G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Atenolol
CAS:29122-68-7
Atenolol (Tenormin) is a selective β1 receptor antagonist.
Formula:
C14H22N2O3
Purity:
99.07%
Color and Shape:
White Crystalline Powder Solid
Molecular weight:
266.3361
Ref: TM-T0007
| 1ml | 54.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
KGA-2727
CAS:666842-36-0
KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity …
Formula:
C26H40N4O8
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
536.62
Ref: TM-T15656
| 1mg | 131.00 € | ||
| 2mg | 180.00 € | ||
| 5mg | 271.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 740.00 € | ||
| 50mg | 1,013.00 € | ||
| 100mg | 1,388.00 € | ||
| 1mL*10mM (DMSO) | 318.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PF-04995274
CAS:1331782-27-4
PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive …
Formula:
C23H32N2O6
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
432.51
Ref: TM-T16481
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 498.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Buflomedil hydrochloride
CAS:35543-24-9
Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of …
Formula:
C17H26ClNO4
Purity:
99.67% - 99.7%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
343.85
Ref: TM-T0317
| 1g | 84.00 € | ||
| 5g | 175.00 € | ||
| 100mg | 41.00 € | ||
| 500mg | 58.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Granisetron hydrochloride
CAS:107007-99-8
Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used …
Formula:
C18H25ClN4O
Purity:
99.88% - 99.94%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
348.87
Ref: TM-T1042
| 10mg | 38.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 81.00 € | ||
| 100mg | 126.00 € | ||
| 200mg | 176.00 € | ||
| 500mg | 300.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Loxapine succinate
CAS:27833-64-3
Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.
Formula:
C22H24ClN3O5
Purity:
99.92%
Color and Shape:
White To Of-White Solid
Molecular weight:
445.9
Ref: TM-T1412
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 82.00 € | ||
| 500mg | 161.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PF429242 dihydrochloride
CAS:2248666-66-0
PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).
Formula:
C25H37Cl2N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
482.49
Ref: TM-T12437
| 1mg | 43.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 606.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Bambuterol hydrochloride
CAS:81732-46-9
Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of …
Formula:
C18H30ClN3O5
Purity:
100% - 99.74%
Color and Shape:
White Solid
Molecular weight:
403.91
Ref: TM-T1446
| 10mg | 52.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 135.00 € | ||
| 500mg | 212.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Droperidol
CAS:548-73-2
Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as …
Formula:
C22H22FN3O2
Purity:
97.16% - 98%
Color and Shape:
Solid
Molecular weight:
379.43
Ref: TM-T0990
| 100mg | 51.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
DREADD agonist 21
CAS:56296-18-5
DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).
Formula:
C17H18N4
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
278.35
Ref: TM-T11095L
| 2mg | 34.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 136.00 € | ||
| 50mg | 214.00 € | ||
| 100mg | 318.00 € | ||
| 200mg | 456.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Haloperidol
CAS:52-86-8
Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve …
Formula:
C21H23ClFNO2
Purity:
99.69% - 99.76%
Color and Shape:
Crystals Solid
Molecular weight:
375.86
Ref: TM-T0025
| 25mg | 40.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 75.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Fluoxetine hydrochloride
CAS:56296-78-7
Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side …
Formula:
C17H19ClF3NO
Purity:
99.6% - 99.98%
Color and Shape:
White To Off-White Crystalline Solid White To Off-White Powder
Molecular weight:
345.787
Ref: TM-T0450L
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 148.00 € | ||
| 500mg | 239.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Carteolol hydrochloride
CAS:51781-21-6
Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.
Formula:
C16H24N2O3·HCl
Purity:
99.91% - 99.97%
Color and Shape:
Solid
Molecular weight:
328.83
Ref: TM-T1282
| 10mg | 37.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 110.00 € | ||
| 200mg | 162.00 € | ||
| 500mg | 265.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Sulfisoxazole
CAS:127-69-5
Sulfisoxazole: a short-acting antibacterial targeting gram-positive/negative bacteria and inhibits breast cancer exosome by affecting endothelin …
Formula:
C11H13N3O3S
Purity:
99.98%
Color and Shape:
White To Cream Powder
Molecular weight:
267.3
Ref: TM-T0750
| 1g | 73.00 € | ||
| 200mg | 37.00 € | ||
| 500mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Pizotifen Malate
CAS:5189-11-7
Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based …
Formula:
C19H21NS·C4H6O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
429.53
Ref: TM-T0225
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Metaraminol tartrate
CAS:33402-03-8
Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.
Formula:
C13H19NO8
Purity:
99.53%
Color and Shape:
White Powder
Molecular weight:
317.29
Ref: TM-T0279
| 50mg | 50.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 90.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Fluoxetine
CAS:54910-89-3
Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.
Formula:
C17H18F3NO
Purity:
99.07% - 99.28%
Color and Shape:
Solid
Molecular weight:
309.33
Ref: TM-T0450
| 10mg | 40.00 € | ||
| 25mg | 53.00 € | ||
| 50mg | 67.00 € | ||
| 100mg | 85.00 € | ||
| 200mg | 124.00 € | ||
| 500mg | 216.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Loperamide hydrochloride
CAS:34552-83-5
Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
Formula:
C29H34Cl2N2O2
Purity:
100% - 99.78%
Color and Shape:
Crystals Practically Insoluble In Water
Molecular weight:
513.498
Ref: TM-T0209
| 100mg | 59.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Quetiapine
CAS:111974-69-7
Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine …
Formula:
C21H25N3O2S
Purity:
100% - 99.14%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
383.51
Ref: TM-T0162
| 10mg | 59.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 118.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Trazodone hydrochloride
CAS:25332-39-2
Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive …
Formula:
C19H23Cl2N5O
Purity:
99.50% - 99.52%
Color and Shape:
Solid
Molecular weight:
408.33
Ref: TM-T1619
| 50mg | 46.00 € | ||
| 100mg | 57.00 € | ||
| 500mg | 83.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
