G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is …
Formula:
C42H61N11O19
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1024.01
Ref: TM-TP1452L1
| 1mg | 251.00 € | ||
| 5mg | 513.00 € | ||
| 10mg | 777.00 € | ||
| 25mg | 1,398.00 € | ||
| 50mg | 2,095.00 € | ||
| 100mg | 3,143.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Ezlopitant
CAS:147116-64-1
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and …
Formula:
C31H38N2O
Purity:
97.03%
Color and Shape:
Liquid
Molecular weight:
454.65
Ref: TM-T68068
| 1mg | 91.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 729.00 € | ||
| 100mg | 1,013.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
4-Thiouridine 5′-triphosphate disodium
CAS:68507-49-3
4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 …
Formula:
C9H11N2Na2O14P3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
546.19
Ref: TM-T79197
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Vibozilimod
CAS:1403232-33-6
Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .
Formula:
C29H36ClN3O5
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
542.07
Ref: TM-T38826
| 1mg | 74.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 223.00 € | ||
| 25mg | 387.00 € | ||
| 50mg | 559.00 € | ||
| 100mg | 765.00 € | ||
| 200mg | 1,012.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Losulazine
CAS:72141-57-2
Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.
Formula:
C27H22F4N4O3S
Purity:
99.80%
Color and Shape:
Liquid
Molecular weight:
558.55
Ref: TM-T68095
| 1mg | 92.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 725.00 € | ||
| 100mg | 1,013.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
(S, R)-LSN 3318839
CAS:2765539-92-0
(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
Formula:
C26H23Cl2N3O2
Purity:
99.57%
Color and Shape:
Soild
Molecular weight:
480.39
Ref: TM-T63166L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PF-03382792
CAS:1400811-63-3
PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.
Formula:
C23H32FN3O4
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
433.52
Ref: TM-T33940
| 1mg | 224.00 € | ||
| 5mg | 558.00 € | ||
| 10mg | 794.00 € | ||
| 25mg | 1,189.00 € | ||
| 50mg | 1,635.00 € | ||
| 100mg | 2,192.00 € | ||
| 500mg | 4,419.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
ITIC-4F
CAS:2097998-59-7
ITIC-4F: a postfullerene IDTT electron acceptor for high-efficiency PSCs, relevant in binary, ternary, and tandem …
Formula:
C94H78F4N4O2S4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1499.92
Ref: TM-T19385
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
(R)-CJ 11974
CAS:187281-35-2
(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.
Formula:
C31H38N2O
Purity:
97.03%
Color and Shape:
Soild
Molecular weight:
454.65
Ref: TM-T68068L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
FSCPX
CAS:156547-56-7
FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting …
Formula:
C23H27FN4O6S
Purity:
98.00%
Color and Shape:
Liquid
Molecular weight:
506.55
Ref: TM-T39039
| 1mg | 176.00 € | ||
| 5mg | 446.00 € | ||
| 10mg | 668.00 € | ||
| 25mg | 1,135.00 € | ||
| 50mg | 1,516.00 € | ||
| 100mg | 2,037.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
DPTN dihydrochloride
CAS:325767-87-1
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 …
Formula:
C22H20Cl2N4OS
Purity:
100%
Color and Shape:
Soild
Molecular weight:
459.39
Ref: TM-T72067
| 1mg | 50.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 162.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 524.00 € | ||
| 100mg | 738.00 € | ||
| 500mg | 1,557.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PZ-1922
PZ-1922 (Compound 16), able to cross the blood-brain barrier, is a dual antagonist for 5-HT6R …
Purity:
98%
Ref: TM-T81335
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Balixafortide TFA (1051366-32-5 free base)
Balixafortide TFA is a selective CXCR4 antagonist with IC50 < 10nM, over 1000x preference for CXCR4, …
Formula:
C82H113N22F3O23S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1896.05
Ref: TM-TP2141
| 5mg | 150.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 875.00 € | ||
| 100mg | To inquire | ||
| 200mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
W140 HBr
CAS:1246817-25-3
[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.
Formula:
C16H28BrN2O4P
Purity:
99.34%
Color and Shape:
Soild
Molecular weight:
423.28
Ref: TM-T60204
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
5-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only …
Formula:
C17H22F2N6O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
364.39
Ref: TM-T79684
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Panaxydol
CAS:72800-72-7
Panaxydol has anti-cancer activity, can inhibit the growth and apoptosis of cancer cells, the signaling …
Formula:
C17H24O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
260.37
Ref: TM-TN2039
| 1mg | 208.00 € | ||
| 5mg | 991.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Ki16198
CAS:355025-13-7
Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. …
Formula:
C24H25ClN2O5S
Purity:
97.6%
Color and Shape:
Solid
Molecular weight:
488.98
Ref: TM-T6347
| 5mg | 52.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 254.00 € | ||
| 100mg | 368.00 € | ||
| 500mg | 799.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Talquetamab
CAS:2226212-40-2
Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment …
Color and Shape:
Liquid
Molecular weight:
144.59 kDa
Ref: TM-T76882
| 1mg | 273.00 € | ||
| 2mg | 413.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 1,094.00 € | ||
| 25mg | 1,622.00 € | ||
| 50mg | 2,188.00 € | ||
| 100mg | 2,951.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
SB-408124
CAS:288150-92-5
SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x …
Formula:
C19H18F2N4O
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
356.37
Ref: TM-T6658
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 201.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
E70K
E70K, a CXCL8 C-terminal peptide, features a lysine (K) substitution for glutamic acid (E) at …
Formula:
C108H178N34O28
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2400.78
Ref: TM-T80525
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
