G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CTCE 9908 acetate
CTCE 9908 acetate is an antagonist of CXCR4 and inhibits migration in CXCR4-expressing ovarian cancer …
Formula:
C88H151N27O25
Purity:
98.47%
Color and Shape:
Liquid
Molecular weight:
1987.31
Ref: TM-TP2051L
| 1mg | 146.00 € | ||
| 5mg | 345.00 € | ||
| 10mg | 517.00 € | ||
| 25mg | 760.00 € | ||
| 50mg | 1,037.00 € | ||
| 100mg | 1,403.00 € | ||
| 200mg | 1,816.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Tolazoline
CAS:59-98-3
Tolazoline (Benzalolin), a vasodilator, treats vessel spasms and reverses 5-HT2A drug overdose effects.
Formula:
C10H12N2
Purity:
97.51%
Color and Shape:
Solid
Molecular weight:
160.22
Ref: TM-T21447
| 500mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Ki16425
CAS:355025-24-0
Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 …
Formula:
C23H23ClN2O5S
Purity:
97.60% - 97.78%
Color and Shape:
Solid
Molecular weight:
474.96
Ref: TM-T6108
| 2mg | 41.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 189.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
PU-H54
CAS:1454619-13-6
PU-H54 is a purine-derived Grp94 inhibitor targeting the S2 subpocket's unique binding region.
Formula:
C18H19N5S
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
337.44
Ref: TM-T8958
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 525.00 € | ||
| 200mg | 712.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, …
Formula:
C43H77N17O12S2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
1088.32
Ref: TM-TP1192L
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 192.00 € | ||
| 100mg | 287.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
3-AQC
CAS:201216-42-4
3-AQC is a competitive antagonist of 5-HT3.
Formula:
C20H21N5O4
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
395.41
Ref: TM-T8475
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 198.00 € | ||
| 200mg | 292.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Empagliflozin
CAS:864070-44-0
Empagliflozin (BI 10773) is an SGLT-2 inhibitor (IC50=3.1 nM) that is potent and selective, with …
Formula:
C23H27ClO7
Purity:
98% - 99.89%
Color and Shape:
Solid
Molecular weight:
450.91
Ref: TM-T1766
| 1g | 277.00 € | ||
| 5mg | 46.00 € | ||
| 10mg | 60.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 142.00 € | ||
| 500mg | 185.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
AVN-101
CAS:1061354-48-0
AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.
Formula:
C21H25ClN2
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
340.89
Ref: TM-T26690
| 1mg | 36.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 575.00 € | ||
| 200mg | 822.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
tcY-NH2 TFA(327177-34-4 free base)
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced …
Formula:
C42H50F3N7O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
853.9
Ref: TM-TP1925L
| 1mg | 101.00 € | ||
| 5mg | 219.00 € | ||
| 10mg | 329.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 708.00 € | ||
| 100mg | 943.00 € | ||
| 200mg | 1,272.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
PD-168077 maleate
CAS:630117-19-0
PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)
Formula:
C24H26N4O5
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
450.49
Ref: TM-T5047
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 402.00 € | ||
| 100mg | 600.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Verucerfont
CAS:885220-61-1
Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .
Formula:
C22H26N6O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
406.48
Ref: TM-T7361
| 1mg | 63.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 135.00 € | ||
| 10mg | 214.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 598.00 € | ||
| 100mg | 838.00 € | ||
| 1mL*10mM (DMSO) | 149.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
AS1269574
CAS:330981-72-1
AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the …
Formula:
C13H14BrN3O
Purity:
99.99%
Color and Shape:
Solid
Molecular weight:
308.17
Ref: TM-T21623
| 2mg | 48.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 308.00 € | ||
| 100mg | 460.00 € | ||
| 500mg | 1,012.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Levalbuterol tartrate
CAS:661464-94-4
Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and …
Formula:
C17H27NO9
Purity:
98.97% - 99.79%
Color and Shape:
Solid
Molecular weight:
389.39
Ref: TM-T7164
| 1mg | 45.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 308.00 € | ||
| 500mg | 730.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
8-Cyclopentyl-1,3-dimethylxanthine
CAS:35873-49-5
8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
Formula:
C12H16N4O2
Purity:
100% - 98.58%
Color and Shape:
Solid
Molecular weight:
248.28
Ref: TM-T27076
| 10mg | 40.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 109.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
BRL 52537 hydrochloride
CAS:112282-24-3
BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke …
Formula:
C18H25Cl3N2O
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
391.76
Ref: TM-T21757
| 1mg | 41.00 € | ||
| 2mg | 53.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 490.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Canagliflozin
CAS:842133-18-0
Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II …
Formula:
C24H25FO5S
Purity:
100% - 99.76%
Color and Shape:
Solid
Molecular weight:
444.52
Ref: TM-T1782
| 5mg | 51.00 € | ||
| 10mg | 66.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 121.00 € | ||
| 200mg | 172.00 € | ||
| 500mg | 291.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Veralipride
CAS:66644-81-3
Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.
Formula:
C17H25N3O5S
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T7632
| 1mg | 64.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 373.00 € | ||
| 50mg | 579.00 € | ||
| 100mg | 871.00 € | ||
| 1mL*10mM (DMSO) | 153.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
2-Chloroadenosine
CAS:146-77-0
2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, …
Formula:
C10H12ClN5O4
Purity:
99.24%
Color and Shape:
White Powder
Molecular weight:
301.69
Ref: TM-T7736
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 130.00 € | ||
| 500mg | 316.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
Mosapride
CAS:112885-41-3
Mosapride (AS-4370) is a selective 5HT4 agonist
Formula:
C21H25ClFN3O3
Purity:
99.56%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
421.89
Ref: TM-T8128
| 5mg | 44.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 153.00 € | ||
| 200mg | 219.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
CHEMBL241987
CAS:109740-09-2
CHEMBL241987 targets the Adenosine receptor A3 (human)
Formula:
C16H11N3O
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
261.28
Ref: TM-T8598
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 157.00 € | ||
| 100mg | 228.00 € | ||
| 200mg | 337.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 19 Dec 2024
