G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Muscarinic toxin 3
CAS:873336-87-9
Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values …
Formula:
C319H489N89O97S8
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
7379.35
Ref: TM-T80477
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM …
Formula:
C25H30N2O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
438.52
Ref: TM-T78916
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Ac-(d-Arg)-CEH-(d-Phe)-RWC-NH2
CAS:819048-44-7
Ac-DArg-c[Cys-Glu-His-DPhe-Arg-Trp-Cys]-NH2 is a synthetic cyclic octapeptide that exhibits melanocortin-4 receptor (MC4R) agonism and has been …
Formula:
C51H70N18O11S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1175.35
Ref: TM-T80121
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
GRP (14-27) (human, porcine, canine)
CAS:81608-29-9
GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific …
Formula:
C75H110N24O16S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1667.96
Ref: TM-T80148
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:176714-12-8
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
Formula:
C52H76N14O11S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1137.38
Ref: TM-T80137
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
(Val3,Pro8)-Oxytocin
CAS:2134138-89-7
(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced …
Formula:
C41H60N12O12S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
977.12
Ref: TM-T80140
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Capeserod
CAS:769901-96-4
Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive …
Formula:
C23H25ClN4O4
Purity:
98.82% - 99.37%
Color and Shape:
Liquid
Molecular weight:
456.92
Ref: TM-T68035
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,004.00 € | ||
| 50mg | 1,385.00 € | ||
| 100mg | 1,831.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(D-Arg8)-Inotocin
CAS:745816-74-4
'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), …
Formula:
C39H68N14O11S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
973.17
Ref: TM-T80138
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Invopressin
CAS:1488411-60-4
Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in …
Formula:
C110H161N31O27S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2413.78
Ref: TM-T80270
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Vasopressin Dimer (parallel) (TFA)
Vasopressin Dimer (parallel) TFA, a parallel dimer of Vasopressin, has the capability to activate four …
Formula:
C94H131F3N30O26S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2282.49
Ref: TM-T80197
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Galanin-Like Peptide (rat)
CAS:245114-97-0
Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating …
Formula:
C288H461N87O83S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
6502.34
Ref: TM-T80146
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is …
Formula:
C162H262N50O52S2·C2HF3O2
Purity:
98%
Color and Shape:
Liquid
Ref: TM-T78540
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Vasopressin Dimer (anti-parallel) (TFA)
Vasopressin Dimer (anti-parallel) TFA, an anti-parallel dimer form of vasopressin, has the capability to activate …
Formula:
C94H131F3N30O26S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2282.49
Ref: TM-T80198
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
CXCR4-IN-2
CXCR4-IN-2 (compound A1), a potent bifunctional fluorinated small molecule, inhibits CXCR4 and exhibits anticancer properties …
Formula:
C21H20F6N4S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
474.47
Ref: TM-T78879
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Vilanterol
CAS:503068-34-6
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and …
Formula:
C24H33Cl2NO5
Purity:
98.09% - 99.46%
Color and Shape:
Solid
Molecular weight:
486.43
Ref: TM-T2645
| 1mg | 48.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ridazolol HCl
CAS:83394-57-4
Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.
Formula:
C15H19Cl3N4O3
Purity:
99.58%
Color and Shape:
Soild
Molecular weight:
409.7
Ref: TM-T26081L
| Undefined size | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Sigma-1 receptor antagonist 4
Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's …
Formula:
C22H26N2O
Color and Shape:
Liquid
Molecular weight:
334.45
Ref: TM-T74813
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
REV 5901A
CAS:92532-23-5
REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial …
Formula:
C22H26ClNO2
Purity:
99.74%
Color and Shape:
Soild
Molecular weight:
371.90
Ref: TM-T21821L
| 1mg | 182.00 € | ||
| 5mg | 450.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,388.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Relenopride
CAS:1221416-43-8
YKP 10811 (Relenopride) is a novel 5-HT4 receptor partial agonist, which can be used to …
Formula:
C24H30ClFN4O4
Purity:
98.91% - 99.20%
Color and Shape:
Soild
Molecular weight:
492.97
Ref: TM-T83981
| 1mg | 125.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,351.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(S)-(-)-Atenolol
CAS:93379-54-5
(S)-(-)-Atenolol has beta-adrenergic blocking effects.
Formula:
C14H22N2O3
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
266.34
Ref: TM-T35833
| 1mg | 73.00 € | ||
| 5mg | 151.00 € | ||
| 10mg | 213.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 763.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
