G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Tolamolol
CAS:38103-61-6
Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of …
Formula:
C19H24N2O4
Purity:
97.58%
Color and Shape:
Solid
Molecular weight:
344.4
Ref: TM-T68164
| 1mg | 101.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 613.00 € | ||
| 100mg | 910.00 € | ||
| 500mg | 1,831.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values …
Formula:
C28H42N6O5
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
542.67
Ref: TM-T16738L
| 1mg | 63.00 € | ||
| 1ml | 162.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 315.00 € | ||
| 50mg | 451.00 € | ||
| 100mg | 622.00 € | ||
| 200mg | 838.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CI 169369
CAS:85273-96-7
CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and …
Formula:
C19H21ClN2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.9
Ref: TM-T84289
| 1mg | 199.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 692.00 € | ||
| 25mg | 1,080.00 € | ||
| 50mg | 1,489.00 € | ||
| 100mg | 1,907.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![5-Bromoimidazo[1,2-A]Pyrazine](https://static.cymitquimica.com/products/TM/thumb/T77641.jpg)
5-Bromoimidazo[1,2-A]Pyrazine
CAS:87597-26-0
5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.
Formula:
C6H4BrN3
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
198.02
Ref: TM-T77641
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,431.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Retatrutide
CAS:2381089-83-2
Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used …
Formula:
C221H342N46O68
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
4731.33
Ref: TM-T76279
| 1mg | 231.00 € | ||
| 5mg | 581.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,374.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,513.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PAR-4 Agonist Peptide, amide acetate
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
Formula:
C36H52N8O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
740.86
Ref: TM-T7623L
| 1mg | 96.00 € | ||
| 5mg | 287.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 833.00 € | ||
| 50mg | 1,249.00 € | ||
| 100mg | 1,873.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Homoeriodictyol
CAS:446-71-9
Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food …
Formula:
C16H14O6
Purity:
99.34% - 99.96%
Color and Shape:
Solid
Molecular weight:
302.28
Ref: TM-TN1740
| 1mg | 126.00 € | ||
| 5mg | 262.00 € | ||
| 10mg | 428.00 € | ||
| 25mg | 684.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
YNT-185
CAS:1804978-81-1
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values …
Formula:
C33H37N5O5S
Purity:
98.6%
Color and Shape:
Solid
Molecular weight:
615.74
Ref: TM-T39229
| 1mg | 65.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 446.00 € | ||
| 50mg | 717.00 € | ||
| 100mg | 975.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Meclinertant
CAS:146362-70-1
Meclinertant: selective NTS1 antagonist, blocks Ca2+ mobilization, with anxiolytic and anti-addictive properties.
Formula:
C32H31ClN4O5
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
587.07
Ref: TM-T16034
| 1mg | 86.00 € | ||
| 2mg | 131.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 546.00 € | ||
| 25mg | 857.00 € | ||
| 50mg | 1,170.00 € | ||
| 100mg | 1,569.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Donetidine
CAS:99248-32-5
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
Formula:
C20H25N5O3S
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
415.51
Ref: TM-T68056
| 1mg | 125.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,748.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Relamorelin
CAS:661472-41-9
Relamorelin (RM-131) is a growth hormone-releasing peptide/growth hormone secretagogue receptor agonist, a 5 amino acid …
Formula:
C43H50N8O5S
Purity:
99.26% - 99.85%
Color and Shape:
Solid
Molecular weight:
790.97
Ref: TM-T34281
| 1mg | 468.00 € | ||
| 5mg | 1,082.00 € | ||
| 10mg | 1,458.00 € | ||
| 25mg | 2,163.00 € | ||
| 50mg | 2,793.00 € | ||
| 100mg | 3,940.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Kushenol A
CAS:99217-63-7
Kushenol A is a kind of Adenosine 3', 5'-cyclic monophosphate(cAMP)phosphodiesterase inhibitiors, it shows selective alpha-glucosidase …
Formula:
C25H28O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
408.49
Ref: TM-TN1841
| 1ml | 1,021.00 € | ||
| 5mg | 741.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Eldelumab
CAS:946414-98-8
Eldelumab (BMS-936557) is an anti-IP-10 IgG 1 monoclonal antibody.Eldelumab has anti-inflammatory activity and is used …
Purity:
95%
Color and Shape:
Solid
Ref: TM-T76741
| 1mg | 226.00 € | ||
| 2mg | 333.00 € | ||
| 5mg | 554.00 € | ||
| 10mg | 841.00 € | ||
| 25mg | 1,273.00 € | ||
| 50mg | 1,716.00 € | ||
| 100mg | 2,310.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Thioperamide maleate
CAS:148440-81-7
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = …
Formula:
C19H28N4O4S
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
408.52
Ref: TM-T41247
| 1mg | 42.00 € | ||
| 1ml | 98.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Pafenolol
CAS:75949-61-0
Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an …
Formula:
C18H31N3O3
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
337.46
Ref: TM-T68124
| 1mg | 93.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 1,019.00 € | ||
| 500mg | 2,070.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tolnapersine TFA
Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
Formula:
C23H27F3N2O3
Purity:
98.10%
Color and Shape:
Soild
Molecular weight:
436.47
Ref: TM-T68023L
| 1mg | 182.00 € | ||
| 5mg | 399.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,267.00 € | ||
| 100mg | 1,710.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
S1R agonist 2
CAS:150085-21-5
S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for …
Formula:
C21H27NO
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
309.45
Ref: TM-T72059
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 600.00 € | ||
| 500mg | 1,268.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Saterinone
CAS:102669-89-6
Saterinone: PDE III inhibitor, α-1-adrenoceptor antagonist, vasodilator, used for acute chronic heart failure, IC50 2.3x10^-5 …
Formula:
C27H30N4O4
Purity:
98.23%
Color and Shape:
Solid
Molecular weight:
474.55
Ref: TM-T68138
| 1mg | 152.00 € | ||
| 1ml | 433.00 € | ||
| 5mg | 365.00 € | ||
| 10mg | 548.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,606.00 € | ||
| 500mg | 3,212.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
IRL-1038 acetate
IRL-1038 acetate is a potent ETB endothelin receptor antagonist.
Formula:
C70H96N14O17S2
Purity:
97.51%
Color and Shape:
Soild
Molecular weight:
1469.73
Ref: TM-TP2262L
| 1mg | 407.00 € | ||
| 5mg | 940.00 € | ||
| 10mg | 1,406.00 € | ||
| 25mg | 2,407.00 € | ||
| 50mg | 3,237.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
REV 5901A
CAS:92532-23-5
REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial …
Formula:
C22H26ClNO2
Purity:
99.74%
Color and Shape:
Soild
Molecular weight:
371.90
Ref: TM-T21821L
| 1mg | 182.00 € | ||
| 5mg | 450.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,388.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
