G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Difelikefalin acetate
Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.
Formula:
C38H57N7O8
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
739.9
Ref: TM-TP2501
| 1mg | 95.00 € | ||
| 5mg | 191.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 483.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 895.00 € | ||
| 200mg | 1,180.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ipragliflozin
CAS:761423-87-4
Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.
Formula:
C21H21FO5S
Purity:
99.37% - 99.97%
Color and Shape:
Solid
Molecular weight:
404.45
Ref: TM-T2385
| 1ml | 53.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 91.00 € | ||
| 100mg | 132.00 € | ||
| 200mg | 204.00 € | ||
| 500mg | 429.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BisfluoroModafinil
CAS:90280-13-0
CRL-40940 is a selective dopaminergic reuptake inhibitor
Formula:
C15H13F2NO2S
Purity:
97.61%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T4262
| 1ml | 68.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 312.00 € | ||
| 200mg | 438.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GSK189254A
CAS:720690-73-3
GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and …
Formula:
C21H25N3O2
Purity:
98.04% - 98.71%
Color and Shape:
Solid
Molecular weight:
351.44
Ref: TM-TQ0066
| 1mg | 52.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 122.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 495.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ref: 4Z-G-053001
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
RS-127445 hydrochloride
CAS:199864-86-3
RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : …
Formula:
C17H17ClFN3
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
317.79
Ref: TM-T7519
| 1ml | 35.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 177.00 € | ||
| 200mg | 264.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BIM-23190 aceate
BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be …
Formula:
C59H83N13O14S2
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
1262.5
Ref: TM-T39262L
| 1mg | 182.00 € | ||
| 1ml | 813.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 604.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,738.00 € | ||
| 500mg | 3,468.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = …
Formula:
C59H82F3N13O14
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1254.36
Ref: TM-TP1933
| 1mg | 147.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 455.00 € | ||
| 25mg | 728.00 € | ||
| 50mg | 1,013.00 € | ||
| 100mg | 1,380.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML-097
CAS:743456-83-9
ML-097 (CID-2160985) is a pan activator of Ras-related GTPases
Formula:
C14H11BrO3
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
307.139
Ref: TM-T21970
| 1ml | 45.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 122.00 € | ||
| 100mg | 175.00 € | ||
| 200mg | 256.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MCH(human, mouse, rat)
CAS:128315-56-0
MCH(human, mouse, rat) is a potent endogenous agonist at melanin-concentration hormone (MCH) receptors. MCH increases …
Formula:
C105H160N30O26S4
Purity:
99.55% - 99.55%
Color and Shape:
White Powder
Molecular weight:
2386.84
Ref: TM-TP1996
| 1mg | 212.00 € | ||
| 5mg | 527.00 € | ||
| 10mg | 731.00 € | ||
| 25mg | 1,096.00 € | ||
| 50mg | 1,448.00 € | ||
| 100mg | 1,953.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MBX-2982
CAS:1037792-44-1
MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.
Formula:
C22H24N8OS
Purity:
98% - 99.96%
Color and Shape:
Solid
Molecular weight:
448.54
Ref: TM-T1793
| 1mg | 34.00 € | ||
| 1ml | 73.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 201.00 € | ||
| 50mg | 307.00 € | ||
| 100mg | 432.00 € | ||
| 200mg | 603.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Temanogrel
CAS:887936-68-7
Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
Formula:
C24H28N4O4
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
436.5
Ref: TM-T17033
| 1mg | 67.00 € | ||
| 1ml | 165.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 217.00 € | ||
| 25mg | 363.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 699.00 € | ||
| 200mg | 906.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nitroprusside disodium dihydrate
CAS:13755-38-9
Nitroprusside disodium dihydrate (Sodium Nitroprusside Dihydrate) is a potent vasodilator working through releasing NO spontaneously …
Formula:
C5H4FeN6Na2O3
Purity:
98%
Color and Shape:
Bright Red
Molecular weight:
297.95
Ref: TM-T6991
| 1ml | 53.00 € | ||
| 500mg | 49.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MSX-122
CAS:897657-95-3
MSX-122 is a novel small molecule and partial CXCR4 antagonist, with potent inhibition of CXCR4/CXCL12 …
Formula:
C16H16N6
Purity:
97.02% - 98.78%
Color and Shape:
Solid
Molecular weight:
292.34
Ref: TM-T3992
| 5mg | 63.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 476.00 € | ||
| 500mg | 1,003.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![[Lys8, Lys9]-Neurotensin (8-13) acetate](https://static.cymitquimica.com/products/TM/thumb/T38807L.jpg)
[Lys8, Lys9]-Neurotensin (8-13) acetate
[Lys8, Lys9]-Neurotensin (8-13) acetate, a Neurotensin analog, exerts its analgesic effects through activation of the …
Formula:
C40H68N8O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
821.02
Ref: TM-T38807L
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 464.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,420.00 € | ||
| 1ml*10 (DMSO) | 491.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Men 10376 TFA(135306-85-3,free)
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor …
Formula:
C59H69F3N12O12
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
1195.25
Ref: TM-TP1086
| 1mg | 168.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,762.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LP-211
CAS:1052147-86-0
LP-211 is a brain penetrant selective agonist for a 5-HT7 receptor (Ki: 0.58 nM), and …
Formula:
C30H34N4O
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
466.62
Ref: TM-T5387
| 1ml | 77.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 476.00 € | ||
| 200mg | 680.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
R 396 acetate
R 396 acetate is an NK-2 Tachykinin Receptor Antagonist.
Formula:
C41H55N9O12
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
865.93
Ref: TM-T24697L
| 1mg | 111.00 € | ||
| 2mg | 157.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 356.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 759.00 € | ||
| 100mg | 1,017.00 € | ||
| 200mg | 1,356.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB-203186 hydrochloride
CAS:207572-69-8
SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist
Formula:
C16H20N2O2·HCl
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
308.81
Ref: TM-T23310
| 5mg | 39.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 274.00 € | ||
| 500mg | 603.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LY255283
CAS:117690-79-6
LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of …
Formula:
C19H28N4O3
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
360.45
Ref: TM-T22946
| 1mg | 41.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 630.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
