G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Esprolol
CAS:396654-09-4
Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.
Formula:
C17H27NO4
Purity:
100% - 99.16%
Color and Shape:
Soild
Molecular weight:
309.4
Ref: TM-T27286L
| 1mg | 125.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 436.00 € | ||
| 25mg | 717.00 € | ||
| 50mg | 1,007.00 € | ||
| 100mg | 1,351.00 € | ||
| 500mg | 2,692.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)
PACAP (6-27) is an antagonist for PACAP receptors with varying IC50s; blocks cAMP in neuroblastoma …
Ref: TM-T36427
| 500µg | 422.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PACAP-related Peptide (human) (trifluoroacetate salt)
Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some …
Ref: TM-T36428
| 1mg | 839.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Romergoline 2HCl
Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's …
Formula:
C20H24Cl2N4O2
Purity:
100% - 98.33%
Color and Shape:
Soild
Molecular weight:
423.34
Ref: TM-T71707L
| 1mg | 181.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 639.00 € | ||
| 25mg | 998.00 € | ||
| 50mg | 1,376.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PACAP-related Peptide (rat) (trifluoroacetate salt)
PRP, a 29-amino acid peptide in the secretin/glucagon family, is found in rat brain regions …
Color and Shape:
Liquid
Ref: TM-T37435
| 1mg | 473.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Corticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.
Purity:
98.30%
Ref: TM-TP1144L
| 1mg | 143.00 € | ||
| 5mg | 465.00 € | ||
| 10mg | 694.00 € | ||
| 25mg | 1,246.00 € | ||
| 50mg | 1,854.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PACAP-38 (31-38), human, mouse, rat acetate
PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.
Formula:
C49H87N17O13
Purity:
99.92%
Color and Shape:
Liquid
Molecular weight:
1122.32
Ref: TM-TP1618L
| 1mg | 135.00 € | ||
| 5mg | 391.00 € | ||
| 10mg | 567.00 € | ||
| 25mg | 904.00 € | ||
| 50mg | 1,224.00 € | ||
| 100mg | 1,641.00 € | ||
| 500mg | 3,240.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PA-8
CAS:878437-15-1
PA-8: Selective PAC1 antagonist, orally active, blocks CREB phosphorylation & cAMP increase (IC50=2nM), reduces pain …
Formula:
C17H18N4O4
Purity:
97.64%
Color and Shape:
Liquid
Molecular weight:
342.35
Ref: TM-T41005
| 5mg | 46.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 254.00 € | ||
| 100mg | 446.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PACAP (6-38), human, ovine, rat acetate
PACAP (6-38), human, ovine, rat acetate is a potent PACAP receptor antagonist with IC50s of …
Purity:
99.84%
Color and Shape:
Soild
Ref: TM-TP1722L
| 1mg | 94.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 515.00 € | ||
| 50mg | 697.00 € | ||
| 100mg | 943.00 € | ||
| 200mg | 1,272.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TAK-448 acetate
CAS:1470374-22-1
TAK-448 acetate (MVT-602 acetate) is a KISS1R agonist, a synthetic peptide similar to kisspeptin.
Formula:
C60H84N16O16
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
1285.41
Ref: TM-TP1093
| 1mg | 94.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 601.00 € | ||
| 50mg | 843.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DuP 747 HCl
CAS:115904-74-0
DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two …
Formula:
C24H29Cl3N2O2
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
483.86
Ref: TM-T25354L
| 1mg | 241.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,279.00 € | ||
| 50mg | 1,727.00 € | ||
| 100mg | 2,334.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Y1 receptor antagonist 1
CAS:221697-09-2
Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.
Formula:
C28H33N5O3
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
487.59
Ref: TM-T12155
| 1mg | 331.00 € | ||
| 5mg | 557.00 € | ||
| 25mg | 869.00 € | ||
| 50mg | 1,179.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonist
Formula:
C7H13N3O2
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
171.2
Ref: TM-T23038L
| 1mg | 187.00 € | ||
| 5mg | 462.00 € | ||
| 10mg | 662.00 € | ||
| 25mg | 1,033.00 € | ||
| 50mg | 1,425.00 € | ||
| 100mg | 1,885.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lintopride HCl
CAS:268548-31-8
Lintopride HCl is a 5HT-4 antagonist.
Formula:
C14H20Cl2N4O2
Purity:
97.70% - 98.42%
Color and Shape:
Soild
Molecular weight:
347.24
Ref: TM-T15760L
| 1mg | 96.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 292.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 713.00 € | ||
| 100mg | 998.00 € | ||
| 500mg | 2,004.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dazmegrel HCl
Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and …
Formula:
C16H18ClN3O2
Purity:
98.63%
Color and Shape:
Liquid
Molecular weight:
319.79
Ref: TM-T31213L
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMY 25368 HCl
CAS:86134-36-3
BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated …
Formula:
C19H26ClN3O3
Purity:
98.73% - 99.81%
Color and Shape:
Soild
Molecular weight:
379.88
Ref: TM-T23811L
| 1mg | 96.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 496.00 € | ||
| 50mg | 717.00 € | ||
| 100mg | 1,007.00 € | ||
| 500mg | 2,013.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to …
Formula:
C19H26F2N2O3
Purity:
96.15%
Color and Shape:
Soild
Molecular weight:
368.42
Ref: TM-T12416L
| Undefined size | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Sarizotan 2HCl
CAS:177976-12-4
Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant …
Formula:
C22H23Cl2FN2O
Purity:
98.83%
Color and Shape:
Soild
Molecular weight:
421.34
Ref: TM-T70044L
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,836.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
YT 146
CAS:90596-75-1
YT 146 is a biochemical.
Formula:
C18H25N5O4
Purity:
98.81% - 99.72%
Color and Shape:
Solid
Molecular weight:
375.42
Ref: TM-T35282
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,572.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tirzepatide
CAS:2023788-19-2
Tirzepatide (LY-3298176) is a dual agonist of GIP and GLP-1 receptors with neuroprotective activity and …
Formula:
C225H348N48O68
Purity:
99.52% - 99.99%
Color and Shape:
Solid
Molecular weight:
4813.45
Ref: TM-TP1111
| 1mg | 247.00 € | ||
| 5mg | 648.00 € | ||
| 10mg | 927.00 € | ||
| 25mg | 1,372.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
