G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Bosentan
CAS:147536-97-8
Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.
Formula:
C27H29N5O6S
Purity:
100% - 99.8%
Color and Shape:
Pale Yellow To Off-White Solid
Molecular weight:
551.614
Ref: TM-T6264
| 1ml | 88.00 € | ||
| 10mg | 38.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 80.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 202.00 € | ||
| 500mg | 304.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cebranopadol
CAS:863513-91-1
Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, …
Formula:
C24H27FN2O
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
378.48
Ref: TM-T5167
| 1ml | 43.00 € | ||
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 236.00 € | ||
| 200mg | 342.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
Formula:
C31H60N10O9
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
716.88
Ref: TM-TP1046L
| 1mg | 84.00 € | ||
| 5mg | 191.00 € | ||
| 10mg | 341.00 € | ||
| 25mg | 575.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,105.00 € | ||
| 500mg | 2,261.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
DORA-22
CAS:1088991-95-0
DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on …
Formula:
C23H22F2N4O2
Purity:
97.67%
Color and Shape:
Solid
Molecular weight:
424.44
Ref: TM-T5500
| 1mg | 129.00 € | ||
| 1ml | 330.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 697.00 € | ||
| 50mg | 976.00 € | ||
| 100mg | 1,319.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Acrivastine
CAS:87848-99-5
Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.
Formula:
C22H24N2O2
Purity:
100% - 99.85%
Color and Shape:
Solid
Molecular weight:
348.44
Ref: TM-T4551
| 1g | 774.00 € | ||
| 1ml | 41.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 222.00 € | ||
| 500mg | 541.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Palosuran hydrochloride 540769-28-6(free base)
Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human …
Formula:
C25H31ClN4O2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
454.99
Ref: TM-T4689
| 1mg | 65.00 € | ||
| 1ml | 181.00 € | ||
| 2mg | 104.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 281.00 € | ||
| 25mg | 456.00 € | ||
| 50mg | 653.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
5-HT1A modulator 2 hydrochloride
CAS:3880-76-0
5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM …
Formula:
C11H16ClNO
Purity:
97%
Color and Shape:
Solid
Molecular weight:
213.7
Ref: TM-T37197
| 1ml | 50.00 € | ||
| 50mg | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SR 57227 hydrochloride
CAS:77145-61-0
SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. …
Formula:
C10H14ClN3·HCl
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
248.15
Ref: TM-T23394
| 1ml | 52.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 300.00 € | ||
| 200mg | 427.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CAY10471 Racemate
CAS:844639-57-2
CAY10471 Racemate is a potent CRTH2/DP2 antagonist with Ki of 0.6 nM; less active on …
Formula:
C21H21FN2O4S
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
416.47
Ref: TM-T7359
| 1ml | 50.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 136.00 € | ||
| 50mg | 196.00 € | ||
| 100mg | 290.00 € | ||
| 200mg | 419.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Midodrine
CAS:42794-76-3
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
Formula:
C12H18N2O4
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
254.28
Ref: TM-T22369
| 1ml | 51.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 214.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Gramine
CAS:87-52-5
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active …
Formula:
C11H14N2
Purity:
97.23% - 98.44%
Color and Shape:
White Crystalline Powder
Molecular weight:
174.24
Ref: TM-T6519
| 1g | 157.00 € | ||
| 1ml | 39.00 € | ||
| 50mg | 38.00 € | ||
| 100mg | 50.00 € | ||
| 500mg | 107.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.
Formula:
C154H256N44O44
Purity:
98%
Color and Shape:
Solid
Molecular weight:
3428.01
Ref: TM-TP2328L
| 1mg | 128.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 423.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,319.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
EST64454 hydrochloride
CAS:1950569-11-5
EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the …
Formula:
C18H23ClF2N4O2
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
400.85
Ref: TM-T8834
| 1mg | 51.00 € | ||
| 1ml | 117.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 318.00 € | ||
| 50mg | 515.00 € | ||
| 100mg | 817.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nonapeptide-1 acetate salt (158563-45-2 free base)
Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a …
Formula:
C63H91N15O11S
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
1266.58
Ref: TM-TP1101
| 1mg | 68.00 € | ||
| 2mg | 94.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 243.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 587.00 € | ||
| 100mg | 820.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CP 376395
CAS:175140-00-8
CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.
Formula:
C21H30N2O
Purity:
99.83% - 99.96%
Color and Shape:
Solid
Molecular weight:
326.48
Ref: TM-T4329
| 1mg | 41.00 € | ||
| 1ml | 91.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 133.00 € | ||
| 25mg | 262.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 661.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ML-18
CAS:1422269-30-4
ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.
Formula:
C32H35N5O5
Purity:
100% - 98.53%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-T4540
| 1mg | 35.00 € | ||
| 1ml | 78.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 434.00 € | ||
| 200mg | 598.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Protease-Activated Receptor-1, PAR-1 Agonist acetate
PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.
Formula:
C37H62N10O11
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
822.95
Ref: TM-T38836L
| 1mg | 83.00 € | ||
| 2mg | 102.00 € | ||
| 5mg | 152.00 € | ||
| 10mg | 213.00 € | ||
| 25mg | 357.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 693.00 € | ||
| 200mg | 904.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Lurasidone
CAS:367514-87-2
Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It …
Formula:
C28H36N4O2S
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
492.68
Ref: TM-T21337
| 5mg | 46.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 203.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PRE-084 hydrochloride
CAS:75136-54-8
PRE-084 hydrochloride is a selective agonist of σ1(IC50:44 nM, in the sigma receptor assay).
Formula:
C19H28ClNO3
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
353.88
Ref: TM-T3198L
| 1ml | 72.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 364.00 € | ||
| 200mg | 553.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Scopine
CAS:498-45-3
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy …
Formula:
C8H13NO2
Purity:
100% - ≥98%
Color and Shape:
Solid
Molecular weight:
155.19
Ref: TM-T6662
| 1ml | 49.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 290.00 € | ||
| 200mg | 433.00 € | ||
| 500mg | 694.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
