G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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HJC0197
CAS:1383539-73-8
HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.
Formula:
C19H21N3OS
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
339.45
Ref: TM-T15485
| 2mg | 37.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 272.00 € | ||
| 200mg | 411.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BP 897 hydrochloride
CAS:314776-92-6
BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low …
Formula:
C26H32ClN3O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T14767
| 1mg | 36.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Iloperidone
CAS:133454-47-4
Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.
Formula:
C24H27FN2O4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
426.48
Ref: TM-T1539
| 25mg | 47.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 95.00 € | ||
| 200mg | 138.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Zolmitriptan
CAS:139264-17-8
Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, …
Formula:
C16H21N3O2
Purity:
98.8% - 99.91%
Color and Shape:
White Or Kind Of White Powder
Molecular weight:
287.36
Ref: TM-T1092
| 10mg | 62.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 217.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Vilazodone
CAS:163521-12-8
Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.
Formula:
C26H27N5O2
Purity:
99.83%
Color and Shape:
Light Yellow Solid
Molecular weight:
441.52
Ref: TM-T1279
| 1mg | 59.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | 306.00 € | ||
| 1mL*10mM (DMSO) | 151.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Promazine hydrochloride
CAS:53-60-1
Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
Formula:
C17H21ClN2S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
320.88
Ref: TM-T0766
| 500mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Cetirizine dihydrochloride
CAS:83881-52-1
Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.
Formula:
C21H27Cl3N2O3
Purity:
100% - 99.4%
Color and Shape:
Solid
Molecular weight:
461.81
Ref: TM-T0089
| 50mg | 47.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 83.00 € | ||
| 500mg | 103.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Chlorpheniramine maleate
CAS:113-92-8
Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, …
Formula:
C20H23ClN2O4
Purity:
99.67%
Color and Shape:
Odorless White Crystalline Solid Or White Powder With A Bitter Taste
Molecular weight:
390.87
Ref: TM-T1553
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Carbinoxamine Maleate Salt
CAS:3505-38-2
Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and …
Formula:
C20H23ClN2O5
Purity:
99.81%
Color and Shape:
Off-White Solid
Molecular weight:
406.86
Ref: TM-T2222
| 25mg | 46.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 72.00 € | ||
| 200mg | 95.00 € | ||
| 500mg | 181.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BTRX-335140
CAS:2244614-14-8
BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic …
Formula:
C25H32FN5O2
Purity:
98% - 98.45%
Color and Shape:
Solid
Molecular weight:
453.55
Ref: TM-T14835
| 1mg | 105.00 € | ||
| 2mg | 154.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 404.00 € | ||
| 25mg | 835.00 € | ||
| 50mg | 1,368.00 € | ||
| 100mg | 1,867.00 € | ||
| 200mg | 2,612.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Glycerol phenylbutyrate
CAS:611168-24-2
Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is …
Formula:
C33H38O6
Purity:
99.00% - 99.74%
Color and Shape:
Solid
Molecular weight:
530.65
Ref: TM-T15393
| 10mg | 46.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 203.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Clomipramine hydrochloride
CAS:17321-77-6
Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the …
Formula:
C19H23ClN2·HCl
Purity:
99.07% - 99.47%
Color and Shape:
White To Slightly Yellow Crystalline Powder
Molecular weight:
351.31
Ref: TM-T0255
| 25mg | 43.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 72.00 € | ||
| 500mg | 94.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Maprotiline hydrochloride
CAS:10347-81-6
Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.
Formula:
C20H24ClN
Purity:
100% - 99.84%
Color and Shape:
White Powder
Molecular weight:
313.864
Ref: TM-T0172
| 50mg | 45.00 € | ||
| 100mg | 58.00 € | ||
| 200mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Amisulpride
CAS:71675-85-9
Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the …
Formula:
C17H27N3O4S
Purity:
100%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
369.48
Ref: TM-T0811
| 1g | 346.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 68.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 138.00 € | ||
| 500mg | 238.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Timonacic
CAS:444-27-9
Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.
Formula:
C4H7NO2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
133.17
Ref: TM-T0221
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dexpramipexole dihydrochloride
CAS:104632-27-1
Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline …
Formula:
C10H19Cl2N3S
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
284.25
Ref: TM-T11011
| 5mg | 52.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 149.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 369.00 € | ||
| 200mg | 541.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pramipexole
CAS:104632-26-0
Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not …
Formula:
C10H17N3S
Purity:
98% - 99.96%
Color and Shape:
Solid
Molecular weight:
211.33
Ref: TM-T1476
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Triprolidine hydrochloride monohydrate
CAS:6138-79-0
Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
Formula:
C19H25ClN2O
Purity:
99.68% - ≥95%
Color and Shape:
White Crystalline Powder
Molecular weight:
332.87
Ref: TM-T1030
| 10mg | 35.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 138.00 € | ||
| 500mg | 331.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Benztropine mesylate
CAS:132-17-2
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in …
Formula:
C21H25NO·CH4SO3
Purity:
100% - 99.52%
Color and Shape:
White Crystalline Powder; Odourless Or Almost Odourless
Molecular weight:
403.53
Ref: TM-T1336
| 500mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AMG 487
CAS:473719-41-4
AMG 487: potent CXCR3 antagonist, blocks CXCL10/CXCL11 binding, IC50s: 8.0/8.2 nM.
Formula:
C32H28F3N5O4
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
603.59
Ref: TM-T10297L
| 1mg | 52.00 € | ||
| 2mg | 75.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 262.00 € | ||
| 50mg | 391.00 € | ||
| 100mg | 577.00 € | ||
| 1mL*10mM (DMSO) | 153.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
