G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PF-06882961
CAS:2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C31H30FN5O4
Purity:
95.1% - 99.54%
Color and Shape:
Solid
Molecular weight:
555.6
Ref: TM-T12431
| 1mg | 50.00 € | ||
| 1ml | 109.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 427.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Prasugrel
CAS:150322-43-3
Prasugrel (CS-747) is a piperazine derivative and PLATELET AGGREGATION INHIBITOR that is used to prevent …
Formula:
C20H20FNO3S
Purity:
98.62% - 99.76%
Color and Shape:
White Solid
Molecular weight:
373.44
Ref: TM-T0230
| 1ml | 55.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 76.00 € | ||
| 200mg | 117.00 € | ||
| 500mg | 190.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Evocalcet
CAS:870964-67-3
Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).
Formula:
C24H26N2O2
Purity:
98.41% - 99.83%
Color and Shape:
Solid
Molecular weight:
374.48
Ref: TM-T15261
| 1ml | 63.00 € | ||
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 366.00 € | ||
| 500mg | 847.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Pranlukast
CAS:103177-37-3
Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.
Formula:
C27H23N5O4
Purity:
99.85%
Color and Shape:
Off-White Solid
Molecular weight:
481.5
Ref: TM-T0694
| 1ml | 55.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 124.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Tripelennamine hydrochloride
CAS:154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent …
Formula:
C16H21N3·HCl
Purity:
100% - 100%
Color and Shape:
White Solid
Molecular weight:
291.82
Ref: TM-T1269
| 1g | 141.00 € | ||
| 1ml | 34.00 € | ||
| 25mg | 39.00 € | ||
| 50mg | 34.00 € | ||
| 100mg | 45.00 € | ||
| 500mg | 93.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Molindone hydrochloride
CAS:15622-65-8
Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking …
Formula:
C16H24N2O2·HCl
Purity:
99% - 99.93%
Color and Shape:
Solid
Molecular weight:
312.84
Ref: TM-T0716
| 1ml | 51.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 101.00 € | ||
| 100mg | 133.00 € | ||
| 200mg | 179.00 € | ||
| 500mg | 291.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Anamorelin
CAS:249921-19-5
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
Formula:
C31H42N6O3
Purity:
99.35% - 99.88%
Color and Shape:
Solid
Molecular weight:
546.7
Ref: TM-T10319
| 1ml | 73.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 175.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Aripiprazole Lauroxil
CAS:1259305-29-7
Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.
Formula:
C36H51Cl2N3O4
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
660.71
Ref: TM-T14319
| 1ml | 49.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 127.00 € | ||
| 200mg | 184.00 € | ||
| 500mg | 312.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Amiselimod hydrochloride
CAS:942398-84-7
Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.
Formula:
C19H31ClF3NO3
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
413.9
Ref: TM-T10305
| 1mg | 38.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 499.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
ONC206
CAS:1638178-87-6
ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the …
Formula:
C23H22F2N4O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
408.44
Ref: TM-T16392
| 1ml | 50.00 € | ||
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Antazoline hydrochloride
CAS:2508-72-7
Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and …
Formula:
C17H19N3·HCl
Purity:
98% - 99.76%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
301.82
Ref: TM-T0092
| 1g | 113.00 € | ||
| 1ml | 34.00 € | ||
| 100mg | 41.00 € | ||
| 500mg | 87.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Citalopram hydrobromide
CAS:59729-32-7
Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal …
Formula:
C20H22BrFN2O
Purity:
99.35%
Color and Shape:
White Crystalline Powder
Molecular weight:
405.304
Ref: TM-T1483
| 10mg | 52.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 113.00 € | ||
| 200mg | 156.00 € | ||
| 500mg | 242.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
CD80-IN-3
CAS:486449-65-4
CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 …
Formula:
C17H10FN3O3
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
323.28
Ref: TM-T10722
| 1mg | 79.00 € | ||
| 1ml | 202.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 482.00 € | ||
| 50mg | 666.00 € | ||
| 100mg | 828.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Roluperidone
CAS:359625-79-9
Roluperidone (CYR-101) is a novel cyclic amide derivative.
Formula:
C22H23FN2O2
Purity:
96.46% - 97.77%
Color and Shape:
Solid
Molecular weight:
366.43
Ref: TM-T15034
| 1mg | 36.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 369.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
BIBO3304 TFA
CAS:191868-14-1
BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).
Formula:
C31H36F3N7O5
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
643.66
Ref: TM-T10539
| 1mg | 95.00 € | ||
| 1ml | 329.00 € | ||
| 2mg | 143.00 € | ||
| 5mg | 218.00 € | ||
| 10mg | 385.00 € | ||
| 25mg | 640.00 € | ||
| 50mg | 908.00 € | ||
| 100mg | 1,226.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
(±) Clopidogrel hydrogen sulfate
CAS:135046-48-9
(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, …
Formula:
C16H16ClNO2S·H2SO4
Purity:
98.67% - 99.04%
Color and Shape:
Colorless To Light Yellow Liquid
Molecular weight:
419.9
Ref: TM-T0182L2
| 1g | 101.00 € | ||
| 1ml | 34.00 € | ||
| 100mg | 34.00 € | ||
| 200mg | 52.00 € | ||
| 500mg | 78.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Clorprenaline hydrochloride
CAS:6933-90-0
Clorprenaline hydrochloride (Clorprenaline HCl) is a beta-2 adrenergic agonist with bronchodilator activity.
Formula:
C11H17Cl2NO
Purity:
100% - 98.65%
Color and Shape:
Solid
Molecular weight:
250.16
Ref: TM-T0248
| 1ml | 55.00 € | ||
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 74.00 € | ||
| 200mg | 94.00 € | ||
| 500mg | 153.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
GTS-21 dihydrochloride
CAS:156223-05-1
GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by …
Formula:
C19H20N2O2·2HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
381.3
Ref: TM-T2663
| 1ml | 57.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 320.00 € | ||
| 500mg | 532.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Triflupromazine hydrochloride
CAS:1098-60-8
Triflupromazine hydrochloride (Fluopromazine hydrochloride), an antipsychotic medication, is Dopamine D1/D2 receptor antagonists.
Formula:
C18H20ClF3N2S
Purity:
99.73% - 99.73%
Color and Shape:
Crystals
Molecular weight:
388.88
Ref: TM-T0302
| 1g | 112.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 34.00 € | ||
| 200mg | 51.00 € | ||
| 500mg | 87.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Terazosin hydrochloride
CAS:63074-08-8
Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.
Formula:
C19H26ClN5O4
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
423.89
Ref: TM-T0197
| 1ml | 55.00 € | ||
| 50mg | 43.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 88.00 € | ||
| 500mg | 132.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
