G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ganirelix Acetate
CAS:123246-29-7
Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist
Formula:
C82H117ClN18O15
Purity:
96.05%
Color and Shape:
Solid
Molecular weight:
1630.4
Ref: TM-TP2337
| 1mg | 84.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 408.00 € | ||
| 50mg | 574.00 € | ||
| 100mg | 776.00 € | ||
| 200mg | 1,029.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Eltoprazine hydrochloride
CAS:98206-09-8
Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B …
Formula:
C12H17ClN2O2
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
256.73
Ref: TM-T7498
| 5mg | 47.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 253.00 € | ||
| 100mg | 369.00 € | ||
| 500mg | 862.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Porcine dynorphin A(1-13) acetate
Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like …
Formula:
C77H130N24O17
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
1664
Ref: TM-TP1179L
| 1mg | 48.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 532.00 € | ||
| 200mg | 720.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Guanfacine hydrochloride
CAS:29110-48-3
Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
Formula:
C9H10Cl3N3O
Purity:
99.72% - 99.89%
Color and Shape:
Solid
Molecular weight:
282.55
Ref: TM-T2150
| 10mg | 35.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 90.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 193.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
PACAP 1-38 acetate
PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), …
Purity:
98.16%
Molecular weight:
N/A
Ref: TM-TP1878L
| 1mg | 157.00 € | ||
| 5mg | 443.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,012.00 € | ||
| 50mg | 1,364.00 € | ||
| 100mg | 1,848.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Dexmedetomidine hydrochloride
CAS:145108-58-3
Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.
Formula:
C13H16N2·HCl
Purity:
100.00% - 99.86%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
236.74
Ref: TM-T6466
| 5mg | 41.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 157.00 € | ||
| 100mg | 222.00 € | ||
| 200mg | 333.00 € | ||
| 500mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
(S)-Amisulpride
CAS:71675-92-8
(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.
Formula:
C17H27N3O4S
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
369.48
Ref: TM-T26375
| 1mg | 49.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 326.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 699.00 € | ||
| 200mg | 898.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
TC-G 1005
CAS:1415407-60-1
TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).
Formula:
C25H25N3O2
Purity:
98.2% - 99.23%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T8818
| 1mg | 35.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 414.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Plecanatide
CAS:467426-54-6
Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) …
Formula:
C65H104N18O26S4
Purity:
97.51%
Color and Shape:
Solid
Molecular weight:
1681.89
Ref: TM-T9080
| 1mg | 78.00 € | ||
| 5mg | 178.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 825.00 € | ||
| 100mg | 1,107.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Methylene Blue
CAS:61-73-4
Methylene Blue (Tetramethylthionine chloride) (IC50 of 1.9 μM) inhibits tau filament formation. And methylene Blue …
Formula:
C16H18ClN3S
Purity:
96.82%
Color and Shape:
Dark Green Crystals Or Powder From Chloroform-Ethyl Ether Green Fine Crystalline Powder
Molecular weight:
319.85
Ref: TM-T6888
| 50mg | 40.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 87.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Guanabenz hydrochloride
CAS:23113-43-1
Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.
Formula:
C8H9Cl3N4
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
267.54
Ref: TM-T21957
| 50mg | 44.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 102.00 € | ||
| 500mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Rotigotine Hydrochloride
CAS:125572-93-2
Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formula:
C19H26ClNOS
Purity:
99.53% - 99.66%
Color and Shape:
Almost White To White Crystalline Powder
Molecular weight:
351.93
Ref: TM-T21446
| 5mg | 43.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 222.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Procaterol hydrochloride
CAS:81262-93-3
Short-acting β2-adrenergic receptor agonist used to treat asthma.
Formula:
C32H48Cl2N4O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
671.65
Ref: TM-T4548
| 1mg | 64.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 777.00 € | ||
| 1mL*10mM (DMSO) | 186.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino …
Formula:
C76H103N15O28S
Purity:
99.35% - 99.82%
Color and Shape:
Solid
Molecular weight:
1706.78
Ref: TM-TP1821L
| 1mg | 170.00 € | ||
| 5mg | 629.00 € | ||
| 10mg | 1,007.00 € | ||
| 25mg | 1,825.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Grp94 Inhibitor-1
CAS:2234897-35-7
Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor (IC50 : 2 nM).
Formula:
C22H28N2O2
Purity:
97.02%
Color and Shape:
Solid
Molecular weight:
352.47
Ref: TM-T7261
| 5mg | 48.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 328.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Terutroban
CAS:165538-40-9
Terutroban, a thromboxane prostaglandin receptor antagonist, affects the progression of atherosclerosis.
Formula:
C20H22ClNO4S
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
407.91
Ref: TM-T5505
| 5mg | 50.00 € | ||
| 10mg | 76.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Talnetant
CAS:174636-32-9
Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and …
Formula:
C25H22N2O2
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
382.45
Ref: TM-T7549
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 479.00 € | ||
| 100mg | 728.00 € | ||
| 1mL*10mM (DMSO) | 142.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.
Formula:
C46H74N14O11
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
999.17
Ref: TM-TP1940L1
| 1mg | 274.00 € | ||
| 2mg | 412.00 € | ||
| 5mg | 620.00 € | ||
| 10mg | 926.00 € | ||
| 25mg | 1,375.00 € | ||
| 50mg | 1,855.00 € | ||
| 100mg | 2,499.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Phenelzine
CAS:51-71-8
Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.
Formula:
C8H12N2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
136.19
Ref: TM-T9540
| 5mg | To inquire | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 200mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Friday 20 Dec 2024
ML339
CAS:2579689-83-9
ML339 a selective inhibitor of CXCR6(IC50 = 140 nM) with no response when screened against …
Formula:
C26H32ClN3O5
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
502
Ref: TM-T9721
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
