G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CAY10678
CAS:1268709-57-4
CAY10678 is an mPGES-1 inhibitor that inhibits PD-1.CAY10678 reduces collagen deposition and T-cell depletion, and …
Formula:
C23H34N4O
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
382.54
Ref: TM-T38369
| 1mg | 52.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 523.00 € | ||
| 100mg | 737.00 € | ||
| 500mg | 1,515.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SB 216641
CAS:170230-39-4
SB 216641 is a 5-HT (1B/1D) antagonist with anxiolytic activity for the study of anxiety …
Formula:
C28H30N4O4
Purity:
98.01%
Color and Shape:
Liquid
Molecular weight:
486.56
Ref: TM-T85323
| 1mg | 196.00 € | ||
| 5mg | 486.00 € | ||
| 10mg | 682.00 € | ||
| 25mg | 1,064.00 € | ||
| 50mg | 1,467.00 € | ||
| 100mg | 1,878.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
TAK-448 acetate
CAS:1470374-22-1
TAK-448 acetate (MVT-602 acetate) is a KISS1R agonist, a synthetic peptide similar to kisspeptin.
Formula:
C60H84N16O16
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
1285.41
Ref: TM-TP1093
| 1mg | 94.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 601.00 € | ||
| 50mg | 843.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Pobilukast
CAS:107023-41-6
Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study …
Formula:
C26H34O5S
Purity:
99.65% - 99.84%
Color and Shape:
Solid
Molecular weight:
458.61
Ref: TM-T68130
| 1mg | 317.00 € | ||
| 5mg | 751.00 € | ||
| 10mg | 1,065.00 € | ||
| 25mg | 1,584.00 € | ||
| 50mg | 2,068.00 € | ||
| 100mg | 2,647.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PF-06655075 TFA
PF-06655075 (TFA) is the trifluoroacetic acid (TFA) salt of PF-06655075, a novel, non-brain-penetrant oxytocin receptor …
Purity:
98%
Ref: TM-T81501
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
KB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8
Formula:
C24H32N2O8
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
476.52
Ref: TM-T62396L
| 5mg | 62.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 189.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Misoprostol
CAS:59122-46-2
Misoprostol is a useful organic compound for research related to life sciences. The catalog number …
Formula:
C22H38O5
Purity:
100%
Color and Shape:
Water-Soluble Viscous Liquid
Molecular weight:
382.53
Ref: TM-T2573
| 1mg | 59.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 551.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
DPDPE
CAS:88373-73-3
DPDPE is selective δ-opioid receptor agonist peptide.
Formula:
C30H39N5O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
645.79
Ref: TM-TP2036
| 1mg | 376.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GPCR agonist-2
CAS:291528-35-3
GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.
Formula:
C10H10N2O4
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
222.2
Ref: TM-T60074
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
TDI-10229
CAS:2810887-45-5
TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.
Formula:
C16H16ClN5
Purity:
97.77%
Color and Shape:
Soild
Molecular weight:
313.78
Ref: TM-T64355
| 1mg | 41.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 903.00 € | ||
| 200mg | 1,246.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
DuP 747 HCl
CAS:115904-74-0
DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two …
Formula:
C24H29Cl3N2O2
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
483.86
Ref: TM-T25354L
| 1mg | 241.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,279.00 € | ||
| 50mg | 1,727.00 € | ||
| 100mg | 2,334.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
![4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-me…](https://static.cymitquimica.com/products/TM/thumb/T60126.jpg)
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine
CAS:2649012-21-3
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine is an enantiomeric
Formula:
C27H28ClFN2OS
Purity:
99.02%
Color and Shape:
Soild
Molecular weight:
483.04
Ref: TM-T60126
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 302.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] …
Formula:
C96H140N20O25S·xNH3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2006.32 (free base)
Ref: TM-T78096
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Octodrine
CAS:543-82-8
Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as …
Formula:
C8H19N
Purity:
99.98%
Color and Shape:
Clear Colorless To Light Yellow Liquid
Molecular weight:
129.24
Ref: TM-T0043
| 1g | 77.00 € | ||
| 5g | 166.00 € | ||
| 500mg | 51.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has …
Purity:
98%
Ref: TM-T81798
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Adrenorphin
CAS:88377-68-8
Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C44H69N15O9S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
984.18
Ref: TM-T7567
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:71800-37-8
Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].
Formula:
C47H75N13O11
Purity:
98%
Color and Shape:
Solid
Molecular weight:
998.18
Ref: TM-T80117
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
BMS-903452
CAS:1339944-47-6
BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe …
Formula:
C21H19Cl2FN4O4S
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
513.37
Ref: TM-T67791
| 1mg | 149.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 510.00 € | ||
| 25mg | 766.00 € | ||
| 50mg | 1,035.00 € | ||
| 100mg | 1,398.00 € | ||
| 500mg | 2,739.00 € | ||
| 1mL*10mM (DMSO) | 426.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ABT 724 trihydrochloride
CAS:587870-77-7
ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.
Formula:
C17H22Cl3N5
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
402.75
Ref: TM-T22019
| 5mg | 39.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 272.00 € | ||
| 200mg | 405.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
UCM-1306
CAS:2258608-78-3
UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive …
Formula:
C14H14FNO2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
279.33
Ref: TM-T67729
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 464.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
