Salts and Derivatives of Active Pharmaceutical Ingredients (API)
The salts of Active Pharmaceutical Ingredients (APIs) are compounds formed by the reaction of an acid with a base, resulting in an ionic equilibrium. These salts often improve the solubility and stability of APIs, facilitating their absorption in the body. API derivatives are chemical variants of an active ingredient that may have enhanced or modified properties to optimise therapeutic efficacy. API salts are used in the formulation of oral, injectable, and topical medications. Additionally, API derivatives can improve the pharmacokinetics of drugs, such as enabling controlled release of active substances.
At CymitQuimica, we provide API salts and derivatives with the necessary purity and quality for research and pharmaceutical formulation development.
Found 79171 products of "Salts and Derivatives of Active Pharmaceutical Ingredients (API)"
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Selexipag
CAS:Controlled Product<p>Applications Selexipag is an orally available, highly selective, long-acting prostacyclin (IP) receptor agonist prodrug. It is a potential drug for the treatment of various vascular disorders such as pulmonary arterial hypertension and arteriosclerosis obliterans.<br>References Kuwano, K., et al.: J. Pharm. Exp. Ther., 322, 1181 (2007);<br></p>Formula:C26H32N4O4SColor and Shape:Light YellowMolecular weight:496.62Bosentan-d4
CAS:Controlled Product<p>Applications Labelled Bosentan (B675900). A mixed endothelin receptor antagonist. Used as a vasodilator. Antihypertensive.<br>References Clozel, M., et al.: J. Pharmacol. Exp. Ther., 270, 228 (1994), Gutsch, G., et al.: Cardiovasc. Drugs Ther., 10, 717 (1996), Weber, C., et al.: Clin Pharmacol. Ther., 60, 124 (1996), Krum, H., et al.: N. Engl. J. Med., 338, 784 (1998)<br></p>Formula:C27H25D4N5O6SColor and Shape:NeatMolecular weight:555.64Ethyl 2-(3-Formyl-4-hydroxyphenyl)-4-methylthiazole-5-carboxylate
CAS:Formula:C14H13NO4SColor and Shape:NeatMolecular weight:291.322,5-Ethyl Acetate Febuxostat
CAS:Controlled Product<p>Applications Febuxostat (F229000) is the parent compound for 2,5-Ethyl Acetate Febuxostat. Used for treatment of hyperuricemia and chronic gout. 40-120 mg/day febuxostat was proven effective in lowering serum urate levels when administered to manage hyperuricemia in patients with gout.<br>References Osada, Y., et al.: Eur. J. Pharmacol., 241, 183 (1993), Okamoto, K., et al.: J. Biol. Chem., 278, 1848 (2003), Mayer, M.D., et al.: Am. J. Therap., 12, 22 (2005), Tomlinson, B., et al.: Curr. Opin. Invest. Drugs, 6, 1168 (2005),<br></p>Formula:C20H25NO5SColor and Shape:NeatMolecular weight:391.48Diclofenac Carboxylic Acid (Diclofenac Metabolite)
CAS:Controlled Product<p>Applications Metabolite of Diclofenac.<br>References Duffy, J.C., et al.: J. Pharm. Pharmacol., 48, 883 (1996), Oza, V., et al.: J. Med. Chem., 45, 321 (2002), Bajaj, S., et al.: Bioorg. Med. Chem., 12, 3695 (2004), Teffera, Y., et al.: Drug Metabolism Lett., 2, 35 (2008),<br></p>Formula:C13H9Cl2NO2Color and Shape:Off-WhiteMolecular weight:282.12Cyclosporin D
CAS:Controlled Product<p>Applications A group of nonpolar cyclic oligopeptides with immunosupppressant activity.<br>References van Wartburg, A., et al.: Prog. Med. Chem., 25, 1 (1988), Jorgensen, K.A., et al.: Scand. J. Imunol., 57, 93 (2003), Vollenbroeker, et al.: Transplant. Proc., 37, 1741 (2005),<br></p>Formula:C63H113N11O12Color and Shape:Off-WhiteMolecular weight:1216.64methyl (Z)-1-acetyl-3-(methoxy(phenyl)methylene)-2-oxoindoline-6-carboxylate
CAS:Formula:C20H17NO5Molecular weight:351.36Lanicemine dihydrochloride
CAS:<p>Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be used to study neurological diseases.</p>Formula:C13H16Cl2N2Purity:98.37%Color and Shape:SolidMolecular weight:271.193”-O-Demethyl Ivermectin
CAS:<p>Applications 3”-O-Demethyl Ivermectin is an impurity of Ivermectin (I940800), an antiparasitic drug that is active against a wide variety of nematode and arthropod parasites and is used to treat scabies and lice in humans. An invitro inhibitor of SARS-CoV-2/ Covid-19.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Campbell, W., et al.: Science, 221, 823 (1983); Glaziou, P., et al.: Trop. Med. Parasitol., 45, 253 (1994); Meinking, T., et al.: New Engl. J. Med., 333, 26 (1995); Caly, L., et al.: Antivir. Res., 178<br></p>Formula:C47H72O14Color and Shape:NeatMolecular weight:861.07(1S)-4,5-Dimethoxy-1-[(methylamino)methyl]benzocyclobutane Hydrochloride
CAS:Controlled ProductFormula:C12H17NO2·ClHColor and Shape:NeatMolecular weight:243.735-Chloro-3-(NMethylsulfamoyl)Thiophene2-Carboxylic Acid
CAS:Formula:C7H8ClNO3S2Molecular weight:253.7
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