G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Pancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.
Purity:
98.61%
Molecular weight:
N/A
Ref: TM-TP1044L
| 1mg | 218.00 € | ||
| 5mg | 520.00 € | ||
| 10mg | 704.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,402.00 € | ||
| 100mg | 1,896.00 € | ||
| 200mg | 2,564.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Guanabenz Acetate
CAS:23256-50-0
Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.
Formula:
C8H8Cl2N4·C2H4O2
Purity:
99% - 99.83%
Color and Shape:
White Solid From Acetonitrile White Solid
Molecular weight:
291.13
Ref: TM-T6522
| 1ml | 36.00 € | ||
| 500mg | 49.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BMY 7378 dihydrochloride
CAS:21102-95-4
BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of …
Formula:
C22H33Cl2N3O3
Purity:
97.67% - 99.08%
Color and Shape:
Solid
Molecular weight:
458.42
Ref: TM-T3046
| 1ml | 55.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 99.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
FK962
CAS:283167-06-6
FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.
Formula:
C14H17FN2O2
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
264.3
Ref: TM-T7829
| 1mg | 36.00 € | ||
| 1ml | 84.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 108.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 403.00 € | ||
| 200mg | 566.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CRF (6-33) acetate(120066-38-8 free base)
CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.
Formula:
C143H235N41O45S
Purity:
97.12%
Color and Shape:
Solid
Molecular weight:
3280.76
Ref: TM-TP2047L
| 1mg | 347.00 € | ||
| 5mg | 784.00 € | ||
| 10mg | 1,077.00 € | ||
| 25mg | 1,604.00 € | ||
| 50mg | 2,155.00 € | ||
| 100mg | 2,905.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Trimethobenzamide hydrochloride
CAS:554-92-7
Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic …
Formula:
C21H29ClN2O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
424.92
Ref: TM-T5009
| 1g | 139.00 € | ||
| 1ml | 45.00 € | ||
| 50mg | 37.00 € | ||
| 100mg | 51.00 € | ||
| 500mg | 95.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ritanserin
CAS:87051-43-2
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: …
Formula:
C27H25F2N3OS
Purity:
99.45% - 99.89%
Color and Shape:
Solid
Molecular weight:
477.57
Ref: TM-T16759
| 1mg | 40.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 403.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PRX-08066
CAS:866206-54-4
PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective …
Formula:
C19H17ClFN5S
Purity:
98.04% - 98.07%
Color and Shape:
Solid
Molecular weight:
401.89
Ref: TM-T16669
| 1mg | 59.00 € | ||
| 1ml | 140.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 732.00 € | ||
| 500mg | 1,514.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AC 187 Acetate
AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective …
Formula:
C129H209N37O42
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
2950.26
Ref: TM-T21581L
| 1mg | 851.00 € | ||
| 5mg | 1,726.00 € | ||
| 10mg | 2,303.00 € | ||
| 25mg | 3,452.00 € | ||
| 50mg | 4,565.00 € | ||
| 100mg | 6,288.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Landiolol hydrochloride
CAS:144481-98-1
Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.
Formula:
C25H40ClN3O8
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
546.05
Ref: TM-T5028
| 1ml | 52.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 102.00 € | ||
| 100mg | 141.00 € | ||
| 200mg | 203.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the …
Formula:
C54H81N15O14
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
1164.31
Ref: TM-TP1819L
| 1mg | 64.00 € | ||
| 5mg | 161.00 € | ||
| 10mg | 240.00 € | ||
| 25mg | 433.00 € | ||
| 50mg | 630.00 € | ||
| 100mg | 899.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Dolasetron Mesylate hydrate
CAS:878143-33-0
Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.
Formula:
C20H26N2O7S
Purity:
99.86% - 99.9%
Color and Shape:
Solid
Molecular weight:
438.49
Ref: TM-T2589
| 1ml | 51.00 € | ||
| 5mg | 34.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML-193
CAS:713121-80-3
ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.
Formula:
C28H25N5O4S
Purity:
97.74%
Color and Shape:
Solid
Molecular weight:
527.59
Ref: TM-T22103
| 1ml | 63.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.
Formula:
C30H39N5O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
597.66
Ref: TM-T8557
| 1mg | 79.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 769.00 € | ||
| 500mg | 1,533.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
WAY-100635 Monomaleate
CAS:1092679-51-0
WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 …
Formula:
C25H34N4O2·C4H4O4
Purity:
100% - 99.68%
Color and Shape:
Solid
Molecular weight:
538.64
Ref: TM-T2631
| 1ml | 50.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 287.00 € | ||
| 200mg | 415.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat …
Purity:
98.42%
Molecular weight:
N/A
Ref: TM-TP1140L
| 1mg | 95.00 € | ||
| 5mg | 228.00 € | ||
| 10mg | 337.00 € | ||
| 25mg | 538.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 971.00 € | ||
| 200mg | 1,310.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as …
Purity:
97.26%
Molecular weight:
N/A
Ref: TM-TP1137L
| 1mg | 185.00 € | ||
| 5mg | 460.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,747.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Detomidine hydrochloride
CAS:90038-01-0
Detomidine hydrochloride (MPV-253 AII) produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 …
Formula:
C12H14N2·HCl
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
222.71
Ref: TM-T6464
| 1ml | 35.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 147.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB225002
CAS:182498-32-4
SB225002 is a potent and selective CXCR2 antagonist inhibiting interleukin IL-8 binding to CXCR2.
Formula:
C13H10BrN3O4
Purity:
96.86% - 98.79%
Color and Shape:
Solid
Molecular weight:
352.14
Ref: TM-T1955
| 1ml | 53.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 395.00 € | ||
| 200mg | 603.00 € | ||
| 500mg | 922.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Niaprazine
CAS:27367-90-4
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.
Formula:
C20H25FN4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
356.44
Ref: TM-T36949
| 1ml | 62.00 € | ||
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 299.00 € | ||
| 200mg | 429.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
