G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ziprasidone hydrochloride
CAS:122883-93-6
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows …
Formula:
C21H22CL2N4OS
Purity:
98.37% - 99.34%
Color and Shape:
Solid
Molecular weight:
449.4
Ref: TM-T0031L
| 5mg | 44.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 91.00 € | ||
| 50mg | 130.00 € | ||
| 100mg | 163.00 € | ||
| 500mg | 388.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Clopidogrel hydrogen sulfate
CAS:120202-66-6
Clopidogrel hydrogen sulfate is a selective P2Y12 receptor blocker that inhibits platelet adhesion and aggregation.
Formula:
C16H16ClNO2S·H2SO4
Purity:
99.51% - 99.57%
Color and Shape:
Solid
Molecular weight:
419.9
Ref: TM-T0182L
| 25mg | 36.00 € | ||
| 50mg | 47.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 63.00 € | ||
| 500mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bromopride
CAS:4093-35-0
Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the …
Formula:
C14H22BrN3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
344.25
Ref: TM-T1175
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 266.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 560.00 € | ||
| 200mg | 781.00 € | ||
| 500mg | 1,180.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MRS-1706
CAS:264622-53-9
MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.
Formula:
C27H29N5O5
Purity:
97.95%
Color and Shape:
Solid
Molecular weight:
503.55
Ref: TM-T16136
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 238.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 678.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Docusate sodium
CAS:577-11-7
Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to …
Formula:
C20H37NaO7S
Purity:
99.77%
Color and Shape:
White Wax-Like Solid With Water (Uscg 1999)
Molecular weight:
444.56
Ref: TM-T0929
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € | ||
| 500mg | 120.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Levocarnitine propionate hydrochloride
CAS:119793-66-7
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, …
Formula:
C10H20ClNO4
Purity:
90% - 98%
Color and Shape:
Solid
Molecular weight:
253.72
Ref: TM-T1182
| 25mg | 35.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 500mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Risperidone
CAS:106266-06-2
Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 …
Formula:
C23H27FN4O2
Purity:
100%
Color and Shape:
Crystalline Solid
Molecular weight:
410.48
Ref: TM-T0351
| 10mg | 55.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 203.00 € | ||
| 500mg | 338.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CD80-IN-3
CAS:486449-65-4
CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 …
Formula:
C17H10FN3O3
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
323.28
Ref: TM-T10722
| 1mg | 79.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 482.00 € | ||
| 50mg | 666.00 € | ||
| 100mg | 828.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
EMPA
CAS:680590-49-2
EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 …
Formula:
C23H26N4O4S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
454.54
Ref: TM-T11186
| 1mg | 51.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 327.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 688.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Cyproheptadine hydrochloride sesquihydrate
CAS:41354-29-4
Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.
Formula:
C21H24ClNO
Purity:
100% - 100%
Color and Shape:
White To Slightly Yellowish Crystalline Solid
Molecular weight:
341.88
Ref: TM-T0174
| 500mg | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pheniramine maleate
CAS:132-20-7
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 …
Formula:
C16H20N2·C4H4O4
Purity:
99.79%
Color and Shape:
Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
Molecular weight:
356.42
Ref: TM-T0370
| 25mg | 36.00 € | ||
| 50mg | 45.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 65.00 € | ||
| 500mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Alarelin Acetate
CAS:79561-22-1
Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis …
Formula:
C56H78N16O12
Purity:
100% - 99.81%
Color and Shape:
White Powder
Molecular weight:
1167.34
Ref: TM-T1494
| 5mg | 57.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 176.00 € | ||
| 500mg | 443.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MP-A08
CAS:219832-49-2
MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 …
Formula:
C27H25N3O4S2
Purity:
98.04%
Color and Shape:
Solid
Molecular weight:
519.64
Ref: TM-T16128
| 1mg | 46.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 302.00 € | ||
| 100mg | 537.00 € | ||
| 500mg | 1,109.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
2-Bromo-6-methoxynaphthalene
CAS:5111-65-9
2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.
Formula:
C11H9BrO
Purity:
98.8%
Color and Shape:
White To Off-White Powder
Molecular weight:
237.09
Ref: TM-T0663
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ceruletide
CAS:17650-98-5
Ceruletide is a decapeptide that is a safe and effective cholecystokinin and cholecystokinin receptor agonist.Cost-effective …
Formula:
C58H73N13O21S2
Purity:
97.54% - 98.47%
Color and Shape:
Solid
Molecular weight:
1352.4
Ref: TM-T14932
| 1mg | 157.00 € | ||
| 5mg | 425.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,727.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Roxatidine Acetate hydrochloride
CAS:93793-83-0
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits …
Formula:
C19H29ClN2O4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
384.9
Ref: TM-T0157
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Fezagepras
CAS:1002101-19-0
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist …
Formula:
C13H18O2
Purity:
96.73% - 99.38%
Color and Shape:
Solid
Molecular weight:
206.28
Ref: TM-T12883
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Agomelatine
CAS:138112-76-2
Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
Formula:
C15H17NO2
Purity:
99.92%
Color and Shape:
White Solid
Molecular weight:
243.3
Ref: TM-T1445
| 5mg | 67.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 732.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Phenothiazine
CAS:92-84-2
Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.
Formula:
C12H9NS
Purity:
99.94%
Color and Shape:
Yellow Solid Pellets
Molecular weight:
199.27
Ref: TM-T0776
| 1g | 41.00 € | ||
| 5g | 86.00 € | ||
| 10g | 112.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
