G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Degarelix acetate(214766-78-6 free base)
CAS:934016-19-0
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
Formula:
C84H107ClN18O18
Purity:
98.66%
Color and Shape:
Liquid
Molecular weight:
1692.34
Ref: TM-T10988L
| 1mg | 75.00 € | ||
| 2mg | 97.00 € | ||
| 5mg | 162.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 468.00 € | ||
| 50mg | 680.00 € | ||
| 100mg | 920.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Duloxetine hydrochloride
CAS:136434-34-9
Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.
Formula:
C18H20ClNOS
Purity:
100% - 99.97%
Color and Shape:
White Or White Crystalline Powder
Molecular weight:
333.88
Ref: TM-T1471
| 10mg | 52.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 130.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
NEO 376
CAS:496921-73-4
NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing …
Formula:
C20H24ClN3O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
357.88
Ref: TM-T12207
| 1mg | 72.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 208.00 € | ||
| 25mg | 359.00 € | ||
| 50mg | 504.00 € | ||
| 100mg | 676.00 € | ||
| 200mg | 909.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Labetalol hydrochloride
CAS:32780-64-6
Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic …
Formula:
C19H25ClN2O3
Purity:
99.29% - 99.85%
Color and Shape:
Solid
Molecular weight:
364.87
Ref: TM-T0348
| 50mg | 46.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 112.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
NTP42
CAS:2055599-51-2
NTP42 is an antagonist of thromboxane A2 (TXA2) receptor(IC50 of 3.278 nM)
Formula:
C25H23F2N3O5S
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
515.53
Ref: TM-T12268
| 1mg | 62.00 € | ||
| 2mg | 89.00 € | ||
| 5mg | 139.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 534.00 € | ||
| 100mg | 766.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Domperidone
CAS:57808-66-9
Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.
Formula:
C22H24ClN5O2
Purity:
98% - 99.73%
Color and Shape:
Solid
Molecular weight:
425.91
Ref: TM-T0082
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 93.00 € | ||
| 500mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
JP1302 dihydrochloride
CAS:1259314-65-2
JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.
Formula:
C24H26Cl2N4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
441.4
Ref: TM-T11726
| 1mg | 45.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 556.00 € | ||
| 500mg | 1,196.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Azacyclonol
CAS:115-46-8
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
Formula:
C18H21NO
Purity:
99.61%
Color and Shape:
Solid Powder
Molecular weight:
267.37
Ref: TM-T0318
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Chlorprothixene hydrochloride
CAS:6469-93-8
Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.
Formula:
C18H18ClNS·HCl
Purity:
99.16%
Color and Shape:
White Powder
Molecular weight:
352.32
Ref: TM-T0074L
| 100mg | 37.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Famotidine
CAS:76824-35-6
Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.
Formula:
C8H15N7O2S3
Purity:
99.33% - 99.75%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
337.45
Ref: TM-T1627
| 2g | 54.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Itopride hydrochloride
CAS:122892-31-3
Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
Formula:
C20H27ClN2O4
Purity:
99.76%
Color and Shape:
White Or Pale Brownish Crystal
Molecular weight:
394.9
Ref: TM-T1552
| 50mg | 41.00 € | ||
| 100mg | 54.00 € | ||
| 500mg | 85.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Aniracetam
CAS:72432-10-1
Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and …
Formula:
C12H13NO3
Purity:
99.8%
Color and Shape:
White Crystalline Or Crystalline Powde
Molecular weight:
219.24
Ref: TM-T0333
| 1g | 51.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Seltorexant
CAS:1293281-49-8
Seltorexant (JNJ-42847922) crosses the blood-brain barrier and quickly occupies OX2R binding sites in the rat …
Formula:
C21H22FN7O
Purity:
100% - 99.86%
Color and Shape:
Solid
Molecular weight:
407.44
Ref: TM-T12877L
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 149.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 369.00 € | ||
| 500mg | 853.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Tripelennamine hydrochloride
CAS:154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent …
Formula:
C16H21N3·HCl
Purity:
100% - 100%
Color and Shape:
White Solid
Molecular weight:
291.82
Ref: TM-T1269
| 1g | 138.00 € | ||
| 100mg | 37.00 € | ||
| 500mg | 93.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ondansetron hydrochloride dihydrate
CAS:103639-04-9
Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported …
Formula:
C18H19N3O·HCl·2H2O
Purity:
99.71%
Color and Shape:
White Crystal Powder
Molecular weight:
365.86
Ref: TM-T1478
| 25mg | 47.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 64.00 € | ||
| 200mg | 78.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Anamorelin
CAS:249921-19-5
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
Formula:
C31H42N6O3
Purity:
99.35% - 99.88%
Color and Shape:
Solid
Molecular weight:
546.7
Ref: TM-T10319
| 5mg | 59.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 175.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Prochlorperazine Maleate
CAS:84-02-6
Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; …
Formula:
C28H32ClN3O8S
Purity:
99.99%
Color and Shape:
Off-White Powder
Molecular weight:
606.09
Ref: TM-T0385
| 25mg | 45.00 € | ||
| 50mg | 54.00 € | ||
| 100mg | 71.00 € | ||
| 200mg | 114.00 € | ||
| 500mg | 207.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Alfuzosin hydrochloride
CAS:81403-68-1
Alfuzosin hydrochloride (Alfuzosin HCl) is an α1 adrenergic receptor antagonist. It applies to treat benign …
Formula:
C19H27N5O4·HCl
Purity:
99.61%
Color and Shape:
White To Off-White Solid
Molecular weight:
425.91
Ref: TM-T0091
| 10mg | 44.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 103.00 € | ||
| 100mg | 151.00 € | ||
| 200mg | 216.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
2-(1-Piperazinyl)pyrimidine
CAS:20980-22-7
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
Formula:
C8H12N4
Purity:
98.86%
Color and Shape:
Liquid - Crystal - Lump
Molecular weight:
164.21
Ref: TM-T1696
| 1g | 38.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Indacaterol maleate
CAS:753498-25-8
Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
Formula:
C28H32N2O7
Purity:
99.03% - 99.67%
Color and Shape:
Solid
Molecular weight:
508.56
Ref: TM-T1239
| 10mg | 36.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 100.00 € | ||
| 200mg | 149.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
