G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CYM-5520
CAS:1449747-00-5
CYM-5520 is a noncompetitive allosteric agonist of S1P2
Formula:
C21H19N3O2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T22703
| 1mg | 47.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 251.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 554.00 € | ||
| 1mL*10mM (DMSO) | 103.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tetrahydromagnolol
CAS:20601-85-8
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
Formula:
C18H22O2
Purity:
100% - 99.82%
Color and Shape:
Solid
Molecular weight:
270.37
Ref: TM-TN2268
| 5mg | 54.00 € | ||
| 10mg | 84.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Galnon TFA
CAS:1217448-19-5
Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 …
Formula:
C42H47F3N4O8
Purity:
99.47%
Color and Shape:
Liquid
Molecular weight:
792.84
Ref: TM-T8559
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Fasiglifam
CAS:1000413-72-8
Fasiglifam (TAK875) is a potent, selective and orally bioavailable GPR40 agonist.
Formula:
C29H32O7S
Purity:
99.61% - 99.82%
Color and Shape:
Solid
Molecular weight:
524.63
Ref: TM-T2351
| 1mg | 49.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 459.00 € | ||
| 100mg | 554.00 € | ||
| 200mg | 802.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
DOPEXAMINE
CAS:86197-47-9
Dopexamine is a dopaminergic agonist
Formula:
C22H32N2O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
356.5
Ref: TM-T8653
| 1mg | 128.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 697.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,319.00 € | ||
| 1mL*10mM (DMSO) | 305.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Lodoxamide
CAS:53882-12-5
Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in …
Formula:
C11H6ClN3O6
Purity:
99.13% - 99.81%
Color and Shape:
Solid
Molecular weight:
311.63
Ref: TM-T4566
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 319.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Benorilate
CAS:5003-48-5
Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and …
Formula:
C17H15NO5
Purity:
98.39% - 99.56%
Color and Shape:
Solid
Molecular weight:
313.3
Ref: TM-T3276
| 1g | 38.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Olcegepant
CAS:204697-65-4
Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist …
Formula:
C38H47Br2N9O5
Purity:
96.08%
Color and Shape:
Solid
Molecular weight:
869.65
Ref: TM-T12293L
| 1mg | 37.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 188.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TG4-155
CAS:1164462-05-8
TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective …
Formula:
C23H26N2O4
Purity:
97.20%
Color and Shape:
Solid
Molecular weight:
394.46
Ref: TM-T5482
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 377.00 € | ||
| 100mg | 560.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Niaprazine
CAS:27367-90-4
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.
Formula:
C20H25FN4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
356.44
Ref: TM-T36949
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 299.00 € | ||
| 200mg | 429.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SB225002
CAS:182498-32-4
SB225002 is a potent and selective CXCR2 antagonist inhibiting interleukin IL-8 binding to CXCR2.
Formula:
C13H10BrN3O4
Purity:
96.86% - 98.79%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T1955
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 395.00 € | ||
| 200mg | 603.00 € | ||
| 500mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ML-193
CAS:713121-80-3
ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.
Formula:
C28H25N5O4S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
527.59
Ref: TM-T22103
| 5mg | 46.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dolasetron Mesylate hydrate
CAS:878143-33-0
Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.
Formula:
C20H26N2O7S
Purity:
99.86% - 99.9%
Color and Shape:
Solid
Molecular weight:
438.49
Ref: TM-T2589
| 5mg | 34.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PRX-08066
CAS:866206-54-4
PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective …
Formula:
C19H17ClFN5S
Purity:
98.04% - 98.07%
Color and Shape:
Solid
Molecular weight:
401.89
Ref: TM-T16669
| 1mg | 59.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 732.00 € | ||
| 500mg | 1,514.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ritanserin
CAS:87051-43-2
Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective …
Formula:
C27H25F2N3OS
Purity:
99.45% - 99.89%
Color and Shape:
Solid
Molecular weight:
477.57
Ref: TM-T16759
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 403.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Trimethobenzamide hydrochloride
CAS:554-92-7
Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic …
Formula:
C21H29ClN2O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
424.92
Ref: TM-T5009
| 50mg | 59.00 € | ||
| 100mg | 88.00 € | ||
| 200mg | 110.00 € | ||
| 500mg | 162.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
CRF (6-33) acetate(120066-38-8 free base)
CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.
Formula:
C143H235N41O45S
Purity:
97.12%
Color and Shape:
Solid
Molecular weight:
3280.76
Ref: TM-TP2047L
| 1mg | 354.00 € | ||
| 5mg | 796.00 € | ||
| 10mg | 1,101.00 € | ||
| 25mg | 1,632.00 € | ||
| 50mg | 2,201.00 € | ||
| 100mg | 2,969.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ML417
CAS:1386162-69-1
ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).
Formula:
C22H25N3O3
Purity:
98.81% - 99.42%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T8423
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 181.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 495.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Nociceptin (1-13) amide TFA
Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat …
Formula:
C63H101F3N22O17
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1495.61
Ref: TM-TP1793L
| 1mg | 130.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 425.00 € | ||
| 25mg | 701.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MIPS521
CAS:1146188-19-3
MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.
Formula:
C19H10ClF6NOS
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
449.8
Ref: TM-T9330
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 500.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
