G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GV-150013X
CAS:151386-96-8
GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKi
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Soild
Molecular weight:
534.65
Ref: TM-T27503L
| 1mg | 183.00 € | ||
| 1ml | 638.00 € | ||
| 5mg | 444.00 € | ||
| 10mg | 608.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,235.00 € | ||
| 100mg | 1,625.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
OX04528
CAS:3028055-45-7
OX04528 is an orally active and potent GPR84 biased agonist.OX04528 inhibits cAMP signaling and may …
Formula:
C16H13F6NO2
Purity:
99.74%
Color and Shape:
Soild
Molecular weight:
365.27
Ref: TM-T84313
| 1mg | 198.00 € | ||
| 5mg | 490.00 € | ||
| 10mg | 687.00 € | ||
| 25mg | 1,072.00 € | ||
| 50mg | 1,479.00 € | ||
| 100mg | 1,894.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Isocupressic acid
CAS:1909-91-7
Isocupressic acid triggers cow abortions in the last trimester by halting angiogenesis and inducing corpus …
Formula:
C20H32O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
320.47
Ref: TM-TN4277
| 1ml | To inquire | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Picumeterol
CAS:130641-36-0
Picumeterol(GR 114297A) is a potent and selective β2 adrenergic receptor agonist. In vitro and in …
Formula:
C21H29Cl2N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
426.38
Ref: TM-T68129
| Undefined size | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GSK270822A
CAS:864082-23-5
GSK270822A is a selective ROCK1 inhibitor. GSK270822A exhibits IC50 of 9nM, 1100nM, 1550nM for ROCK1, …
Formula:
C24H20N4O2
Purity:
98.13% - 98.77%
Color and Shape:
Solid
Molecular weight:
396.44
Ref: TM-T27467
| 1mg | 222.00 € | ||
| 1ml | 564.00 € | ||
| 5mg | 542.00 € | ||
| 10mg | 721.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,461.00 € | ||
| 100mg | 1,964.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
BMS-193885
CAS:186185-03-5
BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a …
Formula:
C33H42N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.71
Ref: TM-T14671
| 1mg | 34.00 € | ||
| 1ml | 90.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 472.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
NF-56-EJ40 hydrochloride
CAS:2728500-80-7
NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 …
Formula:
C27H31Cl2N3O3
Purity:
97.02%
Color and Shape:
Soild
Molecular weight:
516.46
Ref: TM-T12216L
| 5mg | 54.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 402.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
IRL-1038 TFA
IRL-1038 TFA is an ETB receptor antagonist used in the study of cardiovascular disease.
Formula:
C70H93F3N14O17S2
Color and Shape:
Solid
Molecular weight:
1523.7
Ref: TM-TP2262L1
| 1mg | 38.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 82.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
![[Leu13]-Motilin](https://static.cymitquimica.com/products/TM/thumb/T78563.jpg)
[Leu13]-Motilin
CAS:59530-69-7
[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in …
Formula:
C121H190N34O35
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2681.01
Ref: TM-T78563
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
BM213 acetate
BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization …
Formula:
C45H74N12O12
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
975.14
Ref: TM-T35399L
| 1mg | 54.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 336.00 € | ||
| 50mg | 493.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PACAP-38 (31-38), human, mouse, rat acetate
PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.
Formula:
C49H87N17O13
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1122.32
Ref: TM-TP1618L
| 1mg | 132.00 € | ||
| 5mg | 383.00 € | ||
| 10mg | 555.00 € | ||
| 25mg | 891.00 € | ||
| 50mg | 1,203.00 € | ||
| 100mg | 1,606.00 € | ||
| 500mg | 3,240.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(Rac)-Norcisapride
CAS:84946-16-7
Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.
Formula:
C14H20ClN3O3
Purity:
99.13%
Color and Shape:
Soild
Molecular weight:
313.78
Ref: TM-T68116L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 593.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,438.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
L 152804
CAS:6508-43-6
L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese …
Formula:
C23H26O4
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
366.45
Ref: TM-T15679
| 1mg | 36.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 429.00 € | ||
| 500mg | 931.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
N-Desmethyl Pimavanserin
CAS:639863-77-7
N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment …
Formula:
C24H32FN3O2
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
413.53
Ref: TM-T37979
| 1mg | 69.00 € | ||
| 1ml | 238.00 € | ||
| 2mg | 117.00 € | ||
| 5mg | 263.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 631.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Survodutide
CAS:2805997-46-8
Survodutide (BI 456906) is a dual agonist of glucagon and glucagon-like peptide 1 (GLP-1) receptor …
Formula:
C192H289N47O61
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
4231.62
Ref: TM-T76559
| 1mg | 102.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 535.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
β-Endorphin (6-31), human
CAS:77761-27-4
β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid …
Formula:
C131H218N34O40
Purity:
98%
Color and Shape:
Solid
Molecular weight:
2909.38
Ref: TM-T76285
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
AM-8123
CAS:2049973-02-4
AM-8123: oral APJ agonist, potent, inhibits cAMP, activates Gα, key for cardiovascular research.
Formula:
C27H33N7O5S
Purity:
99.59% - 99.76%
Color and Shape:
Solid
Molecular weight:
567.66
Ref: TM-T39442
| 1mg | 272.00 € | ||
| 2mg | 404.00 € | ||
| 5mg | 670.00 € | ||
| 10mg | 915.00 € | ||
| 25mg | 1,409.00 € | ||
| 50mg | 1,836.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Talquetamab
CAS:2226212-40-2
Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment …
Color and Shape:
Solid
Ref: TM-T76882
| 1mg | 273.00 € | ||
| 2mg | 413.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 1,094.00 € | ||
| 25mg | 1,622.00 € | ||
| 50mg | 2,188.00 € | ||
| 100mg | 2,951.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Nociceptin (1-13), amide
CAS:178064-02-3
Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 …
Formula:
C61H100N22O15
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1381.59
Ref: TM-TP1793
| 5mg | 98.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 323.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Hemopressin(human, mouse) TFA
CAS:1431329-48-4
Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.
Formula:
C52H80F3N13O14
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1168.27
Ref: TM-T75799
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
