G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CAY10526
CAS:938069-71-7
CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB …
Formula:
C12H7BrO3S
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
311.15
Ref: TM-T23861
| 1mg | 59.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 209.00 € | ||
| 25mg | 419.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Pridopidine
CAS:346688-38-8
Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's …
Formula:
C15H23NO2S
Purity:
95.2% - 99.89%
Color and Shape:
Solid
Molecular weight:
281.41
Ref: TM-T7352
| 2mg | 40.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 467.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
AZ3451
CAS:2100284-59-9
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
Formula:
C30H27BrN4O3
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
571.46
Ref: TM-TQ0012
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 228.00 € | ||
| 50mg | 402.00 € | ||
| 100mg | 596.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
lumateperone Tosylate
CAS:1187020-80-9
lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors …
Formula:
C31H36FN3O4S
Purity:
95.83% - 98.57%
Color and Shape:
Solid
Molecular weight:
565.7
Ref: TM-TQ0084
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 334.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Antalarmin
CAS:157284-96-3
Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.
Formula:
C24H34N4
Color and Shape:
Liquid
Molecular weight:
378.55
Ref: TM-T70433
| 25mg | 1,397.00 € | ||
| 50mg | 1,820.00 € | ||
| 100mg | 2,297.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
ZM241385
CAS:139180-30-6
ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
Formula:
C16H15N7O2
Purity:
95.28% - 99.69%
Color and Shape:
Solid
Molecular weight:
337.34
Ref: TM-T7021
| 5mg | 56.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 228.00 € | ||
| 100mg | 423.00 € | ||
| 200mg | 638.00 € | ||
| 500mg | 1,009.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Bradykinin (acetate)
CAS:6846-03-3
Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.
Formula:
C52H77N15O13
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1120.26
Ref: TM-T21610
| 1mg | 43.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 399.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
(-)-Isocorypalmine
CAS:483-34-1
(-)-Isocorypalmine ((S)-Tetrahydrocolumbamine), a natural product isolated from Corydalis chaerophylla, has significant antifungal activity.
Formula:
C20H23NO4
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
341.4
Ref: TM-TQ0176
| 1mg | 78.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 233.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
JNJ-63533054
CAS:1802326-66-4
JNJ-63533054 is a potent and selective agonist of hGPR139 with an EC50 = 16 nM.
Formula:
C17H17ClN2O2
Purity:
98.38% - 99.87%
Color and Shape:
Solid
Molecular weight:
316.78
Ref: TM-T3119
| 1mg | 35.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 481.00 € | ||
| 500mg | 1,003.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
SCH442416
CAS:316173-57-6
SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).
Formula:
C20H19N7O2
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
389.41
Ref: TM-T23336
| 1mg | 47.00 € | ||
| 2mg | 62.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 650.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Elinzanetant
CAS:929046-33-3
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive …
Formula:
C33H35F7N4O3
Purity:
98% - 99.13%
Color and Shape:
Odour Color
Molecular weight:
668.64
Ref: TM-T38144
| 1mg | 94.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 782.00 € | ||
| 1mL*10mM (DMSO) | 298.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
EST73502 HCl
CAS:2307458-82-6
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of …
Formula:
C19H27ClF2N2O2
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
388.88
Ref: TM-T39284
| 1mg | 89.00 € | ||
| 5mg | 176.00 € | ||
| 10mg | 251.00 € | ||
| 25mg | 413.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 770.00 € | ||
| 200mg | 1,044.00 € | ||
| 1mL*10mM (DMSO) | 193.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Latanoprost
CAS:130209-82-4
Latanoprost (Xalatan) is a prostaglandin F2alpha analogue and a prostanoid selective FP receptor agonist with …
Formula:
C26H40O5
Purity:
99.69% - 99.78%
Color and Shape:
Pale Yellow Oil
Molecular weight:
432.59
Ref: TM-T2528
| 1mg | 46.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 404.00 € | ||
| 100mg | 595.00 € | ||
| 500mg | 1,263.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Lerisetron
CAS:143257-98-1
Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.
Formula:
C18H20N4
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
292.38
Ref: TM-T8441
| 1mg | 64.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 320.00 € | ||
| 50mg | 470.00 € | ||
| 100mg | 675.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Hemokinin 1 (human) acetate(491851-53-7 free base)
Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.
Formula:
C56H88N14O16S
Purity:
97.82%
Color and Shape:
Solid
Molecular weight:
1245.45
Ref: TM-TP1899L1
| 1mg | 98.00 € | ||
| 5mg | 214.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 779.00 € | ||
| 100mg | 1,068.00 € | ||
| 500mg | 2,126.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Asimadoline hydrochloride
CAS:185951-07-9
Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.
Formula:
C27H31ClN2O2
Purity:
98.63% - 98.94%
Color and Shape:
Solid
Molecular weight:
451.01
Ref: TM-T4691
| 1mg | 35.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 488.00 € | ||
| 500mg | 1,048.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Metoclopramide hydrochloride hydrate
CAS:54143-57-6
Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug …
Formula:
C14H25Cl2N3O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
354.27
Ref: TM-T8385
| 1g | 123.00 € | ||
| 50mg | 37.00 € | ||
| 100mg | 51.00 € | ||
| 500mg | 95.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
Timapiprant
CAS:851723-84-7
Timapiprant (OC000459) is a potent and selective D prostanoid receptor 2 (DP2) antagonist (IC50: 13 …
Formula:
C21H17FN2O2
Purity:
98.4% - 99.89%
Color and Shape:
Solid
Molecular weight:
348.37
Ref: TM-T2664
| 2mg | 41.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 371.00 € | ||
| 200mg | 553.00 € | ||
| 500mg | 879.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
TY-52156
CAS:934369-14-9
TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).
Formula:
C18H19Cl2N3O
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
364.27
Ref: TM-T17183
| 2mg | 40.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 292.00 € | ||
| 100mg | 499.00 € | ||
| 200mg | 668.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
BD-1047 dihydrobromide
CAS:138356-21-5
BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in …
Formula:
C13H22Br2Cl2N2
Purity:
98.13% - 99.39%
Color and Shape:
Solid
Molecular weight:
437.04
Ref: TM-T1740
| 1mg | 36.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 481.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Tuesday 17 Dec 2024
