G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).
Formula:
C114H174N34O31
Purity:
99.05%
Color and Shape:
Liquid
Molecular weight:
2516.81
Ref: TM-TP2279L
| 1mg | 115.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 627.00 € | ||
| 50mg | 893.00 € | ||
| 100mg | 1,216.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and …
Formula:
C76H117N19O22S
Purity:
95.43%
Color and Shape:
Solid
Molecular weight:
1680.94
Ref: TM-TP1930L1
| 1mg | 114.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,074.00 € | ||
| 200mg | 1,444.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
SDZ WAG 994
CAS:130714-47-5
SDZ WAG 994 is an A1 adenosine receptor agonist.
Formula:
C17H25N5O4
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
363.41
Ref: TM-T23347
| 1mg | 66.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 175.00 € | ||
| 25mg | 316.00 € | ||
| 50mg | 455.00 € | ||
| 100mg | 620.00 € | ||
| 200mg | 835.00 € | ||
| 1mL*10mM (DMSO) | 127.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Melanotan (MT)-II
CAS:121062-08-6
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone …
Formula:
C50H69N15O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1024.18
Ref: TM-TP1324
| 2mg | 49.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 264.00 € | ||
| 100mg | 444.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
FAUC-365
CAS:474432-66-1
FAUC-365 is a D3 dopamine receptor agonist.
Formula:
C23H25Cl2N3OS
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
462.44
Ref: TM-T21667
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 323.00 € | ||
| 50mg | 512.00 € | ||
| 100mg | 740.00 € | ||
| 500mg | 1,539.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
AVN-492
CAS:1220646-23-0
AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
Formula:
C17H21N5O2S
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
359.45
Ref: TM-T5179
| 1mg | 39.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 510.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Zafirlukast
CAS:107753-78-6
Zafirlukast (ICI 204219) is an orally leukotriene D4 receptor (LTD4) antagonist. Zafirlukast has anti-asthmatic and …
Formula:
C31H33N3O6S
Purity:
99% - 99.31%
Color and Shape:
Solid
Molecular weight:
575.68
Ref: TM-T6736
| 25mg | 48.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 92.00 € | ||
| 200mg | 148.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Vorapaxar sulfate
CAS:705260-08-8
Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.
Formula:
C29H35FN2O8S
Purity:
99.46% - 99.9%
Color and Shape:
Solid
Molecular weight:
590.66
Ref: TM-T3098
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 528.00 € | ||
| 500mg | 1,159.00 € | ||
| 1mL*10mM (DMSO) | 99.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
(±)-Ibipinabant
CAS:362519-49-1
(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and …
Formula:
C23H20Cl2N4O2S
Purity:
99.28% - 99.83%
Color and Shape:
Solid
Molecular weight:
487.4
Ref: TM-T4654
| 5mg | 50.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 424.00 € | ||
| 200mg | 588.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.
Formula:
C51H79N15O16
Purity:
95.54%
Color and Shape:
Solid
Molecular weight:
1158.26
Ref: TM-TP1882L1
| 1mg | 159.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 520.00 € | ||
| 25mg | 838.00 € | ||
| 50mg | 1,130.00 € | ||
| 100mg | 1,549.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Cyproheptadine hydrochloride
CAS:969-33-5
Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine …
Formula:
C21H21N·HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
323.86
Ref: TM-T6814
| 100mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
Purity:
98%
Molecular weight:
N/A
Ref: TM-TP1148L
| 1mg | 378.00 € | ||
| 5mg | 850.00 € | ||
| 10mg | 1,273.00 € | ||
| 25mg | 2,292.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formula:
C51H65N9O10
Purity:
97.86%
Color and Shape:
Liquid
Molecular weight:
964.12
Ref: TM-T22811L
| 1mg | 363.00 € | ||
| 2mg | 515.00 € | ||
| 5mg | 775.00 € | ||
| 10mg | 1,035.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,090.00 € | ||
| 100mg | 2,822.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist
Formula:
C37H48F6N8O11
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
894.81
Ref: TM-T7740
| 1mg | 48.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 411.00 € | ||
| 100mg | 607.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Vipadenant
CAS:442908-10-3
Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for …
Formula:
C16H15N7O
Purity:
97.25% - 97.36%
Color and Shape:
Solid
Molecular weight:
321.34
Ref: TM-T2373
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € | ||
| 500mg | 1,130.00 € | ||
| 1mL*10mM (DMSO) | 359.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Almorexant
CAS:871224-64-5
Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for …
Formula:
C29H31F3N2O3
Purity:
97.75% - 98.02%
Color and Shape:
Solid
Molecular weight:
512.56
Ref: TM-T2613
| 1mg | 47.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 316.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 758.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Oxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
Purity:
99.24%
Molecular weight:
N/A
Ref: TM-TP1976L
| 1mg | 175.00 € | ||
| 5mg | 517.00 € | ||
| 10mg | 842.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 2,270.00 € | ||
| 100mg | 3,068.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Pergolide mesylate
CAS:66104-23-2
Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve …
Formula:
C20H30N2O3S2
Purity:
99.09%
Color and Shape:
White To Off-White Solid
Molecular weight:
410.59
Ref: TM-T2226
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
PNU 22394 hydrochloride
CAS:15923-42-9
PNU 22394 hydrochloride is a 5-HT2C agonist and partial 5-HT2A/5-HT2B agonist
Formula:
C13H17ClN2
Purity:
97.83%
Color and Shape:
Solid
Molecular weight:
236.74
Ref: TM-T23168
| 1mg | 54.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 103.00 € | ||
| 10mg | 148.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 378.00 € | ||
| 100mg | 540.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Fexofenadine hydrochloride
CAS:153439-40-8
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the …
Formula:
C32H39NO4·HCl
Purity:
99.39% - ≥95%
Color and Shape:
Solid
Molecular weight:
538.13
Ref: TM-T1470
| 10mg | 49.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 96.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
