G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Almotriptan
CAS:154323-57-6
Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and …
Formula:
C17H25N3O2S
Purity:
99.85%
Color and Shape:
Light Yellow Or White Power
Molecular weight:
335.46
Ref: TM-T21231
| 1ml | 58.00 € | ||
| 5mg | 43.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 228.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy …
Formula:
C61H88N16O14
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
1269.45
Ref: TM-TP1434L
| 1mg | 74.00 € | ||
| 5mg | 128.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 315.00 € | ||
| 100mg | 479.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Flupentixol dihydrochloride
CAS:2413-38-9
Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive …
Formula:
C23H27Cl2F3N2OS
Purity:
100% - 99.44%
Color and Shape:
White Or Off-White Solid
Molecular weight:
507.43
Ref: TM-T5135
| 1ml | 52.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 92.00 € | ||
| 50mg | 132.00 € | ||
| 100mg | 182.00 € | ||
| 500mg | 467.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ONO-AE3-208
CAS:402473-54-5
ONO-AE3-208 (AE 3-208) is an EP4 antagonist. It suppresses cell migration, invasion, and metastasis of …
Formula:
C24H21FN2O3
Purity:
98% - 98.04%
Color and Shape:
Solid
Molecular weight:
404.43
Ref: TM-TQ0290
| 1ml | 68.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Nelociguat
CAS:625115-52-8
Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.
Formula:
C19H17FN8O2
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
408.39
Ref: TM-T7201
| 1mg | 36.00 € | ||
| 1ml | 84.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 331.00 € | ||
| 200mg | 422.00 € | ||
| 500mg | 554.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C50H72N15O15S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1326.26
Ref: TM-T7567L
| 1mg | 47.00 € | ||
| 1ml | 180.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 450.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 836.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cinacalcet hydrochloride
CAS:364782-34-3
Cinacalcet hydrochloride (AMG-073 hydrochloride) is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity …
Formula:
C22H23ClF3N
Purity:
99.9% - 99.94%
Color and Shape:
Off-White To Tan Solid
Molecular weight:
393.87
Ref: TM-T2406
| 1ml | 53.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 182.00 € | ||
| 500mg | 304.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
HTMT dimaleate
CAS:195867-54-0
HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.
Formula:
C27H33F3N4O9
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
614.57
Ref: TM-T22842
| 1mg | 74.00 € | ||
| 2mg | 94.00 € | ||
| 5mg | 146.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 463.00 € | ||
| 50mg | 671.00 € | ||
| 100mg | 916.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Bimatoprost acid
CAS:38344-08-0
Bimatoprost acid (17-phenyl trinor PGF2α) is a metabolically stable analog of PGF2α and has a …
Formula:
C23H32O5
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
388.5
Ref: TM-T20939
| 1mg | 130.00 € | ||
| 1ml | 319.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 442.00 € | ||
| 25mg | 724.00 € | ||
| 50mg | 1,002.00 € | ||
| 100mg | 1,355.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Ebastine
CAS:90729-43-4
Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.
Formula:
C32H39NO2
Purity:
100% - 99.93%
Color and Shape:
White To Off-White Powder
Molecular weight:
469.66
Ref: TM-T2335
| 1ml | 57.00 € | ||
| 500mg | 56.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
THIQ
CAS:312637-48-2
THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 …
Formula:
C33H41ClN6O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
589.17
Ref: TM-T8485
| 1mg | 52.00 € | ||
| 1ml | 133.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 557.00 € | ||
| 100mg | 829.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
H2L 5765834
CAS:420841-84-5
H2L 5765834 is a lysophosphatidic acid receptors antagonist
Formula:
C21H12N2O7
Purity:
99.47% - ≥98%
Color and Shape:
Solid
Molecular weight:
404.33
Ref: TM-T22834
| 1mg | 60.00 € | ||
| 1ml | 130.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 730.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
PF3274167
CAS:900510-03-4
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
Formula:
C19H19ClFN5O3
Purity:
99.67% - 99.88%
Color and Shape:
Solid
Molecular weight:
419.84
Ref: TM-T3347
| 1ml | 57.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 382.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Spinorphin
CAS:137201-62-8
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
Formula:
C45H64N8O10
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
877
Ref: TM-T8455
| 1mg | 84.00 € | ||
| 5mg | 145.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 520.00 € | ||
| 100mg | 704.00 € | ||
| 200mg | 904.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
MCOPPB triHydrochloride
CAS:1108147-88-1
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
Formula:
C26H43Cl3N4
Purity:
99.89% - 99.91%
Color and Shape:
Solid
Molecular weight:
518.01
Ref: TM-T2071
| 1ml | 56.00 € | ||
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 516.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Propionylpromazine hydrochloride
CAS:7681-67-6
Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.
Formula:
C20H25ClN2OS
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
376.94
Ref: TM-T9228
| 1mg | 38.00 € | ||
| 1ml | 92.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 276.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AZD1981
CAS:802904-66-1
AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma …
Formula:
C19H17ClN2O3S
Purity:
98.59% - 99.54%
Color and Shape:
Solid
Molecular weight:
388.87
Ref: TM-T6399
| 1ml | 34.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 265.00 € | ||
| 200mg | 386.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Cariprazine
CAS:839712-12-8
Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 …
Formula:
C21H32Cl2N4O
Purity:
99.68% - 99.75%
Color and Shape:
Solid
Molecular weight:
427.41
Ref: TM-T4577
| 1mg | 51.00 € | ||
| 1ml | 108.00 € | ||
| 2mg | 78.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 312.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 646.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the …
Formula:
C61H78N18O16
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
1319.38
Ref: TM-TP1700L
| 1mg | 128.00 € | ||
| 5mg | 281.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,327.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
LIT927
CAS:2172879-52-4
LIT927 (LIT-927) is an orally active CXCL12 neutraligand (Ki: 267 nM for CXCL12 binding to …
Formula:
C17H13ClN2O3
Purity:
99.57% - 99.73%
Color and Shape:
Solid
Molecular weight:
328.75
Ref: TM-T5207
| 1ml | 68.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 330.00 € | ||
| 500mg | 779.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
