G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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L-(R,S)-Tetrahydropalmatine
CAS:10097-84-4
L-(R,S)-Tetrahydropalmatine (Rotundine) is extracted from Corydalis yanhusuo W. T. Wang.
Formula:
C21H25NO4
Purity:
99.63% - 99.76%
Color and Shape:
Solid
Molecular weight:
355.43
Ref: TM-T2714
| 1g | 142.00 € | ||
| 50mg | 34.00 € | ||
| 100mg | 49.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 97.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Leuphasyl TFA
CAS:67586-27-0
Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.
Formula:
C31H40F3N5O9
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
683.67
Ref: TM-T20435L
| 1mg | 86.00 € | ||
| 2mg | 111.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 598.00 € | ||
| 100mg | 810.00 € | ||
| 200mg | 1,074.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Ansofaxine hydrochloride
CAS:916918-84-8
Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).
Formula:
C24H32ClNO3
Purity:
99.57% - 99.77%
Color and Shape:
Solid
Molecular weight:
417.97
Ref: TM-T5380
| 1mg | 78.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 264.00 € | ||
| 25mg | 512.00 € | ||
| 50mg | 723.00 € | ||
| 100mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 178.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Tropisetron
CAS:89565-68-4
Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of …
Formula:
C17H20N2O2
Purity:
99.95%
Color and Shape:
White Solid
Molecular weight:
284.35
Ref: TM-T22448
| 10mg | 47.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 126.00 € | ||
| 100mg | 188.00 € | ||
| 500mg | 487.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Taminadenant
CAS:1337962-47-6
Taminadenant is an adenosine receptor antagonist.
Formula:
C10H8BrN7
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
306.12
Ref: TM-T16980
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 250.00 € | ||
| 200mg | 374.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Riociguat
CAS:625115-55-1
Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth …
Formula:
C20H19FN8O2
Purity:
99.28% - 99.95%
Color and Shape:
Solid
Molecular weight:
422.42
Ref: TM-T6968
| 5mg | 43.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 246.00 € | ||
| 200mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Tolnapersine
CAS:70312-00-4
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Formula:
C21H26N2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
322.44
Ref: TM-T68023
| 1mg | 126.00 € | ||
| 5mg | 304.00 € | ||
| 10mg | 447.00 € | ||
| 25mg | 873.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,843.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Etrasimod
CAS:1206123-37-6
Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: …
Formula:
C26H26F3NO3
Purity:
99.17% - 99.77%
Color and Shape:
Solid
Molecular weight:
457.48
Ref: TM-TQ0227
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Asapiprant
CAS:932372-01-5
Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited …
Formula:
C24H27N3O7S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
501.55
Ref: TM-T5386
| 1mg | 40.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 284.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 730.00 € | ||
| 200mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Etilevodopa hydrochloride
CAS:39740-30-2
Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric …
Formula:
C11H16ClNO4
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
261.7
Ref: TM-T24047
| 10mg | 52.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 250.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Ropinirole
CAS:91374-21-9
Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.
Formula:
C16H24N2O
Purity:
99.68%
Color and Shape:
Liquid
Molecular weight:
260.38
Ref: TM-T60418
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy …
Formula:
C61H88N16O14
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
1269.45
Ref: TM-TP1434L
| 1mg | 74.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 487.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Flupentixol dihydrochloride
CAS:2413-38-9
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive …
Formula:
C23H27Cl2F3N2OS
Purity:
100% - ≥95%
Color and Shape:
White Or Off-White Solid
Molecular weight:
507.43
Ref: TM-T5135
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 185.00 € | ||
| 500mg | 477.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Nelociguat
CAS:625115-52-8
Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formula:
C19H17FN8O2
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
408.39
Ref: TM-T7201
| 5mg | 48.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 129.00 € | ||
| 100mg | 202.00 € | ||
| 200mg | 259.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Cinacalcet hydrochloride
CAS:364782-34-3
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity …
Formula:
C22H23ClF3N
Purity:
99.9% - 99.94%
Color and Shape:
Off-White To Tan Solid
Molecular weight:
393.87
Ref: TM-T2406
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 144.00 € | ||
| 200mg | 185.00 € | ||
| 500mg | 309.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
THIQ
CAS:312637-48-2
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 …
Formula:
C33H41ClN6O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
589.17
Ref: TM-T8485
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 374.00 € | ||
| 50mg | 567.00 € | ||
| 100mg | 848.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
PF3274167
CAS:900510-03-4
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
Formula:
C19H19ClFN5O3
Purity:
99.67% - 99.88%
Color and Shape:
Solid
Molecular weight:
419.84
Ref: TM-T3347
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 235.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
MCOPPB triHydrochloride
CAS:1108147-88-1
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
Formula:
C26H43Cl3N4
Purity:
99.89% - 99.91%
Color and Shape:
Solid
Molecular weight:
518.01
Ref: TM-T2071
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 375.00 € | ||
| 200mg | 535.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Neurokinin A
CAS:86933-74-6
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from …
Formula:
C50H80N14O14S
Purity:
100%
Color and Shape:
White To Off-White Lyophilized Solid
Molecular weight:
1133.32
Ref: TM-TP1008
| 1mg | 62.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 341.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 722.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
APD597
CAS:897732-93-3
APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes.
Formula:
C21H29N5O6S
Purity:
99.63% - 99.78%
Color and Shape:
Solid
Molecular weight:
479.55
Ref: TM-T3176
| 5mg | 70.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 354.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
