
Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65615 products of "Quinazoline and Quinoline Derivatives"
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3-(4-Bromo-pyrazol-1-yl)-propionic acid
CAS:Formula:C6H7BrN2O2Color and Shape:SolidMolecular weight:219.038Ranolazine Dihydrochloride
CAS:<p>Stability Hygroscopic<br>Applications Ranolazine Dihydrochloride is an anti-ischemic agent which modulates myocardial metabolism. Antianginal.<br>References Chaitman, B.R., et al.: J. Am. Coll. Cardial., 43, 1375 (2004); McCormack, J.G., et al.: Gen. Pharmacol., 30, 639 (1998); Schofield, J.A.H., et al.: Expert Opin. Invest. Drugs, 11, 117 (2002)<br></p>Formula:C24H35Cl2N3O4Color and Shape:NeatMolecular weight:500.46Ondansetron-d3
CAS:Controlled Product<p>Applications Ondansetron-d3 is a labeled specific serotonin (5-HT3) receptor antagonist. Antiemetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Kris, M.G., et al.: J. Clin. Oncol., 6, 659 (1988); Faris, P..L., et al.: Lances, 355, 792 (2000)<br></p>Formula:C18H16D3N3OColor and Shape:NeatMolecular weight:296.382,2-Diphenylglycine
CAS:Controlled Product<p>Impurity Phenytoin USP Related Compound A 2,2-Diphenylglycine<br>Stability Hygroscopic<br>Applications 2,2-Diphenylglycine (Phenytoin USP Related Compound A 2,2-Diphenylglycine) is a decomposition product of Phenytoin (D491650), which reduces incidence of grand mal seizures; appears to stabilize excitable membranes perhaps through effects on Na+, K+, and Ca2+ channels.<br>References Shah, V. et al.: J. Pharm. Sci., 75, 1113 (1986); Faucette, S., et al.: J. Pharmacol. Exp. Ther., 320, 72 (2007); Raymond, H. et al.: Teratol., 10, 237 (1974);<br></p>Formula:C14H13NO2Color and Shape:White To Off-WhiteMolecular weight:227.26Ribociclib nitroso impurity 1
Controlled ProductFormula:C23H29N9O2Color and Shape:NeatMolecular weight:419.495Ethyl 3-(2-(chloromethyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanoate
CAS:Purity:98%Molecular weight:400.85998535156254-Defluoro-2-fluoro Haloperidol
CAS:<p>Applications 4-Defluoro-2-fluoro Haloperidol is a positional isomer and impurity of the antipsychotic agent Haloperidol (H103700).<br></p>Formula:C21H23ClFNO2Color and Shape:NeatMolecular weight:375.86Bupivacaine
CAS:<p>Applications Bupivacaine is a sodium channel blocker, local anesthetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Wilson, T.D., et al.: Anal. Profiles Drug Subs., 19, 59 (1990), McClellan, K.J., et al.: Drugs, 56, 355 (1998),<br></p>Formula:C18H28N2OColor and Shape:NeatMolecular weight:288.43Gabapentin-d10
CAS:Controlled Product<p>Applications Gabapentin-d10 is the labelled analogue of Gabapentin (G117250), an amino acid structurally related to γ-Aminobutyric Acid (GABA), designed to cross the blood brain barrier. Used as an anticonvulsant.<br>References Vollmer, K.-O. et al.: Arzneimittel-Forshc., 36, 830 (1986), Saletu, B., et al.: Int. J. Clin. Pharmacol. Ther. Toxicol., 24, 362 (1986)<br></p>Formula:C92H10H7NO2Color and Shape:White To Off-WhiteMolecular weight:181.30N-Ethyl-N-methyl-3-vinylphenyl Carbamate
CAS:Controlled Product<p>Impurity Rivastigmine USP Related Compound F<br>Stability Light Sensitive<br>Applications A related compound of Rivastigmine (R541000), a cholinesterase inhibitor. Rivastigmine USP Related Compound F.<br></p>Formula:C12H15NO2Color and Shape:White SolidMolecular weight:205.252-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl Methanesulfonate
CAS:<p>Applications 2-[2-(2,2,2-Trifluoroethoxy)phenoxy]ethyl Methanesulfonate is an intermediate of Silodosin (S465000) which is an α1a-adrenoceptor antagonist and used in the treatment of benign prostatic hypertophy.<br>References Francesco, C., et al.: Eur. J. Org. Chem., 27, 6011 (2015)<br></p>Formula:C11H13F3O5SColor and Shape:NeatMolecular weight:314.278(1,3-benzodioxol-5-ylmethyl)(2-pyridinylmethyl)amine dihydrobromide
CAS:Purity:95.0%Molecular weight:404.101989746093754-Desmethoxypropoxyl-4-chloro Rabeprazole
CAS:Controlled Product<p>Impurity Rabeprazole EP Impurity H (Lansoprazole EP Impurity F)<br>Applications 4-Desmethoxypropoxyl-4-chloro Rabeprazole (Rabeprazole EP Impurity H (Lansoprazole EP Impurity F)) is a process impurity of Rabeprazole (R070500).<br></p>Formula:C14H12ClN3OSColor and Shape:NeatMolecular weight:305.78Desthiazolylmethyl Ritonavir
CAS:Controlled Product<p>Impurity Ritonavir EP Impurity L<br>Applications Desthiazolylmethyl Ritonavir (Ritonavir EP Impurity L) is an analogue of the selective HIV protease inhibitor Ritonavir (R535000). It is a COVID19-related research product.<br>References Brittain, H., et al.: Pharm. Res., 8, 963 (1991), Sham, H., et al.: J. Med. Chem., 39, 392 (1996), Phadnis, N., et al.: J. Pharm. Sci.,86, 1256 (1997), Bauer, J., et al.: Pharma. Res., 18, 859 (2001),<br></p>Formula:C33H43N5O4SColor and Shape:White To Off-WhiteMolecular weight:605.79Minoxidil Sulfate
CAS:Controlled ProductFormula:C9H15N5O4SColor and Shape:NeatMolecular weight:289.311-[3-(Trifluoromethyl)pyridin-2-yl]piperazine hydrochloride
CAS:Purity:97.0%Molecular weight:267.67999267578125(2R,4R)-2-(2,4-Dichlorophenyl)-2-(1H-imidazol-1-ylmethyl)-1,3-dioxolane-4-methanol 4-(4-Methylbenzenesulfonate)
CAS:Controlled ProductFormula:C21H20Cl2N2O5SColor and Shape:NeatMolecular weight:483.3652'-Hydroxy-3'-methoxyacetophenone
CAS:Controlled Product<p>Applications 2'-Hydroxy-3'-methoxyacetophenone, is an intermediate used for he synthesis of various chemical compounds. It can be used for the synthesis of 4'-Hydroxy-3-methoxyflavones with potent antipicornavirus activity.<br>References Nadine, d. M., et al.: J. Med. Chem., 34, 736 (1991);<br></p>Formula:C9H10O3Color and Shape:NeatMolecular weight:166.18Sodium (S)-6-methoxy-2-(((4-methoxy-3,5-dimethylpyridin-2-yl)methyl)sulfinyl)benzo[d]imidazol-1-ide
CAS:Purity:95.0%Molecular weight:367.39999389648448-[2-(Diphenylmethoxy)-N-methylethylamino]-1,3-dimethylxanthine
CAS:<p>Applications 8-[2-(Diphenylmethoxy)-N-methylethylamino]-1,3-dimethylxanthine is an impurity of Dimenhydrinate (D460520), an antihistamine with antiemetic properties used to prevent nausea and motion sicknes composed of two drugs 8-Chlorotheophylline (C411440) and Diphenhydramine (D486900).<br>References Doege, U., et al.: Pharmazie., 62, 174 (2007); Santoro, R.S., et al.: J. Pharmaceut. Sci., 60, 791 (1971);<br></p>Formula:C23H25N5O3Color and Shape:White To Off-WhiteMolecular weight:419.484-(2-(Pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl)quinolin-7-ol
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:328.3754-(methylthio)-N-(pyridin-3-ylmethyl)benzo[d]thiazol-2-amine
CAS:Purity:95.0%Molecular weight:287.3999938964844rac-erythro Methylphenidate Hydrochloride
CAS:Controlled Product<p>Applications The erythro isomers have been shown to exhibit very little therapeutic effect and contribute mainly to the toxic hypertensive effects of this drug.Controlled substance.<br>References Greenblatt, E.N., et al.: J. Pharmacol. Exp. Ther., 131, 115 (1961), Padmanabhan, G.R., et al.: Anal. Profiles Drug Subs., 10, 473 (1981), Kuczenski, R., et al.: J. Pharmacol. Exp. Ther., 296, 876 (2001), Pelham, W.E., et al.: J. Consult. Clin. Psychol., 61, 506 (1993), Srinivas, N.R., et al.: Pharm. Res., 10, 14 (1993),<br></p>Formula:C14H19NO2·ClHColor and Shape:NeatMolecular weight:269.77Diphenylglycoluril
CAS:Controlled Product<p>Applications Diphenylglycoluril is a bicyclic bis-urea derivative. Studies suggest that it has potential anticonvulsant activity.Diphenylglycoluril is also an impurity found in the synthesis of Phenytoin (D491650).<br>References Khlebnikov, A.I. et al.: Pharm. Chem. J., 36, 240 (2002); Babkibayev, A.A. et al.: Pharm. Chem. J., 8, 15 (1994);<br></p>Formula:C16H14N4O2Color and Shape:NeatMolecular weight:294.314-((4-Bromo-2-fluorophenyl)amino)-6-methoxyquinazolin-7-ol hydrochloride
CAS:Purity:98%Molecular weight:400.6300048828125Trametinib Impurity-I
CAS:Controlled ProductFormula:C26H23FIN5O5Color and Shape:NeatMolecular weight:631.394Cyamemazine-d6
CAS:Controlled Product<p>Applications Labelled Cyamemazine is an anxiolytic antipsychotic, which reduces ethanol withdrawal symptoms.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Robinson, et al.: J. Pharm. Pharmacol., 18, 19 (1966), Miller, L., et al.: J. Pharmacol. Exp. Ther., 246, 170 (1988), Podhorna, J., et al.: Curr. Pharm. Des., 8, 23 (2002), Hameg, A., et al.: Biochem. Pharmacol., 65, 435 (2003),<br></p>Formula:C19H15D6N3SColor and Shape:NeatMolecular weight:329.49Rivaroxaban Diol
CAS:Controlled Product<p>Applications A metabolite of Rivaroxaban (R538000).<br>References Kubitza, D., et al.: Clin. Pharmacol. Ther., 78, 412 (2005), Roehrig, S., et al.: J. Med. Chem., 48, 5900 (2005), Biemond, B., et al.: Thromb. Haemost., 97, 471 (2007), Lang, D., et al.: Drug Metab. Dispos., 37, 1046 (2009),<br></p>Formula:C19H20ClN3O6SColor and Shape:White To Off-WhiteMolecular weight:453.92,6-Dimethylaniline-d6
CAS:Controlled Product<p>Applications Labelled Bupivacaine (B689560) impurity.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Lepage, F., et al.: Eur. J. Med. Chem., 27, 581 (1992), Thummel, K.E., et al.: Drug Metab. Dispos., 21, 350 (1993)<br></p>Formula:C82H6H5NColor and Shape:BrownMolecular weight:127.22Darunavir-d9
CAS:Controlled Product<p>Applications Second generation HIV-1-protease inhibitor; structurally similar to amprenavir. Antiviral. It is a COVID19-related research product.<br>References Koh, Y., et al.: Antimicrob. Agents Chemother., 47, 3123 (2003), Arasteh, K., et al.: AIDS, 19, 943 (2005), Surleraux, D.L.N.G., et al.: J. Med. Chem., 48, 1813 (2005),<br></p>Formula:C272H9H28N3O7SColor and Shape:Off-White To Light BeigeMolecular weight:556.724-[3-(methoxycarbonyl)-5-(thiophen-2-yl)-1H-pyrazol-1-yl]benzoic acid
CAS:Purity:95.0%Molecular weight:328.3399963378906Dihydro-Axitinib
CAS:<p>Applications Dihydro-Axitinib is a useful intermediate for the preparation of axitinib; an antitumor agent.<br>References Chekal, B. P., et al.: Org. Process Res. Dev., 18, 266 (2014)<br></p>Formula:C22H20N4OSColor and Shape:White To Off-WhiteMolecular weight:388.49rac N-Propyl-2-cyanimidopyrrolidine-5-acetic Acid
CAS:Controlled Product<p>Applications rac N-Propyl-2-cyanimidopyrrolidine-5-acetic Acid is a potent peptidic renin inhibitor. Pramipexole Related Compound<br></p>Formula:C10H15N3O2Color and Shape:NeatMolecular weight:209.24(R)-Lisinopril Sodium Salt
CAS:<p>Applications R,S,S-Isomer of Lisinopril (L468985).<br>References Goa, K.L., et al.: Drugs, 52, 564 (1996), Chaturvedi, N., et al.: Lancet, 351, 28 (1998)<br></p>Formula:C21H31N3NaO5Color and Shape:NeatMolecular weight:428.48Lansoprazole-d4
CAS:Controlled ProductFormula:C162H4H10F3N3O2SColor and Shape:NeatMolecular weight:373.39Dipyridamole Tri(diethanolamine)
CAS:Controlled Product<p>Impurity Dipyridamole EP Impurity B<br>Applications Dipyridamole Tri(diethanolamine) (Dipyridamole EP Impurity B) Dipyridamole (D492625) impurity.<br>References Gerlach, E., et al.: Arzneim.-Forsch., 15, 558 (1965),<br></p>Formula:C23H40N8O6Color and Shape:NeatMolecular weight:524.61Linagliptin
CAS:<p>Applications Linagliptin is a novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.<br>References Prabavathy, N. et al.: Int. J. Pharm. Bio. Sci., 2, 438 (2011); Deacon, C.F.: Diab. Obes. Metab., 13, 7 (2011);<br></p>Formula:C25H28N8O2Color and Shape:White To OrangeMolecular weight:472.541-Methoxy-Empagliflozin Tetraacetoxy
CAS:Formula:C32H37ClO12Color and Shape:NeatMolecular weight:649.082(R)-Tamsulosin-d4 Hydrochloride
CAS:Controlled Product<p>Applications (R)-Tamsulosin-d4 Hydrochloride is the labeled analogue of (R)-Tamsulosin Hydrochloride (T006350), a specific α1-adrenoceptor antagonist. It is used in the treatment of benign prostatic hypertrophy.<br>References Kawabe, K., et al.: J. Urol., 144, 908 (1990); Abrams, P., et al.: Br. J. Urol., 76, 325 (1995); Michel, M.C., Expert Opin. Pharmacother., 5, 151 (2004)<br></p>Formula:C20H25D4ClN2O5SColor and Shape:NeatMolecular weight:449.05-Hydroxy Omeprazole Sodium Salt
CAS:<p>Stability Hygroscopic<br>Applications The main metabolite of Omeprazole.<br>References Renberg, L., et al.: Drug Metab. Dispos., 17, 69 (1989), Calabresi, L., et al.: Pharmacol. Res., 49, 493 (2004), Yin, O., et al.: J. Clin. Pharmacol., 44, 582 (2004),<br></p>Formula:C17H18N3NaO4SColor and Shape:White To Light YellowMolecular weight:383.40Teneligliptin Sulfoxide (Mixture of Diastereomers)
Controlled Product<p>Applications Teneligliptin Sulfoxide, is an impurity of Teneligliptin (T018300) which is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. Tenegliptin is eliminated from the via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Formula:C22H30N6O2SColor and Shape:NeatMolecular weight:442.58N1,N3-Bis[2-(3,4-dimethoxyphenyl)ethyl]-N1,N3-dimethyl-1,3-propanediamine Dihydrochloride
CAS:Controlled Product<p>Impurity Verapamil EP Impurity A DIHCL<br>Stability Hygroscopic<br>Applications N1,N3-Bis[2-(3,4-dimethoxyphenyl)ethyl]-N1,N3-dimethyl-1,3-propanediamine Dihydrochloride (Verapamil EP Impurity A DIHCL) is an impurity of Verapamil (V125000), a calcium channel blocker. Antihypertensive; antianginal; antiarrhythmic (class IV).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Atlas, D, and Adler, M.: Proc. Natl. Acad. Sci. USA, 78, 1237 (1981), Janis, R., et al.: Adv. Drug. Res., 16, 309 (1987)<br></p>Formula:C25H38N2O4·2ClHColor and Shape:NeatMolecular weight:503.514-Amino-2,6-dichloro-α-(4-chlorophenyl)benzeneacetonitrile
CAS:Controlled Product<p>Applications This compound is used in the synthesis of Diclazuril (D436200) and diclazuril derivatives.<br></p>Formula:C14H9Cl3N2Color and Shape:NeatMolecular weight:311.59Methyl 4-(((4-(pyridin-3-yl)pyrimidin-2-yl)amino)methyl)benzoate
CAS:Purity:95+%Molecular weight:320.35198974609375Metaflumizone
CAS:<p>Applications Metaflumizone is a semicarbazone insecticide that works by blocking sodium channel in target insects resulting in paralyzation associated with blocking nerve activity. Metaflumizone is useful as a heartworm control treatment.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Zhang, Zhe,, et al.: J. Integrat. Agri. 11, 1145 (2012); Kuhn, D., et al.: Modern. Crop. Protect. Compound., 3, 1273 (2012);<br></p>Formula:C24H16F6N4O2Color and Shape:WhiteMolecular weight:506.402-Ethyl-2-methylsuccinic Acid
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications 2-Ethyl-2-methylsuccinic Acid is an inhibitor of plasmid-borne IMP-1 metallo-β-lactamase.<br>References Toney, J., et. al.: J. Biol. Chem., 276, 31913 (2001)<br></p>Formula:C7H12O4Color and Shape:NeatMolecular weight:160.1682-(2-methoxyphenyl)-8-methylquinoline-4-carboxylic acid
CAS:Purity:95.0%Molecular weight:293.32199096679694-bromo-2-(5-pyridin-3-yl-4,5-dihydro-1H-pyrazol-3-yl)phenol
CAS:Purity:95.0%Molecular weight:318.17401123046875Sulindac Sulfide
CAS:<p>Stability Hygroscopic<br>Applications An active metabolite of Sulindac. Inhibits cyclooxygenase, but induces apoptosis by a cyclooxygenase-independent mechanism. Inhibition of Ras activation of Ref-1. Impairs nucleotide exchange on Ras by CDC25 and accelerates Ras hydrolysis of GTP by p120GAP.<br>References Hermann, C., et al.: Oncogene, 17, 1769 (1998), Lim, T.J., et al.: Biochem. Pharmacol., 58, 1097 (1999), Zhang, Z. and DuBois, R.N.: Gastroenterology, 118, 1012 (2000),<br></p>Formula:C20H17FO2SColor and Shape:Yellow-OrangeMolecular weight:340.411-(4-Fluorophenyl)-4-(4-(pyridin-2-yl)piperazin-1-yl)butan-1-one
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:327.403015136718752-Hydroxy-6-methylpyridine-3,4-dicarboxylic acid
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:197.145996093753-Picoline
CAS:Controlled Product<p>Applications A useful precursor to agrochemicals and antidotes for organophosphate poisoning.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Qiao, L., et al.: Bioorg. Med. Chem. Lett., 19, 6122 (2009), Giri, A., et al.: Food Chem., 120, 621 (2010), Farrer, N., et al.: Chem. Res. Toxicol., 23, 413 (2010),<br></p>Formula:C6H7NColor and Shape:ColourlessMolecular weight:93.13Quinoxyfen
CAS:Controlled Product<p>Applications Agricultural fungicide.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Corrales, M., et al.: Food Chem. Toxicol., 48, 3471 (2010), Lagunas-Allue, L., et al.: Anal. Bioanal. Chem., 398, 1509 (2010), Wong, J., et al.: J. Agric. Food Chem., 58, 5897 (2010),<br></p>Formula:C15H8Cl2FNOColor and Shape:Off-WhiteMolecular weight:308.13N-Boc-L-cis-4,5-Methanoprolineamide
CAS:Controlled Product<p>Applications N-Boc-L-cis-4,5-Methanoprolineamide is an intermediate used to prepare methanoprolinenitrile-contg. dipeptide mimetics as DPP-IV inhibitors and as antidiabetic agents.<br>References Magnin, D., et al.: J. Med. Chem., 47, 2587 (2004)<br></p>Formula:C11H18N2O3Color and Shape:NeatMolecular weight:226.272Ranitidine-d6 Hydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A histamine H2-receptor antagonist which inhibits gastric acid secretion. Antiulcerative.<br>References Bradshaw, J., et al.: Brit. J. Pharmacol., 66, 464 (1979), Berstad, A., et al.: Scand. J. Gastroenterol, 15, 637 (1980), Hohnjec, M., et al.: Anal. Profiles Drug Subs., 15, 533 (1986),<br></p>Formula:C132H6H16N4O3S·ClHPurity:>90%Color and Shape:NeatMolecular weight:356.903-(4-Fluorophenyl)-1-phenyl-1H-pyrazole-4-carboxaldehyde
CAS:Purity:95.0%Molecular weight:266.27499389648442-Amino-4-(4-cyclohexyl-phenyl)-thiophene-3-carboxylic acid methyl ester
CAS:Formula:C18H21NO2SPurity:97%Color and Shape:SolidMolecular weight:315.431-N-Boc-4-(4-Pyridylmethylamino)piperidine
CAS:Formula:C16H25N3O2Purity:98.0%Color and Shape:Solid, No data available.Molecular weight:291.39510-Oxo Mirtazapine (Mirtazapine Impurity F)
CAS:Controlled Product<p>Impurity Mirtazapine EP Impurity F<br>Applications 10-Oxo Mirtazapine (Mirtazapine Impurity F) is an impurity of Mirtazapine. Mirtazapine EP Impurity F.<br>References De Boer, T., et al.: Neuropharmacol., 27, 399 (1988), Vindevogel, J., et al.: Anal. Chem., 63, 1530 (1991), Wynia, G., et al.: J. Chromatogr., 773, 339 (1997),<br></p>Formula:C17H17N3OColor and Shape:NeatMolecular weight:279.34N-Benzyl Hydroxymedetomidine
CAS:Controlled Product<p>Applications N-Benzyl Hydroxymedetomidine is an impurity of Medetomidine (M203250, HCl); an α2-adrenergic agonist, sedative, and analgesic.<br>References Scheinin, M., et al.: Br. J. Clin. Pharmacol., 24, 443 (1987); Stenberg, D., et al.: J. Vet. Pharmacol. Ther., 10, 319 (1987); Virtanen, R., et al.: Eur. J. Pharmacol., 150, 9 (1988); Cullen, L.K., et al.: Br. Vet. J., 152, 519 (1996)<br></p>Formula:C20H22N2OColor and Shape:NeatMolecular weight:306.4N-(2,6-Dimethylphenyl)-1-piperazineacetamide
CAS:Formula:C14H21N3OColor and Shape:NeatMolecular weight:247.34Bupivacaine Hydrochloride Monohydrate
CAS:<p>Applications Sodium channel blocker, local anesthetic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Wilson, T.D., et al.: Anal. Profiles Drug Subs., 19, 59 (1990), McClellan, K.J., et al.: Drugs, 56, 355 (1998),<br></p>Formula:C18H28N2O·ClH·H2OColor and Shape:WhiteMolecular weight:324.89Levetiracetam-d6
CAS:Controlled Product<p>Applications Levetiracetam-d6 is a labelled (S)-enantiomer of the ethyl analog of Piracetam (P500800), an anticonvulsant.<br>References Gower, A.J., et al.: Eur. J. Pharmacol., 222, 193 (1992), Kasteleijn-Noist Trenite, D.G.A., et al.: Epilepsy Res., 25, 225 (1996), Patsalos, P.N., et al.: Pharmacol. Ther., 85, 77 (2000),<br></p>Formula:C8D6H8N2O2Color and Shape:NeatMolecular weight:176.25Benzydamine-d6 N-Oxide
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A labelled metabolite of Benzydamine (B209950).<br>References Beaty, N., et al.: J. Biol. Chem., 255, 3817 (1980), Tugnait, M., et al.: Drug Metab. Dispos., 25, 524 (1997), Ubeaud, G., et al.: Eur. J. Pharm. Sci., 8, 255 (1999),<br></p>Formula:C19H17D6N3O2Color and Shape:NeatMolecular weight:331.44Ofloxacin N-Oxide Acetic Acid Salt (Mixture of Diastereomers)
CAS:Controlled Product<p>Applications A metabolite of Ofloxacin.<br>References Uematsu, T., et al.: Eur. J. Clin. Pharmacol., 40, 581 (1991), Uematsu, T., et al.: Ther. Drug Monit., 17, 101 (1995), Ballesteros, O., et al.: J. Pharm. Biomed. Anal., 30, 1103 (2002), Kitade, T., et al.: Chem. Pharm. Bull., 51, 53 (2003),<br></p>Formula:C18H20FN3O5·ClHColor and Shape:NeatMolecular weight:437.419N”Nitrosoketamine
CAS:Controlled ProductFormula:C13H15ClN2O2Color and Shape:White To Light YellowMolecular weight:266.7232-(2,6-Dimethylbenzoyl)-5-(1,3-dioxolan-2-yl)thiophene
CAS:Purity:97.0%Molecular weight:288.3599853515625Prochlorperazine Sulfoxide-d3
CAS:Controlled Product<p>Applications A labelled metabolite of Prochlorperazine.<br>References Finn, A., et al.: J. Clin. Pharmacol., 45, 1383 (2005),<br></p>Formula:C202H3H21ClN3OSColor and Shape:Off WhiteMolecular weight:392.96α-Hydroxy Montelukast
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A hydroxylated impurity of the selective leukotriene D4-receptor antagonist, Montelukast (M568000).<br></p>Formula:C35H36ClNO4SColor and Shape:NeatMolecular weight:602.18Pentoxifylline-d6
CAS:Controlled Product<p>Applications A labelled metabolite of Pentifylline. Methylxanthine derivative that improves blood flow by decreasing blood viscosity. Phosphodiesterase inhibitor. Inhibits the synthesis of tumor necrosis factor α (TNF-α).<br>References Ward, A., et al.: Drugs, 34, 50 (1987), Samlaska, C.P., et al.: J. Am. Acad. Dermatol., 30, 603 (1994), Poulakis, et al.: Respir. Med., 93, 52 (1999), Reuter, et al.: Am J. Physiol., 277, 854 (1999),<br></p>Formula:C132H6H12N4O3Color and Shape:NeatMolecular weight:284.342-(CHLOROMETHYL)-4-(2,2,3,3,4,4,4-HEPTAFLUOROBUTOXY)PYRIDINE
CAS:Purity:95.0%Molecular weight:325.60998535156254-methoxy-7-methyl-N-(pyridin-3-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Purity:95.0%Molecular weight:285.36999511718751-des(piperidin-3R-amino)-1-chloro-Alogliptin
CAS:Controlled Product<p>Impurity Alogliptin 6-Chloro Impurity<br>Applications Alogliptin (A575425) intermediate.<br></p>Formula:C13H10ClN3O2Color and Shape:NeatMolecular weight:275.692,4-Difluoro-α-(1H-1,2,4-triazolyl)acetophenone
CAS:Controlled Product<p>Impurity Voriconazole EP Impurity A; Voriconazole USP Related Compound C<br>Applications 2,4-Difluoro-α-(1H-1,2,4-triazolyl)acetophenone (Voriconazole EP Impurity A; Voriconazole USP Related Compound C) is an antifungal activity, particularly toward Candida albicans and Candida parapsilosis<br>References Upadhayaya, R., et al.: Eur. J. Med. Chem., 39, 579 (2004), Sheng, C., et al.: J. Med. Chem., 49, 2512 (2006),<br></p>Formula:C10H7F2N3OColor and Shape:BeigeMolecular weight:223.18Adrafinil
CAS:Controlled ProductFormula:C15H15NO3SColor and Shape:Off-White Light Orange ColourMolecular weight:289.35Primidone
CAS:<p>Applications Primidone is an Anticonvulsant.<br>References Bogue, C., et al.: Br. J. Pharmacol., 8, 230 (1953), Daley, R.D., Anal. Profiles Drug Subs., 2, 409 (1973),<br></p>Formula:C12H14N2O2Color and Shape:White To Off-WhiteMolecular weight:218.25N,N'-Methylene Ambroxol Hydrochloride
CAS:Controlled Product<p>Impurity Ambroxol EP Impurity B Hydrochloride<br>Stability Hygroscopic<br>Applications Ambroxol Cyclic Impurity is a metabolite as well as an impurity of the bronchosecretolytic drug, Ambroxol (A575900).<br>References Hammer, R. et al.: Arzneim.-Forsch., 28, 899 (1978); Nieder, M. et al.: HRC & CC, 9, 561 (1986); Huq, F. et al.: J. Pharmacol. Toxicol., 3, 147 (2008);<br></p>Formula:C14H18Br2N2O·ClHColor and Shape:White To Off-WhiteMolecular weight:426.574-(3-Aminophenyl)-3-morpholinone
CAS:Controlled Product<p>Applications 4-(3-Aminophenyl)-3-morpholinone is an intermediate during the preparation of imidazothiazoles as protein kinase inhibitors for treating cancers.<br>References Bamaung, N., et al.: PCT Int. Appl. (2009), WO 2009070516 A1 20090604.<br></p>Formula:C10H12N2O2Color and Shape:NeatMolecular weight:192.2141-[3-(4-tert-Butylbenzoyl)propyl]-4-hydroxypiperidine
CAS:Controlled ProductFormula:C19H29NO2Color and Shape:WhiteMolecular weight:303.44Edoxaban-d6
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Edoxaban-d6 is the isotope labelled analog of Edoxaban (E555520); an anticoagulant drug which acts as a direct factor Xa inhibitor.<br>References Ruff, C., et al.: Am. Heart J., 160, 635 (2010); Ogata, K., et al.: J. Clin. Pharm., 50, 73 (2010)<br></p>Formula:C24H24D6ClN7O4SColor and Shape:Light Beige To Light BrownMolecular weight:554.09


