G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Temanogrel
CAS:887936-68-7
Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).
Formula:
C24H28N4O4
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
436.5
Ref: TM-T17033
| 1mg | 67.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 217.00 € | ||
| 25mg | 363.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 699.00 € | ||
| 200mg | 906.00 € | ||
| 1mL*10mM (DMSO) | 165.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MBX-2982
CAS:1037792-44-1
MBX-2982 is a selective, orally-available GPR119 agonist, used for the treatment of diabetes.
Formula:
C22H24N8OS
Purity:
98% - 99.96%
Color and Shape:
Solid
Molecular weight:
448.54
Ref: TM-T1793
| 1mg | 50.00 € | ||
| 2mg | 71.00 € | ||
| 5mg | 106.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 525.00 € | ||
| 100mg | 738.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ipragliflozin
CAS:761423-87-4
Ipragliflozin (ASP1941) is under investigation in Type 2 Diabetes and Diabetes Mellitus, Type 2.
Formula:
C21H21FO5S
Purity:
99.37% - 99.97%
Color and Shape:
Solid
Molecular weight:
404.45
Ref: TM-T2385
| 25mg | 56.00 € | ||
| 50mg | 91.00 € | ||
| 100mg | 132.00 € | ||
| 200mg | 204.00 € | ||
| 500mg | 429.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TC14012 acetate
TC14012 acetate is a serum-stable derivative of T140 which is a selective and peptidomimetic CXCR4 …
Formula:
C92H144N34O21S2
Purity:
98.33% - 99.71%
Color and Shape:
Solid
Molecular weight:
2126.47
Ref: TM-TP2112L
| 1mg | 83.00 € | ||
| 5mg | 275.00 € | ||
| 10mg | 442.00 € | ||
| 25mg | 721.00 € | ||
| 50mg | 1,019.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GSK2018682
CAS:1034688-30-6
GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).
Formula:
C22H21ClN4O4
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
440.88
Ref: TM-T7360
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 398.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
T-1095
CAS:209746-59-8
T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) …
Formula:
C26H28O11
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
516.49
Ref: TM-T9590
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 387.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
idalopirdine
CAS:467459-31-0
Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for …
Formula:
C20H19F5N2O
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
398.37
Ref: TM-T7103
| 1mg | 88.00 € | ||
| 2mg | 117.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 251.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | 622.00 € | ||
| 100mg | 887.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MEN 10207 acetate
MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.
Formula:
C59H72N14O12
Purity:
99.18%
Color and Shape:
Liquid
Molecular weight:
1169.29
Ref: TM-T24446L
| 1mg | 143.00 € | ||
| 5mg | 314.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 737.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,412.00 € | ||
| 500mg | 2,767.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[Leu31,Pro34]-Neuropeptide Y (porcine)](https://static.cymitquimica.com/products/TM/thumb/TP2206.jpg)
[Leu31,Pro34]-Neuropeptide Y (porcine)
CAS:125580-28-1
[Leu31,Pro34]-Neuropeptide Y (porcine), is a selective and high affinity agonist of neuropeptide Y (NPY) Y1 …
Formula:
C190H286N54O56
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
4223
Ref: TM-TP2206
| 1mg | 63.00 € | ||
| 5mg | 180.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 456.00 € | ||
| 50mg | 608.00 € | ||
| 100mg | 830.00 € | ||
| 500mg | 1,662.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Oxytocin acetate
CAS:6233-83-6
Oxytocin acetate (α-Hypophamine acetate) is a mammalian neurohypophysial hormone, a ligand of oxytocin receptor.
Formula:
C45H70N12O14S2
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
1067.23
Ref: TM-T5145
| 5mg | 49.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 185.00 € | ||
| 1mL*10mM (DMSO) | 80.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
yangonin
CAS:500-62-9
Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.
Formula:
C15H14O4
Purity:
98.82% - 99.55%
Color and Shape:
Pale Yellow Powder
Molecular weight:
258.27
Ref: TM-T3S0738
| 1mg | 69.00 € | ||
| 5mg | 133.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 721.00 € | ||
| 1mL*10mM (DMSO) | 176.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Melitracen hydrochloride
CAS:10563-70-9
Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist …
Formula:
C21H26ClN
Purity:
99.82%
Color and Shape:
Crystalline Solid
Molecular weight:
327.9
Ref: TM-T4274
| 10mg | 46.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 114.00 € | ||
| 200mg | 167.00 € | ||
| 500mg | 272.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
2,3-Butanediol
CAS:513-85-9
2,3-Butanediol is a butanediol derived from the bioconversion of natural resources which has great potential …
Formula:
C4H10O2
Purity:
98.64% - ≥95%
Color and Shape:
Nearly Colorless Crystalline Solid Or Liquid Solid
Molecular weight:
90.12
Ref: TM-T19094
| 1g | 116.00 € | ||
| 100mg | 47.00 € | ||
| 500mg | 89.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AM-2232
CAS:335161-19-8
AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.
Formula:
C24H20N2O
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
352.43
Ref: TM-T21450
| 1ml | 220.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Urotensin II (114-124), human acetate
Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor …
Formula:
C66H89N13O20S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1448.63
Ref: TM-TP1737L
| 1mg | 182.00 € | ||
| 5mg | 454.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,012.00 € | ||
| 50mg | 1,384.00 € | ||
| 100mg | 1,838.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DJ-V-159
CAS:2253744-53-3
DJ-V-159 is a GPRC6A agonist, targeting the G protein-coupled receptor family C group 6 member …
Formula:
C24H12F6N4O2
Purity:
99.85% - 99.96%
Color and Shape:
Solid
Molecular weight:
502.37
Ref: TM-T5100
| 2mg | 36.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 427.00 € | ||
| 500mg | 931.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Nuciferine
CAS:475-83-2
Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.
Formula:
C19H21NO2
Purity:
98.76% - 99.18%
Color and Shape:
Solid
Molecular weight:
295.38
Ref: TM-T3369
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 251.00 € | ||
| 500mg | 611.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Naratriptan
CAS:121679-13-8
Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment …
Formula:
C17H25N3O2S
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
335.47
Ref: TM-T8666
| 1mg | 41.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 374.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tesmilifene fumarate
CAS:1185241-83-1
Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
Formula:
C23H29NO5
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T22746
| 5mg | 45.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 240.00 € | ||
| 200mg | 355.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Secretin (33-59), rat
CAS:121028-49-7
Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a …
Formula:
C129H216N42O42
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
3027.35
Ref: TM-TP1039
| 1mg | 100.00 € | ||
| 5mg | 239.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 539.00 € | ||
| 50mg | 748.00 € | ||
| 100mg | 1,010.00 € | ||
| 200mg | 1,356.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
