G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Reparixin
CAS:266359-83-5
Reparixin inhibits CXCR1 (IC50=1 nM) strongly, CXCR2 weakly (IC50=100 nM), and it's a CXCL8 receptor …
Formula:
C14H21NO3S
Purity:
98% - 99.89%
Color and Shape:
Solid
Molecular weight:
283.39
Ref: TM-T4163
| 1mg | 52.00 € | ||
| 2mg | 78.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 384.00 € | ||
| 50mg | 578.00 € | ||
| 100mg | 817.00 € | ||
| 500mg | 1,626.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
S 38093 HCl
CAS:1222097-72-4
S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.
Formula:
C17H25ClN2O2
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
324.85
Ref: TM-T4087
| 1mg | 50.00 € | ||
| 2mg | 69.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 469.00 € | ||
| 200mg | 634.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Xaliproden hydrochloride
CAS:90494-79-4
Xaliproden is a compound that mimics the effects of nerve growth factor and is also …
Formula:
C24H23ClF3N
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
417.89
Ref: TM-T9272
| 1mg | 40.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 372.00 € | ||
| 100mg | 534.00 € | ||
| 200mg | 447.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
11-Keto-β-boswellic acid
CAS:17019-92-0
11-Keto-beta-boswellic acid, a novel Nrf2 activator, and a selective 5-lipoxygenase (5-LOX) inhibitor, exerts dose dependent …
Formula:
C30H46O4
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
470.68
Ref: TM-TN1182
| 1mg | 59.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 517.00 € | ||
| 100mg | 733.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
PF-06291874
CAS:1393124-08-7
PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist …
Formula:
C26H28F3N3O4
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
503.51
Ref: TM-TQ0239
| 5mg | 60.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Velneperit
CAS:342577-38-2
Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment …
Formula:
C17H24F3N3O3S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
407.45
Ref: TM-T17222
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 634.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Cerlapirdine
CAS:925448-93-7
Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.
Formula:
C22H23N3O3S
Purity:
98.60%
Color and Shape:
Solid
Molecular weight:
409.5
Ref: TM-T30798
| 1mg | 81.00 € | ||
| 2mg | 68.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 771.00 € | ||
| 100mg | 1,060.00 € | ||
| 200mg | 837.00 € | ||
| 1mL*10mM (DMSO) | 196.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Cariprazine hydrochloride
CAS:1083076-69-0
Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial …
Formula:
C21H33Cl3N4O
Purity:
100% - 98.52%
Color and Shape:
Solid
Molecular weight:
463.87
Ref: TM-T8382
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 168.00 € | ||
| 500mg | 402.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.
Formula:
C38H64F3N11O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
891.98
Ref: TM-TP1378
| 1mg | 54.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 482.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
BW-180C
CAS:63631-40-3
BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid …
Formula:
C29H39N5O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1905
| 1mg | 46.00 € | ||
| 2mg | 61.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 392.00 € | ||
| 100mg | 582.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
MSX-130
CAS:4051-59-6
MSX-130 is CXCR4 Antagonist.
Formula:
C36H26N4
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
514.62
Ref: TM-T4033
| 1mg | 36.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 223.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 580.00 € | ||
| 200mg | 822.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Parmodulin 2
CAS:423735-93-7
ML161 (Parmodulin 2) inhibits PAR1, blocking platelet activation and thrombin-induced activity (IC50: 0.26μM).
Formula:
C17H17BrN2O2
Purity:
96.72% - 99.95%
Color and Shape:
Solid
Molecular weight:
361.23
Ref: TM-T1893
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 157.00 € | ||
| 50mg | 239.00 € | ||
| 100mg | 371.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
DAMGO TFA (78123-71-4(Free base))
DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and …
Formula:
C28H36F3N5O8
Purity:
98.67% - 99.76%
Color and Shape:
Solid
Molecular weight:
627.6
Ref: TM-T4411
| 1mg | 63.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 282.00 € | ||
| 25mg | 536.00 € | ||
| 50mg | 733.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Diquafosol tetrasodium
CAS:211427-08-6
Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular …
Formula:
C18H22N4Na4O23P4
Purity:
98.7% - 99.97%
Color and Shape:
Solid
Molecular weight:
878.23
Ref: TM-T7423
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 179.00 € | ||
| 50mg | 307.00 € | ||
| 100mg | 462.00 € | ||
| 500mg | 1,003.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Ditolylguanidine
CAS:97-39-2
Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).
Formula:
C15H17N3
Purity:
98.42%
Color and Shape:
White To Pinkish Solid Powder
Molecular weight:
239.32
Ref: TM-T5969
| 1g | 35.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Org 27569
CAS:868273-06-7
Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state …
Formula:
C24H28ClN3O
Purity:
100% - ≥95%
Color and Shape:
Solid
Molecular weight:
409.95
Ref: TM-T2635
| 2mg | 36.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 412.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Midodrine
CAS:42794-76-3
Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.
Formula:
C12H18N2O4
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
254.28
Ref: TM-T22369
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 148.00 € | ||
| 100mg | 214.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
DORA-22
CAS:1088991-95-0
DORA-22 is a dual orexin receptor antagonist, improves mild stress-induced insomnia with minimal effect on …
Formula:
C23H22F2N4O2
Purity:
97.67%
Color and Shape:
Solid
Molecular weight:
424.44
Ref: TM-T5500
| 1mg | 129.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 697.00 € | ||
| 50mg | 976.00 € | ||
| 100mg | 1,319.00 € | ||
| 1mL*10mM (DMSO) | 330.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
CAY10526
CAS:938069-71-7
CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB …
Formula:
C12H7BrO3S
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
311.15
Ref: TM-T23861
| 1mg | 59.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 209.00 € | ||
| 25mg | 419.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
Pridopidine
CAS:346688-38-8
Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's …
Formula:
C15H23NO2S
Purity:
95.2% - 99.89%
Color and Shape:
Solid
Molecular weight:
281.41
Ref: TM-T7352
| 2mg | 40.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 467.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Monday 2 Dec 2024
