G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Brexpiprazole S-oxide
CAS:1191900-51-2
Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial …
Formula:
C25H27N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
449.57
Ref: TM-T10612
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Spiroglumide
CAS:137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 …
Formula:
C21H26Cl2N2O4
Purity:
98.34%
Color and Shape:
Soild
Molecular weight:
441.35
Ref: TM-T68016
| 1mg | 152.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 876.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,214.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Sigma-1 receptor antagonist 4
Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's …
Formula:
C22H26N2O
Color and Shape:
Solid
Molecular weight:
334.45
Ref: TM-T74813
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Dalcotidine
CAS:120958-90-9
Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, …
Formula:
C18H29N3O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
319.44
Ref: TM-T31195
| 1mg | 138.00 € | ||
| 1ml | 338.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,486.00 € | ||
| 500mg | 2,971.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Seganserin
CAS:87729-89-3
Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.
Formula:
C29H27F2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
471.54
Ref: TM-T68141
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,438.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.
Formula:
C22H30N2O7S
Purity:
97.05% - 99.47%
Color and Shape:
Soild
Molecular weight:
466.55
Ref: TM-T68161L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,415.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Fargesone B
CAS:116424-70-5
Fargesone B inhibits the vascular smooth muscle contraction by suppressing the voltage- and receptor-activated calcium …
Formula:
C21H24O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.417
Ref: TM-TN4051
| 1ml | 576.00 € | ||
| 5mg | 557.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Eledoisin Related Peptide
CAS:2990-43-4
Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.
Formula:
C34H58N8O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
706.94
Ref: TM-T7631
| 1mg | 153.00 € | ||
| 5mg | 641.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Bucumolol
CAS:58409-59-9
Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and …
Formula:
C17H23NO4
Purity:
99.70%
Color and Shape:
Soild
Molecular weight:
305.37
Ref: TM-T30606L
| 1mg | 193.00 € | ||
| 5mg | 477.00 € | ||
| 10mg | 670.00 € | ||
| 25mg | 1,045.00 € | ||
| 50mg | 1,442.00 € | ||
| 100mg | 1,846.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
CAS:1366000-58-9
ANP, a guanylate cyclase stimulator, protects cardiomyocytes and stimulates exercise-linked lipolysis.
Formula:
C129H207N45O41S3
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
3140.5
Ref: TM-TP1219
| 1mg | 212.00 € | ||
| 2mg | 357.00 € | ||
| 5mg | 760.00 € | ||
| 10mg | 1,003.00 € | ||
| 25mg | 1,514.00 € | ||
| 50mg | 2,031.00 € | ||
| 100mg | 2,759.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Donitriptan hydrochloride
CAS:170911-68-9
Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis …
Formula:
C23H26ClN5O2
Purity:
99.8% - 99.8%
Color and Shape:
Solid
Molecular weight:
439.94
Ref: TM-T21666
| 1ml | 76.00 € | ||
| 2mg | 40.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 332.00 € | ||
| 200mg | 430.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tiaprost
CAS:71116-82-0
Tiaprost is a analog of prostaglandin F2α .
Formula:
C20H28O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
396.5
Ref: TM-T17092
| 1mg | 162.00 € | ||
| 5mg | 650.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tirzepatide monosodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective …
Formula:
C225H347N48O68Na
Purity:
99.69%
Color and Shape:
Soild
Molecular weight:
4835.51
Ref: TM-TP1111L1
| 1mg | 249.00 € | ||
| 5mg | 652.00 € | ||
| 10mg | 1,069.00 € | ||
| 25mg | 1,598.00 € | ||
| 50mg | 2,193.00 € | ||
| 100mg | 2,959.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Mazdutide acetate(2259884-03-0 free base)
Mazdutide acetate is a potent (GLP-1R and GCGR agonist that stimulates insulin secretion from mouse …
Purity:
98.41%
Ref: TM-T78097L
| 1mg | 95.00 € | ||
| 5mg | 252.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 681.00 € | ||
| 50mg | 1,083.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Enrasentan
CAS:167256-08-8
Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure …
Formula:
C29H30O8
Purity:
97.90% - 97.96%
Color and Shape:
Solid
Molecular weight:
506.54
Ref: TM-T31640
| 1mg | 181.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 640.00 € | ||
| 25mg | 1,004.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
1-Oleoyl Lysophosphatidic Acid
CAS:65528-98-5
1-Oleoyl Lysophosphatidic Acid (1-Oleoyl LPA) is a biologically active phospholipid that can be used to …
Formula:
C21H41O7P
Color and Shape:
Solid
Molecular weight:
436.52
Ref: TM-T36907
| 22.91mM*1 | 379.00 € | ||
| 22.91mM*100 | 68.00 € | ||
| 22.91mM*2.5 | 795.00 € | ||
| 22.91mM*500 | 231.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Ro60-0175
CAS:169675-08-5
Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.
Formula:
C11H12ClFN2
Purity:
97.09%
Color and Shape:
Solid
Molecular weight:
226.68
Ref: TM-T39161
| 1mg | 96.00 € | ||
| 1ml | 193.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 606.00 € | ||
| 50mg | 828.00 € | ||
| 100mg | 1,141.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
O-Desethyl Dapagliflozin
CAS:864070-37-1
O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.
Formula:
C19H21ClO6
Purity:
97.09%
Color and Shape:
Solid
Molecular weight:
380.82
Ref: TM-T67849
| 1mg | 56.00 € | ||
| 1ml | 132.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 460.00 € | ||
| 100mg | 667.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
LY 344864 racemate
CAS:186543-64-6
LY 344864 racemate is a 5-HT1F receptor agonist.
Formula:
C21H22FN3O
Purity:
99.47%
Color and Shape:
Soild
Molecular weight:
351.42
Ref: TM-T2344L
| 1ml | 36.00 € | ||
| 5mg | 45.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Upacicalcet HCl
Upacicalcet HCl, a calcium mimetic, reduces blood PTH by targeting parathyroid receptors; treats secondary hyperparathyroidism.
Formula:
C11H15Cl2N3O6S
Purity:
98.56%
Color and Shape:
Soild
Molecular weight:
388.22
Ref: TM-T29067L
| 1mg | 172.00 € | ||
| 5mg | 424.00 € | ||
| 10mg | 621.00 € | ||
| 25mg | 989.00 € | ||
| 50mg | 1,337.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
