G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Docusate sodium
CAS:577-11-7
Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to …
Formula:
C20H37NaO7S
Purity:
99.77%
Color and Shape:
White Wax-Like Solid With Water (Uscg 1999)
Molecular weight:
444.56
Ref: TM-T0929
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € | ||
| 500mg | 120.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Cyproheptadine hydrochloride sesquihydrate
CAS:41354-29-4
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
Formula:
C21H24ClNO
Purity:
100% - 100%
Color and Shape:
White To Slightly Yellowish Crystalline Solid
Molecular weight:
341.88
Ref: TM-T0174
| 500mg | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Risperidone
CAS:106266-06-2
Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 …
Formula:
C23H27FN4O2
Purity:
100%
Color and Shape:
Crystalline Solid
Molecular weight:
410.48
Ref: TM-T0351
| 10mg | 55.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 203.00 € | ||
| 500mg | 338.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
EMPA
CAS:680590-49-2
EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 …
Formula:
C23H26N4O4S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
454.54
Ref: TM-T11186
| 1mg | 51.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 327.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 688.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pheniramine maleate
CAS:132-20-7
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 …
Formula:
C16H20N2·C4H4O4
Purity:
99.79%
Color and Shape:
Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
Molecular weight:
356.42
Ref: TM-T0370
| 25mg | 36.00 € | ||
| 50mg | 45.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 65.00 € | ||
| 500mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Roxatidine Acetate hydrochloride
CAS:93793-83-0
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits …
Formula:
C19H29ClN2O4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
384.9
Ref: TM-T0157
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
2-Bromo-6-methoxynaphthalene
CAS:5111-65-9
2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.
Formula:
C11H9BrO
Purity:
98.8%
Color and Shape:
White To Off-White Powder
Molecular weight:
237.09
Ref: TM-T0663
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MP-A08
CAS:219832-49-2
MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 …
Formula:
C27H25N3O4S2
Purity:
98.04%
Color and Shape:
Solid
Molecular weight:
519.64
Ref: TM-T16128
| 1mg | 46.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 302.00 € | ||
| 100mg | 537.00 € | ||
| 500mg | 1,109.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Agomelatine
CAS:138112-76-2
Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
Formula:
C15H17NO2
Purity:
99.92%
Color and Shape:
White Solid
Molecular weight:
243.3
Ref: TM-T1445
| 5mg | 67.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 732.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Levocarnitine propionate hydrochloride
CAS:119793-66-7
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, …
Formula:
C10H20ClNO4
Purity:
90% - 98%
Color and Shape:
Solid
Molecular weight:
253.72
Ref: TM-T1182
| 25mg | 35.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 500mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Duloxetine hydrochloride
CAS:136434-34-9
Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.
Formula:
C18H20ClNOS
Purity:
100% - 99.97%
Color and Shape:
White Or White Crystalline Powder
Molecular weight:
333.88
Ref: TM-T1471
| 10mg | 52.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 130.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Fezagepras
CAS:1002101-19-0
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist …
Formula:
C13H18O2
Purity:
96.73% - 99.38%
Color and Shape:
Solid
Molecular weight:
206.28
Ref: TM-T12883
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Degarelix acetate(214766-78-6 free base)
CAS:934016-19-0
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
Formula:
C84H107ClN18O18
Purity:
98.66%
Color and Shape:
Liquid
Molecular weight:
1692.34
Ref: TM-T10988L
| 1mg | 75.00 € | ||
| 2mg | 97.00 € | ||
| 5mg | 162.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 468.00 € | ||
| 50mg | 680.00 € | ||
| 100mg | 920.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MRGPRX1 agonist 1
CAS:2377379-39-8
MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
Formula:
C23H21N3O4S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
435.5
Ref: TM-T12104
| 1mg | 87.00 € | ||
| 5mg | 206.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 599.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 228.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BIBO3304 TFA
CAS:191868-14-1
BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).
Formula:
C31H36F3N7O5
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
643.66
Ref: TM-T10539
| 1mg | 95.00 € | ||
| 2mg | 143.00 € | ||
| 5mg | 218.00 € | ||
| 10mg | 385.00 € | ||
| 25mg | 640.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,226.00 € | ||
| 1mL*10mM (DMSO) | 329.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Domperidone
CAS:57808-66-9
Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.
Formula:
C22H24ClN5O2
Purity:
98% - 99.73%
Color and Shape:
Solid
Molecular weight:
425.91
Ref: TM-T0082
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 93.00 € | ||
| 500mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NEO 376
CAS:496921-73-4
NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing …
Formula:
C20H24ClN3O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
357.88
Ref: TM-T12207
| 1mg | 72.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 208.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 504.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 909.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Labetalol hydrochloride
CAS:32780-64-6
Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic …
Formula:
C19H25ClN2O3
Purity:
99.29% - 99.85%
Color and Shape:
Solid
Molecular weight:
364.87
Ref: TM-T0348
| 50mg | 46.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 112.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NTP42
CAS:2055599-51-2
NTP42 is an antagonist of thromboxane A2 (TXA2) receptor(IC50 of 3.278 nM)
Formula:
C25H23F2N3O5S
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
515.53
Ref: TM-T12268
| 1mg | 62.00 € | ||
| 2mg | 89.00 € | ||
| 5mg | 139.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 766.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
