G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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FFN246
CAS:2210244-83-8
FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 …
Formula:
C15H13FN2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
256.27
Ref: TM-T78684
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Estimated delivery in United States, on Monday 16 Dec 2024
(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:77327-45-8
(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the …
Formula:
C48H74N12O12S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1075.3
Ref: TM-T80126
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Estimated delivery in United States, on Monday 16 Dec 2024
Emoghrelin
CAS:928262-58-2
Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the …
Formula:
C24H22O13
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
518.42
Ref: TM-T80006
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Estimated delivery in United States, on Monday 16 Dec 2024
PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, …
Formula:
C10H15F2N3O13P3S·xC6H15N
Purity:
98%
Color and Shape:
Liquid
Ref: TM-T78080
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Estimated delivery in United States, on Monday 16 Dec 2024
PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting …
Formula:
C18H20N5O7S2·NH4·75H2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
532.09
Ref: TM-T78084
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Estimated delivery in United States, on Monday 16 Dec 2024
D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor …
Formula:
C27H37NO5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
455.59
Ref: TM-T78736
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Estimated delivery in United States, on Monday 16 Dec 2024
Galanin-Like Peptide (human)
CAS:245114-99-2
Galanin-Like Peptide (human) is a neuropeptide consisting of 60 amino acids, instrumental in regulating feeding, …
Formula:
C292H451N83O84S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6500.28
Ref: TM-T80144
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Estimated delivery in United States, on Monday 16 Dec 2024
Stressin I TFA
Stressin I (Cyclo(31-34)[DPhe12, Nle21, 38, Glu31, Lys34]Ac-hCRF(4-41)) TFA, with a K i of 1.7 nM, …
Purity:
98%
Ref: TM-T81081
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Estimated delivery in United States, on Monday 16 Dec 2024
ACTH (7-38) (human)
CAS:68563-24-6
ACTH (7-38) (human) is a fragment (7-38) of the full human adrenocorticotropic hormone (ACTH (1-39)), …
Formula:
C167H257N47O46
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3659.11
Ref: TM-T80125
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Estimated delivery in United States, on Monday 16 Dec 2024
Atrial natriuretic peptide (3-28) (human)
CAS:102686-43-1
Atrial natriuretic peptide (3-28) (human) (ANP (3-28) (human)), a peptide hormone produced by the atrial …
Formula:
C118H187N43O36S3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2880.21
Ref: TM-T80438
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Estimated delivery in United States, on Monday 16 Dec 2024
4-Methylhistamine
CAS:36507-31-0
4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for …
Formula:
C6H11N3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
125.17
Ref: TM-T80645
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Estimated delivery in United States, on Monday 16 Dec 2024
NXT-10796
NXT-10796 is an orally active, intestinally restricted agonist of the EP4 receptor [1].
Formula:
C23H31N3O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
445.51
Ref: TM-T79432
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Estimated delivery in United States, on Monday 16 Dec 2024
Ala5-Galanin (2-11)
CAS:859843-84-8
Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity …
Formula:
C54H81N13O13
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1120.3
Ref: TM-T80517
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Estimated delivery in United States, on Monday 16 Dec 2024
(Leu31,Pro34)-Peptide YY (human) (TFA)
"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a …
Formula:
C195H296N54O56·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
4292.75 (free base)
Ref: TM-T80087
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Estimated delivery in United States, on Monday 16 Dec 2024
Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has …
Purity:
98%
Ref: TM-T81798
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Estimated delivery in United States, on Monday 16 Dec 2024
Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:71800-37-8
Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].
Formula:
C47H75N13O11
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
998.18
Ref: TM-T80117
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Estimated delivery in United States, on Monday 16 Dec 2024
A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 …
Formula:
C28H34N6O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
550.61
Ref: TM-T79372
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Estimated delivery in United States, on Monday 16 Dec 2024
AD186
AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for …
Formula:
C22H28N2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
320.47
Ref: TM-T78915
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Estimated delivery in United States, on Monday 16 Dec 2024
Galanin-Like Peptide (porcine)
CAS:245114-96-9
Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.
Formula:
C281H443N81O78
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6204.02
Ref: TM-T80145
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Estimated delivery in United States, on Monday 16 Dec 2024
D3R/MOR antagonist 2
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM …
Formula:
C25H31ClN2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
410.98
Ref: TM-T78779
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Estimated delivery in United States, on Monday 16 Dec 2024
