G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
9-FLUORENOL
CAS:1689-64-1
9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite …
Formula:
C13H10O
Purity:
99.98%
Color and Shape:
Off-White Crystalline Powder
Molecular weight:
182.22
Ref: TM-T8633
| 1g | 34.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
2-(pentylsulfanyl)pyrimidine-4,6-diol
CAS:489403-70-5
2-(pentylsulfanyl)pyrimidine-4,6-diol is a novel GRP84 agonist.
Formula:
C9H14N2O2S
Purity:
97.58%
Color and Shape:
Solid
Molecular weight:
214.28
Ref: TM-T50078
| 1mg | 81.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 240.00 € | ||
| 25mg | 394.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pregnenolone acetate
CAS:1778-02-5
Pregnenolone acetate inhibits CB1 receptors, blocking THC effects and shielding the brain from cannabis intoxication.
Formula:
C23H34O3
Purity:
99.66%
Color and Shape:
White To Light Yellow Crystalline Powder
Molecular weight:
358.51
Ref: TM-TC0019
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 163.00 € | ||
| 200mg | 232.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Uridine-5'-diphosphate disodium salt
CAS:27821-45-0
UDP disodium salt is a P2Y6 agonist (EC50 = 13 nM), enhances inflammation, phagocytosis, vasoconstriction, …
Formula:
C9H12N2Na2O12P2
Purity:
100% - 98.6%
Color and Shape:
White Fine Crystals
Molecular weight:
448.12
Ref: TM-T4706
| 1ml | 53.00 € | ||
| 50mg | 38.00 € | ||
| 100mg | 49.00 € | ||
| 500mg | 94.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
L-(R,S)-Tetrahydropalmatine
CAS:10097-84-4
L-(R,S)-Tetrahydropalmatine (Rotundine) is extracted from Corydalis yanhusuo W. T. Wang.
Formula:
C21H25NO4
Purity:
99% - 99.97%
Color and Shape:
Solid
Molecular weight:
355.43
Ref: TM-T2714
| 1g | 137.00 € | ||
| 1ml | 33.00 € | ||
| 50mg | 33.00 € | ||
| 100mg | 48.00 € | ||
| 200mg | 61.00 € | ||
| 500mg | 93.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Leuphasyl TFA
CAS:67586-27-0
Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.
Formula:
C31H40F3N5O9
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
683.67
Ref: TM-T20435L
| 1mg | 83.00 € | ||
| 2mg | 107.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ansofaxine hydrochloride
CAS:916918-84-8
Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).
Formula:
C24H32ClNO3
Purity:
99.57% - 99.77%
Color and Shape:
Solid
Molecular weight:
417.97
Ref: TM-T5380
| 1mg | 76.00 € | ||
| 1ml | 175.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 500.00 € | ||
| 50mg | 707.00 € | ||
| 100mg | 916.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 …
Formula:
C118H190N36O30S2
Purity:
96.86%
Color and Shape:
Solid
Molecular weight:
2657.12
Ref: TM-T21611L
| 1mg | 235.00 € | ||
| 2mg | 328.00 € | ||
| 5mg | 489.00 € | ||
| 10mg | 705.00 € | ||
| 25mg | 1,095.00 € | ||
| 50mg | 1,467.00 € | ||
| 100mg | 1,990.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![[D-Ala2]leucine-enkephalin](https://static.cymitquimica.com/products/TM/thumb/TP1367.jpg)
[D-Ala2]leucine-enkephalin
CAS:64963-01-5
[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta …
Formula:
C29H39N5O7
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1367
| 5mg | 39.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 191.00 € | ||
| 100mg | 269.00 € | ||
| 200mg | 376.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Capadenoson
CAS:544417-40-5
Capadenoson (BAY 68-4986) is a selective adenosine-A1 receptor agonist.
Formula:
C25H18ClN5O2S2
Purity:
98.85% - 99.62%
Color and Shape:
Solid
Molecular weight:
520.03
Ref: TM-TQ0125
| 1ml | 47.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Tropisetron
CAS:89565-68-4
Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of …
Formula:
C17H20N2O2
Purity:
99.95%
Color and Shape:
White Solid
Molecular weight:
284.35
Ref: TM-T22448
| 1ml | 50.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 124.00 € | ||
| 100mg | 185.00 € | ||
| 500mg | 478.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Taminadenant
CAS:1337962-47-6
Taminadenant is an adenosine receptor antagonist.
Formula:
C10H8BrN7
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
306.12
Ref: TM-T16980
| 1ml | 34.00 € | ||
| 5mg | 34.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 102.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 232.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
S1RA hydrochloride
CAS:1265917-14-3
S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, …
Formula:
C20H24ClN3O2
Purity:
98% - 99.78%
Color and Shape:
Solid
Molecular weight:
373.87
Ref: TM-T4229
| 1mg | 38.00 € | ||
| 1ml | 88.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 508.00 € | ||
| 500mg | 1,004.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Riociguat
CAS:625115-55-1
Riociguat (BAY 632521) is a stimulator of guanylate cyclase which causes relaxation of vascular smooth …
Formula:
C20H19FN8O2
Purity:
99.91% - 99.95%
Color and Shape:
Solid
Molecular weight:
422.42
Ref: TM-T6968
| 1ml | 69.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 161.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 401.00 € | ||
| 500mg | 912.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
APD597
CAS:897732-93-3
APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes.
Formula:
C21H29N5O6S
Purity:
99.63% - 99.87%
Color and Shape:
Solid
Molecular weight:
479.55
Ref: TM-T3176
| 1ml | 45.00 € | ||
| 5mg | 44.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 135.00 € | ||
| 100mg | 203.00 € | ||
| 200mg | 303.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SR59230A hydrochloride
CAS:1135278-41-9
SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue …
Formula:
C21H28ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
361.91
Ref: TM-T13016L
| 1mg | 45.00 € | ||
| 1ml | 93.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 261.00 € | ||
| 100mg | 386.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Uridine 5′-diphosphoglucose disodium salt
CAS:28053-08-9
Uridine 5′-diphosphoglucose disodium salt (UDP-Glucose sodium salt) is an endogenous nucleotide sugar involved in glycosyltransferase …
Formula:
C15H22N2Na2O17P2
Purity:
100% - 99.83%
Color and Shape:
Solid
Molecular weight:
610.27
Ref: TM-T4743
| 100mg | 50.00 € | ||
| 500mg | 92.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Etrasimod
CAS:1206123-37-6
Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: …
Formula:
C26H26F3NO3
Purity:
99.17% - 99.77%
Color and Shape:
Solid
Molecular weight:
457.48
Ref: TM-TQ0227
| 1mg | 52.00 € | ||
| 1ml | 111.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 237.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 414.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Asapiprant
CAS:932372-01-5
Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited …
Formula:
C24H27N3O7S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
501.55
Ref: TM-T5386
| 1mg | 61.00 € | ||
| 1ml | 169.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 248.00 € | ||
| 25mg | 468.00 € | ||
| 50mg | 742.00 € | ||
| 100mg | 1,207.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
SNAP 94847 hydrochloride
CAS:1781934-47-1
SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)
Formula:
C29H33ClF2N2O2
Purity:
100% - 99.85%
Color and Shape:
Solid
Molecular weight:
515.03
Ref: TM-T8004
| 1ml | 69.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 181.00 € | ||
| 50mg | 306.00 € | ||
| 100mg | 440.00 € | ||
| 200mg | 613.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
