G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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S 38093
CAS:862896-30-8
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
Formula:
C17H24N2O2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
288.38
Ref: TM-T4099
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Prucalopride Succinate
CAS:179474-85-2
Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM …
Formula:
C18H26ClN3O3·C4H6O4
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
485.96
Ref: TM-T6958
| 10mg | 47.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 111.00 € | ||
| 200mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and …
Purity:
98.27%
Molecular weight:
N/A
Ref: TM-TP2071L
| 1mg | 299.00 € | ||
| 5mg | 654.00 € | ||
| 10mg | 881.00 € | ||
| 25mg | 1,312.00 € | ||
| 50mg | 1,783.00 € | ||
| 100mg | 2,411.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Protease-Activated Receptor-2, amide
CAS:190383-13-2
Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)
Formula:
C28H54N8O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
614.78
Ref: TM-T7513
| 2mg | 52.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 282.00 € | ||
| 100mg | 421.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Deltorphin I
CAS:122752-15-2
Deltorphin I is an agonist of δ-opioid receptor.
Formula:
C37H52N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
768.86
Ref: TM-T7637
| 1mg | 62.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 505.00 € | ||
| 100mg | 720.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Etelcalcetide hydrochloride
CAS:1334237-71-6
Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary …
Formula:
C38H73N21O10S2HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1353.33
Ref: TM-TP1236
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 535.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Bradykinin (2-9)
CAS:16875-11-9
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.
Formula:
C44H61N11O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
904.02
Ref: TM-TP1181
| 1mg | 52.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 162.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 394.00 € | ||
| 100mg | 572.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
VUF10460
CAS:1028327-66-3
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Formula:
C15H19N5
Purity:
98.68% - 99.53%
Color and Shape:
Solid
Molecular weight:
269.34
Ref: TM-T3963
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 365.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Vanoxerine dihydrochloride
CAS:67469-78-7
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 …
Formula:
C28H34Cl2F2N2O
Purity:
97.1%
Color and Shape:
White Solid
Molecular weight:
523.49
Ref: TM-T7153
| 10mg | 51.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 172.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Desmopressin acetate (16679-58-6 free base)
CAS:62288-83-9
Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine …
Formula:
C48H68N14O14S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1129.26
Ref: TM-T5144
| 1mg | 49.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 527.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
MK-1064
CAS:1207253-08-4
MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).
Formula:
C24H20ClN5O3
Purity:
99.19% - 99.88%
Color and Shape:
Solid
Molecular weight:
461.9
Ref: TM-T3722
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 453.00 € | ||
| 100mg | 730.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Oxytocin acetate
CAS:6233-83-6
Oxytocin acetate (α-Hypophamine acetate) is a mammalian neurohypophysial hormone, a ligand of oxytocin receptor.
Formula:
C45H70N12O14S2
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
1067.23
Ref: TM-T5145
| 5mg | 49.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 185.00 € | ||
| 1mL*10mM (DMSO) | 80.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Vortioxetine hydrobromide
CAS:960203-27-4
Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 …
Formula:
C18H22N2S·HBr
Purity:
100% - 99.89%
Color and Shape:
Solid
Molecular weight:
379.36
Ref: TM-T2395L
| 25mg | 41.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | 81.00 € | ||
| 500mg | 204.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
M617 acetate
M617 acetate is a selective agonist of galanin receptor 1 (GAL1).
Formula:
C112H161N29O28
Purity:
96.02%
Color and Shape:
Liquid
Molecular weight:
2361.65
Ref: TM-TP1993L
| 1mg | 261.00 € | ||
| 5mg | 548.00 € | ||
| 10mg | 731.00 € | ||
| 25mg | 1,090.00 € | ||
| 50mg | 1,466.00 € | ||
| 100mg | 1,988.00 € | ||
| 200mg | 2,683.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
SHU 9119 acetate
SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, …
Formula:
C56H75N15O11
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
1134.29
Ref: TM-T16879L
| 1mg | 96.00 € | ||
| 5mg | 357.00 € | ||
| 10mg | 534.00 € | ||
| 25mg | 858.00 € | ||
| 50mg | 1,174.00 € | ||
| 1mL*10mM (DMSO) | 611.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Vericiguat
CAS:1350653-20-1
Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.
Formula:
C19H16F2N8O2
Purity:
98.86% - 99.6%
Color and Shape:
Solid
Molecular weight:
426.38
Ref: TM-T17226
| 1mg | 47.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 256.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 591.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
SRT3109
CAS:1204707-71-0
SRT3109 is a CXCR2 ligand used in the treatment of chemokine mediated diseases and conditions.
Formula:
C18H23F2N5O4S2
Purity:
99.65% - 99.92%
Color and Shape:
Solid
Molecular weight:
475.53
Ref: TM-T3047
| 2mg | 41.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 299.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
PEN (human) aceate
PEN (human) aceate, one of the most abundant hypothalamic neuropeptide and derived from the proprotein …
Formula:
C99H163N27O34
Purity:
99.25%
Color and Shape:
Liquid
Molecular weight:
2275.51
Ref: TM-TP1949L
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 464.00 € | ||
| 25mg | 834.00 € | ||
| 50mg | 1,264.00 € | ||
| 100mg | 1,866.00 € | ||
| 200mg | 2,778.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Tandospirone citrate
CAS:112457-95-1
Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : …
Formula:
C27H37N5O9
Purity:
97.84% - 99.83%
Color and Shape:
Solid
Molecular weight:
575.61
Ref: TM-T7412
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 362.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.
Formula:
C60H94N16O15S2
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
1343.61
Ref: TM-TP1922L1
| 1mg | 130.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 425.00 € | ||
| 25mg | 702.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
