G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Formula:
C38H39ClFN3O12
Purity:
95%
Color and Shape:
Solid
Molecular weight:
784.18
Ref: TM-T9579L
| 1mg | 181.00 € | ||
| 1ml | 635.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,738.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial …
Formula:
C102H163N31O26
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
2239.58
Ref: TM-TP2075L
| 1mg | 303.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 1,033.00 € | ||
| 25mg | 1,838.00 € | ||
| 50mg | 2,755.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Asenapine
CAS:65576-45-6
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic …
Formula:
C17H16ClNO
Purity:
99.16%
Color and Shape:
Coa
Molecular weight:
285.77
Ref: TM-T21360
| 1mg | 38.00 € | ||
| 1ml | 86.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 341.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Rotigotine
CAS:92206-54-7
Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.
Formula:
C19H25NOS
Purity:
98.84% - 99.82%
Color and Shape:
Solid
Molecular weight:
315.47
Ref: TM-T9237
| 1ml | 36.00 € | ||
| 10mg | 45.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 132.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Kynurenic acid
CAS:492-27-3
Kynurenic acid (Quinurenic acid) is an NMDA, glutamate, α7 nicotinic acetylcholine receptor triple antagonist and …
Formula:
C10H7NO3
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
189.17
Ref: TM-T65135
| 50mg | 36.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SB-674042
CAS:483313-22-0
SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is …
Formula:
C24H21FN4O2S
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
448.51
Ref: TM-T16854
| 1mg | 49.00 € | ||
| 1ml | 92.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Tamsulosin
CAS:106133-20-4
Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.
Formula:
C20H28N2O5S
Purity:
99.94%
Color and Shape:
White Crystals
Molecular weight:
408.51
Ref: TM-T0210L
| 1ml | 57.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Apraclonidine hydrochloride
CAS:73218-79-8
Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.
Formula:
C9H11Cl3N4
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
281.57
Ref: TM-T21371
| 1ml | 52.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 274.00 € | ||
| 500mg | 596.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Clopidogrel thiolactone
CAS:1147350-75-1
Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.
Formula:
C16H16ClNO3S
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T5501
| 1ml | 309.00 € | ||
| 2mg | 166.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 439.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Atipamezole
CAS:104054-27-5
Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in …
Formula:
C14H16N2
Purity:
99.76%
Color and Shape:
Off-White To Light Yellow Crystal Powder
Molecular weight:
212.29
Ref: TM-T6766
| 1ml | 55.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 353.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GR79236
CAS:124555-18-6
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has …
Formula:
C15H21N5O5
Color and Shape:
Solid
Molecular weight:
351.36
Ref: TM-TQ0136
| 2mg | 53.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
LP-533401 hydrochloride
CAS:1040526-12-2
LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can …
Formula:
C27H23ClF4N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
562.94
Ref: TM-T15779
| 1mg | 40.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SB-277011 hydrochloride
CAS:215804-67-4
SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.
Formula:
C28H31ClN4O
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
475.03
Ref: TM-T63096
| 2mg | 51.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
WAY-100635 maleate
CAS:634908-75-1
WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).
Formula:
C25H34N4O2·xC4H4O4
Purity:
100%
Color and Shape:
White Solid
Molecular weight:
538.645
Ref: TM-T3453
| 1ml | 79.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 223.00 € | ||
| 100mg | 329.00 € | ||
| 500mg | 789.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Ketanserin tartrate
CAS:83846-83-7
Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study …
Formula:
C26H28FN3O9
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
545.51
Ref: TM-T1066L
| 1ml | 36.00 € | ||
| 25mg | 37.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 68.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Meclizine
CAS:569-65-3
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that …
Formula:
C25H27ClN2
Purity:
95.16%
Color and Shape:
Solid
Molecular weight:
390.95
Ref: TM-T40652
| 1mg | 182.00 € | ||
| 5mg | 419.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,291.00 € | ||
| 100mg | 1,757.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Sumatriptan
CAS:103628-46-2
Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in …
Formula:
C14H21N3O2S
Purity:
98%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
295.4
Ref: TM-T23405
| 1ml | 41.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 67.00 € | ||
| 100mg | 96.00 € | ||
| 500mg | 199.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
SB-269970 hydrochloride
CAS:261901-57-9
SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist …
Formula:
C18H28N2O3S·HCl
Purity:
98.45%
Color and Shape:
Solid
Molecular weight:
388.95
Ref: TM-T6655
| 1ml | 75.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 251.00 € | ||
| 50mg | 440.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Clothiapine
CAS:2058-52-8
Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
Formula:
C18H18ClN3S
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
343.87
Ref: TM-T23900
| 1mg | 96.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
MS 15203
CAS:73912-52-4
MS 15203 is a GPR171 agonist that reduces chronic neuropathic and inflammatory pain in male …
Formula:
C12H11NO5
Color and Shape:
Solid
Molecular weight:
249.22
Ref: TM-T37131
| 1ml | 71.00 € | ||
| 2mg | 43.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 100.00 € | ||
| 25mg | 201.00 € | ||
| 50mg | 297.00 € | ||
| 100mg | 446.00 € | ||
| 500mg | 969.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
