G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Trimipramine maleate
CAS:521-78-8
Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.
Formula:
C24H30N2O4
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
410.51
Ref: TM-T1045
| 1ml | 55.00 € | ||
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 73.00 € | ||
| 500mg | 108.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Pericyazine
CAS:2622-26-6
Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.
Formula:
C21H23N3OS
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
365.49
Ref: TM-T16472
| 1mg | 45.00 € | ||
| 1ml | 77.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 380.00 € | ||
| 100mg | 554.00 € | ||
| 500mg | 1,198.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
GSK256073
CAS:862892-90-8
GSK256073 is an orally active GPR109A agonist.
Formula:
C10H13ClN4O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
256.69
Ref: TM-T15432
| 1mg | 72.00 € | ||
| 1ml | 168.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 633.00 € | ||
| 100mg | 900.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Pizotifen
CAS:15574-96-6
Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available …
Formula:
C19H21NS
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
295.44
Ref: TM-T1442
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 77.00 € | ||
| 500mg | 121.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Motixafortide TFA(664334-36-5,Free)
Motixafortide TFA is a CXCR4 antagonist with ~1 nM IC50, promoting AML apoptosis by modulating …
Formula:
C99H145F4N33O21S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
2273.54
Ref: TM-T14665L
| 1mg | 72.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 272.00 € | ||
| 25mg | 435.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 817.00 € | ||
| 200mg | 1,080.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
N6-Cyclohexyladenosine
CAS:36396-99-3
N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.
Formula:
C16H23N5O4
Purity:
99.84% - 99.98%
Color and Shape:
Solid
Molecular weight:
349.38
Ref: TM-T12160
| 1ml | 34.00 € | ||
| 10mg | 34.00 € | ||
| 25mg | 60.00 € | ||
| 50mg | 101.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 213.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Proglumide
CAS:6620-60-6
Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal …
Formula:
C18H26N2O4
Purity:
99.44%
Color and Shape:
White Crystalline Powder
Molecular weight:
334.41
Ref: TM-T1052
| 1ml | 57.00 € | ||
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 117.00 € | ||
| 500mg | 182.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
MRS-1706
CAS:264622-53-9
MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.
Formula:
C27H29N5O5
Purity:
97.95%
Color and Shape:
Solid
Molecular weight:
503.55
Ref: TM-T16136
| 1ml | 51.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 397.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Fexofenadine hydrochloride
CAS:138452-21-8
Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor …
Formula:
C32H40ClNO4
Purity:
100%
Color and Shape:
White Crystalline Powder
Molecular weight:
538.12
Ref: TM-T1470L
| 1ml | 53.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 104.00 € | ||
| 100mg | 138.00 € | ||
| 200mg | 187.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Anandamide
CAS:94421-68-8
Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but …
Formula:
C22H37NO2
Purity:
98.76%
Color and Shape:
Light Yellow Oil
Molecular weight:
347.53
Ref: TM-T14046
| 1ml | 87.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 426.00 € | ||
| 100mg | 625.00 € | ||
| 500mg | 1,333.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Alverine citrate
CAS:5560-59-8
Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.
Formula:
C26H35NO7
Purity:
100% - 99.83%
Color and Shape:
Coa
Molecular weight:
473.57
Ref: TM-T0428
| 1g | 80.00 € | ||
| 1ml | 49.00 € | ||
| 500mg | 48.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Atenolol
CAS:29122-68-7
Atenolol (Tenormin) is a selective β1 receptor antagonist.
Formula:
C14H22N2O3
Purity:
99.07%
Color and Shape:
White Crystalline Powder Solid
Molecular weight:
266.3361
Ref: TM-T0007
| 1ml | 54.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Metipranolol
CAS:22664-55-7
Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic …
Formula:
C17H27NO4
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
309.4
Ref: TM-T8899
| 1ml | 85.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 290.00 € | ||
| 100mg | 473.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Vincamine
CAS:1617-90-9
Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain …
Formula:
C21H26N2O3
Purity:
99.52%
Color and Shape:
White To Almost White Fine Crystalline Powder
Molecular weight:
354.44
Ref: TM-T1286
| 1g | 66.00 € | ||
| 500mg | 53.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Salbutamol
CAS:18559-94-9
Salbutamol (Albuterol) stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that …
Formula:
C13H21NO3
Purity:
91.59% - 99.90%
Color and Shape:
White To Off-White Crystalline Solid Solid
Molecular weight:
239.31
Ref: TM-T1139
| 1g | 133.00 € | ||
| 1ml | 49.00 € | ||
| 50mg | 35.00 € | ||
| 100mg | 49.00 € | ||
| 500mg | 93.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ursodeoxycholic acid
CAS:128-13-2
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
Formula:
C24H40O4
Purity:
98% - 99.8%
Color and Shape:
White - Almost White Solid Powder
Molecular weight:
392.57
Ref: TM-T0700
| 1g | 54.00 € | ||
| 5g | 111.00 € | ||
| 1ml | 65.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Promazine hydrochloride
CAS:53-60-1
Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
Formula:
C17H21ClN2S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
320.88
Ref: TM-T0766
| 1ml | 55.00 € | ||
| 500mg | 54.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
TSHR antagonist S37
CAS:1217616-61-9
TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
Formula:
C25H20N2O3S2
Purity:
98.35%
Color and Shape:
Solid
Molecular weight:
460.57
Ref: TM-T13216
| 1mg | 67.00 € | ||
| 1ml | 175.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 384.00 € | ||
| 50mg | 573.00 € | ||
| 100mg | 817.00 € | ||
| 500mg | 1,653.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ziprasidone hydrochloride
CAS:122883-93-6
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows …
Formula:
C21H22CL2N4OS
Purity:
98.37% - 99.34%
Color and Shape:
Solid
Molecular weight:
449.4
Ref: TM-T0031L
| 1ml | 55.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 163.00 € | ||
| 500mg | 388.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Levocetirizine
CAS:130018-77-8
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a …
Formula:
C21H25ClN2O3
Purity:
98% - 99.9%
Color and Shape:
White Powder
Molecular weight:
388.89
Ref: TM-T1469
| 1ml | 58.00 € | ||
| 5mg | 38.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 169.00 € | ||
| 200mg | 253.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
