G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Benorilate
CAS:5003-48-5
Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and …
Formula:
C17H15NO5
Purity:
98.39% - 99.56%
Color and Shape:
Solid
Molecular weight:
313.3
Ref: TM-T3276
| 1g | 38.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Lodoxamide
CAS:53882-12-5
Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in …
Formula:
C11H6ClN3O6
Purity:
99.13% - 99.81%
Color and Shape:
Solid
Molecular weight:
311.63
Ref: TM-T4566
| 1ml | 51.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 319.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
DOPEXAMINE
CAS:86197-47-9
Dopexamine is a dopaminergic agonist
Formula:
C22H32N2O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
356.5
Ref: TM-T8653
| 1mg | 128.00 € | ||
| 1ml | 305.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 697.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,319.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Fasiglifam
CAS:1000413-72-8
Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.
Formula:
C29H32O7S
Purity:
99.61% - 99.82%
Color and Shape:
Solid
Molecular weight:
524.63
Ref: TM-T2351
| 1mg | 49.00 € | ||
| 1ml | 123.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 459.00 € | ||
| 100mg | 554.00 € | ||
| 200mg | 802.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Galnon TFA
CAS:1217448-19-5
Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 …
Formula:
C42H47F3N4O8
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
792.84
Ref: TM-T8559
| 1mg | 85.00 € | ||
| 1ml | 113.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tetrahydromagnolol
CAS:20601-85-8
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
Formula:
C18H22O2
Purity:
100% - 99.82%
Color and Shape:
Solid
Molecular weight:
270.37
Ref: TM-TN2268
| 1ml | 67.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 84.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CYM-5520
CAS:1449747-00-5
CYM-5520 is a noncompetitive allosteric agonist of S1P2
Formula:
C21H19N3O2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T22703
| 1mg | 47.00 € | ||
| 1ml | 103.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 251.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 554.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Histrelin acetate
CAS:220810-26-4
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.
Formula:
C68H90N18O14
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
1383.55
Ref: TM-TP2107L
| 1mg | 87.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 455.00 € | ||
| 50mg | 637.00 € | ||
| 100mg | 900.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GSK163090
CAS:844903-58-8
GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for …
Formula:
C25H29N5O
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
415.53
Ref: TM-TQ0311
| 1mg | 36.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Buserelin Acetate (57982-77-1 free base)
CAS:68630-75-1
Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
Formula:
C62H90N16O15
Purity:
99.23% - 99.78%
Color and Shape:
Solid
Molecular weight:
1299.48
Ref: TM-TP1307
| 1mg | 41.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Mosapride Citrate
CAS:112885-42-4
Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.
Formula:
C21H25ClFN3O3·C6H8O7
Purity:
99.88%
Color and Shape:
White Powder
Molecular weight:
614.02
Ref: TM-T6597
| 1ml | 53.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 248.00 € | ||
| 500mg | 417.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Vanoxerine dihydrochloride
CAS:67469-78-7
Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 …
Formula:
C28H34Cl2F2N2O
Purity:
97.1%
Color and Shape:
White Solid
Molecular weight:
523.49
Ref: TM-T7153
| 1ml | 37.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 172.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS:4815-38-7
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)
Formula:
C14H15NO2S
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
261.34
Ref: TM-T8603
| 1ml | 50.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 226.00 € | ||
| 200mg | 335.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Intepirdine
CAS:607742-69-8
Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment …
Formula:
C19H19N3O2S
Purity:
95.19% - 98.99%
Color and Shape:
Solid
Molecular weight:
353.44
Ref: TM-T1774
| 1ml | 43.00 € | ||
| 5mg | 39.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 250.00 € | ||
| 200mg | 355.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Enavogliflozin
CAS:1415472-28-4
Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.
Formula:
C24H27ClO6
Purity:
97.81%
Color and Shape:
Solid
Molecular weight:
446.92
Ref: TM-T38843
| 1mg | 153.00 € | ||
| 1ml | 413.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 580.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,374.00 € | ||
| 100mg | 1,830.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GR 125743
CAS:148547-33-5
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
Formula:
C25H28N4O2
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
416.52
Ref: TM-T8737
| 1mg | 42.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 510.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MF-766
CAS:1050656-06-8
MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with …
Formula:
C27H21F3N2O3
Purity:
98% - 98.06%
Color and Shape:
Solid
Molecular weight:
478.46
Ref: TM-T9622
| 1mg | 51.00 € | ||
| 1ml | 110.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 164.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 451.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 839.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SHU 9119 acetate
SHU 9119 acetate: hMC3R & hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, …
Formula:
C56H75N15O11
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
1134.29
Ref: TM-T16879L
| 1mg | 96.00 € | ||
| 1ml | 611.00 € | ||
| 5mg | 357.00 € | ||
| 10mg | 534.00 € | ||
| 25mg | 858.00 € | ||
| 50mg | 1,174.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
R 59-022
CAS:93076-89-2
R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus …
Formula:
C27H26FN3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
459.58
Ref: TM-T16709
| 1mg | 37.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 775.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
FAUC 213
CAS:337972-47-1
FAUC 213 is a selective full antagonist of the dopamine D4 receptor.
Formula:
C18H19ClN4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
326.82
Ref: TM-T24055
| 1mg | 45.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
