G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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4-Deoxypyridoxine hydrochloride
CAS:148-51-6
4-Deoxypyridoxine HCl halts S1P breakdown by blocking SPL, reducing apoptosis in insulinoma cells like S1P.
Formula:
C8H12ClNO2
Purity:
99.86%
Color and Shape:
White To Off White Crystalline Powder
Molecular weight:
189.64
Ref: TM-T38294
| 100mg | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Reboxetine mesylate
CAS:98769-84-7
Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).
Formula:
C19H23NO3·CH4O3S
Purity:
99.24% - 99.72%
Color and Shape:
Tan Or Off-White Cyrstalline Solid
Molecular weight:
409.5
Ref: TM-T6963
| 5mg | 42.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 286.00 € | ||
| 100mg | 457.00 € | ||
| 500mg | 989.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Anisotropine Methylbromide
CAS:80-50-2
Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm …
Formula:
C17H32BrNO2
Purity:
99.73%
Color and Shape:
Crystals From Acetone Solid
Molecular weight:
362.35
Ref: TM-T4981
| 5mg | 96.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 194.00 € | ||
| 50mg | 286.00 € | ||
| 100mg | 426.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Tetradecyl Phosphonate
CAS:4671-75-4
Tetradecyl phosphonate is a pan-antagonist of lysophosphatidic acid 1 (LPA1), LPA2, and LPA3 receptors.
Formula:
C14H31O3P
Purity:
≥95%
Color and Shape:
White To Off-White Powder
Molecular weight:
278.37
Ref: TM-T7689
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 165.00 € | ||
| 200mg | 240.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
ABT-702 dihydrochloride
CAS:1188890-28-9
ABT-702 dihydrochloride is a potent adenosine kinase (AK) inhibitor.
Formula:
C22H21BrCl2N6O
Purity:
98.89% - 99%
Color and Shape:
Solid
Molecular weight:
536.25
Ref: TM-T4668
| 1mg | 61.00 € | ||
| 2mg | 85.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 520.00 € | ||
| 100mg | 732.00 € | ||
| 500mg | 1,542.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
A-381393
CAS:726174-00-1
A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for …
Formula:
C20H24N4
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
320.43
Ref: TM-T5397
| 1mg | 39.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 292.00 € | ||
| 100mg | 422.00 € | ||
| 200mg | 593.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BMS986188
CAS:1776115-10-6
BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.
Formula:
C30H31BrO4
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
535.47
Ref: TM-T8992
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 191.00 € | ||
| 100mg | 284.00 € | ||
| 200mg | 397.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS:960404-48-2
Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal …
Formula:
C24H35ClO9
Purity:
99.39% - 99.94%
Color and Shape:
Solid
Molecular weight:
502.98
Ref: TM-T4460
| 10mg | 43.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 74.00 € | ||
| 500mg | 161.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
![1-[(5-methylisoxazol-3-yl)methyl]piperazine](https://static.cymitquimica.com/products/TM/thumb/T8582.jpg)
1-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:173850-51-6
1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.
Formula:
C9H15N3O
Purity:
95%
Color and Shape:
Solid
Molecular weight:
181.23
Ref: TM-T8582
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Hydroxyzine dihydrochloride
CAS:2192-20-3
Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.
Formula:
C21H27ClN2O2·2HCl
Purity:
99.79% - 99.79%
Color and Shape:
Oil Powder
Molecular weight:
447.83
Ref: TM-T2200
| 1g | 51.00 € | ||
| 100mg | 34.00 € | ||
| 200mg | 34.00 € | ||
| 500mg | 41.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
VKGILS-NH2 Acetate
VKGILS-NH2 Acetate is a reversed amino acid sequence control peptide for SLIGKV-NH2, a protease-activated receptor …
Formula:
C30H58N8O9
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
674.83
Ref: TM-T21699L
| 1mg | 34.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 337.00 € | ||
| 200mg | 479.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
CGS 21680 Hydrochloride
CAS:124431-80-7
CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in …
Formula:
C23H29N7O6·HCl
Purity:
96.74% - 98.81%
Color and Shape:
Solid
Molecular weight:
535.98
Ref: TM-T6441
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | 593.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Ropinirole hydrochloride
CAS:91374-20-8
Ropinirole HCl (SKF-101468A) is a selective D2 dopamine agonist (Ki: 29 nM) with antiparkinsonian effects.
Formula:
C16H24N2O·HCl
Purity:
99.87% - 99.98%
Color and Shape:
Off-White Solid
Molecular weight:
296.84
Ref: TM-T2592
| 25mg | 47.00 € | ||
| 50mg | 61.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 109.00 € | ||
| 500mg | 170.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Derenofylline
CAS:251945-92-3
Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)
Formula:
C18H20N4O
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
308.38
Ref: TM-T8312
| 5mg | 49.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 360.00 € | ||
| 200mg | 491.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
D3-βArr
CAS:662164-09-2
D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of …
Formula:
C20H23N5
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
333.43
Ref: TM-T5383
| 5mg | 47.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 230.00 € | ||
| 100mg | 342.00 € | ||
| 500mg | 802.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Doxazosin
CAS:74191-85-8
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat …
Formula:
C23H25N5O5
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
451.48
Ref: TM-T22316
| 5mg | 52.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 133.00 € | ||
| 100mg | 195.00 € | ||
| 200mg | 302.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Brimonidine
CAS:59803-98-4
Brimonidine (Bromoxidine) is a drug used as eye drops under the brand names Alphagan and …
Formula:
C11H10BrN5
Purity:
98.60%
Color and Shape:
Yellow Solid
Molecular weight:
292.13
Ref: TM-T20157
| 5mg | 56.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 331.00 € | ||
| 100mg | 495.00 € | ||
| 500mg | 1,096.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Peptide YY (PYY) (3-36), human
CAS:126339-09-1
Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY …
Formula:
C176H272N52O54
Purity:
97.76%
Color and Shape:
Solid
Molecular weight:
3980.42
Ref: TM-TP1059
| 1mg | 83.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 716.00 € | ||
| 100mg | 926.00 € | ||
| 200mg | 713.00 € | ||
| 500mg | 1,839.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
NNC-0640
CAS:307986-98-7
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 …
Formula:
C29H31N7O4S
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
573.67
Ref: TM-T7364
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 644.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Syrosingopine
CAS:84-36-6
Syrosingopine is a dual inhibitor of MCT1 and MCT4, 60 times more potent against MCT4, …
Formula:
C35H42N2O11
Purity:
99.25% - 99.78%
Color and Shape:
Solid
Molecular weight:
666.71
Ref: TM-TN2252
| 1mg | 71.00 € | ||
| 5mg | 146.00 € | ||
| 10mg | 213.00 € | ||
| 25mg | 361.00 € | ||
| 50mg | 536.00 € | ||
| 100mg | 740.00 € | ||
| 1mL*10mM (DMSO) | 200.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
