G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Donetidine
CAS:99248-32-5
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
Formula:
C20H25N5O3S
Purity:
99.12%
Color and Shape:
Liquid
Molecular weight:
415.51
Ref: TM-T68056
| 1mg | 125.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,748.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Homoeriodictyol
CAS:446-71-9
Homoeriodictyol, a naturally occurring, bitter-masking flavanone, as a promising agent to increase appetite and food …
Formula:
C16H14O6
Purity:
98.16% - 99.96%
Color and Shape:
Solid
Molecular weight:
302.28
Ref: TM-TN1740
| 1mg | 126.00 € | ||
| 5mg | 262.00 € | ||
| 10mg | 428.00 € | ||
| 25mg | 684.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
YNT-185
CAS:1804978-81-1
YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values …
Formula:
C33H37N5O5S
Purity:
98.6%
Color and Shape:
Liquid
Molecular weight:
615.74
Ref: TM-T39229
| 1mg | 65.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 446.00 € | ||
| 50mg | 717.00 € | ||
| 100mg | 975.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PAR-4 Agonist Peptide, amide acetate
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
Formula:
C36H52N8O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
740.86
Ref: TM-T7623L
| 1mg | 96.00 € | ||
| 5mg | 287.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 833.00 € | ||
| 50mg | 1,249.00 € | ||
| 100mg | 1,873.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
CI 169369
CAS:85273-96-7
CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and …
Formula:
C19H21ClN2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
344.9
Ref: TM-T84289
| 1mg | 199.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 692.00 € | ||
| 25mg | 1,080.00 € | ||
| 50mg | 1,489.00 € | ||
| 100mg | 1,907.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Vilanterol
CAS:503068-34-6
Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and …
Formula:
C24H33Cl2NO5
Purity:
98.09% - 99.46%
Color and Shape:
Solid
Molecular weight:
486.43
Ref: TM-T2645
| 1mg | 48.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Thioperamide maleate
CAS:148440-81-7
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = …
Formula:
C19H28N4O4S
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
408.52
Ref: TM-T41247
| 1mg | 42.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 98.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.
Formula:
C22H30N2O7S
Purity:
97.05% - 99.47%
Color and Shape:
Soild
Molecular weight:
466.55
Ref: TM-T68161L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,415.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
IRL-1038 acetate
IRL-1038 acetate is a potent ETB endothelin receptor antagonist.
Formula:
C70H96N14O17S2
Purity:
97.51%
Color and Shape:
Soild
Molecular weight:
1469.73
Ref: TM-TP2262L
| 1mg | 407.00 € | ||
| 5mg | 940.00 € | ||
| 10mg | 1,406.00 € | ||
| 25mg | 2,407.00 € | ||
| 50mg | 3,237.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
AC265347
CAS:1253901-26-6
AC265347 is a potent calcium-sensitive receptor (CaSR) agonist and ago-PAM orthosteric modulator with antitumour activity …
Formula:
C17H17NOS
Purity:
100%
Color and Shape:
Solid
Molecular weight:
283.39
Ref: TM-T29541
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 341.00 € | ||
| 100mg | 503.00 € | ||
| 500mg | 1,076.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
![[Leu13]-Motilin](https://static.cymitquimica.com/products/TM/thumb/T78563.jpg)
[Leu13]-Motilin
CAS:59530-69-7
[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in …
Formula:
C121H190N34O35
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2681.01
Ref: TM-T78563
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
PF-06478939
PF-06478939 is a peptide that functions as an agonist at the oxytocin (OT) receptor and …
Formula:
C78H134N14O22S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1684.11
Ref: TM-T79173
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial …
Formula:
C102H163N31O26
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
2239.58
Ref: TM-TP2075L
| 1mg | 303.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 1,033.00 € | ||
| 25mg | 1,838.00 € | ||
| 50mg | 2,755.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Y1 receptor antagonist 1
CAS:221697-09-2
Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.
Formula:
C28H33N5O3
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
487.59
Ref: TM-T12155
| 1mg | 331.00 € | ||
| 5mg | 557.00 € | ||
| 25mg | 869.00 € | ||
| 50mg | 1,179.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
![4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-me…](https://static.cymitquimica.com/products/TM/thumb/T60126.jpg)
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine
CAS:2649012-21-3
4-(2-chloro-4-methoxy-5-methylphenyl)-N-[(1A)-2-cyclopropyl-1-(3-fluoro-4-methylphenyl)ethyl]-5-methyl-N-(2-propyn-1-yl)-2-thiazolamine is an enantiomeric
Formula:
C27H28ClFN2OS
Purity:
99.02%
Color and Shape:
Soild
Molecular weight:
483.04
Ref: TM-T60126
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 302.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
PF-06655075
PF-06655075 is a novel, non-brain-penetrant oxytocin receptor agonist that demonstrates enhanced selectivity for the oxytocin …
Formula:
C75H130N14O22S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1644.05
Ref: TM-T79172
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Zalospirone
CAS:114298-18-9
Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and …
Formula:
C24H29N5O2
Purity:
100% - 99%
Color and Shape:
Liquid
Molecular weight:
419.52
Ref: TM-T68172
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,336.00 € | ||
| 500mg | 4,564.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
DuP 747 HCl
CAS:115904-74-0
DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two …
Formula:
C24H29Cl3N2O2
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
483.86
Ref: TM-T25354L
| 1mg | 241.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,279.00 € | ||
| 50mg | 1,727.00 € | ||
| 100mg | 2,334.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
CSD-CH2(1,8)-NH2
CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of …
Formula:
C76H125N25O15S2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1693.09
Ref: TM-T80421
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Avexitide acetate
CAS:2051593-46-3
Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the …
Formula:
C155H246N40O53S
Purity:
96.64%
Color and Shape:
Liquid
Molecular weight:
3549.91
Ref: TM-TP2100L
| 1mg | 162.00 € | ||
| 5mg | 457.00 € | ||
| 10mg | 641.00 € | ||
| 25mg | 991.00 € | ||
| 50mg | 1,342.00 € | ||
| 100mg | 1,805.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
