G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.
Formula:
C32H51F3N8O9
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
748.79
Ref: TM-T7674
| 1mg | 45.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 516.00 € | ||
| 200mg | 703.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Perospirone hydrochloride
CAS:129273-38-7
Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.
Formula:
C23H31ClN4O2S
Purity:
99.37%
Color and Shape:
White Solid
Molecular weight:
463
Ref: TM-T8136
| 5mg | 35.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 91.00 € | ||
| 100mg | 133.00 € | ||
| 200mg | 185.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Ablukast
CAS:96566-25-5
Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.
Formula:
C28H34O8
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
498.56
Ref: TM-T26519
| 1mg | 48.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 654.00 € | ||
| 200mg | 881.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
LML134
CAS:1542135-76-1
LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg …
Formula:
C19H29N5O3
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
375.47
Ref: TM-T8514
| 1mg | 79.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 265.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 1,081.00 € | ||
| 1mL*10mM (DMSO) | 182.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Talinolol
CAS:57460-41-0
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Formula:
C20H33N3O3
Purity:
98.80%
Color and Shape:
Solid
Molecular weight:
363.49
Ref: TM-T21640
| 1mg | 73.00 € | ||
| 2mg | 97.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 296.00 € | ||
| 25mg | 534.00 € | ||
| 50mg | 768.00 € | ||
| 100mg | 1,054.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Ibutamoren Mesylate
CAS:159752-10-0
Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
Formula:
C28H40N4O8S2
Purity:
97.98% - ≥98%
Color and Shape:
Solid
Molecular weight:
624.77
Ref: TM-T7112
| 1g | 150.00 € | ||
| 5mg | 40.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 60.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 81.00 € | ||
| 500mg | 102.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SR59230A hydrochloride
CAS:1135278-41-9
SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue …
Formula:
C21H28ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
361.91
Ref: TM-T13016L
| 1mg | 45.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 261.00 € | ||
| 100mg | 386.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SB-334867 free base
CAS:792173-99-0
SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.
Formula:
C17H13N5O2
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
319.32
Ref: TM-T6140
| 2mg | 42.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 224.00 € | ||
| 100mg | 333.00 € | ||
| 200mg | 496.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Avexitide
CAS:133514-43-9
Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 …
Formula:
C149H234N40O47S
Purity:
98% - 98.76%
Color and Shape:
Solid
Molecular weight:
3369.76
Ref: TM-TP2100
| 1mg | 187.00 € | ||
| 5mg | 484.00 € | ||
| 10mg | 689.00 € | ||
| 25mg | 1,033.00 € | ||
| 50mg | 1,399.00 € | ||
| 100mg | 1,810.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Questiomycin A
CAS:1916-59-2
Questiomycin A: crème fraiche antibiotic with antibacterial, anticancer effects; inhibits GRP78.
Formula:
C12H8N2O2
Purity:
98% - 99.07%
Color and Shape:
Solid
Molecular weight:
212.2
Ref: TM-T36818
| 10mg | 55.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 176.00 € | ||
| 200mg | 251.00 € | ||
| 500mg | 244.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
SNAP 94847
CAS:487051-12-7
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM).
Formula:
C29H32F2N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
478.57
Ref: TM-T5406
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 310.00 € | ||
| 50mg | 528.00 € | ||
| 100mg | 892.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BD1063 dhydrochloride
CAS:206996-13-6
BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).
Formula:
C13H20Cl4N2
Purity:
99.52% - ≥95%
Color and Shape:
Solid
Molecular weight:
346.12
Ref: TM-T7488
| 2mg | 48.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 335.00 € | ||
| 100mg | 493.00 € | ||
| 200mg | 693.00 € | ||
| 500mg | 1,050.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
JNJ-5207852
CAS:398473-34-2
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat …
Formula:
C20H32N2O
Purity:
97.19%
Color and Shape:
Solid
Molecular weight:
316.48
Ref: TM-T7413
| 5mg | 49.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 379.00 € | ||
| 200mg | 539.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
IPSU
CAS:1373765-19-5
IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus …
Formula:
C23H27N5O2
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
405.49
Ref: TM-T5503
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 196.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 653.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tiprenolol
CAS:26481-51-6
Tiprenolol is a beta adrenergic receptor antagonist.[1]
Formula:
C13H21NO2S
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
255.38
Ref: TM-T50081
| 1mg | 81.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 241.00 € | ||
| 25mg | 398.00 € | ||
| 50mg | 543.00 € | ||
| 100mg | 760.00 € | ||
| 200mg | 1,000.00 € | ||
| 1mL*10mM (DMSO) | 152.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BAR 501 impurity
CAS:1632118-70-7
BAR501 impurity boosts luciferase in GP-BAR1 assay by 150% at 10 μM, acting as a …
Formula:
C26H46O3
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
406.64
Ref: TM-T8752
| 1mg | 85.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
β-Neoendorphin acetate(77739-21-0 free base)
CAS:78658-39-6
beta-Neoendorphin acetate is an agonist of κ-opioid receptor
Formula:
C56H81N13O14
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
1160.34
Ref: TM-TP2322L
| 1mg | 130.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 425.00 € | ||
| 25mg | 701.00 € | ||
| 50mg | 985.00 € | ||
| 100mg | 1,332.00 € | ||
| 200mg | 1,044.00 € | ||
| 500mg | 2,627.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
CVN424
CAS:2254706-21-1
CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.
Formula:
C24H29F2N5O3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
473.52
Ref: TM-T9346
| 1mg | 94.00 € | ||
| 5mg | 239.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 878.00 € | ||
| 100mg | 1,189.00 € | ||
| 1mL*10mM (DMSO) | 251.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Pre-084
CAS:138847-85-5
Pre-084 is a high affinity, selective σ1 agonist.
Formula:
C19H28ClNO3
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
353.88
Ref: TM-T3198
| 10mg | 469.00 € | ||
| 50mg | 1,878.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Cetirizine Impurity B dihydrochloride
CAS:1000690-91-4
Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.
Formula:
C19H23Cl3N2O2
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
417.76
Ref: TM-T9084
| 10mg | 35.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 120.00 € | ||
| 1mL*10mM (DMSO) | 40.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
