G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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LY2795050
CAS:1346133-08-1
LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).
Formula:
C23H22ClN3O2
Purity:
97.77%
Color and Shape:
Solid
Molecular weight:
407.89
Ref: TM-TQ0091
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 292.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Methiothepin mesylate
CAS:74611-28-2
Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an …
Formula:
C21H28N2O3S3
Purity:
98% - 99.92%
Color and Shape:
Solid
Molecular weight:
452.65
Ref: TM-T2190
| 5mg | 36.00 € | ||
| 10mg | 54.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dolasetron
CAS:115956-12-2
Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and …
Formula:
C19H20N2O3
Purity:
99.74% - 99.86%
Color and Shape:
White Powder
Molecular weight:
324.37
Ref: TM-T4568
| 5mg | 47.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 276.00 € | ||
| 500mg | 680.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
5-Hydroxy-1-methylhydantoin
CAS:84210-26-4
5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.
Formula:
C4H6N2O3
Purity:
99.99%
Color and Shape:
Solid
Molecular weight:
130.1
Ref: TM-T28222
| 1g | 1,097.00 € | ||
| 2mg | 36.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 349.00 € | ||
| 500mg | 815.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ESI-09
CAS:263707-16-0
ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and …
Formula:
C16H15ClN4O2
Purity:
98.48% - 99.57%
Color and Shape:
Solid
Molecular weight:
330.77
Ref: TM-T2244
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 297.00 € | ||
| 100mg | 448.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neurotensin
CAS:39379-15-2
Neurotensin, a 13 amino acid peptide, regulates LH and prolactin, interacts with dopamine system.
Formula:
C78H121N21O20
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1672.92
Ref: TM-TP1310
| 1mg | 56.00 € | ||
| 2mg | 87.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 426.00 € | ||
| 50mg | 612.00 € | ||
| 100mg | 859.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Arformoterol Tartrate
CAS:200815-49-2
Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.
Formula:
C23H30N2O10
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
494.49
Ref: TM-T22245
| 5mg | 60.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 147.00 € | ||
| 50mg | 217.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 476.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ANP(1-28) Acetate (human, porcine)
CAS:1366000-58-9
Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.
Formula:
C129H207N45O41S3
Purity:
98.24%
Color and Shape:
Solid
Molecular weight:
3140.5
Ref: TM-TP1220L
| 25mg | 62.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMS 182874 hydrochloride
CAS:1215703-04-0
BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.
Formula:
C17H20ClN3O3S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
381.88
Ref: TM-T21790
| 1mg | 79.00 € | ||
| 2mg | 93.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 208.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 486.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 912.00 € | ||
| 1mL*10mM (DMSO) | 149.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
5-Benzyloxygramine
CAS:1453-97-0
5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus …
Formula:
C18H20N2O
Purity:
96.33%
Color and Shape:
Solid
Molecular weight:
280.36
Ref: TM-T35841
| 100mg | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TCS-OX2-29
CAS:372523-75-6
TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold …
Formula:
C23H31N3O3
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
397.51
Ref: TM-T4965
| 2mg | 46.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 261.00 € | ||
| 100mg | 467.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CCG-50014
CAS:883050-24-6
CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.
Formula:
C16H13FN2O2S
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
316.35
Ref: TM-T6434
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 393.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dazoxiben
CAS:74226-22-5
Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase
Formula:
C12H13ClN2O3
Purity:
99.99%
Color and Shape:
Solid
Molecular weight:
268.7
Ref: TM-T7968
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 248.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 508.00 € | ||
| 500mg | 1,085.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
S1p receptor agonist 1
CAS:1514888-56-2
S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.
Formula:
C23H24FN3O3
Purity:
99.07% - 99.90%
Color and Shape:
Solid
Molecular weight:
409.45
Ref: TM-T4031
| 1mg | 46.00 € | ||
| 5mg | 127.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 540.00 € | ||
| 100mg | 743.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AR 231453
CAS:733750-99-7
Azenosertib (ZN-c3) is an orally active, specific GPR119 agonist. Cost-effective and quality-assured.
Formula:
C21H24FN7O5S
Purity:
99.31% - 99.45%
Color and Shape:
Solid
Molecular weight:
505.52
Ref: TM-T8329
| 1mg | 35.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 330.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TRAP-6
CAS:141136-83-6
TRAP-6 (Thrombin Receptor Activator Peptide 6)(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
Formula:
C34H56N10O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
748.87
Ref: TM-T7625
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 405.00 € | ||
| 100mg | 587.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Netupitant
CAS:290297-26-6
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).
Formula:
C30H32F6N4O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
578.59
Ref: TM-T6905
| 5mg | 51.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 195.00 € | ||
| 100mg | 351.00 € | ||
| 200mg | 519.00 € | ||
| 500mg | 826.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
β-CGRP, human acetate
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying …
Formula:
C164H271N51O50S3
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
3853.46
Ref: TM-TP2167
| 1mg | 355.00 € | ||
| 5mg | 799.00 € | ||
| 10mg | 1,096.00 € | ||
| 25mg | 1,634.00 € | ||
| 50mg | 2,201.00 € | ||
| 100mg | 2,965.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Batefenterol
CAS:743461-65-6
Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).
Formula:
C40H42ClN5O7
Purity:
97.94% - 98.4%
Color and Shape:
Solid
Molecular weight:
740.24
Ref: TM-T7079
| 1mg | 48.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 602.00 € | ||
| 1mL*10mM (DMSO) | 151.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
RG7713
CAS:920022-47-5
RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.
Formula:
C25H28ClN3O2
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
437.96
Ref: TM-T4141
| 1mg | 59.00 € | ||
| 5mg | 117.00 € | ||
| 10mg | 196.00 € | ||
| 25mg | 332.00 € | ||
| 50mg | 495.00 € | ||
| 100mg | 717.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
