G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Intepirdine
CAS:607742-69-8
Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment …
Formula:
C19H19N3O2S
Purity:
95.19% - 98.99%
Color and Shape:
Solid
Molecular weight:
353.44
Ref: TM-T1774
| 5mg | 39.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 250.00 € | ||
| 200mg | 355.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS:4815-38-7
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)
Formula:
C14H15NO2S
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
261.34
Ref: TM-T8603
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 226.00 € | ||
| 200mg | 335.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Mosapride Citrate
CAS:112885-42-4
Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.
Formula:
C21H25ClFN3O3·C6H8O7
Purity:
99.88%
Color and Shape:
White Powder
Molecular weight:
614.02
Ref: TM-T6597
| 10mg | 50.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 248.00 € | ||
| 500mg | 417.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Buserelin Acetate (57982-77-1 free base)
CAS:68630-75-1
Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
Formula:
C62H90N16O15
Purity:
99.23% - 99.78%
Color and Shape:
Solid
Molecular weight:
1299.48
Ref: TM-TP1307
| 1mg | 41.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
GSK163090
CAS:844903-58-8
GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for …
Formula:
C25H29N5O
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
415.53
Ref: TM-TQ0311
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Histrelin acetate
CAS:220810-26-4
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.
Formula:
C68H90N18O14
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
1383.55
Ref: TM-TP2107L
| 1mg | 87.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 459.00 € | ||
| 50mg | 644.00 € | ||
| 100mg | 909.00 € | ||
| 200mg | 727.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
CYM-5520
CAS:1449747-00-5
CYM-5520 is a noncompetitive allosteric agonist of S1P2
Formula:
C21H19N3O2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T22703
| 1mg | 47.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 251.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 554.00 € | ||
| 1mL*10mM (DMSO) | 103.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Tetrahydromagnolol
CAS:20601-85-8
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
Formula:
C18H22O2
Purity:
100% - 99.82%
Color and Shape:
Solid
Molecular weight:
270.37
Ref: TM-TN2268
| 5mg | 54.00 € | ||
| 10mg | 84.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Galnon TFA
CAS:1217448-19-5
Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 …
Formula:
C42H47F3N4O8
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
792.84
Ref: TM-T8559
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Fasiglifam
CAS:1000413-72-8
Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.
Formula:
C29H32O7S
Purity:
99.61% - 99.82%
Color and Shape:
Solid
Molecular weight:
524.63
Ref: TM-T2351
| 1mg | 49.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 459.00 € | ||
| 100mg | 554.00 € | ||
| 200mg | 802.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
DOPEXAMINE
CAS:86197-47-9
Dopexamine is a dopaminergic agonist
Formula:
C22H32N2O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
356.5
Ref: TM-T8653
| 1mg | 128.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 697.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,319.00 € | ||
| 1mL*10mM (DMSO) | 305.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Lodoxamide
CAS:53882-12-5
Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in …
Formula:
C11H6ClN3O6
Purity:
99.13% - 99.81%
Color and Shape:
Solid
Molecular weight:
311.63
Ref: TM-T4566
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 319.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Benorilate
CAS:5003-48-5
Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and …
Formula:
C17H15NO5
Purity:
98.39% - 99.56%
Color and Shape:
Solid
Molecular weight:
313.3
Ref: TM-T3276
| 1g | 38.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Olcegepant
CAS:204697-65-4
Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist …
Formula:
C38H47Br2N9O5
Purity:
96.08%
Color and Shape:
Solid
Molecular weight:
869.65
Ref: TM-T12293L
| 1mg | 37.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 188.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
TG4-155
CAS:1164462-05-8
TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective …
Formula:
C23H26N2O4
Purity:
97.20%
Color and Shape:
Solid
Molecular weight:
394.46
Ref: TM-T5482
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 377.00 € | ||
| 100mg | 560.00 € | ||
| 200mg | 459.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Niaprazine
CAS:27367-90-4
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.
Formula:
C20H25FN4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
356.44
Ref: TM-T36949
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 299.00 € | ||
| 200mg | 429.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
SB225002
CAS:182498-32-4
SB225002 is a potent and selective CXCR2 antagonist inhibiting interleukin IL-8 binding to CXCR2.
Formula:
C13H10BrN3O4
Purity:
96.86% - 98.79%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T1955
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 395.00 € | ||
| 200mg | 603.00 € | ||
| 500mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
ML-193
CAS:713121-80-3
ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.
Formula:
C28H25N5O4S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
527.59
Ref: TM-T22103
| 5mg | 46.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Dolasetron Mesylate hydrate
CAS:878143-33-0
Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.
Formula:
C20H26N2O7S
Purity:
99.86% - 99.9%
Color and Shape:
Solid
Molecular weight:
438.49
Ref: TM-T2589
| 5mg | 34.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PRX-08066
CAS:866206-54-4
PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective …
Formula:
C19H17ClFN5S
Purity:
98.04% - 98.07%
Color and Shape:
Solid
Molecular weight:
401.89
Ref: TM-T16669
| 1mg | 59.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 732.00 € | ||
| 500mg | 1,514.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
