G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Galanin Receptor Ligand M35 TFA
Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 …
Formula:
C109H154N27F3O28
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
2347.62
Ref: TM-TP1704
| 1mg | 107.00 € | ||
| 5mg | 308.00 € | ||
| 10mg | 433.00 € | ||
| 25mg | 676.00 € | ||
| 50mg | 912.00 € | ||
| 100mg | 1,217.00 € | ||
| 200mg | 1,629.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.
Formula:
C35H47FN10O8
Purity:
97.97%
Color and Shape:
Solid
Molecular weight:
754.85
Ref: TM-TP1127L1
| 1mg | 117.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 385.00 € | ||
| 25mg | 641.00 € | ||
| 50mg | 911.00 € | ||
| 100mg | 1,233.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Carazolol
CAS:57775-29-8
Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) …
Formula:
C18H22N2O2
Purity:
98.54% - 99.08%
Color and Shape:
Yellowish Solid
Molecular weight:
298.38
Ref: TM-T3284
| 25mg | 60.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 113.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
HT-2157
CAS:303149-14-6
HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective …
Formula:
C21H13F3N2O
Purity:
98.33% - 98.55%
Color and Shape:
Solid
Molecular weight:
366.34
Ref: TM-T5455
| 5mg | 55.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 295.00 € | ||
| 100mg | 495.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
L-732138
CAS:148451-96-1
L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)
Formula:
C22H18F6N2O3
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
472.38
Ref: TM-T8235
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 553.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Amperozide
CAS:75558-90-6
Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.
Formula:
C23H29F2N3O
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
401.49
Ref: TM-T23733
| 1mg | 91.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 513.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 995.00 € | ||
| 500mg | 1,979.00 € | ||
| 1mL*10mM (DMSO) | 337.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
M871 acetate
M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 …
Formula:
C110H167N27O30
Purity:
99.84%
Color and Shape:
Liquid
Molecular weight:
2347.67
Ref: TM-TP1994L
| 1mg | 259.00 € | ||
| 5mg | 547.00 € | ||
| 10mg | 730.00 € | ||
| 25mg | 1,089.00 € | ||
| 50mg | 1,464.00 € | ||
| 100mg | 1,985.00 € | ||
| 200mg | 2,681.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GSK1292263
CAS:1032823-75-8
GSK1292263 is a GPR119 agonist and has been investigated for the treatment of DIABETES MELLITUS, …
Formula:
C23H28N4O4S
Purity:
98.34% - 99.46%
Color and Shape:
Solid
Molecular weight:
456.56
Ref: TM-T2701
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 292.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Eltoprazine hydrochloride
CAS:98206-09-8
Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B …
Formula:
C12H17ClN2O2
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
256.73
Ref: TM-T7498
| 5mg | 47.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 253.00 € | ||
| 100mg | 369.00 € | ||
| 500mg | 862.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Guanfacine hydrochloride
CAS:29110-48-3
Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
Formula:
C9H10Cl3N3O
Purity:
99.72% - 99.89%
Color and Shape:
Solid
Molecular weight:
282.55
Ref: TM-T2150
| 10mg | 35.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 90.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 193.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Plecanatide
CAS:467426-54-6
Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) …
Formula:
C65H104N18O26S4
Purity:
97.51%
Color and Shape:
Solid
Molecular weight:
1681.89
Ref: TM-T9080
| 1mg | 78.00 € | ||
| 5mg | 178.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 825.00 € | ||
| 100mg | 1,107.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Phenelzine
CAS:51-71-8
Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.
Formula:
C8H12N2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
136.19
Ref: TM-T9540
| 5mg | To inquire | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 200mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Desmopressin acetate (16679-58-6 free base)
CAS:62288-83-9
Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine …
Formula:
C48H68N14O14S2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1129.26
Ref: TM-T5144
| 1mg | 49.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 527.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
MK-1064
CAS:1207253-08-4
MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).
Formula:
C24H20ClN5O3
Purity:
99.19% - 99.88%
Color and Shape:
Solid
Molecular weight:
461.9
Ref: TM-T3722
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 453.00 € | ||
| 100mg | 730.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Vortioxetine hydrobromide
CAS:960203-27-4
Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 …
Formula:
C18H22N2S·HBr
Purity:
100% - 99.89%
Color and Shape:
Solid
Molecular weight:
379.36
Ref: TM-T2395L
| 25mg | 41.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | 81.00 € | ||
| 500mg | 204.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Zatebradine
CAS:85175-67-3
Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).
Formula:
C26H36N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
456.57
Ref: TM-T13387
| 2mg | 95.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Azaphen dihydrochloride monohydrate
CAS:63302-99-8
Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used …
Formula:
C16H23Cl2N5O2
Color and Shape:
Liquid
Molecular weight:
388.29
Ref: TM-T61741
| 10mg | 43.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 121.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
R 59-022
CAS:93076-89-2
R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus …
Formula:
C27H26FN3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
459.58
Ref: TM-T16709
| 1mg | 37.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 775.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Myristyl nicotinate
CAS:273203-62-6
Myristyl nicotinate (Tetradecyl nicotinate) is an ester prodrug being developed for delivery of nicotinic acid …
Formula:
C20H33NO2
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
319.48
Ref: TM-T19438
| 100mg | 34.00 € | ||
| 200mg | 44.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Tolnapersine
CAS:70312-00-4
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
Formula:
C21H26N2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
322.44
Ref: TM-T68023
| 1mg | 125.00 € | ||
| 5mg | 301.00 € | ||
| 10mg | 442.00 € | ||
| 25mg | 864.00 € | ||
| 50mg | 1,176.00 € | ||
| 100mg | 1,824.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
