G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Latanoprost
CAS:130209-82-4
Latanoprost (Xalatan) is a prostaglandin F2alpha analogue and a prostanoid selective FP receptor agonist with …
Formula:
C26H40O5
Purity:
99.69% - 99.78%
Color and Shape:
Pale Yellow Oil
Molecular weight:
432.59
Ref: TM-T2528
| 1mg | 46.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 404.00 € | ||
| 100mg | 595.00 € | ||
| 500mg | 1,263.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SORT-PGRN interaction inhibitor 1
CAS:100957-85-5
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
Formula:
C15H18N2O2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
258.32
Ref: TM-T9044
| 10mg | 34.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML382
CAS:1646499-97-9
ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).
Formula:
C18H20N2O4S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
360.43
Ref: TM-T8538
| 1ml | 49.00 € | ||
| 5mg | 47.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 323.00 € | ||
| 200mg | 451.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
EST73502 HCl
CAS:2307458-82-6
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of …
Formula:
C19H27ClF2N2O2
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
388.88
Ref: TM-T39284
| 1mg | 149.00 € | ||
| 1ml | 327.00 € | ||
| 5mg | 295.00 € | ||
| 10mg | 420.00 € | ||
| 25mg | 692.00 € | ||
| 50mg | 979.00 € | ||
| 100mg | 1,299.00 € | ||
| 500mg | 2,636.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Elinzanetant
CAS:929046-33-3
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive …
Formula:
C33H35F7N4O3
Purity:
98% - 99.13%
Color and Shape:
Odour Color
Molecular weight:
668.64
Ref: TM-T38144
| 1mg | 94.00 € | ||
| 1ml | 298.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 782.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JD-5037
CAS:1392116-14-1
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
Formula:
C27H27Cl2N5O3S
Purity:
98.14% - 98.87%
Color and Shape:
Solid
Molecular weight:
572.51
Ref: TM-T4453
| 1mg | 43.00 € | ||
| 1ml | 106.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 538.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SCH442416
CAS:316173-57-6
SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).
Formula:
C20H19N7O2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
389.41
Ref: TM-T23336
| 1mg | 47.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 275.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 643.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
3-CPMT
CAS:14008-79-8
3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
Formula:
C21H25Cl2NO
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
378.33
Ref: TM-T22508
| 1mg | 44.00 € | ||
| 1ml | 91.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 417.00 € | ||
| 100mg | 616.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JNJ-63533054
CAS:1802326-66-4
JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
Formula:
C17H17ClN2O2
Purity:
98.38% - 99.87%
Color and Shape:
Solid
Molecular weight:
316.78
Ref: TM-T3119
| 1ml | 45.00 € | ||
| 5mg | 42.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 272.00 € | ||
| 200mg | 393.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
(-)-Isocorypalmine
CAS:483-34-1
(-)-Isocorypalmine ((S)-Tetrahydrocolumbamine), a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.
Formula:
C20H23NO4
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
341.4
Ref: TM-TQ0176
| 1mg | 78.00 € | ||
| 5mg | 164.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bradykinin (acetate)
CAS:6846-03-3
Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.
Formula:
C52H77N15O13
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1120.26
Ref: TM-T21610
| 1mg | 43.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 399.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ZM241385
CAS:139180-30-6
ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
Formula:
C16H15N7O2
Purity:
95.28% - 99.69%
Color and Shape:
Solid
Molecular weight:
337.34
Ref: TM-T7021
| 1ml | 57.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 228.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 638.00 € | ||
| 500mg | 1,009.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Antalarmin
CAS:157284-96-3
Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.
Formula:
C24H34N4
Color and Shape:
Solid
Molecular weight:
378.55
Ref: TM-T70433
| 25mg | 1,397.00 € | ||
| 50mg | 1,820.00 € | ||
| 100mg | 2,297.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
5-O-Demethylnobiletin
CAS:2174-59-6
5-O-Demethylnobiletin is a natural anti-inflammatory that inhibits 5-LOX without altering COX-2 expression.
Formula:
C20H20O8
Purity:
98% - 99.83%
Color and Shape:
Solid
Molecular weight:
388.37
Ref: TM-T5714
| 1mg | 64.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 204.00 € | ||
| 25mg | 357.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 739.00 € | ||
| 500mg | 1,613.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JMS-17-2
CAS:1380392-05-1
JMS-17-2 is a potent and selective antagonist of CX3CR1( IC50 : 0.32 nM).
Formula:
C25H26ClN3O
Purity:
98.70% - ≥98%
Color and Shape:
Solid
Molecular weight:
419.95
Ref: TM-T5849
| 1mg | 40.00 € | ||
| 1ml | 96.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 337.00 € | ||
| 100mg | 500.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
lumateperone Tosylate
CAS:1187020-80-9
lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors …
Formula:
C31H36FN3O4S
Purity:
98% - 98.57%
Color and Shape:
Solid
Molecular weight:
565.7
Ref: TM-TQ0084
| 1ml | 65.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 334.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AZ3451
CAS:2100284-59-9
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
Formula:
C30H27BrN4O3
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
571.46
Ref: TM-TQ0012
| 1ml | 50.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 139.00 € | ||
| 50mg | 236.00 € | ||
| 100mg | 349.00 € | ||
| 200mg | 496.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cotadutide acetate
Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 …
Formula:
C169H256N42O57
Purity:
98.28%
Color and Shape:
Solid
Molecular weight:
3788.14
Ref: TM-TP1103
| 1mg | 148.00 € | ||
| 5mg | 432.00 € | ||
| 10mg | 580.00 € | ||
| 25mg | 925.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pridopidine
CAS:346688-38-8
Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's …
Formula:
C15H23NO2S
Purity:
95.2% - 99.89%
Color and Shape:
Solid
Molecular weight:
281.41
Ref: TM-T7352
| 1ml | 51.00 € | ||
| 5mg | 47.00 € | ||
| 10mg | 76.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 274.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CAY10526
CAS:938069-71-7
CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB …
Formula:
C12H7BrO3S
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
311.15
Ref: TM-T23861
| 1mg | 62.00 € | ||
| 1ml | 150.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 231.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 727.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
