G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formula:
C51H65N9O10
Purity:
97.86%
Color and Shape:
Liquid
Molecular weight:
964.12
Ref: TM-T22811L
| 1mg | 351.00 € | ||
| 2mg | 497.00 € | ||
| 5mg | 749.00 € | ||
| 10mg | 1,000.00 € | ||
| 25mg | 1,495.00 € | ||
| 50mg | 2,018.00 € | ||
| 100mg | 2,724.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
Formula:
C37H48F6N8O11
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
894.81
Ref: TM-T7740
| 1mg | 47.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 407.00 € | ||
| 100mg | 599.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Vipadenant
CAS:442908-10-3
Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for …
Formula:
C16H15N7O
Purity:
97.25% - 97.36%
Color and Shape:
Solid
Molecular weight:
321.34
Ref: TM-T2373
| 1mg | 40.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 211.00 € | ||
| 50mg | 348.00 € | ||
| 100mg | 515.00 € | ||
| 500mg | 1,105.00 € | ||
| 1mL*10mM (DMSO) | 357.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Almorexant
CAS:871224-64-5
Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for …
Formula:
C29H31F3N2O3
Purity:
97.75% - 98.02%
Color and Shape:
Solid
Molecular weight:
512.56
Ref: TM-T2613
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 310.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 742.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Oxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
Purity:
99.24%
Molecular weight:
N/A
Ref: TM-TP1976L
| 1mg | 174.00 € | ||
| 5mg | 510.00 € | ||
| 10mg | 830.00 € | ||
| 25mg | 1,488.00 € | ||
| 50mg | 2,236.00 € | ||
| 100mg | 3,021.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Pergolide mesylate
CAS:66104-23-2
Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve …
Formula:
C20H30N2O3S2
Purity:
99.09%
Color and Shape:
White To Off-White Solid
Molecular weight:
410.59
Ref: TM-T2226
| 5mg | 56.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 174.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PNU 22394 hydrochloride
CAS:15923-42-9
PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
Formula:
C13H17ClN2
Purity:
97.83%
Color and Shape:
Solid
Molecular weight:
236.74
Ref: TM-T23168
| 1mg | 52.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 100.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 364.00 € | ||
| 100mg | 521.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Fexofenadine hydrochloride
CAS:153439-40-8
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the …
Formula:
C32H39NO4·HCl
Purity:
99.39% - ≥95%
Color and Shape:
Solid
Molecular weight:
538.13
Ref: TM-T1470
| 10mg | 49.00 € | ||
| 25mg | 77.00 € | ||
| 50mg | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Maropitant
CAS:147116-67-4
Maropitant is a selective neurokinin (NK1) receptor antagonist.
Formula:
C32H40N2O
Purity:
97.35% - 99.75%
Color and Shape:
Solid
Molecular weight:
468.67
Ref: TM-T7209
| 5mg | 49.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 303.00 € | ||
| 200mg | 435.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
VUF 10166
CAS:155584-74-0
VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 …
Formula:
C13H15ClN4
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
262.74
Ref: TM-T6728
| 10mg | 47.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
NIBR189
CAS:1599432-08-2
NIBR189 is a potent and selective antagonist of EBI2 (GPR183) receptor (IC50 of 11 and …
Formula:
C21H21BrN2O3
Purity:
97%
Color and Shape:
Colourless
Molecular weight:
429.31
Ref: TM-T7156
| 1mg | 35.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 242.00 € | ||
| 50mg | 427.00 € | ||
| 100mg | 631.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Lurasidone
CAS:367514-87-2
Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It …
Formula:
C28H36N4O2S
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
492.68
Ref: TM-T21337
| 5mg | 46.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 203.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Nonapeptide-1 acetate salt (158563-45-2 free base)
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a …
Formula:
C63H91N15O11S
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
1266.58
Ref: TM-TP1101
| 1mg | 69.00 € | ||
| 2mg | 94.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 401.00 € | ||
| 50mg | 593.00 € | ||
| 100mg | 828.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
SR 57227 hydrochloride
CAS:77145-61-0
SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. …
Formula:
C10H14ClN3·HCl
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
248.15
Ref: TM-T23394
| 5mg | 49.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 300.00 € | ||
| 200mg | 427.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Acrivastine
CAS:87848-99-5
Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.
Formula:
C22H24N2O2
Purity:
100% - 99.85%
Color and Shape:
Solid
Molecular weight:
348.44
Ref: TM-T4551
| 1g | 774.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 222.00 € | ||
| 500mg | 541.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
Formula:
C31H60N10O9
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
716.88
Ref: TM-TP1046L
| 1mg | 84.00 € | ||
| 5mg | 191.00 € | ||
| 10mg | 341.00 € | ||
| 25mg | 575.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,105.00 € | ||
| 500mg | 2,261.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
A-582941 dihydrochloride
CAS:848591-90-2
A-582941 dihydrochloride (A 582941) is a Selective agonist of α7 nAChR partial
Formula:
C17H22Cl2N4
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
353.29
Ref: TM-T22016
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 522.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ONO-8130
CAS:459841-96-4
ONO-8130 is an orally available antagonist of EP1 receptor.
Formula:
C25H28N2O5S2
Purity:
97.82%
Color and Shape:
Solid
Molecular weight:
500.63
Ref: TM-T21976
| 1mg | 156.00 € | ||
| 5mg | 337.00 € | ||
| 10mg | 551.00 € | ||
| 25mg | 880.00 € | ||
| 50mg | 1,202.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BP 897
CAS:192384-87-5
BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 …
Formula:
C26H31N3O2
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
417.54
Ref: TM-T9100
| 1mg | 78.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 219.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 521.00 € | ||
| 100mg | 704.00 € | ||
| 200mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 172.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Elagolix sodium
CAS:832720-36-2
Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of …
Formula:
C32H29F5N3NaO5
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
653.57
Ref: TM-T5031
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 415.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
