G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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BD1063 dhydrochloride
CAS:206996-13-6
BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).
Formula:
C13H20Cl4N2
Purity:
98% - 99.52%
Color and Shape:
Solid
Molecular weight:
346.12
Ref: TM-T7488
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 196.00 € | ||
| 100mg | 289.00 € | ||
| 200mg | 406.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
8-Cyclopentyl-1,3-dimethylxanthine
CAS:35873-49-5
8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.
Formula:
C12H16N4O2
Purity:
100% - 98.58%
Color and Shape:
Solid
Molecular weight:
248.28
Ref: TM-T27076
| 10mg | 40.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 109.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Exendin-4 acetate
CAS:914454-01-6
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 …
Formula:
C186H286N50O62S
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
4247
Ref: TM-T8748
| 1mg | 67.00 € | ||
| 5mg | 135.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 412.00 € | ||
| 100mg | 607.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SNAP 94847
CAS:487051-12-7
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM).
Formula:
C29H32F2N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
478.57
Ref: TM-T5406
| 1mg | 49.00 € | ||
| 1ml | 109.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 310.00 € | ||
| 50mg | 528.00 € | ||
| 100mg | 892.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nastorazepide
CAS:209219-38-5
Nastorazepide is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic …
Formula:
C29H36N4O5
Purity:
99.60%
Color and Shape:
Solid
Molecular weight:
520.62
Ref: TM-TQ0062
| 1mg | 52.00 € | ||
| 1ml | 121.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 516.00 € | ||
| 100mg | 744.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Relugolix
CAS:737789-87-6
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) …
Formula:
C29H27F2N7O5S
Purity:
98.64% - 99.67%
Color and Shape:
Solid
Molecular weight:
623.63
Ref: TM-T3630
| 1mg | 36.00 € | ||
| 1ml | 95.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 500.00 € | ||
| 500mg | 1,075.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Questiomycin A
CAS:1916-59-2
Questiomycin A: crème fraiche antibiotic with antibacterial, anticancer effects; inhibits GRP78.
Formula:
C12H8N2O2
Purity:
98% - 99.07%
Color and Shape:
Solid
Molecular weight:
212.2
Ref: TM-T36818
| 10mg | 34.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 82.00 € | ||
| 100mg | 106.00 € | ||
| 200mg | 150.00 € | ||
| 500mg | 244.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BRL 52537 hydrochloride
CAS:112282-24-3
BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke …
Formula:
C18H25Cl3N2O
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
391.76
Ref: TM-T21757
| 1mg | 41.00 € | ||
| 2mg | 53.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 490.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Canagliflozin
CAS:842133-18-0
Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II …
Formula:
C24H25FO5S
Purity:
100% - 99.76%
Color and Shape:
Solid
Molecular weight:
444.52
Ref: TM-T1782
| 1ml | 53.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 66.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 121.00 € | ||
| 200mg | 172.00 € | ||
| 500mg | 291.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Veralipride
CAS:66644-81-3
Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.
Formula:
C17H25N3O5S
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T7632
| 1mg | 64.00 € | ||
| 1ml | 154.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 573.00 € | ||
| 100mg | 861.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
2-Chloroadenosine
CAS:146-77-0
2-Chloroadenosine (CADO) is a metabolically stable analog of adenosine that binds to adenosine A1, A2A, …
Formula:
C10H12ClN5O4
Purity:
99.24%
Color and Shape:
White Powder
Molecular weight:
301.69
Ref: TM-T7736
| 1ml | 34.00 € | ||
| 25mg | 44.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 85.00 € | ||
| 500mg | 185.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Mosapride
CAS:112885-41-3
Mosapride (AS-4370) is a selective 5HT4 agonist
Formula:
C21H25ClFN3O3
Purity:
99.56%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
421.89
Ref: TM-T8128
| 1ml | 55.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 153.00 € | ||
| 200mg | 219.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CHEMBL241987
CAS:109740-09-2
CHEMBL241987 targets the Adenosine receptor A3 (human)
Formula:
C16H11N3O
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
261.28
Ref: TM-T8598
| 1ml | 49.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 157.00 € | ||
| 100mg | 228.00 € | ||
| 200mg | 337.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Avexitide
CAS:133514-43-9
Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 …
Formula:
C149H234N40O47S
Purity:
98% - 98.76%
Color and Shape:
Solid
Molecular weight:
3369.76
Ref: TM-TP2100
| 1mg | 187.00 € | ||
| 5mg | 484.00 € | ||
| 10mg | 689.00 € | ||
| 25mg | 1,033.00 € | ||
| 50mg | 1,399.00 € | ||
| 100mg | 1,810.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GLP-1 receptor agonist 9
CAS:2401892-71-3
1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
Formula:
C32H31ClFN3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
592.06
Ref: TM-T9579
| 1mg | 95.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 436.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 836.00 € | ||
| 200mg | 1,118.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JNJ-37822681
CAS:935776-74-2
JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation …
Formula:
C17H17F5N4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
372.34
Ref: TM-T27677
| 1mg | 94.00 € | ||
| 2mg | 120.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 446.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SB-334867 free base
CAS:792173-99-0
SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.
Formula:
C17H13N5O2
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
319.32
Ref: TM-T6140
| 1mg | 38.00 € | ||
| 1ml | 75.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 535.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pitolisant hydrochloride
CAS:903576-44-3
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki …
Formula:
C17H27Cl2NO
Purity:
99.26% - 99.72%
Color and Shape:
Solid
Molecular weight:
332.31
Ref: TM-T7176
| 1ml | 53.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 305.00 € | ||
| 200mg | 460.00 € | ||
| 500mg | 731.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Clomipramine
CAS:303-49-1
Clomipramine treats OCD, depression, chronic pain, and may lower suicide risk in seniors; works by …
Formula:
C19H23ClN2
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
314.85
Ref: TM-T21013
| 1ml | 87.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 398.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ibutamoren Mesylate
CAS:159752-10-0
Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
Formula:
C28H40N4O8S2
Purity:
97.98% - ≥98%
Color and Shape:
Solid
Molecular weight:
624.77
Ref: TM-T7112
| 1ml | 87.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 83.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 122.00 € | ||
| 500mg | 170.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
