G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AL 34662
CAS:210580-75-9
AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM …
Formula:
C10H13N3O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
191.23
Ref: TM-T22029
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 212.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.
Purity:
> 95%
Ref: TM-T77053
| 1mg | 247.00 € | ||
| 5mg | 647.00 € | ||
| 10mg | 1,013.00 € | ||
| 25mg | 1,529.00 € | ||
| 50mg | 2,045.00 € | ||
| 100mg | 2,795.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM …
Formula:
C25H30N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.52
Ref: TM-T78916
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
(Iso)-Landipirdine
CAS:1000308-09-7
(Iso)-Landipirdine((Iso)-RO5025181) is a selective and potent 5-HT6R antagonist.
Formula:
C18H19FN2O3S
Purity:
97.27%
Color and Shape:
Soild
Molecular weight:
362.42
Ref: TM-T27795L
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,384.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
BF-1
CAS:518980-66-0
BF-1 blocks 5-HT2B, may prevent migraines by hindering BW723C86/mCPP in guinea pigs.
Formula:
C22H25NO2S
Purity:
100% - 99.25%
Color and Shape:
Solid
Molecular weight:
367.50
Ref: TM-T26781
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,423.00 € | ||
| 50mg | 1,869.00 € | ||
| 100mg | 2,605.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
S1PR1 modulator 1
CAS:2328109-05-1
S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.
Formula:
C23H24N2O3S
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
408.51
Ref: TM-T12821
| 1mg | 64.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 394.00 € | ||
| 100mg | 584.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Myriceric acid C
CAS:162059-94-1
Myriceric acid C has cytotoxic activity against human lung carcinoma and breast carcinoma.
Formula:
C48H60O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
796.98
Ref: TM-TN4606
| 5mg | 670.00 € | ||
| 1mL*10mM (DMSO) | 1,020.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
S1R agonist 2
CAS:150085-21-5
S1R agonist 2 is a selective S1R agonist with a Ki of 88 nM for …
Formula:
C21H27NO
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
309.45
Ref: TM-T72059
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 600.00 € | ||
| 500mg | 1,268.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ALX 40-4C acetate
ALX 40-4C acetate is a CXCR4 inhibitor (Ki=1μM), blocks X4 HIV-1, and antagonizes APJ receptor …
Formula:
C58H117N37O12
Purity:
98.94% - 99%
Color and Shape:
Solid
Molecular weight:
1524.79
Ref: TM-TP1364L
| 1mg | 206.00 € | ||
| 5mg | 715.00 € | ||
| 10mg | 1,069.00 € | ||
| 25mg | 1,860.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
DALDA TFA
DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant …
Formula:
C30H45N9O5·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
611.74 (free base)
Ref: TM-T80086
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Saterinone
CAS:102669-89-6
Saterinone: PDE III inhibitor, α-1-adrenoceptor antagonist, vasodilator, used for acute chronic heart failure, IC50 2.3x10^-5 …
Formula:
C27H30N4O4
Purity:
98.23%
Color and Shape:
Liquid
Molecular weight:
474.55
Ref: TM-T68138
| 1mg | 152.00 € | ||
| 5mg | 365.00 € | ||
| 10mg | 548.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,606.00 € | ||
| 500mg | 3,212.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Neurokinin B acetate(86933-75-7 free base)
Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological …
Formula:
C57H83N13O16S2
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
1270.48
Ref: TM-TP1363L
| 1mg | 86.00 € | ||
| 5mg | 309.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 880.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
D3R/MOR antagonist 2
Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM …
Formula:
C25H31ClN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
410.98
Ref: TM-T78779
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Spiroglumide
CAS:137795-35-8
Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 …
Formula:
C21H26Cl2N2O4
Purity:
98.34%
Color and Shape:
Soild
Molecular weight:
441.35
Ref: TM-T68016
| 1mg | 152.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 876.00 € | ||
| 50mg | 1,196.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,214.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
(Leu31,Pro34)-Peptide YY (human) (TFA)
"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a …
Formula:
C195H296N54O56·xC2HF3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
4292.75 (free base)
Ref: TM-T80087
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
CI 169369
CAS:85273-96-7
CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and …
Formula:
C19H21ClN2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.9
Ref: TM-T84289
| 1mg | 199.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 692.00 € | ||
| 25mg | 1,080.00 € | ||
| 50mg | 1,489.00 € | ||
| 100mg | 1,907.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Dalcotidine
CAS:120958-90-9
Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, …
Formula:
C18H29N3O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
319.44
Ref: TM-T31195
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,486.00 € | ||
| 500mg | 2,971.00 € | ||
| 1mL*10mM (DMSO) | 338.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Cortistatin-14
CAS:186901-48-4
Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.
Formula:
C81H114N20O18S2
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
1720.03
Ref: TM-TP1570
| 1mg | 97.00 € | ||
| 5mg | 374.00 € | ||
| 10mg | 671.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
AMI-193
CAS:510-74-7
AMI-193 (Spiramide) is a selective 5-HT2 & D2 receptor antagonist with antipsychotic properties.
Formula:
C22H26FN3O2
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T21855
| 5mg | 45.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 310.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
cAC 253 acetate
cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin …
Formula:
C128H206N42O42S2
Purity:
98.16% - 99.99%
Color and Shape:
Soild
Molecular weight:
3069.39
Ref: TM-TP2135L
| 1mg | 182.00 € | ||
| 5mg | 415.00 € | ||
| 10mg | 616.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,290.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
