G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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NOX-6-18
CAS:898211-21-7
NOX-6-18 (GPR132-B-160) is a GPR132 antagonist with insulin-promoting activity and reduced weight gain.
Formula:
C18H17NO5S
Purity:
99.29%
Color and Shape:
Soild
Molecular weight:
359.4
Ref: TM-T83972
| 1mg | 75.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 809.00 € | ||
| 100mg | 1,290.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
KB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8
Formula:
C24H32N2O8
Purity:
98.54%
Color and Shape:
Liquid
Molecular weight:
476.52
Ref: TM-T62396L
| 5mg | 62.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 189.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pobilukast
CAS:107023-41-6
Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study …
Formula:
C26H34O5S
Purity:
99.65% - 99.84%
Color and Shape:
Liquid
Molecular weight:
458.61
Ref: TM-T68130
| 1mg | 317.00 € | ||
| 5mg | 751.00 € | ||
| 10mg | 1,065.00 € | ||
| 25mg | 1,584.00 € | ||
| 50mg | 2,068.00 € | ||
| 100mg | 2,647.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CAY10678
CAS:1268709-57-4
CAY10678 is an mPGES-1 inhibitor that inhibits PD-1.CAY10678 reduces collagen deposition and T-cell depletion, and …
Formula:
C23H34N4O
Purity:
99.66%
Color and Shape:
Liquid
Molecular weight:
382.54
Ref: TM-T38369
| 1mg | 52.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 523.00 € | ||
| 100mg | 737.00 € | ||
| 500mg | 1,515.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VUF-11222
CAS:1414376-84-3
VUF-11222 is an agonist of high affinity non-peptide CXCR3 agonist (pKi = 7.2).
Formula:
C25H31BrIN
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
552.33
Ref: TM-T35085
| 1mg | 140.00 € | ||
| 2mg | 187.00 € | ||
| 5mg | 329.00 € | ||
| 10mg | 491.00 € | ||
| 25mg | 796.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,482.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BM213 acetate
BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization …
Formula:
C45H74N12O12
Purity:
99.88%
Color and Shape:
Liquid
Molecular weight:
975.14
Ref: TM-T35399L
| 1mg | 54.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 336.00 € | ||
| 50mg | 493.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Vazegepant
CAS:1337918-83-8
Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.
Formula:
C36H46N8O3
Purity:
98.61%
Color and Shape:
Solid
Molecular weight:
638.80
Ref: TM-T38734
| 1mg | 102.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 599.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Somatostatin acetate
Somatostatin acetate is an endogenously secreted inhibitor of cell proliferation with potential antitumor activity for …
Ref: TM-TP1302L
| 1mg | 59.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 282.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 619.00 € | ||
| 500mg | 1,312.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AVN 322 free base
CAS:1194574-33-8
AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the …
Formula:
C17H19N5O2S
Purity:
99.13%
Color and Shape:
Liquid
Molecular weight:
357.43
Ref: TM-T84317
| 1mg | 200.00 € | ||
| 5mg | 494.00 € | ||
| 10mg | 693.00 € | ||
| 25mg | 1,082.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 1,911.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
RS 56812
CAS:143137-37-5
RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive …
Formula:
C18H21N3O2
Purity:
98.78%
Color and Shape:
Soild
Molecular weight:
311.38
Ref: TM-T23264L
| 1mg | 200.00 € | ||
| 2mg | 295.00 € | ||
| 5mg | 494.00 € | ||
| 10mg | 693.00 € | ||
| 25mg | 1,082.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 1,911.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ebalzotan
CAS:149494-37-1
NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 …
Formula:
C19H30N2O2
Purity:
99.08% - 99.41%
Color and Shape:
Liquid
Molecular weight:
318.45
Ref: TM-T68059
| 1mg | 271.00 € | ||
| 5mg | 737.00 € | ||
| 10mg | 1,101.00 € | ||
| 25mg | 2,001.00 € | ||
| 50mg | 2,624.00 € | ||
| 100mg | 3,492.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
WAY-100635 maleate
CAS:634908-75-1
WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).
Formula:
C25H34N4O2·xC4H4O4
Purity:
100%
Color and Shape:
White Solid
Molecular weight:
538.645
Ref: TM-T3453
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 223.00 € | ||
| 100mg | 329.00 € | ||
| 500mg | 789.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GRK6-IN-2
CAS:2677786-27-3
GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 …
Formula:
C21H21FN6
Purity:
98.94%
Color and Shape:
Liquid
Molecular weight:
376.43
Ref: TM-T61556
| 2mg | 61.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 694.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
LAS101057
CAS:925676-48-8
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the …
Formula:
C18H14FN5O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
335.34
Ref: TM-T15715
| 1mg | 41.00 € | ||
| 5mg | 86.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ATI-2341
CAS:1337878-62-2
ATI-2341, pepducin targeting the CXCR4, is an allosteric agonist activating the Gi to promote inhibition …
Formula:
C104H178N26O25S2
Color and Shape:
Solid
Molecular weight:
2256.82
Ref: TM-T6764
| 1mg | 115.00 € | ||
| 2mg | 205.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 593.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Eticlopride hydrochloride
CAS:97612-24-3
Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).
Formula:
C17H25ClN2O3·HCl
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.31
Ref: TM-T4007
| 1mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pramipexole dihydrochloride
CAS:104632-25-9
Pramipexole dihydrochloride could be used to treat Parkinson disease.
Formula:
C10H18ClN3S
Purity:
98%
Color and Shape:
White Crystalline Powder
Molecular weight:
247.79
Ref: TM-T1476L
| 5mg | 36.00 € | ||
| 10mg | 59.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Asenapine
CAS:65576-45-6
Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic …
Formula:
C17H16ClNO
Purity:
99.16%
Color and Shape:
Coa
Molecular weight:
285.77
Ref: TM-T21360
| 1mg | 38.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 341.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(S)-Mirtazapine
CAS:61337-87-9
(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to …
Formula:
C17H19N3
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
265.35
Ref: TM-T12632L
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 857.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Clopidogrel thiolactone
CAS:1147350-75-1
Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.
Formula:
C16H16ClNO3S
Color and Shape:
Solid
Molecular weight:
337.82
Ref: TM-T5501
| 2mg | 166.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 309.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
