G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Alizapride hydrochloride
CAS:59338-87-3
Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea …
Formula:
C16H21N5O2·HCl
Purity:
99.35% - 99.48%
Color and Shape:
Coa
Molecular weight:
351.83
Ref: TM-T2574
| 25mg | 52.00 € | ||
| 50mg | 76.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 162.00 € | ||
| 500mg | 263.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
7-Methoxyrosmanol
CAS:113085-62-4
7-Methoxyrosmanol (7-O-Methylrosmanol) can suppress FSK-induced luciferase expression under the control of the CRE, PEPCK-C and …
Formula:
C21H28O5
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
360.44
Ref: TM-TN1334
| 1mg | 134.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 487.00 € | ||
| 25mg | 774.00 € | ||
| 50mg | 1,040.00 € | ||
| 1mL*10mM (DMSO) | 366.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Amitriptyline
CAS:50-48-6
Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.
Formula:
C20H23N
Purity:
98.24% - 99.64%
Color and Shape:
Crystals Solid
Molecular weight:
277.4
Ref: TM-T22240
| 10mg | 46.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 129.00 € | ||
| 200mg | 185.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Siramesine
CAS:147817-50-3
Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to …
Formula:
C30H31FN2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
454.58
Ref: TM-T4620
| 5mg | 193.00 € | ||
| 10mg | 293.00 € | ||
| 25mg | 447.00 € | ||
| 50mg | 688.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
![[Sar9,Met(O2)11]-Substance P acetate](https://static.cymitquimica.com/products/TM/thumb/TP1369L.jpg)
[Sar9,Met(O2)11]-Substance P acetate
[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but …
Formula:
C67H106N18O17S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1467.75
Ref: TM-TP1369L
| 1mg | 91.00 € | ||
| 5mg | 349.00 € | ||
| 10mg | 518.00 € | ||
| 25mg | 834.00 € | ||
| 50mg | 1,129.00 € | ||
| 100mg | 1,546.00 € | ||
| 200mg | 1,192.00 € | ||
| 500mg | 3,039.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
BD 1008 dihydrobromide
CAS:138356-09-9
BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.
Formula:
C15H24Br2Cl2N2
Purity:
97.81%
Color and Shape:
Solid
Molecular weight:
463.08
Ref: TM-T21788
| 1mg | 64.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 337.00 € | ||
| 50mg | 500.00 € | ||
| 100mg | 712.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
AZD1981
CAS:802904-66-1
AZD1981: selective CRTh2 antagonist, IC50 4 nM, 1000x specificity over 340+ enzymes/receptors, tested in asthma …
Formula:
C19H17ClN2O3S
Purity:
98.59% - 99.54%
Color and Shape:
Solid
Molecular weight:
388.87
Ref: TM-T6399
| 10mg | 50.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 265.00 € | ||
| 200mg | 386.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Almotriptan
CAS:154323-57-6
Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and …
Formula:
C17H25N3O2S
Purity:
99.85%
Color and Shape:
Light Yellow Or White Power
Molecular weight:
335.46
Ref: TM-T21231
| 5mg | 43.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 228.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
APD597
CAS:897732-93-3
APD597 (JNJ-38431055) is a GPR119 agonist, used in the treatment of type 2 diabetes.
Formula:
C21H29N5O6S
Purity:
99.63% - 99.87%
Color and Shape:
Solid
Molecular weight:
479.55
Ref: TM-T3176
| 5mg | 70.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 225.00 € | ||
| 100mg | 349.00 € | ||
| 200mg | 303.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Etilevodopa hydrochloride
CAS:39740-30-2
Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric …
Formula:
C11H16ClNO4
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
261.7
Ref: TM-T24047
| 10mg | 51.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 155.00 € | ||
| 100mg | 241.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
CV 6209
CAS:100488-87-7
Platelet activating factor (PAF) inhibitor
Formula:
C34H60ClN3O6
Purity:
Min. 95%
Molecular weight:
642.31 g/mol
Ref: 3D-FC20594
| 1mg | 501.00 € | ||
| 2mg | 895.00 € | ||
| 5mg | 1,894.00 € | ||
| 10mg | 2,946.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BNP-32 (human)
CAS:124584-08-3
Natriuretic; vasodilatory;diuretic; treats decompensated congestive hear failure
Formula:
C143H244N50O42S4
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
3,464.04 g/mol
Ref: 3D-FB110377
| 1mg | 645.00 € | ||
| 2mg | 934.00 € | ||
| 100µg | 367.00 € | ||
| 250µg | 487.00 € | ||
| 500µg | 544.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Exenatide acetate
CAS:141732-76-5
Agonist of glucagon-like peptide GLP1 which is used for treatment of type 2 diabetes mellitus. …
Formula:
C184H282N50O60S·C2H4O2
Purity:
Min. 95%
Color and Shape:
White Powder
Molecular weight:
4246.63
Ref: 3D-FE23212
| 5mg | 138.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 400.00 € | ||
| 50mg | 602.00 € | ||
| 100mg | 813.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Siponimod
CAS:1230487-00-9
Sphingosine-1-phosphate receptor modulator
Formula:
C29H35F3N2O3
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
516.6 g/mol
Ref: 3D-FS103613
| 10mg | 192.00 € | ||
| 25mg | 271.00 € | ||
| 50mg | 396.00 € | ||
| 100mg | 686.00 € | ||
| 250mg | 1,449.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Baclofen - Bio-X ™
CAS:1134-47-0
Baclofen is a GABA-ergic agonist drug that is used to manage severe spasticity of the …
Formula:
C10H12ClNO2
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
213.66 g/mol
Ref: 3D-BB166152
| 10mg | 136.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Famotidine
CAS:76824-35-6
Famotidine is a selective histamine H2-receptor antagonist used in the treatment of gastric hypersecretory disorders. …
Formula:
C8H15N7O2S3
Purity:
Min. 98 Area-%
Color and Shape:
White Powder
Molecular weight:
337.45 g/mol
Ref: 3D-FF23221
| 100g | 186.00 € | ||
| 250g | 363.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Vismodegib
CAS:879085-55-9
Vismodegib is a Hedgehog (Hh) pathway inhibitor belonging to the 2-arylpyridine class. It acts as …
Formula:
C19H14Cl2N2O3S
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
421.30 g/mol
Ref: 3D-FC28712
| 1g | 378.00 € | ||
| 5g | 1,015.00 € | ||
| 10g | 1,739.00 € | ||
| 250mg | 172.00 € | ||
| 500mg | 271.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Montelukast - Bio-X ™
CAS:158966-92-8
Montelukast is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and …
Formula:
C35H36ClNO3S
Purity:
Min. 98 Area-%
Color and Shape:
Powder
Molecular weight:
586.19 g/mol
Ref: 3D-BM164608
| 50mg | 136.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Fingolimod - Bio-X ™
CAS:162359-55-9
Fingolimod is a sphingosine 1-phosphate receptor modulator that is used in the treatment of relapsing-remitting …
Formula:
C19H33NO2
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
307.47 g/mol
Ref: 3D-BF164460
| 100mg | 137.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Desmopressin acetate
CAS:62288-83-9
Synthetic analog of vasopressin; anti-diuretic; hemostatic
Formula:
C48H68N14O14S2
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
1128.44809
Ref: 3D-FD21366
| 25mg | 136.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 236.00 € | ||
| 250mg | 353.00 € | ||
| 500mg | 550.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
