G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .
Formula:
C46H60F3N13O12S
Purity:
98.49%
Color and Shape:
Solid
Molecular weight:
1076.12
Ref: TM-T7627L
| 1mg | 56.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 334.00 € | ||
| 50mg | 501.00 € | ||
| 100mg | 639.00 € | ||
| 200mg | 925.00 € | ||
| 1mL*10mM (DMSO) | 213.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Rotigotine-
CAS:99755-59-6
Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease …
Formula:
C19H25NOS
Purity:
99.59% - 99.76%
Color and Shape:
Solid
Molecular weight:
315.47
Ref: TM-T6647
| 5mg | 52.00 € | ||
| 10mg | 76.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 369.00 € | ||
| 200mg | 541.00 € | ||
| 500mg | 848.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Sec-O-Glucosylhamaudol
CAS:80681-44-3
Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.
Formula:
C21H26O10
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
438.43
Ref: TM-T5S0581
| 20mg | 86.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Atherosperminine
CAS:5531-98-6
Atherosperminine inhibits AChE/BChE and relaxes trachealis via cAMP phosphodiesterase inhibition.
Formula:
C20H23NO2
Purity:
99.4%
Color and Shape:
Solid
Molecular weight:
309.4
Ref: TM-TN3466
| 1mg | 92.00 € | ||
| 2mg | 138.00 € | ||
| 5mg | 204.00 € | ||
| 10mg | 306.00 € | ||
| 25mg | 522.00 € | ||
| 50mg | 734.00 € | ||
| 1mL*10mM (DMSO) | 210.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Tetrahydropalmatine hydrochloride
CAS:6024-85-7
Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.
Formula:
C21H26ClNO4
Purity:
98% - 99.84%
Color and Shape:
Solid
Molecular weight:
391.888
Ref: TM-T2917
| 25mg | 39.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 72.00 € | ||
| 200mg | 93.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
γ-Mangostin
CAS:31271-07-5
Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an …
Formula:
C23H24O6
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
396.43
Ref: TM-T4S1637
| 1mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 639.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Bindarit
CAS:130641-38-2
Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.
Formula:
C19H20N2O3
Purity:
98.48% - 98.71%
Color and Shape:
Solid
Molecular weight:
324.37
Ref: TM-T6413
| 1mg | 56.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 311.00 € | ||
| 50mg | 464.00 € | ||
| 100mg | 665.00 € | ||
| 500mg | 1,356.00 € | ||
| 1mL*10mM (DMSO) | 135.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
3-chloro-5-hydroxybenzoic Acid
CAS:53984-36-4
3-chloro-5-hydroxy Benzoic Acid (3-chloro-5-hydroxy BA) is an agonist of GPR81 (EC50 : 16 μM)
Formula:
C7H5ClO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
172.57
Ref: TM-T7482
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 68.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
ICI 118,551 hydrochloride
CAS:72795-01-8
ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: …
Formula:
C17H28ClNO2
Purity:
98% - 99.53%
Color and Shape:
Solid
Molecular weight:
313.86
Ref: TM-T11607
| 5mg | 53.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Nafarelin acetate(76932-56-4 free base)
CAS:76932-60-0
Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for …
Formula:
C68H89N17O16
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
1400.56
Ref: TM-T21309
| 5mg | 54.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 267.00 € | ||
| 200mg | 402.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
D-tetrahydropalmatine
CAS:3520-14-7
D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.
Formula:
C21H25NO4
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
355.43
Ref: TM-T4S0779
| 2mg | 43.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 175.00 € | ||
| 50mg | 263.00 € | ||
| 100mg | 378.00 € | ||
| 200mg | 538.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
7,4'-Dihydroxyflavone
CAS:2196-14-7
7,4'-Dihydroxyflavone (4',7-Dihydroxyflavone) can induce transcription of nodulation (nod) genes in Rhizobium meliloti.
Formula:
C15H10O4
Purity:
99.39% - 99.6%
Color and Shape:
Solid
Molecular weight:
254.24
Ref: TM-TN1273
| 2mg | 39.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 130.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Hirsuteine
CAS:35467-43-7
Hirsuteine: natural product; blocks nicotine effects on dopamine by hindering ion flow in receptor channels.
Formula:
C22H26N2O3
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
366.45
Ref: TM-TN1081
| 1mg | 90.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 275.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
N-Oleoyl glycine
CAS:2601-90-3
N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of …
Formula:
C20H37NO3
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
339.51
Ref: TM-T13803
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 147.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 318.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
MK-6892
CAS:917910-45-3
MK-6892 is a selective and full agonist for the high-affinity nicotinic acid receptor GPR109A (Ki: …
Formula:
C19H22N4O5
Purity:
99.01% - 99.03%
Color and Shape:
Solid
Molecular weight:
386.4
Ref: TM-TQ0108
| 1mg | 96.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 466.00 € | ||
| 50mg | 646.00 € | ||
| 100mg | 931.00 € | ||
| 500mg | 1,857.00 € | ||
| 1mL*10mM (DMSO) | 228.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
BMS-986122
CAS:313669-88-4
BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment …
Formula:
C16H15BrClNO3S2
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
448.78
Ref: TM-T26869
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 539.00 € | ||
| 100mg | 772.00 € | ||
| 500mg | 1,537.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
CB1 antagonist 4
CAS:1253641-65-4
TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment …
Formula:
C30H25Cl2F3N4OS
Purity:
100%
Color and Shape:
Solid
Molecular weight:
617.51
Ref: TM-T8511
| 1mg | 60.00 € | ||
| 1ml | 163.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 420.00 € | ||
| 100mg | 616.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Blarcamesine hydrochloride
CAS:195615-84-0
Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).
Formula:
C19H24ClNO
Purity:
98.62% - 99.95%
Color and Shape:
Solid
Molecular weight:
317.85
Ref: TM-T4111
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 640.00 € | ||
| 500mg | 1,379.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Gluten Exorphin C
CAS:142479-62-7
Gluten exorphin C is an opioid peptide derived from wheat gluten.
Formula:
C29H45N5O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
591.7
Ref: TM-TP1832
| 1mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 344.00 € | ||
| 100mg | 504.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Bupranolol
CAS:14556-46-8
Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.
Formula:
C14H22ClNO2
Purity:
95.85%
Color and Shape:
Solid
Molecular weight:
271.78
Ref: TM-T8580
| 1mg | 49.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 593.00 € | ||
| 200mg | 799.00 € | ||
| 1mL*10mM (DMSO) | 98.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
