G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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BML-190
CAS:2854-32-2
BML-190 (Indomethacin morpholinylamide) is a specific CB2 receptor inverse agonist (Ki: 435 nM), with 50-fold …
Formula:
C23H23ClN2O4
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
426.89
Ref: TM-T6417
| 10mg | 46.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 166.00 € | ||
| 200mg | 266.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Cutamesine dihydrochloride
CAS:165377-44-6
Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving …
Formula:
C23H32N2O2·2HCl
Purity:
98.83% - 99%
Color and Shape:
Solid
Molecular weight:
441.43
Ref: TM-T3597
| 2mg | 43.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 418.00 € | ||
| 100mg | 618.00 € | ||
| 500mg | 1,291.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
α-MSH
CAS:581-05-5
α-MSH (MSH, amide) is amide stimulates melanocortin 1 receptor that results in the activation of …
Formula:
C77H109N21O19S
Purity:
100%
Color and Shape:
White Powder
Molecular weight:
1664.89
Ref: TM-T7813
| 1mg | 56.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 263.00 € | ||
| 25mg | 447.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 926.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
Formula:
C65H102N16O25
Purity:
95.55%
Color and Shape:
Solid
Molecular weight:
1507.6
Ref: TM-TP1578L
| 1mg | 72.00 € | ||
| 2mg | 89.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 196.00 € | ||
| 25mg | 358.00 € | ||
| 50mg | 536.00 € | ||
| 100mg | 755.00 € | ||
| 500mg | 1,550.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
N-ACETYLTRYPTAMINE
CAS:1016-47-3
N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination …
Formula:
C12H14N2O
Purity:
98.79%
Color and Shape:
Powder
Molecular weight:
202.25
Ref: TM-T8600
| 10mg | 43.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 107.00 € | ||
| 100mg | 164.00 € | ||
| 200mg | 235.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Bosentan (hydrate)
CAS:157212-55-0
Bosentan hydrate (Ro 47-0203) is a competitive and dual antagonist of endothelin-1 at the endothelin-A …
Formula:
C27H29N5O6S·H2O
Purity:
99.31% - 99.86%
Color and Shape:
White Powder
Molecular weight:
569.63
Ref: TM-T6265
| 25mg | 51.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 99.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Bexagliflozin
CAS:1118567-05-7
Bexagliflozin (EGT1442) is a potent, selective sodium glucose co-transporter 2 (SGLT2) inhibitor with IC50 values …
Formula:
C24H29ClO7
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
464.94
Ref: TM-T7217
| 1mg | 70.00 € | ||
| 2mg | 89.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 384.00 € | ||
| 50mg | 572.00 € | ||
| 100mg | 811.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
GW 405833
CAS:180002-83-9
GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selective
Formula:
C23H24Cl2N2O3
Purity:
99.82% - 99.93%
Color and Shape:
Solid
Molecular weight:
447.35
Ref: TM-T7705
| 1mg | 37.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 483.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Olodaterol hydrochloride
CAS:869477-96-3
Olodaterol hydrochloride (BI-1744 HCl) is a novel, long-acting β2-adrenergic agonist that exerts its pharmacological effect …
Formula:
C21H27ClN2O5
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
422.9
Ref: TM-T5159
| 1mg | 60.00 € | ||
| 2mg | 86.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 512.00 € | ||
| 100mg | 737.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
![[Leu5]-Enkephalin TFA(58822-25-6(free bas))](https://static.cymitquimica.com/products/TM/thumb/T7665.jpg)
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
CAS:73563-78-7
[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago
Formula:
C30H38F3N5O9
Purity:
97.03% - 99.78%
Color and Shape:
Solid
Molecular weight:
669.64
Ref: TM-T7665
| 10mg | 51.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 209.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
GLPG2938
CAS:2130996-00-6
GLPG2938 (1-(2-Ethoxy-6-(trifluoromethyl)pyridin-4-yl)-3-((5-methyl-6-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl)pyridazin-3-yl)methyl)urea) is a potent and
Formula:
C20H19F6N7O2
Purity:
98.25%
Color and Shape:
Solid
Molecular weight:
503.4
Ref: TM-T9199
| 1mg | 83.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,079.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Dioxopromethazine hydrochloride
CAS:15374-15-9
Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
Formula:
C17H20N2O2S·HCl
Purity:
100%
Color and Shape:
Solid
Molecular weight:
352.88
Ref: TM-T3723
| 25mg | 35.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 87.00 € | ||
| 500mg | 227.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
N-Cbz-DL-tryptophan
CAS:13058-16-7
N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
Formula:
C19H18N2O4
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
338.36
Ref: TM-T9343
| 5mg | 41.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 198.00 € | ||
| 200mg | 295.00 € | ||
| 500mg | 495.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
NPS ALX Compound 4a
CAS:299433-10-6
NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of …
Formula:
C25H25N3O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
431.55
Ref: TM-T12262
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 19 Dec 2024
Betahistine
CAS:5638-76-6
Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 …
Formula:
C8H12N2
Purity:
97.92% - 99.87%
Color and Shape:
Yellowish Liquid Liquid Liquid
Molecular weight:
136.19
Ref: TM-T4195
| 100mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Volinanserin
CAS:139290-65-6
Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x …
Formula:
C22H28FNO3
Purity:
98.94% - 99.95%
Color and Shape:
Solid
Molecular weight:
373.46
Ref: TM-T5389
| 5mg | 93.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 234.00 € | ||
| 50mg | 300.00 € | ||
| 200mg | 645.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Escin IB
CAS:26339-90-2
Escin Ib inhibits gastric emptying, at least in part, mediated by capsaicin-sensitive sensory nerves, to …
Formula:
C55H86O24
Purity:
99.09% - 99.73%
Color and Shape:
Solid
Molecular weight:
1131.26
Ref: TM-T5S1389
| 1mg | 69.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 570.00 € | ||
| 50mg | 808.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Tianeptine
CAS:72797-41-2
Tianeptine (Tianeptine sodium) is a selective 5-HT uptake facilitator in vitro and in vivo.
Formula:
C21H25ClN2O4S
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
436.95
Ref: TM-T8140
| 10mg | 36.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 103.00 € | ||
| 500mg | 245.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
SB-222200
CAS:174635-69-9
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
Formula:
C26H24N2O
Purity:
97.13%
Color and Shape:
Solid
Molecular weight:
380.48
Ref: TM-T16849
| 1mg | 39.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 451.00 € | ||
| 100mg | 644.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Tavapadon
CAS:1643489-24-0
Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.
Formula:
C19H16F3N3O3
Purity:
99.33% - 99.8%
Color and Shape:
Solid
Molecular weight:
391.34
Ref: TM-T16999
| 1mg | 80.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 494.00 € | ||
| 50mg | 695.00 € | ||
| 100mg | 917.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
