G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Neurokinin A
CAS:86933-74-6
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from …
Formula:
C50H80N14O14S
Purity:
100%
Color and Shape:
White To Off-White Lyophilized Solid
Molecular weight:
1133.32
Ref: TM-TP1008
| 1mg | 60.00 € | ||
| 5mg | 117.00 € | ||
| 10mg | 195.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 488.00 € | ||
| 100mg | 694.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
RFRP-1 (human) acetate(311309-25-8 free base)
RFRP-1 (human) acetate: potent NPFF2/1 agonist, alters rat/rabbit cardiac functions, and regulates rat prolactin.
Formula:
C69H105N19O16S
Purity:
96.84%
Color and Shape:
Solid
Molecular weight:
1488.77
Ref: TM-TP1937L1
| 1mg | 128.00 € | ||
| 5mg | 281.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 695.00 € | ||
| 50mg | 978.00 € | ||
| 100mg | 1,318.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
BD 1008 dihydrobromide
CAS:138356-09-9
BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.
Formula:
C15H24Br2Cl2N2
Purity:
97.81%
Color and Shape:
Solid
Molecular weight:
463.08
Ref: TM-T21788
| 1mg | 105.00 € | ||
| 1ml | 200.00 € | ||
| 2mg | 132.00 € | ||
| 5mg | 174.00 € | ||
| 10mg | 272.00 € | ||
| 25mg | 395.00 € | ||
| 50mg | 520.00 € | ||
| 100mg | 775.00 € | ||
| 200mg | 1,035.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![[Sar9,Met(O2)11]-Substance P acetate](https://static.cymitquimica.com/products/TM/thumb/TP1369L.jpg)
[Sar9,Met(O2)11]-Substance P acetate
[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but …
Formula:
C67H106N18O17S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1467.75
Ref: TM-TP1369L
| 1mg | 89.00 € | ||
| 5mg | 341.00 € | ||
| 10mg | 509.00 € | ||
| 25mg | 820.00 € | ||
| 50mg | 1,106.00 € | ||
| 100mg | 1,514.00 € | ||
| 500mg | 3,039.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Regadenoson
CAS:313348-27-5
Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a …
Formula:
C15H18N8O5
Purity:
100% - 99.78%
Color and Shape:
Off-White Solid
Molecular weight:
390.35
Ref: TM-T2671
| 1ml | 72.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 407.00 € | ||
| 500mg | 914.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
RS-127445
CAS:199864-87-4
RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of …
Formula:
C17H16FN3
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
281.33
Ref: TM-T6973
| 1ml | 51.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 197.00 € | ||
| 100mg | 292.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Gadolinium chloride
CAS:10138-52-0
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
Formula:
Cl3Gd
Purity:
98%
Color and Shape:
White Crystalline Solid
Molecular weight:
263.61
Ref: TM-T22795
| 25mg | 48.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | 89.00 € | ||
| 200mg | 124.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Neuropeptide S (Mouse) acetate
Neuropeptide S (Mouse) acetate is a bioactive peptide.
Formula:
C95H160N34O29
Purity:
98.25%
Color and Shape:
Solid
Molecular weight:
2242.5
Ref: TM-TP1981L
| 1mg | 143.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 465.00 € | ||
| 25mg | 739.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,411.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
![[D-Phe12,Leu14]-Bombesin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1916L1.jpg)
[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.
Formula:
C77H118N22O20
Purity:
98.41% - 99.14%
Color and Shape:
Solid
Molecular weight:
1671.9
Ref: TM-TP1916L1
| 1mg | 95.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 310.00 € | ||
| 25mg | 488.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 915.00 € | ||
| 200mg | 1,235.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
ELA-11 (human) acetate(1784687-32-6 free base)
ELA-11: potent apelin receptor agonist, Ki=14 nM. Blocks cAMP, boosts β-arrestin. Part of ELA-32.
Formula:
C60H94N16O15S2
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
1343.61
Ref: TM-TP1922L1
| 1mg | 128.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 695.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,319.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Pimavanserin tartrate
CAS:706782-28-7
Pimavanserin tartrate (Nuplazid) is an effective and specific serotonin 5-HT2A inverse agonist (pIC50: 8.73), used …
Formula:
C50H68F2N6O4·C4H6O6
Purity:
100% - 99.98%
Color and Shape:
Solid
Molecular weight:
1005.2
Ref: TM-T6946
| 1ml | 34.00 € | ||
| 25mg | 50.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 141.00 € | ||
| 500mg | 227.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
DAMGO
CAS:78123-71-4
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity …
Formula:
C26H35N5O6
Purity:
98.83% - 99.92%
Color and Shape:
Solid
Molecular weight:
513.59
Ref: TM-T4351
| 1mg | 50.00 € | ||
| 1ml | 88.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 609.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Deslorelin acetate(57773-65-6 free base)
Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)
Formula:
C66H87N17O14
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
1342.5
Ref: TM-TP2323L
| 1mg | 91.00 € | ||
| 2mg | 118.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 591.00 € | ||
| 100mg | 824.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
1-Ethyl-6-aminouracil
CAS:41862-09-3
1-Ethyl-6-aminouracil (6-AMINO-1-ETHYL-1H-PYRIMIDINE-2,4-DIONE) is an intermediate in the synthesis of a series of new substituted Xanthines …
Formula:
C6H9N3O2
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
155.15
Ref: TM-T8613
| 2mg | 54.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 256.00 € | ||
| 100mg | 384.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
F-15599
CAS:635323-95-4
F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).
Formula:
C19H21ClF2N4O
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
394.85
Ref: TM-T7281
| 1mg | 51.00 € | ||
| 1ml | 131.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 489.00 € | ||
| 100mg | 735.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
TUG-891
CAS:1374516-07-0
TUG-891 is a G protein-coupled receptor expressed in intestine, adipocytes, and pro-inflammatory macrophages that is …
Formula:
C23H21FO3
Purity:
98.28% - 99.21%
Color and Shape:
Solid
Molecular weight:
364.41
Ref: TM-T3433
| 1mg | 40.00 € | ||
| 1ml | 93.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 540.00 € | ||
| 500mg | 1,143.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
cangrelor tetrasodium
CAS:163706-36-3
Cangrelor tetrasodium is a reversible and selective antagonist of platelet P2Y12, with prompt and potent …
Formula:
C17H21Cl2F3N5Na4O12P3S2
Purity:
100% - 99.15%
Color and Shape:
Solid
Molecular weight:
864.29
Ref: TM-T5036
| 1mg | 46.00 € | ||
| 1ml | 134.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 425.00 € | ||
| 100mg | 611.00 € | ||
| 500mg | 1,262.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
JNJ-10229570
CAS:524923-88-4
JNJ-10229570 (UNII-N9IX402L35) is an antagonist of melanocortin receptor 1 (MC1R) and melanocortin receptor 5 (MC5R), …
Formula:
C22H19N3O2S
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
389.47
Ref: TM-T5464
| 1mg | 108.00 € | ||
| 1ml | 210.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 461.00 € | ||
| 50mg | 640.00 € | ||
| 100mg | 828.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
AR-M 1000390 hydrochloride
CAS:209808-47-9
ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from …
Formula:
C23H29ClN2O
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
384.94
Ref: TM-T4236
| 1ml | 77.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 368.00 € | ||
| 100mg | 553.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) …
Formula:
C42H69N13O12
Purity:
98.37%
Color and Shape:
Solid
Molecular weight:
948.08
Ref: TM-TP1884L1
| 1mg | 85.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Tuesday 15 Oct 2024
