G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).
Formula:
C114H174N34O31
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
2516.81
Ref: TM-TP2279L
| 1mg | 74.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 217.00 € | ||
| 25mg | 362.00 € | ||
| 50mg | 515.00 € | ||
| 100mg | 703.00 € | ||
| 200mg | 903.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Urotensin II, mouse acetate (9047-55-6 free base)
Urotensin II, mouse acetate (9047-55-6 free base) is an endogenous ligand for the orphan GPR14 …
Formula:
C64H88N14O19S2
Purity:
97.86%
Color and Shape:
Solid
Molecular weight:
1421.61
Ref: TM-TP2165
| 1mg | 96.00 € | ||
| 5mg | 226.00 € | ||
| 10mg | 337.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 974.00 € | ||
| 200mg | 1,301.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
IBC 293
CAS:306935-41-1
IBC 293: Selective GPR109B agonist, favoring it over GPR109A; targets receptor in fat cells.
Formula:
C10H11N3O2
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
205.21
Ref: TM-T19700
| 1ml | 46.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 152.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Methyldopa hydrate
CAS:41372-08-1
Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used …
Formula:
C10H13NO4H2O
Purity:
≥98%
Color and Shape:
White Solid
Molecular weight:
238.24
Ref: TM-T5954
| 1g | 52.00 € | ||
| 1ml | 49.00 € | ||
| 500mg | 48.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Betaxolol
CAS:63659-18-7
Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension …
Formula:
C18H29NO3
Purity:
99.01%
Color and Shape:
White Crystalline Solid
Molecular weight:
307.43
Ref: TM-T6408
| 1ml | 43.00 € | ||
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 90.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
DAMGO TFA (78123-71-4(Free base))
Selective Mu-opioid receptor agonist; antinociceptive, boosts cAMP production, triggers TGF-beta1 chemokines, and raises rat food …
Formula:
C28H36F3N5O8
Purity:
98.67% - 99.76%
Color and Shape:
Solid
Molecular weight:
627.6
Ref: TM-T4411
| 1mg | 63.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 282.00 € | ||
| 25mg | 536.00 € | ||
| 50mg | 733.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and …
Formula:
C76H117N19O22S
Purity:
95.43%
Color and Shape:
Solid
Molecular weight:
1680.94
Ref: TM-TP1930L1
| 1mg | 110.00 € | ||
| 5mg | 246.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 543.00 € | ||
| 50mg | 759.00 € | ||
| 100mg | 1,035.00 € | ||
| 200mg | 1,392.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Talinolol
CAS:57460-41-0
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
Formula:
C20H33N3O3
Purity:
98.80%
Color and Shape:
Solid
Molecular weight:
363.49
Ref: TM-T21640
| 1mg | 73.00 € | ||
| 1ml | 168.00 € | ||
| 2mg | 97.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 296.00 € | ||
| 25mg | 534.00 € | ||
| 50mg | 768.00 € | ||
| 100mg | 1,054.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
GW842166X
CAS:666260-75-9
GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.
Formula:
C18H17Cl2F3N4O2
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
449.25
Ref: TM-T6527
| 1ml | 47.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 192.00 € | ||
| 100mg | 285.00 € | ||
| 200mg | 411.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Deltorphin 2
CAS:122752-16-3
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of …
Formula:
C38H54N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
782.88
Ref: TM-T7639
| 1mg | 39.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 305.00 € | ||
| 50mg | 439.00 € | ||
| 100mg | 598.00 € | ||
| 200mg | 805.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Thonzylamine
CAS:91-85-0
Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy …
Formula:
C16H22N4O
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
286.37
Ref: TM-T4563
| 2mg | 35.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 268.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LML134
CAS:1542135-76-1
LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg …
Formula:
C19H29N5O3
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
375.47
Ref: TM-T8514
| 1mg | 79.00 € | ||
| 1ml | 182.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 265.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 1,081.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Carbetocin
CAS:37025-55-1
Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.
Formula:
C45H69N11O12S
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
988.16
Ref: TM-T7601
| 10mg | 513.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ablukast
CAS:96566-25-5
Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.
Formula:
C28H34O8
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
498.56
Ref: TM-T26519
| 1mg | 73.00 € | ||
| 1ml | 198.00 € | ||
| 5mg | 180.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 575.00 € | ||
| 50mg | 806.00 € | ||
| 100mg | 1,095.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Betahistine dihydrochloride
CAS:5579-84-0
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as …
Formula:
C8H14Cl2N2
Purity:
99.34% - 99.88%
Color and Shape:
White To Light Yellow Crystalline Powder
Molecular weight:
209.12
Ref: TM-T0246
| 1g | 34.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Perospirone hydrochloride
CAS:129273-38-7
Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.
Formula:
C23H31ClN4O2S
Purity:
99.37%
Color and Shape:
White Solid
Molecular weight:
463
Ref: TM-T8136
| 1ml | 34.00 € | ||
| 25mg | 44.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 112.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Zafirlukast
CAS:107753-78-6
Zafirlukast (ICI 204219) is an orally available leukotriene receptor antagonist which is widely used for …
Formula:
C31H33N3O6S
Purity:
99% - 99.31%
Color and Shape:
Solid
Molecular weight:
575.68
Ref: TM-T6736
| 1ml | 65.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 91.00 € | ||
| 200mg | 145.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
KH7
CAS:330676-02-3
KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.
Formula:
C17H15BrN4O2S
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
419.3
Ref: TM-T15658
| 1mg | 43.00 € | ||
| 1ml | 89.00 € | ||
| 2mg | 54.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SDZ WAG 994
CAS:130714-47-5
SDZ WAG 994 is an A1 adenosine receptor agonist.
Formula:
C17H25N5O4
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
363.41
Ref: TM-T23347
| 1mg | 98.00 € | ||
| 1ml | 203.00 € | ||
| 5mg | 191.00 € | ||
| 10mg | 286.00 € | ||
| 25mg | 516.00 € | ||
| 50mg | 741.00 € | ||
| 100mg | 1,013.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.
Formula:
C32H51F3N8O9
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
748.79
Ref: TM-T7674
| 1mg | 45.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 141.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 516.00 € | ||
| 200mg | 703.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
