G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Mifentidine
CAS:83184-43-4
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric …
Formula:
C13H16N4
Purity:
100% - 99.20%
Color and Shape:
Solid
Molecular weight:
228.29
Ref: TM-T68100
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,390.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high …
Formula:
C20H19F3N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
388.39
Ref: TM-T79577
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PF-06655075 TFA
PF-06655075 (TFA) is the trifluoroacetic acid (TFA) salt of PF-06655075, a novel, non-brain-penetrant oxytocin receptor …
Purity:
98%
Ref: TM-T81501
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] …
Formula:
C96H140N20O25S·xNH3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2006.32 (free base)
Ref: TM-T78096
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Senktide acetate
Senktide acetate is a tachykinin NK3 receptor agonist that promotes the consolidation or expression of …
Formula:
C42H59N7O13S
Purity:
95%
Color and Shape:
Solid
Molecular weight:
902.02
Ref: TM-T7633L
| 1mg | 89.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 264.00 € | ||
| 25mg | 447.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 930.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Esprolol
CAS:396654-09-4
Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.
Formula:
C17H27NO4
Purity:
100% - 99.16%
Color and Shape:
Soild
Molecular weight:
309.4
Ref: TM-T27286L
| 1mg | 125.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,351.00 € | ||
| 500mg | 2,692.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(S)-(-)-Atenolol
CAS:93379-54-5
(S)-(-)-Atenolol has beta-adrenergic blocking effects.
Formula:
C14H22N2O3
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
266.34
Ref: TM-T35833
| 1mg | 73.00 € | ||
| 5mg | 151.00 € | ||
| 10mg | 213.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 763.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
15(R)-15-methyl Prostaglandin D2
CAS:210978-26-0
15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) is a synthetic analog of PGD2 and a CRTH2/DP2 receptor …
Formula:
C21H34O5
Color and Shape:
Solid
Molecular weight:
366.49
Ref: TM-T37264
| 1mg | 313.00 € | ||
| 500µg | 185.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Relenopride
CAS:1221416-43-8
YKP 10811 (Relenopride) is a novel 5-HT4 receptor partial agonist, which can be used to …
Formula:
C24H30ClFN4O4
Purity:
98.91% - 99.20%
Color and Shape:
Soild
Molecular weight:
492.97
Ref: TM-T83981
| 1mg | 125.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,351.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Cyclosomatostatin Acetate
Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and …
Formula:
C46H61N7O8
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
840.02
Ref: TM-T21567L
| 1mg | 145.00 € | ||
| 1ml | 548.00 € | ||
| 2mg | 243.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 548.00 € | ||
| 25mg | 814.00 € | ||
| 50mg | 1,090.00 € | ||
| 100mg | 1,475.00 € | ||
| 200mg | 1,988.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
VUF-11222
CAS:1414376-84-3
VUF-11222 is an agonist of high affinity non-peptide CXCR3 agonist (pKi = 7.2).
Formula:
C25H31BrIN
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
552.33
Ref: TM-T35085
| 1mg | 140.00 € | ||
| 2mg | 187.00 € | ||
| 5mg | 329.00 € | ||
| 10mg | 491.00 € | ||
| 25mg | 796.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,482.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
TCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin …
Formula:
C63H87N15O11·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1230.46 (free base)
Ref: TM-T80541
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![Des-Arg9-[Leu8]-Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb/T80072.jpg)
Des-Arg9-[Leu8]-Bradykinin acetate
CAS:115035-45-5
Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal …
Formula:
C43H67N11O12
Purity:
98%
Color and Shape:
Solid
Molecular weight:
930.06
Ref: TM-T80072
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PU-WS13 hydrobromide
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like …
Formula:
C17H21BrCl2N6S
Purity:
98%
Color and Shape:
Soild
Molecular weight:
492.26
Ref: TM-T5351L
| 1mg | 42.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 420.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
BF-1
CAS:518980-66-0
BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.
Formula:
C22H25NO2S
Purity:
100% - 99.25%
Color and Shape:
Solid
Molecular weight:
367.50
Ref: TM-T26781
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,423.00 € | ||
| 50mg | 1,869.00 € | ||
| 100mg | 2,605.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[Ala11,D-Leu15]-Orexin B acetate](https://static.cymitquimica.com/products/TM/thumb/TP1975L.jpg)
[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of …
Formula:
C122H210N44O37S
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
2917.31
Ref: TM-TP1975L
| 1mg | 492.00 € | ||
| 5mg | 1,107.00 € | ||
| 10mg | 1,660.00 € | ||
| 25mg | 2,988.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Oxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.
Formula:
C20H23N5O5S
Purity:
97.34%
Color and Shape:
Soild
Molecular weight:
445.49
Ref: TM-T68122L
| 1mg | 182.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Arotinolol hydrochloride
CAS:68377-91-3
Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.
Formula:
C15H22ClN3O2S3
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
408
Ref: TM-T30140
| 1mg | 52.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 546.00 € | ||
| 500mg | 1,161.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Brefonalol HCl
Brefonalol HCl, ADRA blocker for neurological/cardiovascular issues, treats angina, arrhythmias, hypertension.
Formula:
C22H29ClN2O2
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
388.93
Ref: TM-T30586L
| 1mg | 183.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,415.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
