G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and …
Purity:
98.27%
Molecular weight:
N/A
Ref: TM-TP2071L
| 1mg | 299.00 € | ||
| 5mg | 654.00 € | ||
| 10mg | 881.00 € | ||
| 25mg | 1,312.00 € | ||
| 50mg | 1,783.00 € | ||
| 100mg | 2,411.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as …
Purity:
97.26%
Molecular weight:
N/A
Ref: TM-TP1137L
| 1mg | 185.00 € | ||
| 5mg | 460.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,747.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat …
Purity:
98.42%
Molecular weight:
N/A
Ref: TM-TP1140L
| 1mg | 95.00 € | ||
| 5mg | 228.00 € | ||
| 10mg | 337.00 € | ||
| 25mg | 538.00 € | ||
| 50mg | 726.00 € | ||
| 100mg | 971.00 € | ||
| 200mg | 1,310.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Pancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.
Purity:
98.61%
Molecular weight:
N/A
Ref: TM-TP1044L
| 1mg | 218.00 € | ||
| 5mg | 520.00 € | ||
| 10mg | 704.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,402.00 € | ||
| 100mg | 1,896.00 € | ||
| 200mg | 2,564.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - …
Purity:
95.44% - 96.09%
Molecular weight:
N/A
Ref: TM-TP1199L
| 1mg | 234.00 € | ||
| 5mg | 553.00 € | ||
| 10mg | 746.00 € | ||
| 25mg | 1,103.00 € | ||
| 50mg | 1,486.00 € | ||
| 100mg | 2,009.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Human growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release …
Purity:
99.26%
Molecular weight:
N/A
Ref: TM-TP1155L
| 1mg | 185.00 € | ||
| 5mg | 460.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,747.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
K 41498 aceate
K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for …
Purity:
96.40%
Molecular weight:
N/A
Ref: TM-TP2009L
| 1mg | 308.00 € | ||
| 5mg | 1,054.00 € | ||
| 10mg | 1,417.00 € | ||
| 25mg | 2,108.00 € | ||
| 50mg | 2,843.00 € | ||
| 100mg | 3,833.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
PACAP 1-38 acetate
PACAP 1-38 acetate, a PACAP analog, targets PACAP type I (IC50=4nM) and VIP2 receptors (IC50=1nM), …
Purity:
98.16%
Molecular weight:
N/A
Ref: TM-TP1878L
| 1mg | 157.00 € | ||
| 5mg | 443.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,012.00 € | ||
| 50mg | 1,364.00 € | ||
| 100mg | 1,848.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
PACAP (1-27), human, ovine, rat acetate
PACAP (1-27), human, ovine, rat acetate (PACAP 1-27 acetate) is a novel neuropeptides originally isolated …
Formula:
C144H228N40O41S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
3207.71
Ref: TM-TP1070L
| 1mg | 148.00 € | ||
| 5mg | 418.00 € | ||
| 10mg | 618.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,746.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
ML382
CAS:1646499-97-9
ML382 is a potent and selective MrgX1 positive allosteric modulator(EC50 : 190 nM).
Formula:
C18H20N2O4S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
360.43
Ref: TM-T8538
| 5mg | 47.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 323.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SR59230A hydrochloride
CAS:1135278-41-9
SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue …
Formula:
C21H28ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
361.91
Ref: TM-T13016L
| 1mg | 45.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 261.00 € | ||
| 100mg | 386.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
NLX-204 hydrochloride(2170405-10-2 free base)
NLX-204 hydrochloride is a potent and selective ERK1/2 phosphorylation-preferring serotonin 5 HT1A receptor agonist(pKi = …
Formula:
C20H23Cl2F2N3O2
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
446.32
Ref: TM-T22379L
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
TFLLR-NH2 2TFA(197794-83-5(free base))
TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).
Formula:
C35H55F6N9O10
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
875.87
Ref: TM-T7573L
| 1mL*10mM (DMSO) | 659.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
FTBMT
CAS:1358575-02-6
FTBMT is a GPR52 receptor agonist with an EC50 value of 71 nM. Studies demonstrate …
Formula:
C19H16F4N4O
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
392.35 g/mol
Ref: 3D-BF161243
| 10mg | 374.00 € | ||
| 50mg | 1,046.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Goserelin acetate
CAS:145781-92-6
LHRH analog; GnRH receptor agonist; antineoplastic
Formula:
C59H84N18O14·xH2O
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
1269.41
Ref: 3D-FG44023
| 10mg | 194.00 € | ||
| 25mg | 310.00 € | ||
| 50mg | 436.00 € | ||
| 100mg | 647.00 € | ||
| 250mg | 986.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Oleoyl-L-a-lysophosphatidic acid sodium salt - Bio-X ™
CAS:22556-62-3
OLA is an endogenous agonist of the lysophospholipid receptors LPA1 and LPA2. This chemical compound …
Formula:
C21H40NaO7P
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
458.5 g/mol
Ref: 3D-BO162776
| 1mg | 172.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Cetrorelix acetate
CAS:130143-01-0
Synthetic antagonist of GnRH receptor
Formula:
C70H92ClN17O14
Purity:
Min. 95%
Color and Shape:
White/Off-White Solid
Molecular weight:
1429.66982
Ref: 3D-FC61440
| 2g | 4,863.00 € | ||
| 10mg | 314.00 € | ||
| 50mg | 874.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Melatonin - Bio-X ™
CAS:73-31-4
Melatonin is a neurotransmitter produced by the pineal gland that is involved in the regulation …
Formula:
C13H16N2O2
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
232.28 g/mol
Ref: 3D-BA164660
| 50mg | 136.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Fingolimod phosphate
CAS:402615-91-2
Sphingosine-1-phosphate (S1P) receptor agonist; antineoplastic, immunosppressant
Formula:
C19H34NO5P
Purity:
Min. 95%
Color and Shape:
Powder
Molecular weight:
387.45 g/mol
Ref: 3D-FA27522
| 1mg | 387.00 € | ||
| 2mg | 620.00 € | ||
| 5mg | 1,158.00 € | ||
| 10mg | 1,852.00 € | ||
| 25mg | 3,704.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Terlipressin acetate
CAS:914453-96-6
Vasopressin analog; vasoactive agent
Formula:
C52H74N16O15S2·C2H4O2
Purity:
Min. 98 Area-%
Color and Shape:
Powder
Molecular weight:
1,287.43 g/mol
Ref: 3D-FT35467
| 10mg | 195.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 821.00 € | ||
| 200mg | 1,234.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
