G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Tetradecyl Phosphonate
CAS:4671-75-4
Tetradecyl phosphonate is a pan-antagonist of lysophosphatidic acid 1 (LPA1), LPA2, and LPA3 receptors.
Formula:
C14H31O3P
Purity:
98%
Color and Shape:
White To Off-White Powder
Molecular weight:
278.37
Ref: TM-T7689
| 5mg | 54.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 267.00 € | ||
| 200mg | 402.00 € | ||
| 500mg | 662.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
(±)-Ibipinabant
CAS:362519-49-1
(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and …
Formula:
C23H20Cl2N4O2S
Purity:
99.28% - 99.83%
Color and Shape:
Solid
Molecular weight:
487.4
Ref: TM-T4654
| 1ml | 50.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 409.00 € | ||
| 200mg | 567.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Anisotropine Methylbromide
CAS:80-50-2
Anisotropine Methylbromide is an anticholinergic agent and has been used for relief of gastrointestinal spasm …
Formula:
C17H32BrNO2
Purity:
99.73%
Color and Shape:
Crystals From Acetone Solid
Molecular weight:
362.35
Ref: TM-T4981
| 5mg | 53.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 99.00 € | ||
| 100mg | 125.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Reboxetine mesylate
CAS:98769-84-7
Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).
Formula:
C19H23NO3·CH4O3S
Purity:
99.24% - 99.72%
Color and Shape:
Tan Or Off-White Cyrstalline Solid
Molecular weight:
409.5
Ref: TM-T6963
| 1ml | 53.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 286.00 € | ||
| 100mg | 453.00 € | ||
| 500mg | 989.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SR17018
CAS:2134602-45-0
SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.
Formula:
C19H18Cl3N3O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
410.72
Ref: TM-T4407
| 1ml | 77.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
tcY-NH2 TFA(327177-34-4 free base)
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced …
Formula:
C42H50F3N7O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
853.9
Ref: TM-TP1925L
| 1mg | 101.00 € | ||
| 5mg | 219.00 € | ||
| 10mg | 329.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 708.00 € | ||
| 100mg | 943.00 € | ||
| 200mg | 1,272.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
4-Deoxypyridoxine hydrochloride
CAS:148-51-6
4-Deoxypyridoxine HCl halts S1P breakdown by blocking SPL, reducing apoptosis in insulinoma cells like S1P.
Formula:
C8H12ClNO2
Purity:
99.86%
Color and Shape:
White To Off White Crystalline Powder
Molecular weight:
189.64
Ref: TM-T38294
| 100mg | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cetirizine Impurity B dihydrochloride
CAS:1000690-91-4
Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.
Formula:
C19H23Cl3N2O2
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
417.76
Ref: TM-T9084
| 1ml | 61.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 184.00 € | ||
| 200mg | 272.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pre-084
CAS:138847-85-5
Pre-084 is a high affinity, selective σ1 agonist.
Formula:
C19H28ClNO3
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
353.88
Ref: TM-T3198
| 10mg | 469.00 € | ||
| 50mg | 1,878.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CVN424
CAS:2254706-21-1
CVN424 is a selective and novel GPR6 Inverse agonist effective in models of Parkinson Disease.
Formula:
C24H29F2N5O3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
473.52
Ref: TM-T9346
| 1mg | 94.00 € | ||
| 1ml | 251.00 € | ||
| 5mg | 239.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 878.00 € | ||
| 100mg | 1,189.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PD-168077 maleate
CAS:630117-19-0
PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)
Formula:
C24H26N4O5
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
450.49
Ref: TM-T5047
| 1ml | 56.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 236.00 € | ||
| 100mg | 351.00 € | ||
| 200mg | 499.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
β-Neoendorphin acetate(77739-21-0 free base)
CAS:78658-39-6
beta-Neoendorphin acetate is an agonist of κ-opioid receptor
Formula:
C56H81N13O14
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
1160.34
Ref: TM-TP2322L
| 1mg | 128.00 € | ||
| 5mg | 281.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,324.00 € | ||
| 500mg | 2,627.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Vorapaxar sulfate
CAS:705260-08-8
Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.
Formula:
C29H35FN2O8S
Purity:
99.46% - 99.9%
Color and Shape:
Solid
Molecular weight:
590.66
Ref: TM-T3098
| 1mg | 38.00 € | ||
| 1ml | 98.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 516.00 € | ||
| 500mg | 1,133.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Verucerfont
CAS:885220-61-1
Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .
Formula:
C22H26N6O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
406.48
Ref: TM-T7361
| 1mg | 41.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 491.00 € | ||
| 200mg | 674.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AS1269574
CAS:330981-72-1
AS1269574 is a potent, orally available GPR119 agonist. AS1269574(AS 1269574) has the potential for the …
Formula:
C13H14BrN3O
Purity:
99.99%
Color and Shape:
Solid
Molecular weight:
308.17
Ref: TM-T21623
| 1ml | 88.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 193.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 456.00 € | ||
| 500mg | 1,012.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BAR 501 impurity
CAS:1632118-70-7
BAR501 impurity boosts luciferase in GP-BAR1 assay by 150% at 10 μM, acting as a …
Formula:
C26H46O3
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
406.64
Ref: TM-T8752
| 1mg | 85.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tiprenolol
CAS:26481-51-6
Tiprenolol is a beta adrenergic receptor antagonist.[1]
Formula:
C13H21NO2S
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
255.38
Ref: TM-T50081
| 1mg | 81.00 € | ||
| 1ml | 152.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 241.00 € | ||
| 25mg | 398.00 € | ||
| 50mg | 543.00 € | ||
| 100mg | 760.00 € | ||
| 200mg | 1,000.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
IPSU
CAS:1373765-19-5
IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus …
Formula:
C23H27N5O2
Purity:
97.05%
Color and Shape:
Solid
Molecular weight:
405.49
Ref: TM-T5503
| 1mg | 40.00 € | ||
| 1ml | 92.00 € | ||
| 2mg | 53.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 196.00 € | ||
| 50mg | 293.00 € | ||
| 100mg | 423.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Levalbuterol tartrate
CAS:661464-94-4
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
Formula:
C17H27NO9
Purity:
98% - 99.79%
Color and Shape:
Solid
Molecular weight:
389.39
Ref: TM-T7164
| 1ml | 62.00 € | ||
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 126.00 € | ||
| 100mg | 181.00 € | ||
| 200mg | 264.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JNJ-5207852
CAS:398473-34-2
JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat …
Formula:
C20H32N2O
Purity:
97.19%
Color and Shape:
Solid
Molecular weight:
316.48
Ref: TM-T7413
| 1ml | 50.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 258.00 € | ||
| 100mg | 379.00 € | ||
| 200mg | 539.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
