G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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BRL 52537 hydrochloride
CAS:112282-24-3
BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke …
Formula:
C18H25Cl3N2O
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
391.76
Ref: TM-T21757
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 494.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Canagliflozin
CAS:842133-18-0
Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II …
Formula:
C24H25FO5S
Purity:
100% - 99.76%
Color and Shape:
Solid
Molecular weight:
444.52
Ref: TM-T1782
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 123.00 € | ||
| 200mg | 175.00 € | ||
| 500mg | 298.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Veralipride
CAS:66644-81-3
Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.
Formula:
C17H25N3O5S
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T7632
| 1mg | 65.00 € | ||
| 5mg | 139.00 € | ||
| 10mg | 205.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 587.00 € | ||
| 100mg | 882.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
2-Chloroadenosine
CAS:146-77-0
2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, …
Formula:
C10H12ClN5O4
Purity:
99.23%
Color and Shape:
White Powder
Molecular weight:
301.69
Ref: TM-T7736
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 131.00 € | ||
| 500mg | 319.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Mosapride
CAS:112885-41-3
Mosapride (AS-4370) is a selective 5HT4 agonist
Formula:
C21H25ClFN3O3
Purity:
99.56%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
421.89
Ref: TM-T8128
| 5mg | 44.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 99.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 219.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
CHEMBL241987
CAS:109740-09-2
CHEMBL241987 targets the Adenosine receptor A3 (human)
Formula:
C16H11N3O
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
261.28
Ref: TM-T8598
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 108.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 349.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
GLP-1 receptor agonist 9
CAS:2401892-71-3
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
Formula:
C32H31ClFN3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
592.06
Ref: TM-T9579
| 1mg | 145.00 € | ||
| 5mg | 319.00 € | ||
| 10mg | 472.00 € | ||
| 25mg | 753.00 € | ||
| 50mg | 1,074.00 € | ||
| 100mg | 1,444.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
AVN-492
CAS:1220646-23-0
AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
Formula:
C17H21N5O2S
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
359.45
Ref: TM-T5179
| 1mg | 39.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 510.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Phloretin
CAS:60-82-2
Phloretin (NSC-407292) inhibits eukaryotic urea transporters, has antioxidative properties, and can induce cancer cell apoptosis. …
Formula:
C15H14O5
Purity:
100% - 99.76%
Color and Shape:
Solid
Molecular weight:
274.27
Ref: TM-T2924
| 250mg | 50.00 € | ||
| 500mg | 63.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Lificiguat
CAS:170632-47-0
Lificiguat (YC-1) is an nitric oxide (NO)-independent activator of soluble guanylyl cyclase(sGC) and an inhibitor …
Formula:
C19H16N2O2
Purity:
98.85% - 99.92%
Color and Shape:
Solid
Molecular weight:
304.34
Ref: TM-T4381
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 240.00 € | ||
| 100mg | 410.00 € | ||
| 200mg | 607.00 € | ||
| 500mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Pimavanserin tartrate
CAS:706782-28-7
Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related …
Formula:
C50H68F2N6O4·C4H6O6
Purity:
100% - 99.98%
Color and Shape:
Solid
Molecular weight:
1005.2
Ref: TM-T6946
| 25mg | 50.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 106.00 € | ||
| 200mg | 143.00 € | ||
| 500mg | 230.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
NGB 2904
CAS:189060-98-8
NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes …
Formula:
C28H29Cl2N3O
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
494.46
Ref: TM-T28167
| 2mg | 40.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 394.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Nociceptin
CAS:170713-75-4
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide …
Formula:
C79H129N27O22
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
1809.04
Ref: TM-TP1071
| 1mg | 81.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 617.00 € | ||
| 50mg | 877.00 € | ||
| 100mg | 1,198.00 € | ||
| 500mg | 2,395.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Urotensin II, mouse acetate (9047-55-6 free base)
Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 …
Formula:
C64H88N14O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1421.61
Ref: TM-TP2165
| 1mg | 99.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 351.00 € | ||
| 25mg | 560.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,017.00 € | ||
| 200mg | 1,359.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
IBC 293
CAS:306935-41-1
IBC 293: Selective GPR109B agonist, favoring it over GPR109A; targets receptor in fat cells.
Formula:
C10H11N3O2
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
205.21
Ref: TM-T19700
| 10mg | 52.00 € | ||
| 25mg | 85.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 156.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Methyldopa hydrate
CAS:41372-08-1
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used …
Formula:
C10H13NO4H2O
Purity:
≥98%
Color and Shape:
White Solid
Molecular weight:
238.24
Ref: TM-T5954
| 1g | 52.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Betaxolol
CAS:63659-18-7
Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension …
Formula:
C18H29NO3
Purity:
99.01%
Color and Shape:
White Crystalline Solid
Molecular weight:
307.43
Ref: TM-T6408
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
THIQ
CAS:312637-48-2
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 …
Formula:
C33H41ClN6O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
589.17
Ref: TM-T8485
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 374.00 € | ||
| 50mg | 567.00 € | ||
| 100mg | 848.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
Dynorphin B (1-13) acetate(83335-41-5 free base)
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.
Formula:
C76H119N21O19
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
1630.89
Ref: TM-TP1826L
| 1mg | 93.00 € | ||
| 5mg | 219.00 € | ||
| 10mg | 324.00 € | ||
| 25mg | 523.00 € | ||
| 50mg | 712.00 € | ||
| 100mg | 959.00 € | ||
| 200mg | 1,293.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
GW842166X
CAS:666260-75-9
GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.
Formula:
C18H17Cl2F3N4O2
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
449.25
Ref: TM-T6527
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Friday 4 Apr 2025
