G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SB756050
CAS:447410-57-3
SB756050 is a specific TGR5 agonist.
Formula:
C21H28N2O8S2
Purity:
100% - 98.78%
Color and Shape:
Solid
Molecular weight:
500.59
Ref: TM-T4352
| 5mg | 41.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 203.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Tianeptine sodium salt
CAS:30123-17-2
Tianeptine sodium salt is a selective serotonin reuptake enhancer (SSRE), used to treat major depressive …
Formula:
C21H24ClN2NaO4S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
458.93
Ref: TM-T2402
| 10mg | 46.00 € | ||
| 25mg | 61.00 € | ||
| 50mg | 72.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 136.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BQU57
CAS:1637739-82-2
BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor …
Formula:
C16H13F3N4O
Purity:
98.36% - 98.72%
Color and Shape:
Solid
Molecular weight:
334.3
Ref: TM-T2267
| 5mg | 39.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 203.00 € | ||
| 200mg | 302.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ADL-5859
CAS:850173-95-4
ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against …
Formula:
C24H28N2O3·HCl
Purity:
99.11% - 99.71%
Color and Shape:
Solid
Molecular weight:
428.95
Ref: TM-T6175
| 1mg | 52.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 333.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 739.00 € | ||
| 500mg | 1,514.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Cinacalcet
CAS:226256-56-0
Cinacalcet (AMG 073) is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular …
Formula:
C22H22F3N
Purity:
99.48%
Color and Shape:
Yellow Oil
Molecular weight:
357.41
Ref: TM-T8403
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 143.00 € | ||
| 500mg | 347.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
RO 46-8443
CAS:175556-12-4
RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.
Formula:
C31H35N3O8S
Purity:
98.5% - 99.77%
Color and Shape:
Solid
Molecular weight:
609.69
Ref: TM-T3474
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 348.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,087.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Buclizine dihydrochloride
CAS:129-74-8
Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor …
Formula:
C28H33ClN2·2HCl
Purity:
99.56%
Color and Shape:
Off-White Powder
Molecular weight:
505.95
Ref: TM-T6426
| 50mg | 35.00 € | ||
| 100mg | 49.00 € | ||
| 200mg | 59.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BGC-20-1531 hydrochloride(1186532-61-5 free base)
CAS:1962928-26-2
BGC-20-1531 hydrochloride(1186532-61-5 free base) (GTPL3380 hydrochloride) is a EP4 antagonist for the treatment of acute …
Formula:
C26H25ClN2O6S
Purity:
98.02% - 99.85%
Color and Shape:
Solid
Molecular weight:
529
Ref: TM-T8993L
| 1mg | 129.00 € | ||
| 2mg | 184.00 € | ||
| 5mg | 277.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 698.00 € | ||
| 50mg | 979.00 € | ||
| 1mL*10mM (DMSO) | 365.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Lofexidine
CAS:31036-80-3
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
Formula:
C11H12Cl2N2O
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
259.13
Ref: TM-T7160
| 5mg | 35.00 € | ||
| 50mg | 92.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
a-MSH, amide Acetate(581-05-5 free base)
a-MSH, amide Acetate as an endogenous neuropeptide.
Formula:
C79H113N21O21S
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
1724.94
Ref: TM-TP2212L
| 1mg | 49.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 224.00 € | ||
| 25mg | 482.00 € | ||
| 50mg | 694.00 € | ||
| 100mg | 981.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
WIN 55,212-2 Mesylate
CAS:131543-23-2
WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis …
Formula:
C28H30N2O6S
Purity:
98% - 99.71%
Color and Shape:
White To Off-White Solid
Molecular weight:
522.61
Ref: TM-T4458
| 1ml | 108.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
AdipoRon
CAS:924416-43-3
AdipoRon (SC-396658) is an orally bioavailable adiponectin receptor agonist. It can combine with AdipoR1/2 (KD: …
Formula:
C27H28N2O3
Purity:
98% - 99.86%
Color and Shape:
Solid
Molecular weight:
428.52
Ref: TM-T2257
| 1g | 672.00 € | ||
| 5mg | 40.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 173.00 € | ||
| 100mg | 215.00 € | ||
| 200mg | 277.00 € | ||
| 500mg | 460.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BMS-986020
CAS:1257213-50-5
BMS-986020 (AM152) is a selective antagonist of LPA1.
Formula:
C29H26N2O5
Purity:
100% - 98.82%
Color and Shape:
Solid
Molecular weight:
482.53
Ref: TM-T4016
| 1mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ambrisentan
CAS:177036-94-1
Ambrisentan, an endothelin antagonist for PAH, has a low risk of liver enzyme elevation, not …
Formula:
C22H22N2O4
Purity:
99.65% - 99.86%
Color and Shape:
Solid
Molecular weight:
378.42
Ref: TM-T1655
| 5mg | 35.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 75.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 152.00 € | ||
| 200mg | 218.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
HJC0350
CAS:885434-70-8
HJC0350 is an effective and specific EPAC2 inhibitor (IC50: 0.3 μM), and no inhibition of …
Formula:
C15H19NO2S
Purity:
99.5% - 99.53%
Color and Shape:
Solid
Molecular weight:
277.38
Ref: TM-T6536
| 5mg | 35.00 € | ||
| 10mg | 44.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 216.00 € | ||
| 200mg | 322.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
RU 24969 free base
CAS:66611-26-5
RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.
Formula:
C14H16N2O
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
228.29
Ref: TM-T8593
| 5mg | 61.00 € | ||
| 10mg | 92.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 383.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Conivaptan hydrochloride
CAS:168626-94-6
Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in …
Formula:
C32H26N4O2·HCl
Purity:
100% - 99.86%
Color and Shape:
Solid
Molecular weight:
535.04
Ref: TM-T6453
| 5mg | 43.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 221.00 € | ||
| 100mg | 369.00 € | ||
| 200mg | 557.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Ro 46-2005
CAS:150725-87-4
Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 …
Formula:
C23H27N3O6S
Purity:
98.02% - 98.8%
Color and Shape:
Solid
Molecular weight:
473.54
Ref: TM-T3194
| 5mg | 44.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 292.00 € | ||
| 200mg | 422.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
SORT-PGRN interaction inhibitor 1
CAS:100957-85-5
SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).
Formula:
C15H18N2O2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
258.32
Ref: TM-T9044
| 10mg | 34.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Cotadutide acetate
Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 …
Formula:
C169H256N42O57
Purity:
98.28%
Color and Shape:
Solid
Molecular weight:
3788.14
Ref: TM-TP1103
| 1mg | 148.00 € | ||
| 5mg | 432.00 € | ||
| 10mg | 580.00 € | ||
| 25mg | 925.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
