G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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β-Endorphin (1-27) (human)
CAS:76622-84-9
β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid …
Formula:
C139H217N33O40S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
3022.47
Ref: TM-T80515
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
IRL-1620 acetate
IRL-1620 acetate is an effective and selective agonist of Endothelin B receptor (ETB) with a …
Formula:
C88H121N17O29
Purity:
96.64%
Color and Shape:
Solid
Molecular weight:
1881
Ref: TM-T15595L
| 1mg | 176.00 € | ||
| 5mg | 436.00 € | ||
| 10mg | 638.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,347.00 € | ||
| 100mg | 1,821.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
AMI-193
CAS:510-74-7
AMI-193 (Spiramide) is a selective 5-HT2 & D2 receptor antagonist with antipsychotic properties.
Formula:
C22H26FN3O2
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T21855
| 1ml | 50.00 € | ||
| 5mg | 45.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 310.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Ki16198
CAS:355025-13-7
Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. …
Formula:
C24H25ClN2O5S
Purity:
97.6%
Color and Shape:
Solid
Molecular weight:
488.98
Ref: TM-T6347
| 1ml | 58.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 254.00 € | ||
| 100mg | 368.00 € | ||
| 500mg | 799.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cortistatin-14
CAS:186901-48-4
Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.
Formula:
C81H114N20O18S2
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
1720.03
Ref: TM-TP1570
| 1mg | 97.00 € | ||
| 5mg | 374.00 € | ||
| 10mg | 671.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Avexitide acetate
CAS:2051593-46-3
Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the …
Formula:
C155H246N40O53S
Purity:
96.64%
Color and Shape:
Solid
Molecular weight:
3549.91
Ref: TM-TP2100L
| 1mg | 162.00 € | ||
| 5mg | 457.00 € | ||
| 10mg | 641.00 € | ||
| 25mg | 991.00 € | ||
| 50mg | 1,342.00 € | ||
| 100mg | 1,805.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Corticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.
Purity:
98.30%
Ref: TM-TP1144L
| 1mg | 143.00 € | ||
| 5mg | 465.00 € | ||
| 10mg | 694.00 € | ||
| 25mg | 1,246.00 € | ||
| 50mg | 1,854.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP-related Peptide (rat) (trifluoroacetate salt)
PRP, a 29-amino acid peptide in the secretin/glucagon family, is found in rat brain regions …
Color and Shape:
Solid
Ref: TM-T37435
| 1mg | 473.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cortistatin-8 acetate
Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.
Formula:
C49H72N12O11S2
Purity:
99.01%
Color and Shape:
Soild
Molecular weight:
1069.3
Ref: TM-TP2236L
| 1mg | 223.00 € | ||
| 5mg | 548.00 € | ||
| 10mg | 783.00 € | ||
| 25mg | 1,189.00 € | ||
| 50mg | 1,613.00 € | ||
| 100mg | 2,172.00 € | ||
| 500mg | 4,353.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Setmelanotide Acetate(920014-72-8 free base)
CAS:2759937-80-7
Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human …
Formula:
C51H72N18O11S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1177.35
Ref: TM-T12882L
| 1mg | 128.00 € | ||
| 1ml | 552.00 € | ||
| 5mg | 281.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 695.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,327.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cortistatin 14, human, rat acetate
Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows …
Formula:
C80H112N18O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1693.98
Ref: TM-TP1188L
| 1mg | 106.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 340.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 979.00 € | ||
| 200mg | 1,309.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tamsolusin Hydrochloride
CAS:80223-99-0
Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the …
Formula:
C20H29ClN2O5S
Purity:
99.92%
Color and Shape:
Soild
Molecular weight:
444.97
Ref: TM-T83965
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € | ||
| 100mg | 1,869.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Talastine
CAS:16188-61-7
Talastine is an antihistamine compound that can induce an allergic rash.
Formula:
C19H21N3O
Purity:
99.30% - 99.37%
Color and Shape:
Solid
Molecular weight:
307.39
Ref: TM-T68150
| 1mg | 91.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 289.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 728.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Lanepitant 2HCl
CAS:170508-05-1
Lanepitant 2HCl is a non-peptide neurokinin-1 receptor antagonist that can be used to study painful …
Formula:
C33H47Cl2N5O3
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
632.66
Ref: TM-T25616
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,025.00 € | ||
| 50mg | 1,413.00 € | ||
| 100mg | 1,869.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Ceruletide Ammonium acetate
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist.
Formula:
C60H77N13O23S2
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
1412.46
Ref: TM-T14932L
| 1mg | 234.00 € | ||
| 5mg | 476.00 € | ||
| 10mg | 691.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PF-06478939
PF-06478939 is a peptide that functions as an agonist at the oxytocin (OT) receptor and …
Formula:
C78H134N14O22S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1684.11
Ref: TM-T79173
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tizanidine
CAS:51322-75-9
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) …
Formula:
C9H8ClN5S
Purity:
99.75%
Color and Shape:
White Solid
Molecular weight:
253.71
Ref: TM-T7065
| 1ml | 46.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 104.00 € | ||
| 500mg | 247.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PF-06655075
PF-06655075 is a novel, non-brain-penetrant oxytocin receptor agonist that demonstrates enhanced selectivity for the oxytocin …
Formula:
C75H130N14O22S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1644.05
Ref: TM-T79172
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cericlamine
CAS:112922-55-1
Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.
Formula:
C12H17Cl2NO
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
262.18
Ref: TM-T68040
| 1mg | 125.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 446.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,380.00 € | ||
| 500mg | 2,759.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
EP3 antagonist 4
CAS:2408297-80-1
EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good …
Formula:
C22H20Cl3FN4O3S2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
577.91
Ref: TM-T77630
| 1mg | 184.00 € | ||
| 5mg | 405.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 1,044.00 € | ||
| 50mg | 1,580.00 € | ||
| 100mg | 2,388.00 € | ||
| 500mg | 5,254.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
