G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Metoclopramide
CAS:364-62-5
Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.
Formula:
C14H22ClN3O2
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
299.8
Ref: TM-T4616
| 50mg | 47.00 € | ||
| 100mg | 60.00 € | ||
| 500mg | 120.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
CID 2745687
CAS:264233-05-8
CID 2745687 blocks human GPR35, countering cromolyn disodium & zaprinast effects.
Formula:
C17H19F2N5O2S
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
395.43
Ref: TM-T21874
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 628.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Brexpiprazole
CAS:913611-97-9
Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
Formula:
C25H27N3O2S
Purity:
99.54% - 99.96%
Color and Shape:
Solid
Molecular weight:
433.57
Ref: TM-T2306
| 5mg | 54.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 97.00 € | ||
| 100mg | 102.00 € | ||
| 200mg | 150.00 € | ||
| 500mg | 273.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Zotepine
CAS:26615-21-4
Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and …
Formula:
C18H18ClNOS
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
331.86
Ref: TM-T19680
| 5mg | 36.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 212.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Exo-1
CAS:461681-88-9
Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism …
Formula:
C15H12FNO3
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
273.26
Ref: TM-T9200
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 270.00 € | ||
| 200mg | 405.00 € | ||
| 500mg | 665.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Mebhydrolin
CAS:524-81-2
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
Formula:
C19H20N2
Purity:
99.73% - ≥98%
Color and Shape:
Solid
Molecular weight:
276.38
Ref: TM-T7085
| 100mg | 43.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 124.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Norepinephrine bitartrate salt
CAS:3414-63-9
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
Formula:
C12H17NO9
Purity:
97.32% - 99.97%
Color and Shape:
Solid
Molecular weight:
319.27
Ref: TM-T21066
| 5mg | 44.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 184.00 € | ||
| 500mg | 455.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
LRGILS-NH2 acetate
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
Formula:
C29H56N10O7
Purity:
96.65%
Color and Shape:
Liquid
Molecular weight:
656.82
Ref: TM-T22933L
| 1mg | 41.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 541.00 € | ||
| 200mg | 730.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of …
Formula:
C51H68N12O13
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
1057.16
Ref: TM-TP1404L
| 1mg | 105.00 € | ||
| 5mg | 310.00 € | ||
| 10mg | 556.00 € | ||
| 25mg | 833.00 € | ||
| 50mg | 1,144.00 € | ||
| 100mg | 1,529.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PAR-4 Agonist Peptide, amide TFA
CAS:1228078-65-6
PAR-4 agonist peptide doesn't affect PAR-1/PAR-2; blocked by PAR-4 antagonist.
Formula:
C36H49F3N8O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
794.82
Ref: TM-TP1065
| 1mg | 51.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 232.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 559.00 € | ||
| 100mg | 810.00 € | ||
| 1mL*10mM (DMSO) | 221.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
SKF-83566
CAS:99295-33-7
SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.
Formula:
C17H18BrNO
Purity:
95.00% - 99.82%
Color and Shape:
Solid
Molecular weight:
332.23
Ref: TM-T8702
| 1mg | 53.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
4F 4PP oxalate
CAS:144734-36-1
4F 4PP oxalate is a 5-HT2A antagonist.
Formula:
C22H26FNO·C2H2O4
Purity:
97.34%
Color and Shape:
Solid
Molecular weight:
429.49
Ref: TM-T22514
| 5mg | 44.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 430.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Kisspeptin-10, rat acetate(478507-53-8 free base)
Kisspeptin-10, rat acetate is an endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).
Formula:
C65H87N17O17
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
1378.45
Ref: TM-TP1666L
| 1mg | 90.00 € | ||
| 2mg | 128.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 507.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,016.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BigLEN (mouse) acetate
BigLEN (mouse) acetate is a potent and selective agonist of orphan G protein-coupled receptor 171 …
Formula:
C80H134N24O24
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
1816.07
Ref: TM-TP2073L
| 1mg | 95.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 627.00 € | ||
| 100mg | 843.00 € | ||
| 200mg | 1,127.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.
Formula:
C52H83N13O14
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
1114.29
Ref: TM-TP1900L1
| 1mg | 239.00 € | ||
| 5mg | 532.00 € | ||
| 10mg | 764.00 € | ||
| 25mg | 1,161.00 € | ||
| 50mg | 1,579.00 € | ||
| 100mg | 2,118.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Tasimelteon
CAS:609799-22-6
Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 …
Formula:
C15H19NO2
Purity:
98.08% - 99.93%
Color and Shape:
Solid
Molecular weight:
245.32
Ref: TM-T3495
| 10mg | 44.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 175.00 € | ||
| 500mg | 438.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Terazosin hydrochloride dihydrate
CAS:70024-40-7
Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms …
Formula:
C19H25N5O4·HCl·2H2O
Purity:
99.97%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
459.92
Ref: TM-T6701
| 100mg | 40.00 € | ||
| 200mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
C14TKL-1 acetate
C14TKL-1 acetate is a NK1 receptor agonist.
Formula:
C65H102N20O15S2
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
1467.75
Ref: TM-TP2227L
| 1mg | 130.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 425.00 € | ||
| 25mg | 702.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
DPDPE TFA (88373-73-3 free base)
CAS:172888-59-4
DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and …
Formula:
C32H40F3N5O9S2
Purity:
99.39%
Color and Shape:
Solid
Molecular weight:
759.81
Ref: TM-TP2036L
| 1mg | 72.00 € | ||
| 5mg | 155.00 € | ||
| 10mg | 228.00 € | ||
| 25mg | 372.00 € | ||
| 50mg | 519.00 € | ||
| 100mg | 698.00 € | ||
| 200mg | 904.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Prasugrel Hydrochloride
CAS:389574-19-0
Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis …
Formula:
C20H20FNO3S·HCl
Purity:
99.39% - 99.79%
Color and Shape:
Solid
Molecular weight:
409.9
Ref: TM-T6952
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 129.00 € | ||
| 100mg | 183.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
