G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and …
Formula:
C77H112N20O15
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
1557.84
Ref: TM-T20413L
| 1mg | 127.00 € | ||
| 1ml | 738.00 € | ||
| 5mg | 322.00 € | ||
| 10mg | 517.00 € | ||
| 25mg | 835.00 € | ||
| 50mg | 1,133.00 € | ||
| 100mg | 1,531.00 € | ||
| 500mg | 3,044.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Romergoline 2HCl
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's …
Formula:
C20H24Cl2N4O2
Purity:
100% - 98.33%
Color and Shape:
Soild
Molecular weight:
423.34
Ref: TM-T71707L
| 1mg | 181.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 639.00 € | ||
| 25mg | 998.00 € | ||
| 50mg | 1,376.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tiflucarbine
CAS:89875-86-5
Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity …
Formula:
C16H17FN2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
288.38
Ref: TM-T68162
| 1mg | 260.00 € | ||
| 5mg | 640.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,361.00 € | ||
| 50mg | 1,828.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP-related Peptide (human) (trifluoroacetate salt)
Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some …
Ref: TM-T36428
| 1mg | 839.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)
PACAP (6-27) is an antagonist for PACAP receptors with varying IC50s; blocks cAMP in neuroblastoma …
Ref: TM-T36427
| 500µg | 422.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tiaspirone hydrochloride
CAS:87691-92-7
Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.
Formula:
C24H33ClN4O2S
Purity:
99.98%
Color and Shape:
Soild
Molecular weight:
477.06
Ref: TM-T24885L
| 1mg | 185.00 € | ||
| 1ml | 47.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CSD-CH2(1,8)-NH2
CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of …
Formula:
C76H125N25O15S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1693.09
Ref: TM-T80421
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Besipirdine hydrochloride
CAS:130953-69-4
Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of …
Formula:
C16H18ClN3
Purity:
98.40%
Color and Shape:
Soild
Molecular weight:
287.79
Ref: TM-T26778L
| 1mg | 184.00 € | ||
| 5mg | 456.00 € | ||
| 10mg | 653.00 € | ||
| 25mg | 1,019.00 € | ||
| 50mg | 1,405.00 € | ||
| 100mg | 1,858.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PG 106 acetate
PG 106 acetate: Selective hMC3 receptor antagonist, IC50=210 nM; inactive on hMC5 and hMC4, EC50=9900 …
Formula:
C53H73N13O11
Purity:
98.24%
Color and Shape:
Solid
Molecular weight:
1068.23
Ref: TM-TP1952L
| 1mg | 101.00 € | ||
| 5mg | 328.00 € | ||
| 10mg | 468.00 € | ||
| 25mg | 708.00 € | ||
| 50mg | 944.00 € | ||
| 100mg | 1,292.00 € | ||
| 200mg | 1,722.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Xanthine amine congener trihydrochloride
CAS:2459963-12-1
Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, …
Formula:
C21H29ClN6O4
Purity:
97.85%
Color and Shape:
Solid
Molecular weight:
464.95
Ref: TM-T23535L
| 1mg | 73.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 327.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 648.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
2-Oleoylglycerol
CAS:3443-84-3
2-Oleoylglycerol is a lipid found in palm kernels that acts as a GPR119 agonist with …
Formula:
C21H40O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
356.54
Ref: TM-T37526
| 28mM*100 | 93.00 € | ||
| 28mM*2.5 | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
JPC0323
JPC0323 is a dual positive allosteric modulator of the 5-HT2C and 5-HT2A receptors, featuring on-target …
Formula:
C22H43NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
385.58
Ref: TM-T79524
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
E70K
E70K, a CXCL8 C-terminal peptide, features a lysine (K) substitution for glutamic acid (E) at …
Formula:
C108H178N34O28
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2400.78
Ref: TM-T80525
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
human GALP (3-32)
Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 …
Formula:
C137H213N43O38S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
3102.49
Ref: TM-T80516
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
5-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like …
Formula:
C17H22Cl2N6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
413.37
Ref: TM-T79325
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Pranazepide
CAS:150408-73-4
Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders …
Formula:
C26H19FN4O2
Purity:
98.20%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T34123
| 1mg | 513.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity …
Formula:
C24H26F3N3O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
477.48
Ref: TM-T12054L
| 1mg | 184.00 € | ||
| 5mg | 781.00 € | ||
| 10mg | 1,028.00 € | ||
| 25mg | 1,556.00 € | ||
| 50mg | 2,103.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tetrapeptide-1
CAS:1632354-04-1
Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as …
Formula:
C20H36N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
428.52
Ref: TM-T80202
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
[D-Pro2] Spantide I TFA
[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the …
Formula:
C75H108N20O13·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Ref: TM-T80031
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MRS7925
MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition …
Formula:
C20H26IN5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
511.36
Ref: TM-T79326
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
