G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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N6-Cyclohexyladenosine
CAS:36396-99-3
N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.
Formula:
C16H23N5O4
Purity:
99.84% - 99.98%
Color and Shape:
Solid
Molecular weight:
349.38
Ref: TM-T12160
| 10mg | 34.00 € | ||
| 25mg | 60.00 € | ||
| 50mg | 101.00 € | ||
| 100mg | 150.00 € | ||
| 200mg | 213.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Rupatadine Fumarate
CAS:182349-12-8
Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 …
Formula:
C26H26ClN3·C4H4O4
Purity:
99.64%
Color and Shape:
White Or Almost-White Powder
Molecular weight:
532.03
Ref: TM-T6242
| 1g | 180.00 € | ||
| 25mg | 38.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 69.00 € | ||
| 500mg | 125.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Adrenalone hydrochloride
CAS:62-13-5
Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.
Formula:
C9H11NO3·HCl
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
217.65
Ref: TM-T0948
| 1g | 142.00 € | ||
| 50mg | 35.00 € | ||
| 100mg | 50.00 € | ||
| 500mg | 94.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
hGPR91 antagonist 1
CAS:1314796-00-3
hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).
Formula:
C31H23F4N3O
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
529.53
Ref: TM-T11560
| 1mg | 94.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 293.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 676.00 € | ||
| 100mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 221.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Nicergoline
CAS:27848-84-6
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with …
Formula:
C24H26BrN3O3
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
484.39
Ref: TM-T1132
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 68.00 € | ||
| 50mg | 84.00 € | ||
| 100mg | 103.00 € | ||
| 200mg | 148.00 € | ||
| 500mg | 231.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
NE 52-QQ57
CAS:1401728-56-0
NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory …
Formula:
C24H28N6O
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
416.52
Ref: TM-T11461
| 1mg | 73.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 231.00 € | ||
| 25mg | 386.00 € | ||
| 50mg | 573.00 € | ||
| 100mg | 821.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Solabegron
CAS:252920-94-8
Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese …
Formula:
C23H23ClN2O3
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T12970
| 1mg | 57.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 459.00 € | ||
| 50mg | 621.00 € | ||
| 100mg | 825.00 € | ||
| 200mg | 1,090.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Linaclotide
CAS:851199-59-2
Linaclotide treats IBS-C & chronic constipation; it's a selective guanylate cyclase C agonist.
Formula:
C59H79N15O21S6
Purity:
97.93% - 98.71%
Color and Shape:
Solid
Molecular weight:
1526.74
Ref: TM-T11852
| 1mg | 65.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 480.00 € | ||
| 100mg | 684.00 € | ||
| 1mL*10mM (DMSO) | 268.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
(R)-Terazosin
CAS:109351-34-0
R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 …
Formula:
C19H25N5O4
Purity:
98.87% - 98.96%
Color and Shape:
Solid
Molecular weight:
387.43
Ref: TM-T12643
| 1mg | 46.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 484.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Pizotifen
CAS:15574-96-6
Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available …
Formula:
C19H21NS
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
295.44
Ref: TM-T1442
| 50mg | 42.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 77.00 € | ||
| 500mg | 124.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Tizanidine hydrochloride
CAS:64461-82-1
Tizanidine hydrochloride (Tizanidine HCl), an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
Formula:
C9H9Cl2N5S
Purity:
99.87%
Color and Shape:
Solid White
Molecular weight:
290.17
Ref: TM-T0290
| 10mg | 51.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 131.00 € | ||
| 500mg | 209.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
AB928
CAS:2239273-34-6
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
Formula:
C23H22N8O
Purity:
100% - 98.09%
Color and Shape:
Solid
Molecular weight:
426.47
Ref: TM-T14078
| 1mg | 51.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 388.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 662.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Nadolol
CAS:42200-33-9
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.
Formula:
C17H27NO4
Purity:
99.87% - 99.92%
Color and Shape:
White To Off-White Crystalline Powder Solid
Molecular weight:
309.4
Ref: TM-T1203
| 25mg | 49.00 € | ||
| 50mg | 72.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Evatanepag
CAS:223488-57-1
Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting …
Formula:
C25H28N2O5S
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
468.57
Ref: TM-T15259
| 1mg | 68.00 € | ||
| 5mg | 155.00 € | ||
| 10mg | 241.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 597.00 € | ||
| 100mg | 816.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Sertraline hydrochloride
CAS:79559-97-0
Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the …
Formula:
C17H18Cl3N
Purity:
99.12% - 99.86%
Color and Shape:
Solid Powder
Molecular weight:
342.691
Ref: TM-T0482
| 5mg | 51.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 101.00 € | ||
| 50mg | 176.00 € | ||
| 100mg | 230.00 € | ||
| 200mg | 298.00 € | ||
| 500mg | 507.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Lamotrigine
CAS:84057-84-1
Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.
Formula:
C9H7Cl2N5
Purity:
99.76% - 99.91%
Color and Shape:
White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
Molecular weight:
256.09
Ref: TM-T0680
| 1g | 83.00 € | ||
| 5g | 253.00 € | ||
| 200mg | 41.00 € | ||
| 500mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Evocalcet
CAS:870964-67-3
Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).
Formula:
C24H26N2O2
Purity:
98.41% - 99.83%
Color and Shape:
Solid
Molecular weight:
374.48
Ref: TM-T15261
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 366.00 € | ||
| 500mg | 847.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Adenosine A1 receptor activator T62
CAS:40312-34-3
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it …
Formula:
C15H14ClNOS
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
291.8
Ref: TM-T14127
| 1mg | 95.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 263.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 271.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Terbutaline
CAS:23031-25-6
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite …
Formula:
C12H19NO3
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
225.3
Ref: TM-T8810
| 5mg | 42.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Olopatadine hydrochloride
CAS:140462-76-6
Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in …
Formula:
C21H23NO3·HCl
Purity:
100% - 99.78%
Color and Shape:
White Solid
Molecular weight:
373.87
Ref: TM-T1170
| 5mg | 36.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 160.00 € | ||
| 500mg | 263.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
