G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CGP71683 hydrochloride
CAS:192322-50-2
CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 …
Formula:
C26H30ClN5O2S
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
512.07
Ref: TM-T5587
| 1mg | 50.00 € | ||
| 1ml | 117.00 € | ||
| 5mg | 103.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 252.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 527.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cetrorelix diacetate
CAS:130143-01-0
Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.
Formula:
C74H100ClN17O18
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
1551.17
Ref: TM-T5520L
| 1mg | 52.00 € | ||
| 1ml | 250.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 287.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 628.00 € | ||
| 500mg | 1,327.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Procaterol hydrochloride
CAS:81262-93-3
Short-acting β2-adrenergic receptor agonist used to treat asthma.
Formula:
C32H48Cl2N4O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
671.65
Ref: TM-T4548
| 1mg | 64.00 € | ||
| 1ml | 186.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 777.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino …
Formula:
C76H103N15O28S
Purity:
99.35% - 99.82%
Color and Shape:
Solid
Molecular weight:
1706.78
Ref: TM-TP1821L
| 1mg | 170.00 € | ||
| 5mg | 629.00 € | ||
| 10mg | 1,007.00 € | ||
| 25mg | 1,825.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB 204741
CAS:152239-46-8
SB 204741 is a selective 5-HT2B antagonist with high affinity and pKi value of 7.1.
Formula:
C14H14N4OS
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
286.35
Ref: TM-T23312
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 147.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 384.00 € | ||
| 200mg | 546.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML339
CAS:2579689-83-9
ML339 a selective inhibitor of CXCR6(IC50 = 140 nM) with no response when screened against …
Formula:
C26H32ClN3O5
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
502
Ref: TM-T9721
| 1mg | 45.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
S 38093
CAS:862896-30-8
S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).
Formula:
C17H24N2O2
Purity:
99.98%
Color and Shape:
Solid
Molecular weight:
288.38
Ref: TM-T4099
| 1ml | 51.00 € | ||
| 2mg | 37.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 323.00 € | ||
| 200mg | 451.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Etelcalcetide hydrochloride
CAS:1334237-71-6
Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary …
Formula:
C38H73N21O10S2HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1353.33
Ref: TM-TP1236
| 1mg | 35.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 535.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
UNBS5162
CAS:956590-23-1
UNBS5162 (UNBS-5162) is a novel naphthalimide that decreases CXCL chemokine expression in experimental prostate cancers.
Formula:
C17H18N4O3
Purity:
98.37% - 99.97%
Color and Shape:
Solid
Molecular weight:
326.35
Ref: TM-T2477
| 1mg | 43.00 € | ||
| 1ml | 129.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 417.00 € | ||
| 100mg | 612.00 € | ||
| 500mg | 1,291.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Phentolamine
CAS:50-60-2
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
Formula:
C17H19N3O
Purity:
100% - 99.86%
Color and Shape:
Crystals Solid
Molecular weight:
281.35
Ref: TM-T8348
| 1ml | 53.00 € | ||
| 5mg | 53.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 177.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Methylene Blue trihydrate
CAS:7220-79-3
Dark green, bronze-lustered Methylene Blue trihydrate is a deep blue dye in water/alcohol, used in …
Formula:
C16H24ClN3O3S
Purity:
95.42% - 98.91%
Color and Shape:
Dark Green Solid
Molecular weight:
373.9
Ref: TM-T0006
| 10g | 49.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
Formula:
C25H31N3O7
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
485.53
Ref: TM-T21660L
| 1ml | 57.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 195.00 € | ||
| 200mg | 291.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tyr-Gly-Gly-Phe-Met-OH
CAS:58569-55-4
Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding …
Formula:
C27H35N5O7S
Purity:
98%
Color and Shape:
White Lyophilised Solid
Molecular weight:
573.66
Ref: TM-T7211
| 1ml | 37.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 177.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MIPS521
CAS:1146188-19-3
MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.
Formula:
C19H10ClF6NOS
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
449.8
Ref: TM-T9330
| 1mg | 38.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 500.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tandospirone citrate
CAS:112457-95-1
Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : …
Formula:
C27H37N5O9
Purity:
97.84% - 99.83%
Color and Shape:
Solid
Molecular weight:
575.61
Ref: TM-T7412
| 1ml | 72.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 362.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Eptapirone
CAS:179756-58-2
Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant …
Formula:
C16H23N7O2
Purity:
99.39% - 99.65%
Color and Shape:
Solid
Molecular weight:
345.4
Ref: TM-T3179
| 1ml | 48.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 67.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 194.00 € | ||
| 100mg | 288.00 € | ||
| 200mg | 416.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nociceptin (1-13) amide TFA
Nociceptin (1-13), amide: ORL1 receptor agonist, pEC50 7.9 (mouse vas deferens), Ki 0.75 nM (rat …
Formula:
C63H101F3N22O17
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1495.61
Ref: TM-TP1793L
| 1mg | 128.00 € | ||
| 5mg | 283.00 € | ||
| 10mg | 423.00 € | ||
| 25mg | 698.00 € | ||
| 50mg | 976.00 € | ||
| 100mg | 1,318.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Rotundine
CAS:483-14-7
Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 …
Formula:
C21H25NO4
Purity:
100% - 99.8%
Color and Shape:
Off-White Solid
Molecular weight:
355.43
Ref: TM-T6648
| 1g | 150.00 € | ||
| 50mg | 42.00 € | ||
| 100mg | 57.00 € | ||
| 500mg | 101.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML417
CAS:1386162-69-1
ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).
Formula:
C22H25N3O3
Purity:
98.81% - 99.42%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T8423
| 1ml | 51.00 € | ||
| 5mg | 38.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 195.00 € | ||
| 100mg | 290.00 € | ||
| 200mg | 419.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MDL 100009
CAS:175673-57-1
MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is …
Formula:
C22H28FNO3
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
373.46
Ref: TM-T22359
| 1mg | 143.00 € | ||
| 1ml | 323.00 € | ||
| 2mg | 182.00 € | ||
| 5mg | 272.00 € | ||
| 10mg | 408.00 € | ||
| 25mg | 632.00 € | ||
| 50mg | 851.00 € | ||
| 100mg | 1,126.00 € | ||
| 200mg | 1,537.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
