G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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GLP-1 receptor agonist 9
CAS:2401892-71-3
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
Formula:
C32H31ClFN3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
592.06
Ref: TM-T9579
| 1mg | 144.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 467.00 € | ||
| 25mg | 744.00 € | ||
| 50mg | 1,060.00 € | ||
| 100mg | 1,426.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Urotensin II, mouse acetate (9047-55-6 free base)
Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 …
Formula:
C64H88N14O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1421.61
Ref: TM-TP2165
| 1mg | 96.00 € | ||
| 5mg | 226.00 € | ||
| 10mg | 337.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 974.00 € | ||
| 200mg | 1,301.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
IBC 293
CAS:306935-41-1
IBC 293: Selective GPR109B agonist, favoring it over GPR109A; targets receptor in fat cells.
Formula:
C10H11N3O2
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
205.21
Ref: TM-T19700
| 10mg | 52.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 152.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Methyldopa hydrate
CAS:41372-08-1
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used …
Formula:
C10H13NO4H2O
Purity:
≥98%
Color and Shape:
White Solid
Molecular weight:
238.24
Ref: TM-T5954
| 1g | 52.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Betaxolol
CAS:63659-18-7
Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension …
Formula:
C18H29NO3
Purity:
99.01%
Color and Shape:
White Crystalline Solid
Molecular weight:
307.43
Ref: TM-T6408
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Dynorphin B (1-13) acetate(83335-41-5 free base)
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.
Formula:
C76H119N21O19
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
1630.89
Ref: TM-TP1826L
| 1mg | 90.00 € | ||
| 5mg | 211.00 € | ||
| 10mg | 313.00 € | ||
| 25mg | 505.00 € | ||
| 50mg | 687.00 € | ||
| 100mg | 925.00 € | ||
| 200mg | 1,246.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
GW842166X
CAS:666260-75-9
GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.
Formula:
C18H17Cl2F3N4O2
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
449.25
Ref: TM-T6527
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 327.00 € | ||
| 100mg | 486.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Deltorphin 2
CAS:122752-16-3
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of …
Formula:
C38H54N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
782.88
Ref: TM-T7639
| 1mg | 62.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 521.00 € | ||
| 50mg | 749.00 € | ||
| 100mg | 1,023.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Thonzylamine
CAS:91-85-0
Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy …
Formula:
C16H22N4O
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
286.37
Ref: TM-T4563
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 268.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Carbetocin
CAS:37025-55-1
Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.
Formula:
C45H69N11O12S
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
988.16
Ref: TM-T7601
| 10mg | 513.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Betahistine dihydrochloride
CAS:5579-84-0
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as …
Formula:
C8H14Cl2N2
Purity:
99.34% - 99.88%
Color and Shape:
White To Light Yellow Crystalline Powder
Molecular weight:
209.12
Ref: TM-T0246
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
KH7
CAS:330676-02-3
KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.
Formula:
C17H15BrN4O2S
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
419.3
Ref: TM-T15658
| 1mg | 43.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
CLOZAPINE N-OXIDE
CAS:34233-69-7
View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also …
Formula:
C18H19ClN4O
Purity:
98.43% - 99.94%
Color and Shape:
Solid
Molecular weight:
342.82
Ref: TM-T4494
| 2mg | 40.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 264.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Aticaprant
CAS:1174130-61-0
Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective …
Formula:
C26H27FN2O2
Purity:
99.53% - 99.93%
Color and Shape:
Solid
Molecular weight:
418.5
Ref: TM-TQ0082
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 593.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 …
Formula:
C79H125N23O22
Purity:
98.52%
Color and Shape:
Liquid
Molecular weight:
1748.98
Ref: TM-TP1973L
| 1mg | 269.00 € | ||
| 5mg | 598.00 € | ||
| 10mg | 813.00 € | ||
| 25mg | 1,217.00 € | ||
| 50mg | 1,601.00 € | ||
| 100mg | 2,177.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
MK-0557
CAS:328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 …
Formula:
C22H19FN4O3
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
406.41
Ref: TM-TQ0286
| 1mg | 51.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 159.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 647.00 € | ||
| 200mg | 900.00 € | ||
| 1mL*10mM (DMSO) | 119.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Linzagolix
CAS:935283-04-8
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under …
Formula:
C22H15F3N2O7S
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
508.42
Ref: TM-T27837
| 1mg | 42.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 266.00 € | ||
| 50mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
PW0787
CAS:2624131-45-7
PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).
Formula:
C23H20F4N4O2
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
460.42
Ref: TM-T9452
| 1mg | 56.00 € | ||
| 2mg | 80.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 186.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 581.00 € | ||
| 100mg | 825.00 € | ||
| 1mL*10mM (DMSO) | 143.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ACH-000143
CAS:2225836-30-4
ACH-000143 have been identified as a novel agonist of the melatonin receptors MT1 and MT2.
Formula:
C13H16ClN3O3
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
297.74
Ref: TM-T9193
| 1mg | 51.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 590.00 € | ||
| 200mg | 795.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
NAN-190 hydrobromide
CAS:115338-32-4
NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formula:
C23H28BrN3O3
Purity:
95.92%
Color and Shape:
Solid
Molecular weight:
474.39
Ref: TM-T12172
| 5mg | 43.00 € | ||
| 10mg | 50.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 94.00 € | ||
| 200mg | 167.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
