G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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![[Leu5]-Enkephalin, amide acetate](https://static.cymitquimica.com/products/TM/thumb/TP1113L.jpg)
[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.
Formula:
C30H42N6O8
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
614.69
Ref: TM-TP1113L
| 2mg | 38.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 178.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 401.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MK-3697
CAS:1224846-01-8
MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist …
Formula:
C23H21N5O3S
Purity:
98.15% - 98.4%
Color and Shape:
Solid
Molecular weight:
447.51
Ref: TM-T1913
| 1mg | 52.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 211.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 504.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Metadoxine
CAS:74536-44-0
Metadoxine (Metadoxil) is a neurotransmitter stimulant.
Formula:
C8H11NO3·C5H7NO3
Purity:
100%
Color and Shape:
Off-White Powder
Molecular weight:
298.29
Ref: TM-T3269
| 1g | 110.00 € | ||
| 100mg | 38.00 € | ||
| 200mg | 51.00 € | ||
| 500mg | 83.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TCS 1102
CAS:916141-36-1
TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).
Formula:
C27H26N4O2S
Purity:
99.35% - 99.52%
Color and Shape:
Solid
Molecular weight:
470.59
Ref: TM-T2710
| 5mg | 40.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 178.00 € | ||
| 100mg | 251.00 € | ||
| 200mg | 367.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PD 117519
CAS:96392-15-3
PD 117519 (CI947) is an agonist of adenosine receptor
Formula:
C19H21N5O4
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
383.4
Ref: TM-T7509
| 2mg | 35.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PZM21
CAS:1997387-43-5
PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
Formula:
C19H27N3O2S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
361.5
Ref: TM-T4386
| 1mg | 46.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 295.00 € | ||
| 100mg | 468.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Setipiprant
CAS:866460-33-5
Setipiprant (ACT-129968) is an oral CRTH2 antagonist for asthma/allergy, targeting PGD2-induced inflammation (IC50: 6.0 nM).
Formula:
C24H19FN2O3
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
402.42
Ref: TM-T3520
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 176.00 € | ||
| 200mg | 260.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
TRAP-6 amide acetate
TRAP-6 amide acetate is a PAR-1 thrombin receptor agonist peptide[1].
Formula:
C36H61N11O10
Purity:
98.55%
Color and Shape:
Liquid
Molecular weight:
807.94
Ref: TM-T38852L
| 1mg | 96.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 441.00 € | ||
| 50mg | 628.00 € | ||
| 100mg | 844.00 € | ||
| 200mg | 1,102.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Metiamide
CAS:34839-70-8
Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .
Formula:
C9H16N4S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
244.38
Ref: TM-T7524
| 1mg | 80.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 461.00 € | ||
| 50mg | 675.00 € | ||
| 100mg | 921.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMS986187
CAS:684238-37-7
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
Formula:
C31H34O4
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
470.6
Ref: TM-T8991
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 503.00 € | ||
| 500mg | 1,068.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
M 1145 acetate
M1145 acetate: chimeric peptide, selective GAL2 agonist, Ki=6.55 nM; >90x affinity vs GAL1, 76x vs …
Formula:
C130H209N37O34
Purity:
99.1%
Color and Shape:
Liquid
Molecular weight:
2834.28
Ref: TM-TP1991L
| 1mg | 338.00 € | ||
| 5mg | 726.00 € | ||
| 10mg | 974.00 € | ||
| 25mg | 1,447.00 € | ||
| 50mg | 1,956.00 € | ||
| 100mg | 2,648.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GSK 789472 hydrochloride
CAS:1257326-24-1
GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.
Formula:
C15H22ClN3O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
295.81
Ref: TM-T22817
| 1mg | 43.00 € | ||
| 2mg | 56.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 543.00 € | ||
| 200mg | 717.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GR 125743
CAS:148547-33-5
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
Formula:
C25H28N4O2
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
416.52
Ref: TM-T8737
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 510.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Enavogliflozin
CAS:1415472-28-4
Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.
Formula:
C24H27ClO6
Purity:
97.81%
Color and Shape:
Solid
Molecular weight:
446.92
Ref: TM-T38843
| 1mg | 153.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 580.00 € | ||
| 25mg | 1,009.00 € | ||
| 50mg | 1,374.00 € | ||
| 100mg | 1,830.00 € | ||
| 1mL*10mM (DMSO) | 413.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Intepirdine
CAS:607742-69-8
Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment …
Formula:
C19H19N3O2S
Purity:
95.19% - 98.99%
Color and Shape:
Solid
Molecular weight:
353.44
Ref: TM-T1774
| 5mg | 39.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 250.00 € | ||
| 200mg | 355.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS:4815-38-7
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)
Formula:
C14H15NO2S
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
261.34
Ref: TM-T8603
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 226.00 € | ||
| 200mg | 335.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Mosapride Citrate
CAS:112885-42-4
Mosapride Citrate (TAK-370 citrate), a gastroprokinetic agent, utilizes as a selective 5HT4 agonist.
Formula:
C21H25ClFN3O3·C6H8O7
Purity:
99.88%
Color and Shape:
White Powder
Molecular weight:
614.02
Ref: TM-T6597
| 10mg | 50.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 248.00 € | ||
| 500mg | 417.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Buserelin Acetate (57982-77-1 free base)
CAS:68630-75-1
Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).
Formula:
C62H90N16O15
Purity:
99.23% - 99.78%
Color and Shape:
Solid
Molecular weight:
1299.48
Ref: TM-TP1307
| 1mg | 41.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 435.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GSK163090
CAS:844903-58-8
GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for …
Formula:
C25H29N5O
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
415.53
Ref: TM-TQ0311
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Histrelin acetate
CAS:220810-26-4
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.
Formula:
C68H90N18O14
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
1383.55
Ref: TM-TP2107L
| 1mg | 87.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 459.00 € | ||
| 50mg | 644.00 € | ||
| 100mg | 909.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
