48N8O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
680.79
Ref: TM-T7623
| 1mg | 90.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 398.00 € | ||
| 50mg | 567.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Phoenixin-14
CAS:1415039-79-0
Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH …
Formula:
C75H110N18O20
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1583.78
Ref: TM-T80422
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Semaglutide TFA
Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels …
Formula:
C189H290F3N45O61
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
4225.6482
Ref: TM-T12878
| 1mg | 220.00 € | ||
| 5mg | 762.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
S1R agonist 2
CAS:150085-21-5
S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for …
Formula:
C21H27NO
Purity:
99.04%
Color and Shape:
Liquid
Molecular weight:
309.45
Ref: TM-T72059
| 2mg | 40.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 248.00 € | ||
| 100mg | 366.00 € | ||
| 200mg | 517.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Saterinone
CAS:102669-89-6
Saterinone: PDE III inhibitor, α-1-adrenoceptor antagonist, vasodilator, used for acute chronic heart failure, IC50 2.3x10^-5 …
Formula:
C27H30N4O4
Purity:
98.23%
Color and Shape:
Liquid
Molecular weight:
474.55
Ref: TM-T68138
| 1mg | 94.00 € | ||
| 5mg | 221.00 € | ||
| 10mg | 335.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 979.00 € | ||
| 200mg | 1,320.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
(+/-)-Pinocembrin
CAS:68745-38-0
(+/-)-Pinocembrin (NSC-43318), a natural product from axillary pines, is a GPR120 ligand that promotes wound …
Formula:
C15H12O4
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
256.25
Ref: TM-TN2077
| 1mg | 47.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 557.00 € | ||
| 500mg | 1,169.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Spiroglumide
CAS:137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 …
Formula:
C21H26Cl2N2O4
Purity:
98.34%
Color and Shape:
Soild
Molecular weight:
441.35
Ref: TM-T68016
| 1mg | 94.00 € | ||
| 5mg | 221.00 € | ||
| 10mg | 335.00 € | ||
| 25mg | 537.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Orforglipron
CAS:2212020-52-3
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist …
Formula:
C48H48F2N10O5
Purity:
99.15% - 99.61%
Color and Shape:
Solid
Molecular weight:
882.96
Ref: TM-T11408
| 1mg | 244.00 € | ||
| 5mg | 597.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,882.00 € | ||
| 50mg | 2,593.00 € | ||
| 100mg | 3,505.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Balixafortide
CAS:1051366-32-5
Balixafortide (POL6326), a potent CXCR4 blocker with IC50 < 10 nM, mobilizes HSPCs and is anti-cancer, …
Formula:
C84H118N24O21S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1864.14
Ref: TM-TP2141L
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Mar 2025
MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity …
Formula:
C24H26F3N3O4
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
477.48
Ref: TM-T12054L
| 1mg | 185.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,035.00 € | ||
| 25mg | 1,568.00 € | ||
| 50mg | 2,118.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Dalcotidine
CAS:120958-90-9
Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, …
Formula:
C18H29N3O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
319.44
Ref: TM-T31195
| 1mg | 94.00 € | ||
| 5mg | 205.00 € | ||
| 10mg | 303.00 € | ||
| 25mg | 490.00 € | ||
| 1mL*10mM (DMSO) | 205.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Adrenocorticotropic Hormone (ACTH) (4-10), human
CAS:4037-01-8
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
Formula:
C44H59N13O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
962.09
Ref: TM-T7627
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 227.00 € | ||
| 50mg | 294.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Val9-Oxytocin
CAS:1021701-88-1
Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete …
Formula:
C46H72N12O12S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1049.27
Ref: TM-T80136
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 12 Mar 2025
Seganserin
CAS:87729-89-3
Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.
Formula:
C29H27F2N3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
471.54
Ref: TM-T68141
| 1mg | 185.00 € | ||
| 5mg | 409.00 € | ||
| 10mg | 605.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,293.00 € | ||
| 100mg | 1,738.00 € | ||
| 500mg | 3,496.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
N-0500 HCl
CAS:100935-99-7
N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.
Formula:
C15H22ClNO2
Purity:
98.3% - 98.42%
Color and Shape:
Liquid
Molecular weight:
283.79
Ref: TM-T60107
| 5mg | 35.00 € | ||
| 10mg | 55.00 € |
Estimated delivery in United States, on Wednesday 12 Mar 2025
