G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Pimavanserin
CAS:706779-91-1
Pimavanserin is a potent 5-HT2A inverse agonist, used to treat Parkinson's psychosis.
Formula:
C25H34FN3O2
Purity:
97.84% - 98%
Color and Shape:
Pale Yellow To Pale Orange Solid
Molecular weight:
427.55
Ref: TM-T2076
| 1ml | 34.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 104.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Capromorelin Tartrate
CAS:193273-69-7
Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist …
Formula:
C32H41N5O10
Purity:
97.69%
Color and Shape:
Solid
Molecular weight:
655.7
Ref: TM-TQ0022
| 1ml | 51.00 € | ||
| 5mg | 38.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 307.00 € | ||
| 200mg | 439.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Icatibant Acetate
CAS:138614-30-9
Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of …
Formula:
C61H93N19O15S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1364.57
Ref: TM-T22344
| 1mg | 69.00 € | ||
| 1ml | 373.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 702.00 € | ||
| 100mg | 916.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
(±)-Cannabichromene
CAS:20675-51-8
(±)-Cannabichromene is a major non-psychotropic phytocannabinoid that inhibits endocannabinoid inactivation and activates the TRPA1.
Formula:
C21H30O2
Purity:
96.89% - 99.1%
Color and Shape:
Solid
Molecular weight:
314.46
Ref: TM-TN3575
| 1mg | 167.00 € | ||
| 1ml | 519.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 586.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,233.00 € | ||
| 100mg | 1,662.00 € | ||
| 500mg | 3,333.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
6-fluoro-DL-Tryptophan
CAS:7730-20-3
6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.
Formula:
C11H11FN2O2
Purity:
99.25%
Color and Shape:
Off-White Powder
Molecular weight:
222.22
Ref: TM-T7694
| 1ml | 49.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 71.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nefazodone hydrochloride
CAS:82752-99-6
Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, …
Formula:
C25H33Cl2N5O2
Purity:
99% - 99.86%
Color and Shape:
White Solid
Molecular weight:
506.47
Ref: TM-T3275
| 1ml | 77.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 320.00 € | ||
| 200mg | 465.00 € | ||
| 500mg | 763.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GRK5-IN-2
CAS:1642839-27-7
GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.
Formula:
C20H20N4O4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
380.4
Ref: TM-T9609
| 1ml | 53.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 323.00 € | ||
| 200mg | 451.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GUANABENZ
CAS:5051-62-7
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as …
Formula:
C8H8Cl2N4
Purity:
98.6%
Color and Shape:
White Solid From Acetonitrile Solid
Molecular weight:
231.08
Ref: TM-T5471
| 1ml | 79.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 100.00 € | ||
| 25mg | 175.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 356.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bremelanotide Acetate
CAS:1607799-13-2
Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
Formula:
C52H72N14O12
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1085.22
Ref: TM-T7608
| 1ml | 71.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 193.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as …
Formula:
C40H67N7O10
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
805.9
Ref: TM-TP1085L
| 1mg | 35.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 337.00 € | ||
| 200mg | 479.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Opaganib
CAS:915385-81-8
Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).
Formula:
C23H25ClN2O
Purity:
98.86% - 99.71%
Color and Shape:
Solid
Molecular weight:
380.91
Ref: TM-T6750
| 1mg | 40.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 408.00 € | ||
| 100mg | 602.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BPTU
CAS:870544-59-5
BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).
Formula:
C23H22F3N3O3
Purity:
99.37% - 99.89%
Color and Shape:
Solid
Molecular weight:
445.43
Ref: TM-T4132
| 1mg | 38.00 € | ||
| 1ml | 72.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 233.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 600.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Loxiglumide
CAS:107097-80-3
Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.
Formula:
C21H30Cl2N2O5
Purity:
98% - 99.81%
Color and Shape:
Solid
Molecular weight:
461.38
Ref: TM-T2312
| 1ml | 42.00 € | ||
| 5mg | 40.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 115.00 € | ||
| 50mg | 221.00 € | ||
| 100mg | 389.00 € | ||
| 500mg | 883.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Prazosin
CAS:19216-56-9
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is …
Formula:
C19H21N5O4
Purity:
99.29%
Color and Shape:
White To Tan Powder Solid
Molecular weight:
383.4
Ref: TM-T22406
| 1ml | 52.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 71.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Fuscoside
CAS:131631-89-5
Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
Formula:
C26H31N3O4
Purity:
97.98% - 99.66%
Color and Shape:
Solid
Molecular weight:
449.54
Ref: TM-T4355
| 1ml | 88.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 411.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PSN 375963
CAS:388575-52-8
PSN 375963 (PSN 375963 hydrochloride) hydrochloride is a synthetic agonist of the endogenous ligand for …
Formula:
C17H23N3O
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T23204
| 1ml | 62.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 296.00 € | ||
| 200mg | 422.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Alprenolol hydrochloride
CAS:13707-88-5
Alprenolol hydrochloride is a non-selective blocker of beta, and also is a antagonist of5-HT1A receptor.
Formula:
C15H24ClNO2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
285.81
Ref: TM-T22236
| 1ml | 55.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 68.00 € | ||
| 100mg | 100.00 € | ||
| 200mg | 156.00 € | ||
| 500mg | 333.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Guanabenz hydrochloride
CAS:23113-43-1
Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.
Formula:
C8H9Cl3N4
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
267.54
Ref: TM-T21957
| 1ml | 34.00 € | ||
| 50mg | 44.00 € | ||
| 100mg | 78.00 € | ||
| 200mg | 102.00 € | ||
| 500mg | 169.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
3-Hydroxyoctanoic Acid
CAS:14292-27-4
3-Hydroxyoctanoic Acid, an energy metabolism intermediate, activates orphan receptor GPR109B.
Formula:
C8H16O3
Purity:
97.82% - ≥98%
Color and Shape:
Solid
Molecular weight:
160.21
Ref: TM-T9719
| 5mg | 37.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 187.00 € | ||
| 500mg | 486.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Betazole dihydrochloride
CAS:138-92-1
Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.
Formula:
C5H11Cl2N3
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
184.067
Ref: TM-T8599
| 1mg | 52.00 € | ||
| 1ml | 90.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 502.00 € | ||
| 100mg | 651.00 € | ||
| 200mg | 926.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
