G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Pirenperone
CAS:75444-65-4
Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.
Formula:
C23H24FN3O2
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
393.45
Ref: TM-T2599
| 1mg | 40.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 227.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 530.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
ICI 89406
CAS:53671-71-9
ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.
Formula:
C19H22N4O3
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T22852
| 1mg | 80.00 € | ||
| 5mg | 145.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | 662.00 € | ||
| 100mg | 938.00 € | ||
| 500mg | 1,882.00 € | ||
| 1mL*10mM (DMSO) | 154.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Adenosine amine congener
CAS:96760-69-9
Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.
Formula:
C28H32N8O6
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
576.6
Ref: TM-T7683
| 1mg | 73.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 627.00 € | ||
| 100mg | 893.00 € | ||
| 1mL*10mM (DMSO) | 246.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
USL311
CAS:1373268-67-7
USL311 blocks CXCR4/SDF-1 interaction, inhibits tumor cell growth and migration.
Formula:
C24H34N6O
Purity:
99.56% - 99.73%
Color and Shape:
Solid
Molecular weight:
422.57
Ref: TM-T17208
| 1mg | 42.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 628.00 € | ||
| 500mg | 1,304.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Treprostinil
CAS:81846-19-7
Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).
Formula:
C23H34O5
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
390.51
Ref: TM-T5150
| 2mg | 47.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 457.00 € | ||
| 100mg | 655.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer …
Formula:
C59H80N14O13
Purity:
95.3%
Color and Shape:
Solid
Molecular weight:
1193.35
Ref: TM-TP1913L1
| 1mg | 96.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 279.00 € | ||
| 25mg | 504.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,017.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Binodenoson
CAS:144348-08-3
Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.
Formula:
C17H25N7O4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
391.42
Ref: TM-T9516
| 1mg | 137.00 € | ||
| 5mg | 283.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 702.00 € | ||
| 50mg | 938.00 € | ||
| 100mg | 1,320.00 € | ||
| 1mL*10mM (DMSO) | 310.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.
Formula:
C101H159N31O25
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
2207.58
Ref: TM-TP2040L
| 1mg | 71.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 328.00 € | ||
| 25mg | 553.00 € | ||
| 50mg | 792.00 € | ||
| 100mg | 1,093.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Nelotanserin
CAS:839713-36-9
Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B …
Formula:
C18H15BrF2N4O2
Purity:
98.01% - 98.42%
Color and Shape:
Solid
Molecular weight:
437.24
Ref: TM-T7350
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € | ||
| 500mg | 1,130.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Melanin Concentrating Hormone, salmon acetate
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is …
Formula:
C91H143N27O26S4
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
2157
Ref: TM-TP1104L
| 1mg | 120.00 € | ||
| 5mg | 284.00 € | ||
| 10mg | 420.00 € | ||
| 25mg | 655.00 € | ||
| 50mg | 883.00 € | ||
| 100mg | 1,121.00 € | ||
| 200mg | 1,549.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Eprazinone dihydrochloride
CAS:10402-53-6
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.
Formula:
C24H32N2O2·2HCl
Purity:
99.25%
Color and Shape:
A White Or Almost White Crys
Molecular weight:
453.44
Ref: TM-T3034
| 50mg | 39.00 € | ||
| 100mg | 59.00 € | ||
| 250mg | 97.00 € | ||
| 500mg | 170.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
GLP-1(7-37) acetate(106612-94-6 free base)
CAS:1450806-98-0
Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
Formula:
C151H228N40O47
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
3355.67
Ref: TM-TP1376
| 1mg | 111.00 € | ||
| 5mg | 216.00 € | ||
| 10mg | 329.00 € | ||
| 25mg | 560.00 € | ||
| 50mg | 800.00 € | ||
| 100mg | 1,103.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Ralinepag
CAS:1187856-49-0
Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s …
Formula:
C23H26ClNO5
Purity:
99.41% - 99.85%
Color and Shape:
Solid
Molecular weight:
431.91
Ref: TM-T4635
| 1mg | 60.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 227.00 € | ||
| 25mg | 333.00 € | ||
| 50mg | 497.00 € | ||
| 100mg | 722.00 € | ||
| 500mg | 1,501.00 € | ||
| 1mL*10mM (DMSO) | 135.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Azaperone
CAS:1649-18-9
Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.
Formula:
C19H22FN3O
Purity:
98.73%
Color and Shape:
White Or Off-White Crystalline
Molecular weight:
327.4
Ref: TM-T6398
| 25mg | 42.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 79.00 € | ||
| 200mg | 97.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
BETP
CAS:1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and …
Formula:
C20H17F3N2O2S
Purity:
97.92%
Color and Shape:
Solid
Molecular weight:
406.42
Ref: TM-TQ0124
| 1mg | 48.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 424.00 € | ||
| 100mg | 677.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Phenylbiguanide
CAS:102-02-3
Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)
Formula:
C8H11N5
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
177.21
Ref: TM-T7135
| 1g | 85.00 € | ||
| 200mg | 39.00 € | ||
| 500mg | 58.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Leachianone A
CAS:97938-31-3
Leachianone A (Isokurarinone) is a potential antitoxic agent, it shows inhibitory effects on cadmium- Induced …
Formula:
C26H30O6
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
438.51
Ref: TM-TN1856
| 1mg | 80.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 303.00 € | ||
| 25mg | 507.00 € | ||
| 1mL*10mM (DMSO) | 145.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Pizuglanstat
CAS:1244967-98-3
Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.
Formula:
C27H36N6O4
Purity:
98.96%
Color and Shape:
Solid
Molecular weight:
508.61
Ref: TM-T8883
| 5mg | 52.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 225.00 € | ||
| 100mg | 320.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Selexipag
CAS:475086-01-2
Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.
Formula:
C26H32N4O4S
Purity:
99.69% - 99.92%
Color and Shape:
Solid
Molecular weight:
496.62
Ref: TM-T3216
| 5mg | 49.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 92.00 € | ||
| 50mg | 96.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Diclofensine hydrochloride
CAS:34041-84-4
Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。
Formula:
C17H18Cl3NO
Purity:
98.86% - 99.93%
Color and Shape:
Solid
Molecular weight:
358.69
Ref: TM-T7745
| 5mg | 51.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 406.00 € | ||
| 200mg | 568.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
