G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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LY2940094
CAS:1307245-86-8
LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
Formula:
C22H23ClF2N4O2S
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
480.96
Ref: TM-T15799
| 1mg | 81.00 € | ||
| 2mg | 106.00 € | ||
| 5mg | 163.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 778.00 € | ||
| 100mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Naftopidil
CAS:57149-07-2
Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as …
Formula:
C24H28N2O3
Purity:
99.4% - 99.97%
Color and Shape:
White Crystalline Powder
Molecular weight:
392.49
Ref: TM-T0696
| 1g | 70.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Urapidil hydrochloride
CAS:64887-14-5
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Formula:
C20H29N5O3·HCl
Purity:
99.93%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
423.94
Ref: TM-T0088
| 1g | 137.00 € | ||
| 100mg | 47.00 € | ||
| 200mg | 62.00 € | ||
| 500mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
EHP-101
CAS:1818428-24-8
EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related …
Formula:
C28H35NO3
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
433.58
Ref: TM-T13289
| 1mg | 107.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 620.00 € | ||
| 50mg | 868.00 € | ||
| 100mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Mebhydrolin napadisylate
CAS:6153-33-9
Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, …
Formula:
C19H20N2C10H8O6S2
Purity:
99.35% - 99.77%
Color and Shape:
White Or Almost White Crystalline
Molecular weight:
420.52
Ref: TM-T0113
| 1g | 64.00 € | ||
| 5g | 136.00 € | ||
| 10g | 188.00 € | ||
| 500mg | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
PF429242 dihydrochloride
CAS:2248666-66-0
PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).
Formula:
C25H37Cl2N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
482.49
Ref: TM-T12437
| 1mg | 43.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 432.00 € | ||
| 100mg | 620.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Salmeterol
CAS:89365-50-4
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
Formula:
C25H37NO4
Purity:
99.87% - 99.9%
Color and Shape:
Solid
Molecular weight:
415.57
Ref: TM-T12829
| 5mg | 55.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Solabegron
CAS:252920-94-8
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese …
Formula:
C23H23ClN2O3
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T12970
| 1mg | 58.00 € | ||
| 5mg | 164.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 472.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 848.00 € | ||
| 200mg | 1,121.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Silodosin
CAS:160970-54-7
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as …
Formula:
C25H32F3N3O4
Purity:
99.63% - 99.76%
Color and Shape:
Colorless To Pink Solid
Molecular weight:
495.53
Ref: TM-T1504
| 5mg | 38.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 81.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 106.00 € | ||
| 200mg | 133.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Prochlorperazine Maleate
CAS:84-02-6
Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; …
Formula:
C28H32ClN3O8S
Purity:
99.99%
Color and Shape:
Off-White Powder
Molecular weight:
606.09
Ref: TM-T0385
| 25mg | 46.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 71.00 € | ||
| 200mg | 116.00 € | ||
| 500mg | 210.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
JNJ-18038683
CAS:851376-05-1
JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for …
Formula:
C26H28ClN3O7
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
529.97
Ref: TM-T11720
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 383.00 € | ||
| 200mg | 545.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Alfuzosin hydrochloride
CAS:81403-68-1
Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign …
Formula:
C19H27N5O4·HCl
Purity:
99.61%
Color and Shape:
White To Off-White Solid
Molecular weight:
425.91
Ref: TM-T0091
| 10mg | 46.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 105.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 221.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Loperamide hydrochloride
CAS:34552-83-5
Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
Formula:
C29H34Cl2N2O2
Purity:
100% - 99.78%
Color and Shape:
Crystals Practically Insoluble In Water
Molecular weight:
513.498
Ref: TM-T0209
| 100mg | 55.00 € | ||
| 500mg | 85.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Alosetron hydrochloride
CAS:122852-69-1
Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin …
Formula:
C17H19ClN4O
Purity:
100%
Color and Shape:
Off-White Powder
Molecular weight:
330.81
Ref: TM-T2525
| 10mg | 37.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 113.00 € | ||
| 100mg | 177.00 € | ||
| 200mg | 263.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Terbutaline
CAS:23031-25-6
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite …
Formula:
C12H19NO3
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
225.3
Ref: TM-T8810
| 5mg | 43.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 117.00 € | ||
| 1mL*10mM (DMSO) | 48.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Prucalopride
CAS:179474-81-8
Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these …
Formula:
C18H26ClN3O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
367.87
Ref: TM-T2542
| 10mg | 46.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 111.00 € | ||
| 200mg | 165.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Lamotrigine
CAS:84057-84-1
Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.
Formula:
C9H7Cl2N5
Purity:
99.76% - 99.91%
Color and Shape:
White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
Molecular weight:
256.09
Ref: TM-T0680
| 1g | 79.00 € | ||
| 5g | 258.00 € | ||
| 200mg | 37.00 € | ||
| 500mg | 50.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Ifenprodil
CAS:23210-56-2
Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, …
Formula:
C21H27NO2
Purity:
99.78%
Color and Shape:
White Crystalline Powder
Molecular weight:
325.44
Ref: TM-T1186L
| 1mg | 110.00 € | ||
| 5mg | 215.00 € | ||
| 10mg | 324.00 € | ||
| 25mg | 520.00 € | ||
| 50mg | 702.00 € | ||
| 100mg | 932.00 € | ||
| 200mg | 1,283.00 € | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Pemirolast potassium
CAS:100299-08-9
Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.
Formula:
C10H7KN6O
Purity:
98.91% - 99.63%
Color and Shape:
Crystals From Dimethylformamide Crystalline Solid
Molecular weight:
266.31
Ref: TM-T1425
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 160.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Metaproterenol hemisulfate
CAS:5874-97-5
Metaproterenol hemisulfate (Orciprenaline sulfate) is a beta-2 adrenergic agonist used in the treatment of ASTHMA …
Formula:
C11H17NO3·5H2O4S
Purity:
99.74% - 99.83%
Color and Shape:
Solid
Molecular weight:
260.3
Ref: TM-T0277
| 25mg | 35.00 € | ||
| 50mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
