G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Melanotan (MT)-II
CAS:121062-08-6
Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone …
Formula:
C50H69N15O9
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1024.18
Ref: TM-TP1324
| 2mg | 49.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 434.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CLOZAPINE N-OXIDE
CAS:34233-69-7
View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also …
Formula:
C18H19ClN4O
Purity:
98.43% - 99.94%
Color and Shape:
Solid
Molecular weight:
342.82
Ref: TM-T4494
| 2mg | 40.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 179.00 € | ||
| 100mg | 264.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Medetomidine hydrochloride
CAS:86347-15-1
Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold …
Formula:
C13H16N2·HCl
Purity:
96.72%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.74
Ref: TM-T6579
| 1ml | 55.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 236.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
Formula:
C35H51N9O14
Purity:
100%
Color and Shape:
Solid
Molecular weight:
821.84
Ref: TM-TP1419L
| 1mg | 98.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 431.00 € | ||
| 25mg | 649.00 € | ||
| 50mg | 891.00 € | ||
| 100mg | 1,200.00 € | ||
| 200mg | 1,621.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Aticaprant
CAS:1174130-61-0
Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 …
Formula:
C26H27FN2O2
Purity:
99.53% - 99.93%
Color and Shape:
Solid
Molecular weight:
418.5
Ref: TM-TQ0082
| 1mg | 40.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 593.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
CCG215022
CAS:1813527-81-9
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 …
Formula:
C26H22FN7O3
Purity:
97.46% - 99.69%
Color and Shape:
Solid
Molecular weight:
499.5
Ref: TM-T3498
| 1mg | 94.00 € | ||
| 1ml | 257.00 € | ||
| 2mg | 138.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 877.00 € | ||
| 100mg | 1,196.00 € | ||
| 500mg | 2,385.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ONO-7300243
CAS:638132-34-0
ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).
Formula:
C28H31NO5
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
461.55
Ref: TM-T7393
| 1mg | 45.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 407.00 € | ||
| 100mg | 640.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ivabradine hydrochloride
CAS:148849-67-6
Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN …
Formula:
C27H37ClN2O5
Purity:
98.6% - 99.73%
Color and Shape:
Solid
Molecular weight:
505.05
Ref: TM-T2535
| 1ml | 47.00 € | ||
| 10mg | 39.00 € | ||
| 25mg | 54.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 95.00 € | ||
| 200mg | 143.00 € | ||
| 500mg | 246.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
NAN-190 hydrobromide
CAS:115338-32-4
NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formula:
C23H28BrN3O3
Purity:
95.92%
Color and Shape:
Solid
Molecular weight:
474.39
Ref: TM-T12172
| 1ml | 34.00 € | ||
| 10mg | 34.00 € | ||
| 25mg | 42.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 66.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ACH-000143
CAS:2225836-30-4
ACH-000143 have been identified as a novel agonist of the melatonin receptors MT1 and MT2.
Formula:
C13H16ClN3O3
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
297.74
Ref: TM-T9193
| 1mg | 51.00 € | ||
| 1ml | 123.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 590.00 € | ||
| 200mg | 795.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AVN-492
CAS:1220646-23-0
AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
Formula:
C17H21N5O2S
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
359.45
Ref: TM-T5179
| 1mg | 39.00 € | ||
| 1ml | 90.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 501.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
FAUC-365
CAS:474432-66-1
FAUC-365 is a D3 dopamine receptor agonist.
Formula:
C23H25Cl2N3OS
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
462.44
Ref: TM-T21667
| 1mg | 34.00 € | ||
| 1ml | 80.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 428.00 € | ||
| 200mg | 600.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 …
Formula:
C79H125N23O22
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
1748.98
Ref: TM-TP1973L
| 1mg | 269.00 € | ||
| 5mg | 598.00 € | ||
| 10mg | 813.00 € | ||
| 25mg | 1,217.00 € | ||
| 50mg | 1,601.00 € | ||
| 100mg | 2,177.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MK-0557
CAS:328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 …
Formula:
C22H19FN4O3
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
406.41
Ref: TM-TQ0286
| 1mg | 35.00 € | ||
| 1ml | 78.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 379.00 € | ||
| 200mg | 527.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Linzagolix
CAS:935283-04-8
Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under …
Formula:
C22H15F3N2O7S
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
508.42
Ref: TM-T27837
| 1mg | 52.00 € | ||
| 1ml | 115.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 537.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PW0787
CAS:2624131-45-7
PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).
Formula:
C23H20F4N4O2
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
460.42
Ref: TM-T9452
| 1mg | 36.00 € | ||
| 1ml | 93.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 338.00 € | ||
| 100mg | 480.00 € | ||
| 200mg | 661.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ABT-724
CAS:70006-24-5
ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)
Formula:
C17H19N5
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
293.37
Ref: TM-T7834
| 1ml | 90.00 € | ||
| 5mg | 89.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 251.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Grp94 Inhibitor-1
CAS:2234897-35-7
Grp94 Inhibitor-1 is a potent, selective Grp94 inhibitor (IC50 : 2 nM).
Formula:
C22H28N2O2
Purity:
97.02%
Color and Shape:
Solid
Molecular weight:
352.47
Ref: TM-T7261
| 1ml | 51.00 € | ||
| 5mg | 48.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 317.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
VUF10460
CAS:1028327-66-3
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Formula:
C15H19N5
Purity:
98.68% - 99.53%
Color and Shape:
Solid
Molecular weight:
269.34
Ref: TM-T3963
| 1ml | 39.00 € | ||
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 365.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SRT3109
CAS:1204707-71-0
SRT3109 is a CXCR2 ligand used in the treatment of chemokine mediated diseases and conditions.
Formula:
C18H23F2N5O4S2
Purity:
99.65% - 99.92%
Color and Shape:
Solid
Molecular weight:
475.53
Ref: TM-T3047
| 1ml | 64.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 299.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
