G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AR-M 1896 Acetate
AR-M 1896 Acetate is the selective agonist of GalR2.
Formula:
C56H85N13O16
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
1196.35
Ref: TM-T21646L
| 1mg | 517.00 € | ||
| 2mg | 700.00 € | ||
| 5mg | 1,025.00 € | ||
| 10mg | 1,400.00 € | ||
| 25mg | 2,068.00 € | ||
| 50mg | 2,717.00 € | ||
| 1mL*10mM (DMSO) | 2,132.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ML-184
CAS:794572-10-4
ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.
Formula:
C25H34N4O3S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
470.63
Ref: TM-T8571
| 2mg | 48.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 265.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 720.00 € | ||
| 200mg | 1,011.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
![[Lys5,MeLeu9,Nle10]-NKA(4-10)](https://static.cymitquimica.com/products/TM/thumb/TP1883.jpg)
[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:137565-28-7
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the …
Formula:
C39H65N9O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
803.99
Ref: TM-TP1883
| 1mg | 97.00 € | ||
| 5mg | 234.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 539.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 992.00 € | ||
| 200mg | 1,347.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
AM966
CAS:1228690-19-4
AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.
Formula:
C27H23ClN2O5
Purity:
97.32% - 99.49%
Color and Shape:
Solid
Molecular weight:
490.93
Ref: TM-T4278
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 159.00 € | ||
| 100mg | 246.00 € | ||
| 200mg | 354.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
NIBR-0213
CAS:1233332-14-3
NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.
Formula:
C27H29ClN2O3
Purity:
98.36% - 98.87%
Color and Shape:
Solid
Molecular weight:
464.98
Ref: TM-T28169
| 1mg | 41.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 214.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
2-Pyridylethylamine dihydrochloride
CAS:3343-39-3
2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.
Formula:
C7H12Cl2N2
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
195.09
Ref: TM-T22501
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 143.00 € | ||
| 100mg | 209.00 € | ||
| 200mg | 308.00 € | ||
| 500mg | 513.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Sitaxsentan sodium
CAS:210421-74-2
Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.
Formula:
C18H14ClN2O6S2·Na
Purity:
98.39% - ≥95%
Color and Shape:
Solid
Molecular weight:
476.89
Ref: TM-T6672
| 5mg | 35.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 98.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 263.00 € | ||
| 200mg | 383.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
AM251
CAS:183232-66-8
AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).
Formula:
C22H21Cl2IN4O
Purity:
97.38% - 97.88%
Color and Shape:
A Crystalline Solid
Molecular weight:
555.24
Ref: TM-T1915
| 5mg | 50.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 324.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
GBR 12935 dihydrochloride
CAS:67469-81-2
GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine …
Formula:
C28H36Cl2N2O
Purity:
98.17% - ≥95%
Color and Shape:
Solid
Molecular weight:
487.5
Ref: TM-T1871
| 5mg | 40.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 92.00 € | ||
| 50mg | 108.00 € | ||
| 100mg | 182.00 € | ||
| 200mg | 263.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
H4 Receptor antagonist 1
CAS:848217-00-5
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with …
Formula:
C16H17ClN4O
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
316.79
Ref: TM-T5829
| 2mg | 45.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 302.00 € | ||
| 100mg | 435.00 € | ||
| 500mg | 931.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
LIXIVAPTAN
CAS:168079-32-1
Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
Formula:
C27H21ClFN3O2
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
473.93
Ref: TM-T7303
| 1mg | 42.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 624.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Loxapine
CAS:1977-10-2
Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.
Formula:
C18H18ClN3O
Purity:
99.98%
Color and Shape:
Pale Yellowish Crystals From Petroleum Ether Solid
Molecular weight:
327.81
Ref: TM-T21629
| 50mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 83.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
GLP-1(7-36), amide
CAS:107444-51-9
GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the …
Formula:
C149H226N40O45
Purity:
99.85%
Color and Shape:
White Powder
Molecular weight:
3297.63
Ref: TM-T3984
| 1mg | 173.00 € | ||
| 2mg | 306.00 € | ||
| 5mg | 516.00 € | ||
| 10mg | 741.00 € | ||
| 25mg | 1,152.00 € | ||
| 50mg | 1,539.00 € | ||
| 100mg | 2,095.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Trazodone
CAS:19794-93-5
Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major …
Formula:
C19H22ClN5O
Purity:
99.29%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
371.86
Ref: TM-T22442
| 25mg | 51.00 € | ||
| 50mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ramosetron hydrochloride
CAS:132907-72-3
Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant …
Formula:
C17H18ClN3O
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
315.8
Ref: TM-T4562L
| 5mg | 38.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 77.00 € | ||
| 50mg | 98.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 250.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
(R)-Propranolol hydrochloride
CAS:13071-11-9
(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.
Formula:
C16H22ClNO2
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
295.8
Ref: TM-T20898
| 25mg | 41.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TAK-041
CAS:1929519-13-0
TAK-041 (NBI-1065846) is a potent and selective GPR139 agonist.
Formula:
C18H15F3N4O3
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
392.33
Ref: TM-T9317
| 1mg | 37.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 220.00 € | ||
| 25mg | 442.00 € | ||
| 50mg | 707.00 € | ||
| 100mg | 1,104.00 € | ||
| 200mg | 1,482.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Decloxizine
CAS:3733-63-9
Decloxizine is a H1 receptor antagonist
Formula:
C21H28N2O2
Purity:
98.95%
Color and Shape:
White Or Similar To White Powder
Molecular weight:
340.46
Ref: TM-T22713
| 10mg | 40.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Pramipexole dihydrochloride hydrate
CAS:191217-81-9
Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is …
Formula:
C10H17N3S·2HCl·H2O
Purity:
99.55%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
302.26
Ref: TM-T6951
| 10mg | 51.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 176.00 € | ||
| 200mg | 254.00 € | ||
| 500mg | 421.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Sultopride hydrochloride
CAS:23694-17-9
Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.
Formula:
C17H27ClN2O4S
Purity:
≥95%
Color and Shape:
White Or Yellowish Powder
Molecular weight:
390.93
Ref: TM-T7180
| 1mg | 47.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 606.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
