G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Montelukast
CAS:158966-92-8
Montelukast (Singular), oral asthma med, linked to rare liver injury.
Formula:
C35H36ClNO3S
Purity:
100% - 99.74%
Color and Shape:
Solid
Molecular weight:
586.18
Ref: TM-T1677
| 25mg | 34.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dapiprazole Hydrochloride
CAS:72822-13-0
Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.
Formula:
C19H28ClN5
Purity:
100% - 99.86%
Color and Shape:
Solid
Molecular weight:
361.92
Ref: TM-T3996
| 1ml | 34.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 112.00 € | ||
| 200mg | 169.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bromocriptine mesylate
CAS:22260-51-1
Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with …
Formula:
C33H44BrN5O8S
Purity:
99.76% - 99.87%
Color and Shape:
White Solid
Molecular weight:
750.7
Ref: TM-T5842
| 1ml | 60.00 € | ||
| 100mg | 64.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LUN42518 HCl 47142-51-8(free base)
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
Formula:
C17H20ClN3O
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
317.81
Ref: TM-T8738
| 1mg | 85.00 € | ||
| 1ml | 170.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Hypidone hydrochloride
CAS:1339058-04-6
Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor …
Formula:
C18H23ClN2O2
Purity:
99.82% - 99.93%
Color and Shape:
Solid
Molecular weight:
334.84
Ref: TM-T3648
| 1ml | 81.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 343.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Vortioxetine
CAS:508233-74-7
Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.
Formula:
C18H22N2S
Purity:
99.34% - 99.82%
Color and Shape:
Solid
Molecular weight:
298.45
Ref: TM-T2395
| 1g | 493.00 € | ||
| 1ml | 48.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 121.00 € | ||
| 200mg | 211.00 € | ||
| 500mg | 345.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Atipamezole hydrochloride
CAS:104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist.
Formula:
C14H16N2·HCl
Purity:
96.71%
Color and Shape:
Solid
Molecular weight:
248.75
Ref: TM-T6765
| 1ml | 57.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 231.00 € | ||
| 100mg | 341.00 € | ||
| 200mg | 528.00 € | ||
| 500mg | 824.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nociceptin
CAS:170713-75-4
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide …
Formula:
C79H129N27O22
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
1809.04
Ref: TM-TP1071
| 1mg | 80.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 861.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,341.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Vazegepant hydrochloride
CAS:1414976-20-7
Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine …
Formula:
C36H47ClN8O3
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
675.3
Ref: TM-T8682
| 1mg | 105.00 € | ||
| 1ml | 328.00 € | ||
| 5mg | 224.00 € | ||
| 10mg | 327.00 € | ||
| 25mg | 553.00 € | ||
| 50mg | 791.00 € | ||
| 100mg | 1,093.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![Lys-[Des-Arg9]Bradykinin,TFA](https://static.cymitquimica.com/products/TM/thumb/TP1918L.jpg)
Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 …
Formula:
C54H75F6N13O15
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
1260.24
Ref: TM-TP1918L
| 1mg | 85.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 448.00 € | ||
| 50mg | 644.00 € | ||
| 100mg | 912.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BRL 54443
CAS:57477-39-1
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).
Formula:
C14H18N2O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
230.31
Ref: TM-T2459
| 1ml | 59.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 393.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PF-06882961 Tris
CAS:2230198-03-3
PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C35H41FN6O7
Purity:
98.11% - 99.52%
Color and Shape:
Solid
Molecular weight:
676.7
Ref: TM-T8876
| 1mg | 129.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,318.00 € | ||
| 500mg | 2,626.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous …
Formula:
C51H73N15O11
Purity:
98.60%
Color and Shape:
Solid
Molecular weight:
1072.22
Ref: TM-TP1941L1
| 1mg | 155.00 € | ||
| 5mg | 337.00 € | ||
| 10mg | 506.00 € | ||
| 25mg | 760.00 € | ||
| 50mg | 1,018.00 € | ||
| 100mg | 1,358.00 € | ||
| 200mg | 1,798.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CPI-444
CAS:1202402-40-1
CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse …
Formula:
C20H21N7O3
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
407.43
Ref: TM-T7183
| 1ml | 50.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 305.00 € | ||
| 200mg | 438.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Emedastine
CAS:87233-61-2
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
Formula:
C17H26N4O
Purity:
97.1% - 97.1%
Color and Shape:
Oil
Molecular weight:
302.41
Ref: TM-T3979
| 1mg | 36.00 € | ||
| 1ml | 87.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 409.00 € | ||
| 500mg | 912.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tolnapersine
CAS:70312-00-4
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Formula:
C21H26N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
322.44
Ref: TM-T68023
| 1mg | 125.00 € | ||
| 5mg | 301.00 € | ||
| 10mg | 442.00 € | ||
| 25mg | 864.00 € | ||
| 50mg | 1,176.00 € | ||
| 100mg | 1,824.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![Sar-[D-Phe8]-des-Arg9-Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1917L1.jpg)
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM …
Formula:
C49H70N12O13
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
1035.15
Ref: TM-TP1917L1
| 1mg | 170.00 € | ||
| 5mg | 382.00 € | ||
| 10mg | 566.00 € | ||
| 25mg | 841.00 € | ||
| 50mg | 1,081.00 € | ||
| 100mg | 1,521.00 € | ||
| 200mg | 2,061.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AM281
CAS:202463-68-1
AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and …
Formula:
C21H19Cl2IN4O2
Purity:
100% - 99.2%
Color and Shape:
White To Off-White Solid
Molecular weight:
557.21
Ref: TM-T2264
| 1mg | 49.00 € | ||
| 1ml | 147.00 € | ||
| 2mg | 71.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 164.00 € | ||
| 25mg | 320.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 632.00 € | ||
| 200mg | 849.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CID 16020046
CAS:834903-43-4
CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of …
Formula:
C25H19N3O4
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
425.44
Ref: TM-T4478
| 1ml | 68.00 € | ||
| 2mg | 39.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | 322.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Mizagliflozin
CAS:666843-10-3
Mizagliflozin, a selective SGLT1 inhibitor (Ki 27 nM) with 303x SGLT2 selectivity, is an antidiabetic …
Formula:
C28H44N4O8
Purity:
98.32% - 98.66%
Color and Shape:
Solid
Molecular weight:
564.67
Ref: TM-T16083
| 1mg | 80.00 € | ||
| 1ml | 211.00 € | ||
| 2mg | 103.00 € | ||
| 5mg | 161.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 534.00 € | ||
| 50mg | 764.00 € | ||
| 100mg | 1,049.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
