G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
Formula:
C25H31N3O7
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
485.53
Ref: TM-T21660L
| 1mg | 35.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 221.00 € | ||
| 100mg | 332.00 € | ||
| 200mg | 497.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Methylene Blue trihydrate
CAS:7220-79-3
Dark green, bronze-lustered Methylene Blue trihydrate is a deep blue dye in water/alcohol, used in …
Formula:
C16H24ClN3O3S
Purity:
95.42% - 98.91%
Color and Shape:
Dark Green Solid
Molecular weight:
373.9
Ref: TM-T0006
| 10g | 49.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Phentolamine
CAS:50-60-2
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
Formula:
C17H19N3O
Purity:
100% - 99.86%
Color and Shape:
Crystals Solid
Molecular weight:
281.35
Ref: TM-T8348
| 5mg | 53.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
UNBS5162
CAS:956590-23-1
UNBS5162 (UNBS-5162) is a novel naphthalimide that decreases CXCL chemokine expression in experimental prostate cancers.
Formula:
C17H18N4O3
Purity:
98.37% - 99.97%
Color and Shape:
Solid
Molecular weight:
326.35
Ref: TM-T2477
| 1mg | 39.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 336.00 € | ||
| 100mg | 534.00 € | ||
| 200mg | 778.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
SB 204741
CAS:152239-46-8
SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.
Formula:
C14H14N4OS
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
286.35
Ref: TM-T23312
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 655.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
![1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID](https://static.cymitquimica.com/products/TM/thumb/T8913.jpg)
1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID
CAS:260555-42-8
1-(2,3-DIHYDRO-BENZO[1,4]DIOXIN-6-YL)-5-OXO-PYRROLIDINE-3-CARBOXYLIC ACID targets GRK2.
Formula:
C13H13NO5
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
263.25
Ref: TM-T8913
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 164.00 € | ||
| 200mg | 238.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
GW9508
CAS:885101-89-3
GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in …
Formula:
C22H21NO3
Purity:
97.89% - 99.19%
Color and Shape:
Solid
Molecular weight:
347.41
Ref: TM-T1781
| 10mg | 34.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 83.00 € | ||
| 100mg | 136.00 € | ||
| 200mg | 195.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
ACTH 1-14 acetate(25696-21-3 free base)
ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.
Formula:
C79H113N21O22S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1740.96
Ref: TM-TP1238L
| 1mg | 50.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | 380.00 € | ||
| 100mg | 540.00 € | ||
| 200mg | 713.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Fuscoside
CAS:131631-89-5
Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value …
Formula:
C26H31N3O4
Purity:
97.98% - 99.66%
Color and Shape:
Solid
Molecular weight:
449.54
Ref: TM-T4355
| 2mg | 56.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 411.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
GRK5-IN-2
CAS:1642839-27-7
GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.
Formula:
C20H20N4O4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
380.4
Ref: TM-T9609
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 323.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
(±)-Cannabichromene
CAS:20675-51-8
(±)-Cannabichromene is a major non-psychotropic phytocannabinoid that inhibits endocannabinoid inactivation and activates the TRPA1.
Formula:
C21H30O2
Purity:
96.89% - 99.1%
Color and Shape:
Solid
Molecular weight:
314.46
Ref: TM-TN3575
| 1mg | 167.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 586.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,233.00 € | ||
| 100mg | 1,662.00 € | ||
| 500mg | 3,333.00 € | ||
| 1mL*10mM (DMSO) | 519.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Icatibant Acetate
CAS:138614-30-9
Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of …
Formula:
C61H93N19O15S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1364.57
Ref: TM-T22344
| 1mg | 69.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 702.00 € | ||
| 100mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 373.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
AM281
CAS:202463-68-1
AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and …
Formula:
C21H19Cl2IN4O2
Purity:
100% - 99.2%
Color and Shape:
White To Off-White Solid
Molecular weight:
557.21
Ref: TM-T2264
| 1mg | 84.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,079.00 € | ||
| 500mg | 2,135.00 € | ||
| 1mL*10mM (DMSO) | 242.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Emedastine
CAS:87233-61-2
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
Formula:
C17H26N4O
Purity:
97.1% - 97.1%
Color and Shape:
Oil
Molecular weight:
302.41
Ref: TM-T3979
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 409.00 € | ||
| 500mg | 912.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
![Lys-[Des-Arg9]Bradykinin,TFA](https://static.cymitquimica.com/products/TM/thumb/TP1918L.jpg)
Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 …
Formula:
C54H75F6N13O15
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
1260.24
Ref: TM-TP1918L
| 1mg | 86.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 647.00 € | ||
| 100mg | 921.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Vazegepant hydrochloride
CAS:1414976-20-7
Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine …
Formula:
C36H47ClN8O3
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
675.3
Ref: TM-T8682
| 1mg | 105.00 € | ||
| 5mg | 224.00 € | ||
| 10mg | 327.00 € | ||
| 25mg | 553.00 € | ||
| 50mg | 791.00 € | ||
| 100mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 328.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
LUN42518 HCl 47142-51-8(free base)
LUN42518 HCl is an analogue of phentolamine. Phentolamine is a nonselective alpha-adrenergic antagonist.
Formula:
C17H20ClN3O
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
317.81
Ref: TM-T8738
| 1mg | 85.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Bromocriptine mesylate
CAS:22260-51-1
Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with …
Formula:
C33H44BrN5O8S
Purity:
99.76% - 99.87%
Color and Shape:
White Solid
Molecular weight:
750.7
Ref: TM-T5842
| 100mg | 64.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Men 10376 TFA(135306-85-3,free)
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor …
Formula:
C59H69F3N12O12
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
1195.25
Ref: TM-TP1086
| 1mg | 170.00 € | ||
| 5mg | 421.00 € | ||
| 10mg | 618.00 € | ||
| 25mg | 926.00 € | ||
| 50mg | 1,295.00 € | ||
| 100mg | 1,773.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
MSX-122
CAS:897657-95-3
MSX-122 is a novel small molecule and partial CXCR4 antagonist, with potent inhibition of CXCR4/CXCL12 …
Formula:
C16H16N6
Purity:
97.02% - 98.78%
Color and Shape:
Solid
Molecular weight:
292.34
Ref: TM-T3992
| 5mg | 63.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 186.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 481.00 € | ||
| 500mg | 1,003.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
