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Apoptosis

Apoptosis

Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.

Subcategorías de "Apoptosis"

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Se han encontrado 5622 productos de "Apoptosis"

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  • Levobupivacaine

    CAS:
    <p>Levobupivacaine is an amino-amide local anaesthetic drug belonging to the family of n-alkylsubstituted pipecoloxylidide.</p>
    Fórmula:C18H28N2O
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:288.43
  • AZD-8055

    CAS:
    <p>AZD8055 is an ATP-competitive mTOR inhibitor (IC50: 0.8 nM in MDA-MB-468 cells). It is ~1,000-fold selective for mTOR over all PI3K isoforms.</p>
    Fórmula:C25H31N5O4
    Pureza:98% - 99.69%
    Forma y color:Solid
    Peso molecular:465.54
  • σ1 Receptor antagonist-1

    CAS:
    <p>σ1 Receptor antagonist-1 is a selective sigma 1 receptor antagonist.</p>
    Fórmula:C21H23NOS
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:337.48
  • GSK3326595

    CAS:
    <p>GSK3326595 (EPZ015938) is an inhibitor of protein arginine methyltransferase 5 (PRMT5)(IC50:6.2 nM.).</p>
    Fórmula:C24H32N6O3
    Pureza:97.7% - 99.63%
    Forma y color:Solid
    Peso molecular:452.55
  • Birinapant

    CAS:
    <p>Birinapant (TL32711) is a synthetic small molecule that is both a peptidomimetic of second mitochondrial-derived activator of caspases (SMAC) and inhibitor of</p>
    Fórmula:C42H56F2N8O6
    Pureza:97.08% - ≥95%
    Forma y color:Solid
    Peso molecular:806.94
  • MPP dihydrochloride (289726-02-9 Free base)

    CAS:
    <p>MPP dihydrochloride is a highly selective antagonist of estrogen receptor alpha (ERα).</p>
    Fórmula:C29H33Cl2N3O3
    Forma y color:Solid
    Peso molecular:542.5
  • CVT-11127

    CAS:
    <p>CVT-11127 is an StearoylCoA Desaturase-1 (SCD1) inhibitor.</p>
    Fórmula:C25H23Cl2N5O3
    Pureza:98.32%
    Forma y color:Solid
    Peso molecular:512.39
  • Siramesine hydrochloride

    CAS:
    <p>Siramesine hydrochloride (Lu 28-179 hydrochloride) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibit</p>
    Fórmula:C30H32ClFN2O
    Pureza:99.72% - >99.99%
    Forma y color:Solid
    Peso molecular:491.04
  • Piclidenoson

    CAS:
    <p>Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.</p>
    Fórmula:C18H19IN6O4
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:510.29
  • Glycochenodeoxycholic acid sodium salt

    CAS:
    <p>GCDCA, a bile acid-glycine salt, is a secondary bile acid from colonic microbes.</p>
    Fórmula:C26H42NNaO5
    Pureza:95.48% - 99.82%
    Forma y color:Solid
    Peso molecular:471.61
  • Oxychlororaphine

    CAS:
    <p>Oxychlororaphine (phenazine-1-carboxamide) inhibits strongly the growth of Streptomyces sp. 441.</p>
    Fórmula:C13H9N3O
    Pureza:98.3%
    Forma y color:Green-Yellow Solid
    Peso molecular:223.23
  • Pitavastatin sodium

    CAS:
    <p>Pitavastatin sodium inhibits HMG-CoA reductase, enhances LDL-C receptors, and has various protective effects.</p>
    Fórmula:C25H23FNNaO4
    Forma y color:Solid
    Peso molecular:443.45
  • L67

    CAS:
    <p>L67 (DNA Ligase Inhibitor) is a competitive human DNA ligase inhibitor, inhibits DNA ligases I and III (IC50: 10 μM).</p>
    Fórmula:C16H14Br2N4O4
    Pureza:98.34% - 99.56%
    Forma y color:Solid
    Peso molecular:486.11
  • ALSTERPAULLONE

    CAS:
    Alsterpaullone is a Cyclin-Dependent Kinase Inhibitor, Mediated Toxicity in HeLa Cells Through Apoptosis-Inducing Effec
    Fórmula:C16H11N3O3
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:293.28
  • ENMD-1068 hydrochloride

    CAS:
    <p>ENMD-1068 hydrochloride: selective PAR2 antagonist, counters liver fibrosis, hinders endometrial cell growth, and induces apoptosis in studies.</p>
    Fórmula:C15H30ClN3O2
    Forma y color:Solid
    Peso molecular:319.87
  • Cannabigerol

    CAS:
    Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also
    Fórmula:C21H32O2
    Pureza:99.59% - 99.92%
    Forma y color:Solid
    Peso molecular:316.48
  • Talampanel

    CAS:
    <p>Talampanel (LY-300164), an oral selective AMPA receptor antagonist, exhibits anti-seizure and neuroprotective properties.</p>
    Fórmula:C19H19N3O3
    Pureza:98.3%
    Forma y color:Solid
    Peso molecular:337.37
  • TT-232 TFA(147159-51-1 free base)

    CAS:
    <p>TT2-32 TFA induces a biphasic activation of phosphotyrosine phosphatase activity in human colon tumor cell line, SW620</p>
    Fórmula:C47H59F3N10O11S2
    Pureza:99.27% - 99.8%
    Forma y color:Solid
    Peso molecular:1061.16
  • (Z)-Mirin

    CAS:
    <p>(Z)-Mirin is a potent Mre11–Rad50–Nbs1 (MRN) complex inhibitor, and inhibits Mre11-associated exonuclease activity.</p>
    Fórmula:C10H8N2O2S
    Pureza:99.67% - 99.76%
    Forma y color:Solid
    Peso molecular:220.25
  • Cladribine

    CAS:
    <p>Cladribine (2CdA), an adenosine deaminase inhibitor, is utilized in the treatment of lymphoproliferative diseases.</p>
    Fórmula:C10H12ClN5O3
    Pureza:99.58% - >99.99%
    Forma y color:White Crystalline Solid
    Peso molecular:285.69
  • TCS PrP Inhibitor 13

    CAS:
    <p>TCS PrP Inhibitor 13 (5-(4-Nitrophenyl)-2-Phenyl-4H-Pyrazol-3-One) is an antiprion agent inhibiting protease-resistant prion protein (PrP-res) accumulation.</p>
    Fórmula:C15H11N3O3
    Pureza:99.7%
    Forma y color:Solid
    Peso molecular:281.27
  • Trametinib (DMSO solvate)

    CAS:
    <p>Trametinib (DMSO solvate) (GSK-1120212 (DMSO solvate)) is a Highly Potent and Selective MEK Inhibitor that specifically inhibits MEK1/2(IC50 :2 nM)</p>
    Fórmula:C28H29FIN5O5S
    Pureza:98.82% - 99.92%
    Forma y color:Solid
    Peso molecular:693.53
  • CRT0066101 dihydrochloride

    CAS:
    <p>CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).</p>
    Fórmula:C18H22N6O·2HCl
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:411.33
  • Piperazine Erastin

    CAS:
    <p>Piperazine erastin is an analog of erastin. It causes an iron-dependent form of non-apoptotic cell death termed ferroptosis.</p>
    Fórmula:C35H41ClN6O4
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:645.19
  • Thalidomide-O-C6-NH2 hydrochloride

    CAS:
    <p>Thalidomide-O-C6-NH2 hydrochloride (4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride) is a synthesized E3 ligase ligand-</p>
    Fórmula:C19H24ClN3O5
    Pureza:97.45%
    Forma y color:Solid
    Peso molecular:409.86
  • Pyraclostrobin

    CAS:
    Pyraclostrobin is one of the most heavily used fungicides that inhibits mitochondrial complex III of fungal and mammalian cells.
    Fórmula:C19H18ClN3O4
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:387.82
  • Azathioprine Sodium

    CAS:
    <p>Azathioprine Sodium is a pro-drug converted to 6-MP, inhibiting DNA/RNA synthesis, curbing cell proliferation, especially in lymphocytes.</p>
    Fórmula:C9H6N7NaO2S
    Forma y color:Solid
    Peso molecular:299.24
  • Grape Seed Extract

    CAS:
    <p>Grape Seed Extract (Grape Seed P.E.) is exudate from seeds of the grape plant Vitis vinifera, composed of oils and secondary plant metabolites.</p>
    Fórmula:C32H30O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:590.581
  • Imipramine hydrochloride

    CAS:
    <p>Imipramine HCl: 1st-gen tricyclic antidepressant, inhibits serotonin and norepinephrine uptake, blocks aSMase, reduces MV/exosome secretion.</p>
    Fórmula:C19H25ClN2
    Pureza:99.65% - 99.98%
    Forma y color:White To Off-White /Hydrochloride/ Un 1230 3/Pg 2
    Peso molecular:316.87
  • Thalidomide-O-amido-C4-NH2 TFA

    CAS:
    <p>Thalidomide-O-amido-C4-NH2 TFA (E3 ligase Ligand-Linker Conjugates 19 TFA) is a synthesized E3 ligase ligand-linker conjugate.</p>
    Fórmula:C21H23F3N4O8
    Pureza:95%
    Forma y color:Solid
    Peso molecular:516.42
  • CBL0137 hydrochloride

    CAS:
    <p>CBL0137 hydrochloride (Curaxin-137 hydrochloride) is an inhibitor of the histone chaperone FACT, which also activates p53 and inhibits NF-κB.Cost-effective and quality-assured.</p>
    Fórmula:C21H25ClN2O2
    Pureza:99.35% - 99.86%
    Forma y color:Solid
    Peso molecular:372.88
  • Morroniside

    CAS:
    <p>Morroniside regulates liver inflammation, lipid metabolism, protects against diabetic kidney damage, and guards the brain from ischemic injury.</p>
    Fórmula:C17H26O11
    Pureza:99.70% - 99.84%
    Forma y color:Solid
    Peso molecular:406.38
  • ZYN57939

    CAS:
    <p>ZYN57939 (MTR-106), an RNA polymerase I inhibitor, treats related diseases with a 0.855 μM IC50 against HT-29 cells.</p>
    Fórmula:C28H27N7O2S
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:525.62
  • Calcium dobesilate

    CAS:
    Calcium dobesilate(CaD) has angioprotective properties and protects endothelial cells partly by ameliorating HG induced inflammation.
    Fórmula:C6H5O5SCa0
    Pureza:98.39%
    Forma y color:White Or Almost Powder
    Peso molecular:229.2
  • Bicyclol

    CAS:
    <p>Bicyclol is an oral anti-hepatitis drug, decreasing ALT/AST levels by 50% and inhibiting HBV/HCV, boosting efficacy with interferon/lamivudine/adefovir.</p>
    Fórmula:C19H18O9
    Pureza:99.64% - 99.85%
    Forma y color:Solid
    Peso molecular:390.34
  • Hederacolchiside A1

    CAS:
    <p>Hederacolchiside A1 exhibits anti-leishmanial and anticancer activities by disrupting cell membranes and inducing apoptosis via the PI3K/Akt/mTOR pathway.</p>
    Fórmula:C47H76O16
    Pureza:98.76% - 99.92%
    Forma y color:Solid
    Peso molecular:897.1
  • Almorexant

    CAS:
    <p>Almorexant (ACT 078573), a strong dual orexin receptor antagonist, has Ki of 1.3 nM for OX1 and 0.17 nM for OX2.</p>
    Fórmula:C29H31F3N2O3
    Pureza:97.75% - 98.02%
    Forma y color:Solid
    Peso molecular:512.56
  • Lenaldekar

    CAS:
    <p>Lenaldekar (LDK) inhibits T-cell expansion and autoimmune encephalomyelitis.</p>
    Fórmula:C18H14N4
    Pureza:97.73%
    Forma y color:Solid
    Peso molecular:286.33
  • NSC-87877 disodium

    CAS:
    <p>NSC-87877 disodium (NSC87877) is a cell-permeable inhibitor of both SHP-1 and SHP-2. NSC-87877 also inhibits EGF-induced Erk1/2 activation in HEK293 cells.</p>
    Fórmula:C19H13N3O7S2·2Na
    Pureza:97.89%
    Forma y color:Solid
    Peso molecular:503.42
  • Phenoxyethanol

    CAS:
    <p>Phenoxyethanol (NSC-1864) is germicidal. It often used together with quaternary ammonium compounds.</p>
    Fórmula:C8H10O2
    Pureza:99.47%
    Forma y color:Clear To Practically Clear Colourless Liquid
    Peso molecular:138.16
  • Cytochalasin H

    CAS:
    <p>Cytochalasin H ((16-Benzyl-5,12-dihydroxy-5,7,14-trimethyl-13-methylidene-18-oxo-17-azatricyclo[9.7.0.01,15]octadeca-3,9-dien-2-yl) acetate) is a potent</p>
    Fórmula:C30H39NO5
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:493.63
  • Sertaconazole nitrate

    CAS:
    <p>Sertaconazole nitrate, a broad-spectrum topical antifungal, treats skin and mucosal infections.</p>
    Fórmula:C20H15Cl3N2OS·HNO3
    Pureza:98.66% - 99.65%
    Forma y color:Solid
    Peso molecular:500.78
  • Bendamustine

    CAS:
    <p>Bendamustine (SDX105) for the treatment of Non-Hodgkin Lymphomas and Chronic Lymphocytic Leukemia</p>
    Fórmula:C16H21Cl2N3O2
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:358.26
  • SKLB4771

    CAS:
    <p>SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.</p>
    Fórmula:C25H27N7O3S2
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:537.66
  • 4-Hydroxybenzyl alcohol

    CAS:
    4-Hydroxybenzyl alcohol aids brain injury recovery, boosts Nrf2/Prdx6/PDI, and hinders angiogenesis, showing promise in cancer therapy.
    Fórmula:C7H8O2
    Pureza:97.65% - 98.25%
    Forma y color:Solid
    Peso molecular:124.14
  • Zorifertinib

    CAS:
    Zorifertinib (AZD3759) is an orally active, effective and central nervous system-penetrant EGFR inhibitor.
    Fórmula:C22H23ClFN5O3
    Pureza:98.20% - 99.36%
    Forma y color:White To Off-White Solid
    Peso molecular:459.9
  • 2,4,6-Triiodophenol

    CAS:
    <p>2,4,6-Triiodophenol: iodinated byproduct from sewage chlorination, disrupts thyroid function, used to study deiodinase.</p>
    Fórmula:C6H3I3O
    Pureza:98.11%
    Forma y color:Grey To Tan To Brown Powder
    Peso molecular:471.8
  • 2-Methoxyestradiol

    CAS:
    <p>2-ME2, an estradiol derivative, hinders angiogenesis and tumor growth, causes cell apoptosis, and stops mitosis.</p>
    Fórmula:C19H26O3
    Pureza:98% - 99.95%
    Forma y color:Off-White Solid
    Peso molecular:302.41
  • Asiatic acid

    CAS:
    <p>Asiatic acid (Dammarolic acid) is the aglycone of asiaticoside used in wound healing with antioxidant, anti-inflammatory, and neuroprotective properties.</p>
    Fórmula:C30H48O5
    Pureza:98.01% - 99.52%
    Forma y color:Solid Powder
    Peso molecular:488.7
  • RAD51 Inhibitor B02

    CAS:
    <p>RAD51 Inhibitor B02 (B02) (B02) is an inhibitor of human RAD51 with an IC50 of 27.4 μM.</p>
    Fórmula:C22H17N3O
    Pureza:99.72% - 99.89%
    Forma y color:Solid
    Peso molecular:339.39
  • NVP-TAE 684

    CAS:
    <p>NVP-TAE 684 (TAE684) is a excellently effective and specific ALK inhibitor(IC50=3 nM).</p>
    Fórmula:C30H40ClN7O3S
    Pureza:98% - 99.82%
    Forma y color:Solid
    Peso molecular:614.2
  • ICCB280

    CAS:
    <p>ICCB280 was capable of inducing differentiation and apoptosis of ATRA-resistant patient blasts strongly signify that the activity of this compound can overcome</p>
    Fórmula:C23H18N2O4
    Pureza:98.04%
    Forma y color:Solid
    Peso molecular:386.4
  • Thalidomide-O-amido-C6-NH2 TFA

    CAS:
    Thalidomide-O-amido-C6-NH2 TFA (Cereblon Ligand-Linker Conjugates 11 TFA), a synthesized E3 ligase ligand-linker conjugate containing a Thalidomide-based
    Fórmula:C46H53F6N8O16
    Pureza:95.16%
    Forma y color:Solid
    Peso molecular:1087.95
  • Minodronic acid monohydrate

    CAS:
    <p>Minodronic acid monohydrate 是一种法尼基二磷酸合成酶抑制剂,可作为骨吸收抑制剂。</p>
    Fórmula:C9H14N2O8P2
    Pureza:≥95%
    Forma y color:Solid
    Peso molecular:340.16
  • FB23-2

    CAS:
    <p>FB23-2 is a potent and selective mRNA N6-methyladenosine (m6A) demethylase FTO inhibitor(IC50 : 2.6 μM).</p>
    Fórmula:C18H15Cl2N3O3
    Pureza:97.29% - ≥95%
    Forma y color:Solid
    Peso molecular:392.24
  • BAY 61-3606 HCl

    CAS:
    <p>BAY 61-3606 HCl: a reversible Syk inhibitor, halts mast cell degranulation, cytokines, and sensitizes MCF-7 cells to TRAIL-induced apoptosis.</p>
    Fórmula:C20H19ClN6O3
    Forma y color:Solid
    Peso molecular:426.86
  • Thalidomide-5-OH

    CAS:
    <p>Thalidomide-5-OH (2-(2,6-dioxopiperidin-3-yl)-5-hydroxyisoindoline-1,3-dione) is the Thalidomide-based cereblon ligand that used in the recruitment of CRBN</p>
    Fórmula:C13H10N2O5
    Pureza:98.94%
    Forma y color:Solid
    Peso molecular:274.23
  • ZMC1

    CAS:
    <p>NSC-319726 (ZMC1), a mutant p53R175 reactivator, suppresses growth of fibroblasts that expresses the p53R175 mutation (IC50 = 8 nM).</p>
    Fórmula:C11H14N4S
    Pureza:98.97% - 99.76%
    Forma y color:Solid
    Peso molecular:234.32
  • L-Buthionine-(S,R)-sulfoximine hydrochloride


    <p>L-Buthionine-(S,R)-sulfoximine hydrochloride is a fast, irreversible γ-GCS inhibitor that depletes glutathione. IC50: 1.9-29 μM in various tumors.</p>
    Fórmula:C8H19ClN2O3S
    Forma y color:Solid
    Peso molecular:258.77
  • Buprofezin

    CAS:
    Buprofezin (Applaud) is an insecticide used for control of insect pests such as mealybugs, leafhoppers and whitefly on vegetable crops.
    Fórmula:C16H23N3OS
    Pureza:99.02% - 99.73%
    Forma y color:White To Pale Yellow Crystalline Powder
    Peso molecular:305.44
  • Quiflapon sodium

    CAS:
    <p>Quiflapon sodium (MK591) is a selective inhibitor of 5-Lipoxygenase-activating protein (FLAP).</p>
    Fórmula:C34H35ClN2NaO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:610.16
  • Quizartinib HCl

    CAS:
    <p>Quizartinib (AC220/AC010220) is an oral FLT3/STK1 inhibitor for treating AML, blocking kinase-driven cell proliferation and promoting apoptosis.</p>
    Fórmula:C29H34Cl2N6O4S
    Forma y color:Solid
    Peso molecular:633.59
  • Desloratadine

    CAS:
    <p>Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.</p>
    Fórmula:C19H19ClN2
    Pureza:99.79% - >99.99%
    Forma y color:Solid
    Peso molecular:310.82
  • Sodium Demethylcantharidate

    CAS:
    <p>Sodium Demethylcantharidate (Sodium norcantharidin) is extracted from Mylabris phqlarata pallas and has potent antitumor activity.</p>
    Fórmula:C8H9O5·Na
    Pureza:99.66% - ≥98%
    Forma y color:Solid
    Peso molecular:208.14
  • Thalidomide 4'-ether-alkylC2-amine hydrochloride

    CAS:
    <p>Thalidomide 4'-ether-alkylC2-amine hydrochloride (halidomide-linker 6) is a synthesized E3 ligase ligand-linker conjugate.</p>
    Fórmula:C15H16ClN3O5
    Pureza:98.56%
    Forma y color:Solid
    Peso molecular:353.76
  • Ricolinostat

    CAS:
    <p>Ricolinostat (Rocilinostat) is an orally bioavailable, specific inhibitor of histone deacetylase 6 (HDAC6) with potential antineoplastic activity.</p>
    Fórmula:C24H27N5O3
    Pureza:97.17% - 99.76%
    Forma y color:Solid
    Peso molecular:433.5
  • Rafoxanide

    CAS:
    <p>Rafoxanide as a dual CDK4/6 inhibitor for the treatment of skin cancer.</p>
    Fórmula:C19H11Cl2I2NO3
    Pureza:99.47%
    Forma y color:Slight Yellowish Brown Injectable Solution &White Oral Solution
    Peso molecular:626.01
  • Pyrazoloadenine

    CAS:
    <p>Pyrazoloadenine (4-Aminopyrazolo[3,4-d]pyrimidine) is the inhibitor of human xanthine oxidase.</p>
    Fórmula:C5H5N5
    Pureza:99.02%
    Forma y color:Beige Powder
    Peso molecular:135.13
  • Fenoldopam mesylate

    CAS:
    <p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>
    Fórmula:C16H16ClNO3·CH4O3S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:401.86
  • S-99

    CAS:
    S-99 is a high purity chemical that targets ASK and is important for Immunology, Inflammation, Cancer research.
    Fórmula:C16H15F3N6O
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:364.33
  • RRX-001

    CAS:
    <p>RRx-001 is a potent inhibitor ofglucose 6-phosphate dehydrogenase(G6PD) and with potent antimalarial activity</p>
    Fórmula:C5H6BrN3O5
    Pureza:99.91% - ≥95%
    Forma y color:Solid
    Peso molecular:268.02
  • Nerol

    CAS:
    <p>Nerol (Neryl alcohol) is a monoterpene found in many essential oils, such as lemon balm and hop.Nerol can lessened the severity of ouabain-triggered arrhythmias</p>
    Fórmula:C10H18O
    Pureza:98.59%
    Forma y color:Colorless Oily Liquid Liquid
    Peso molecular:154.25
  • Tazemetostat

    CAS:
    <p>Tazemetostat (EPZ6438): Oral EZH2 inhibitor, blocks histone H3K27 methylation, potential cancer therapy.</p>
    Fórmula:C34H44N4O4
    Pureza:98.24% - ≥95%
    Forma y color:Solid
    Peso molecular:572.74
  • Tangeretin

    CAS:
    <p>Tangeretin (NSC-618905), a flavonoid from citrus fruit peels, has been proven to play an important role in anti-inflammatory responses and neuroprotective</p>
    Fórmula:C20H20O7
    Pureza:98.83% - 98.97%
    Forma y color:Yellow Crystalline
    Peso molecular:372.37
  • Torkinib

    CAS:
    <p>Torkinib (PP 242) (PP 242) is a selective and ATP-competitive mTOR inhibitor (IC50: 8 nM). It also inhibits mTORC1/2 (IC50s: 30/58 nM).</p>
    Fórmula:C16H16N6O
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:308.34
  • CPTH2

    CAS:
    <p>CPTH2 is a histone acetyltransferase inhibitor modulating Gcn5 network.</p>
    Fórmula:C14H14ClN3S
    Pureza:99.81%
    Forma y color:Solid
    Peso molecular:291.8
  • Idasanutlin

    CAS:
    <p>Idasanutlin (Ro 5503781) (RG-7388) is an effective and specific p53-MDM2 inhibitor (IC50: 6 nM).</p>
    Fórmula:C31H29Cl2F2N3O4
    Pureza:99.13% - 99.88%
    Forma y color:Solid
    Peso molecular:616.48
  • HLCL-61 hydrochloride

    CAS:
    HLCL-61 hydrochloride (HLCL-61 HCL) is a potent and selective PRMT5 inhibitor for the treatment of acute myeloid leukemia.
    Fórmula:C23H24N2O·ClH
    Pureza:99.88% - 99.95%
    Forma y color:Solid
    Peso molecular:380.91
  • ABT-751

    CAS:
    ABT-751 (E7010) has been investigated for the treatment of Lung Cancer, Non-Small Cell Lung Cancer, and Non-Small-Cell Lung Cancer.
    Fórmula:C18H17N3O4S
    Pureza:98.84% - 99.50%
    Forma y color:Solid
    Peso molecular:371.41
  • cjoc42

    CAS:
    <p>Cjoc42 blocks gankyrin to prevent p53 reduction, aiding cancer prevention and DNA damage response.</p>
    Fórmula:C20H21N3O5S
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:415.46
  • 4'-bromo-Resveratrol

    CAS:
    <p>4'-bromo-Resveratrolis a potent inhibitor of the deacetylases sirtuin 1 (SIRT1) and 3 (SIRT3)</p>
    Fórmula:C14H11BrO2
    Pureza:99.00%
    Forma y color:Solid
    Peso molecular:291.14
  • Shield-1

    CAS:
    <p>Shield-1 is a specific, high-affinity, and cell-permeable ligand for FK506-binding protein 12 (FKBP).Cost-effective and quality-assured.</p>
    Fórmula:C42H56N2O10
    Pureza:99.08%
    Forma y color:Solid
    Peso molecular:748.9
  • Flupentixol dihydrochloride

    CAS:
    <p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.76% - >99.99%
    Forma y color:White Or Off-White Solid
    Peso molecular:507.43
  • Dacomitinib

    CAS:
    <p>Dacomitinib (PF299) is an oral selective inhibitor of EGFR, ERBB2, ERBB4 with IC50s: 6, 45.7, 73.7 nM.</p>
    Fórmula:C24H25ClFN5O2
    Pureza:99.4% - 99.72%
    Forma y color:Solid
    Peso molecular:469.94
  • Thalidomide-NH-C2-PEG3-OH

    CAS:
    <p>Thalidomide-NH-C2-PEG3-OH (H-Isoindole-1,3(2H)-dione, 2-(2,6-dioxo-3-piperidinyl)-4-[[2-[2-[2-(2-hydroxyethoxy)ethoxy]ethoxy]ethyl]amino]-) is an E3 ligase</p>
    Fórmula:C21H27N3O8
    Pureza:99.06%
    Forma y color:Solid
    Peso molecular:449.45
  • Kinetin riboside

    CAS:
    Kinetin riboside (N6-Furfuryladenosine) can induce apoptosis in cancer cells. It inhibits the proliferation of HCT-15 cells(IC50 of 2.5 μM)
    Fórmula:C15H17N5O5
    Pureza:98.17%
    Forma y color:White Solid
    Peso molecular:347.33
  • Fraxetin

    CAS:
    <p>Fraxetin (7,8-dihydroxy-6-methoxy coumarin) has dual-antioxidative ,hepatoprotective and antihyperglycemic functions, it shows potent protective effects against</p>
    Fórmula:C10H8O5
    Pureza:98% - 99.59%
    Forma y color:Light Yellow Crystalline Flakes
    Peso molecular:208.17
  • C5 Lenalidomide

    CAS:
    <p>C5 Lenalidomide is an chemical weith inconclusive biological activity.</p>
    Fórmula:C13H13N3O3
    Pureza:99.4%
    Forma y color:Solid
    Peso molecular:259.26
  • 8-Bromo-cAMP sodium salt

    CAS:
    <p>8-Bromo-cAMP sodium salt (8-Br-Camp sodium salt) is a long-acting derivative of cyclic AMP. 8-Bromo-cAMP is an activator of cyclic AMP-dependent protein kinase.</p>
    Fórmula:C10H10BrN5NaO6P
    Pureza:98% - 99.94%
    Forma y color:Off-White Powder
    Peso molecular:430.08
  • Ac-DEVD-pNA

    CAS:
    <p>Ac-DEVD-pNA is the preferred peptidic substrate for caspase-3.</p>
    Fórmula:C26H34N6O13
    Pureza:>99.99%
    Forma y color:White
    Peso molecular:638.58
  • Dracorhodin perchlorate

    CAS:
    <p>Dracorhodin perchlorate inhibits cell growth, and induces apoptosis in fibroblasts, arresting cell cycle at G1 phase, may as a candidate for anti-breast cancer.</p>
    Fórmula:C17H15ClO7
    Pureza:98.31% - ≥95%
    Forma y color:Solid
    Peso molecular:366.75
  • RG7112

    CAS:
    <p>RG7112 (RO5045337) (RO5045337) is an orally bioavailable and selective p53-MDM2 inhibitor.</p>
    Fórmula:C38H48Cl2N4O4S
    Pureza:99.66% - 99.9%
    Forma y color:Solid
    Peso molecular:727.78
  • Butein

    CAS:
    Butein is a cAMP-specific PDE inhibitor, protein tyrosine kinase inhibitor, and SIRT1 activator.Cost-effective and quality-assured.
    Fórmula:C15H12O5
    Pureza:98.76% - >99.99%
    Forma y color:Solid
    Peso molecular:272.25
  • Vandetanib hydrochloride

    CAS:
    <p>Vandetanib hydrochloride is an oral VEGFR2 inhibitor with an IC50 of 40 nM, also targeting VEGFR3 (110 nM) and EGFR (500 nM).</p>
    Fórmula:C22H25BrClFN4O2
    Forma y color:Solid
    Peso molecular:511.81
  • Zoledronic acid disodium tetrahydrate

    CAS:
    <p>Zoledronic Acid, a potent bisphosphonate, inhibits osteoclasts and has anti-cancer effects.</p>
    Fórmula:C5H16N2Na2O11P2
    Forma y color:Solid
    Peso molecular:388.113
  • Droxinostat

    CAS:
    <p>Droxinostat (NS 41080) is a selective inhibitor of HDAC, mostly for HDACs 6 and 8 with IC50 of 2.47 μM and 1.46 μM, greater than 8-fold selective against HDAC3</p>
    Fórmula:C11H14ClNO3
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:243.69
  • Ulinastatin

    CAS:
    <p>Ulinastatin is a multivalent Kunitz-type serine protease inhibitor with anti-inflammatory properties.</p>
    Fórmula:C13H16O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:220.10994
  • Ziyuglycoside I

    CAS:
    <p>Ziyuglycoside I (Gouguside 7) has anti-inflammatory activity, could be used as an active ingredient for cosmetics.</p>
    Fórmula:C41H66O13
    Pureza:98.987% - ≥95%
    Forma y color:Solid
    Peso molecular:766.95
  • NADPH tetracyclohexanamine

    CAS:
    <p>NADPH tetracyclohexanamine (NADPH (tetracyclohexanamine)) is a cofactor and biological reducing agent.</p>
    Fórmula:C45H82N11O17P3
    Pureza:98.73% - 99.05%
    Forma y color:Solid
    Peso molecular:1142.12
  • Cinchonine monohydrochloride hydrate

    CAS:
    <p>Cinchonine monohydrochloride hydrate: natural antimalarial, inhibits platelet aggregation &amp; cancer cell growth, blocks fat cell formation.</p>
    Fórmula:C19H25ClN2O2
    Forma y color:Solid
    Peso molecular:348.87
  • Prexasertib Mesylate Hydrate

    CAS:
    <p>Prexasertib Mesylate Hydrate is a potent CHK1 inhibitor (IC50&lt;1nM), also inhibits CHK2, RSK1, induces DNA breaks, apoptosis, and has anti-tumor effects.</p>
    Fórmula:C19H25N7O6S
    Forma y color:Solid
    Peso molecular:479.51
  • Benzoylpaeoniflorin

    CAS:
    <p>1. Benzoylpaeoniflorin is active against cyclooxygenase-1 and cyclooxygenase-2 enzymes.</p>
    Fórmula:C30H32O12
    Pureza:95.86% - 97.28%
    Forma y color:Solid
    Peso molecular:584.57
  • α-Lipoic Acid sodium

    CAS:
    <p>α-Lipoic Acid (Thioctic acid) sodium, an essential cofactor for mitochondrial enzyme complexes, serves as an antioxidant.</p>
    Fórmula:C8H13NaO2S2
    Forma y color:Solid
    Peso molecular:228.31
  • Rhosin hydrochloride

    CAS:
    <p>Rhosin hydrochloride is a specific inhibitor of the RhoA subfamily Rho GTPases.Cost-effective and quality-assured.</p>
    Fórmula:C20H20Cl2N6O
    Pureza:97.33% - 98.92%
    Forma y color:Solid
    Peso molecular:431.318
  • 3'-Hydroxypterostilbene

    CAS:
    <p>3'-Hydroxypterostilbene suppresses colon cancer cell growth (COLO 205, HCT-116, HT-29) by triggering apoptosis and autophagy, affecting key pathways.</p>
    Fórmula:C16H16O4
    Pureza:98.25% - 99.19%
    Forma y color:Solid
    Peso molecular:272.3
  • Meloxicam sodium

    CAS:
    <p>Meloxicam sodium is a non-steroidal anti-inflammatory agent, inhibits COX activity, with IC 50 s of 0.49 μM and 36.6 μM for COX-2 and COX-1, respectively [1].</p>
    Fórmula:C14H12N3NaO4S2
    Forma y color:Solid
    Peso molecular:373.38
  • Siremadlin

    CAS:
    <p>Siremadlin (NVP-HDM 201) is a potent, orally bioavailable and highly specific p53-MDM2 interaction inhibitor.</p>
    Fórmula:C26H24Cl2N6O4
    Pureza:99.30% - 99.76%
    Forma y color:Solid
    Peso molecular:555.41
  • Tofacitinib Citrate

    CAS:
    <p>Tofacitinib Citrate (CP-690550 citrate) is a a potent, cell-permeable inhibitor of JAK1/2/3 (IC50s: 1/20/112 nM).</p>
    Fórmula:C22H28N6O8
    Pureza:99.19% - 99.75%
    Forma y color:Solid
    Peso molecular:504.49
  • Itanapraced

    CAS:
    <p>Itanapraced (CHF5074), a γ-secretase modulator, reduces Aβ42/40 secretion (IC50: 3.6/18.4 μM).</p>
    Fórmula:C16H11Cl2FO2
    Pureza:98% - 99.79%
    Forma y color:Solid
    Peso molecular:325.16
  • Perifosine

    CAS:
    <p>Perifosine (KRX-0401) is an oral-active, alkyl-phosphocholine Akt inhibitor with potential antineoplastic activity.</p>
    Fórmula:C25H52NO4P
    Pureza:99.94% - >99.99%
    Forma y color:Solid
    Peso molecular:461.66
  • Dimethyl malonate

    CAS:
    <p>Dimethyl Malonate is a Succinate Dehydrogenase inhibitor.</p>
    Fórmula:C5H8O4
    Pureza:≥95%
    Forma y color:Liquid
    Peso molecular:132.11
  • Chelerythrine

    CAS:
    <p>1.</p>
    Fórmula:C21H18NO4
    Pureza:98.36%
    Forma y color:Solid
    Peso molecular:348.37
  • Fedratinib

    CAS:
    Fedratinib (TG-101348) (TG101348) is an ATP-competitive inhibitor of JAK2 (IC50: 3 nM) with significantly less potent activity against JAK3.
    Fórmula:C27H36N6O3S
    Pureza:97.31% - 99.96%
    Forma y color:Solid
    Peso molecular:524.68
  • ONO-8130

    CAS:
    <p>ONO-8130 is an orally available antagonist of EP1 receptor.</p>
    Fórmula:C25H28N2O5S2
    Pureza:97.82%
    Forma y color:Solid
    Peso molecular:500.63
  • Mitoxantrone diacetate

    CAS:
    <p>Mitoxantrone diacetate hinders topoisomerase II &amp; PKC, fights tumors &amp; orthopoxviruses (IC50: 8.5μM, EC50: 0.25-0.8μM).</p>
    Fórmula:C26H36N4O10
    Forma y color:Solid
    Peso molecular:564.592
  • Fasentin

    CAS:
    <p>Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.</p>
    Fórmula:C11H9ClF3NO2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:279.64
  • SKLB-163

    CAS:
    <p>SKLB-163 acts by downregulating RhoGDI, activating JNK-1 signaling pathway and caspase-3, and reducing phosphorylated Akt and p44/42 MAPK.</p>
    Fórmula:C18H16ClN3O2S2
    Pureza:99.23%
    Forma y color:Solid
    Peso molecular:405.92
  • MCB-613

    CAS:
    <p>MCB-613 is an effective steroid receptor coactivator (SRC) stimulator.</p>
    Fórmula:C20H20N2O
    Pureza:98.17% - 99.754%
    Forma y color:Solid
    Peso molecular:304.39
  • PFI-1

    CAS:
    <p>PFI-1 (PF-6405761), a specific BET (bromodomain-containing protein) inhibitor for BRD4, is with the IC50 of 0.22 μM in a cell-free assay.</p>
    Fórmula:C16H17N3O4S
    Pureza:98.74% - 99.19%
    Forma y color:Solid
    Peso molecular:347.39
  • Thalidomide-PEG4-Propargyl

    CAS:
    <p>Thalidomide-PEG4-Propargyl is a synthetic E3 ligase ligand for PROTAC with a cereblon ligand and linker.</p>
    Fórmula:C24H28N2O9
    Pureza:97.46%
    Forma y color:Solid
    Peso molecular:488.49
  • SC66

    CAS:
    <p>SC66 is a AKT inhibitor in HepG2, HA22T/VGH, and PLC/PRF/5 cells (IC50: about 0.75 μg/ml, at 72 h).</p>
    Fórmula:C18H16N2O
    Pureza:>99.99% - >99.99%
    Forma y color:Solid
    Peso molecular:276.33
  • Fenobam hydrate

    CAS:
    <p>Fenobam hydrate blocks mGluR5, preventing calcium mobilization, and may reduce stress, anxiety, and pain.</p>
    Fórmula:C11H13ClN4O3
    Forma y color:Solid
    Peso molecular:284.7
  • Asiaticoside

    CAS:
    <p>Asiaticoside, in Centella asiatica, may treat wounds/burns.</p>
    Fórmula:C48H78O19
    Pureza:98% - 99.96%
    Forma y color:Powder
    Peso molecular:959.12
  • Laquinimod sodium

    CAS:
    <p>Laquinimod (ABR-215062) sodium is an oral agent for MS, halting neurodegeneration and inflammation.</p>
    Fórmula:C19H16ClN2NaO3
    Forma y color:Solid
    Peso molecular:378.79
  • Dihydrocapsaicin

    CAS:
    Dihydrocapsaicin, similar to capsaicin, is an irritant found in Capsicum, used in "pure" capsaicin products at about 10%, activates VR1, and is an antioxidant.
    Fórmula:C18H29NO3
    Pureza:99.8% - ≥95%
    Forma y color:White Crystal
    Peso molecular:307.43
  • MK-2206

    CAS:
    <p>MK-2206: selective Akt inhibitor, oral, targets Akt1, Akt2, Akt3; effective in breast cancer, PIK3CA mutants, PTEN-deficient cells.</p>
    Fórmula:C25H22ClN5O
    Forma y color:Solid
    Peso molecular:443.94
  • ML311

    CAS:
    <p>ML311 is a selective inhibitor of the Mcl-1/Bim interaction.</p>
    Fórmula:C23H24F3N3O
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:415.45
  • Milademetan free base

    CAS:
    <p>Milademetan (DS-3032b) is a potent MDM2 inhibitor, potentially blocking cancer growth by targeting p53 protein.</p>
    Fórmula:C37H42Cl2FN5O7S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:790.73
  • Thalidomide-O-C4-NH2 hydrochloride

    CAS:
    <p>Thalidomide-linker 9: a cereblon ligand, E3 ligase conjugate for PROTAC tech.</p>
    Fórmula:C17H20ClN3O5
    Pureza:98.33%
    Forma y color:Solid
    Peso molecular:381.81
  • PI-103

    CAS:
    <p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>
    Fórmula:C19H16N4O3
    Pureza:97.79% - 99.3%
    Forma y color:Solid
    Peso molecular:348.36
  • Benidipine

    CAS:
    <p>Benidipine: potent oral calcium blocker, boosts nitric oxide synthase, enhances coronary flow, protects heart cells post-ischemia.</p>
    Fórmula:C28H31N3O6
    Forma y color:Solid
    Peso molecular:505.56
  • Bardoxolone

    CAS:
    <p>Bardoxolone (CDDO) inhibits iNOS, COX-2 in cells; IC50=0.4nM. Reduces ROS/RNS, DNA damage, &amp; cancer growth; triggers apoptosis &amp; boosts antioxidant genes.</p>
    Fórmula:C31H41NO4
    Pureza:97.9% - 98.97%
    Forma y color:Solid
    Peso molecular:491.66
  • Panobinostat lactate

    CAS:
    <p>Panobinostat lactate: potent, non-selective, oral HDAC inhibitor; treats refractory multiple myeloma.</p>
    Fórmula:C24H29N3O5
    Forma y color:Solid
    Peso molecular:439.512
  • QNZ

    CAS:
    <p>QNZ (EVP4593) (EVP4593) is an effective inhibitor of NF-κB activation and TNF-α production. The IC50 of QNZ for NF-κB and TNF-α is11 nM and 7 nM, respectively.</p>
    Fórmula:C22H20N4O
    Pureza:99.17% - 99.18%
    Forma y color:White Solid
    Peso molecular:356.42
  • JKE-1674

    CAS:
    <p>JKE-1674 is an orally active glutathione peroxidase 4 (GPX4) inhibitor and the active metabolite of ML-210.Cost-effective and quality-assured.</p>
    Fórmula:C20H20Cl2N4O4
    Pureza:98.02% - 98.4%
    Forma y color:Solid
    Peso molecular:451.3
  • LY294002

    CAS:
    <p>LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).</p>
    Fórmula:C19H17NO3
    Pureza:98% - 99.96%
    Forma y color:Pale Yellow Solid
    Peso molecular:307.34
  • Trifloxystrobin

    CAS:
    <p>Trifloxystrobin is a fungicide against R. solani in sugar beets with EC50s: 23.0 μg/L for Daphnia neonates, 1.7 μg/L for embryos.</p>
    Fórmula:C20H19F3N2O4
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:408.37
  • ERK1/2 inhibitor 2

    CAS:
    <p>ERK1/2 inhibitor 2 (ASTX029) is a selective and orally bioavailable ERK 1/2 inhibitor, with potential antineoplastic activity.</p>
    Fórmula:C29H31ClFN5O5
    Pureza:98.99%
    Forma y color:Solid
    Peso molecular:584.04
  • Isolongifolene

    CAS:
    <p>Isolongifolene ((-)-Isolongifolene), a tricyclic sesquiterpene isolated from Murraya koenigii, exhibits antioxidant, anti-inflammatory, anticancer, and</p>
    Fórmula:C15H24
    Pureza:90.13% - 99.46%
    Forma y color:Colorless Or Light Yellow Liquid
    Peso molecular:204.35
  • Topotecan hydrochloride hydrate

    CAS:
    <p>Orally active Topotecan HCl hydrate inhibits Topoisomerase I, blocks G0/G1 &amp; S phases, and induces apoptosis.</p>
    Fórmula:C23H26ClN3O6
    Forma y color:Solid
    Peso molecular:475.93
  • Tomivosertib HCl

    CAS:
    <p>Tomivosertib (eFT508) is a MNK1/2 inhibitor that blocks eIF4E phosphorylation, hindering tumor growth and immune signaling.</p>
    Fórmula:C17H21ClN6O2
    Forma y color:Solid
    Peso molecular:376.845
  • CM-272

    CAS:
    CM-272 is a dual G9a/DNA methyltransferases (DNMTs) inhibitor.
    Fórmula:C28H38N4O3
    Pureza:97.83%
    Forma y color:Solid
    Peso molecular:478.63
  • Lanreotide acetate

    CAS:
    Lanreotide acetate (BIM 23014 acetate) is a somatostatin analogue with antineoplastic activity, used for carcinoid syndrome
    Fórmula:C56H73N11O12S2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1156.39
  • Clodronate disodium tetrahydrate

    CAS:
    <p>Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.</p>
    Fórmula:CH10Cl2Na2O10P2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:360.92
  • Rigosertib

    CAS:
    <p>Rigosertib, a multi-kinase inhibitor targeting PLK1 (IC50: 9 nM), induces apoptosis and G2/M arrest by disrupting PI3K/Akt.</p>
    Fórmula:C21H25NO8S
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:451.49
  • CHIR-124

    CAS:
    CHIR-124 is an effective Chk1 inhibitor (IC50: 0.3 nM). It has 2, 000-fold selectivity against Chk2, 500- to 5, 000-fold less activity against Cdc2 and CDK2/4.
    Fórmula:C23H22ClN5O
    Pureza:96.33% - 98.35%
    Forma y color:Solid
    Peso molecular:419.91
  • AZD1208 hydrochloride

    CAS:
    <p>AZD1208 hydrochloride is a highly selective, potent and orally active PIM inhibitor.</p>
    Fórmula:C21H22ClN3O2S
    Forma y color:Solid
    Peso molecular:415.94
  • Psoralen

    CAS:
    <p>Psoralen (Ficusin) is a furocoumarin that intercalates with DNA, inhibiting DNA synthesis and cell division.</p>
    Fórmula:C11H6O3
    Pureza:99.3% - 99.87%
    Forma y color:Crystals From Ether Crystalline Solid
    Peso molecular:186.16
  • Sertaconazole

    CAS:
    <p>Sertaconazole is a broad-spectrum antifungal.</p>
    Fórmula:C20H15Cl3N2OS
    Pureza:99.483%
    Forma y color:Solid
    Peso molecular:437.77
  • Sepantronium bromide

    CAS:
    <p>Sepantronium bromide (YM155) is a small-molecule proapoptotic agent with potential antineoplastic activity.</p>
    Fórmula:C20H19BrN4O3
    Pureza:99.68% - 99.85%
    Forma y color:Solid
    Peso molecular:443.26
  • Etretinate

    CAS:
    <p>Etretinate (Ro 10-9359), an oral retinoid, treats psoriasis by promoting cell differentiation and reducing cell growth and inflammation.</p>
    Fórmula:C23H30O3
    Pureza:97.89%
    Forma y color:Crystals Crystalline Solid
    Peso molecular:354.48
  • Moexipril hydrochloride

    CAS:
    <p>Moexipril hydrochloride (Moexipril HCl) is a potent orally active nonsulfhydrylangiotensin converting enzyme (ACE)inhibitor, used for the treatment of</p>
    Fórmula:C27H34N2O7·HCl
    Pureza:97.8%
    Forma y color:A Fine White To Off-White Powder
    Peso molecular:535.03
  • Afatinib Dimaleate

    CAS:
    <p>Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the EGFR family, with antineoplastic activity.</p>
    Fórmula:C32H33ClFN5O11
    Pureza:98.11% - 99.87%
    Forma y color:Solid
    Peso molecular:718.08
  • AG1024

    CAS:
    <p>AG1024 (Tyrphostin) suppresses IGF-1R autophosphorylation(IC50=7 μM), and is less potent for IR(IC50=57 μM).</p>
    Fórmula:C14H13BrN2O
    Pureza:98% - 99.37%
    Forma y color:Solid
    Peso molecular:305.17
  • SKI-178

    CAS:
    <p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>
    Fórmula:C21H22N4O4
    Pureza:97.09%
    Forma y color:Solid
    Peso molecular:394.42
  • BIX01294 (hydrochloride hydrate)

    CAS:
    <p>BIX01294 inhibits G9a HMTase (IC50=1.7μM), less effective on GLP, and aids in induced pluripotent stem cell generation.</p>
    Fórmula:C28H43Cl3N6O3
    Forma y color:Solid
    Peso molecular:618.04
  • Sacubitril/Valsartan

    CAS:
    <p>Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for treatment of hypertension and heart failure.</p>
    Fórmula:C48H55N6O8Na3·5H2O
    Pureza:99.75% - >99.99%
    Forma y color:Solid
    Peso molecular:957.99
  • Tandutinib hydrochloride

    CAS:
    <p>Tandutinib hydrochloride: FLT3 inhibitor (IC50 0.22 μM), targets c-Kit, PDGFR, treats AML, crosses blood-brain barrier.</p>
    Fórmula:C31H43ClN6O4
    Forma y color:Solid
    Peso molecular:599.16
  • Niraparib tosylate monohyrate

    CAS:
    Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.
    Fórmula:C26H30N4O5S
    Pureza:97.7% - 99.99%
    Forma y color:Solid
    Peso molecular:510.61
  • BAY 87-2243

    CAS:
    BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).
    Fórmula:C26H26F3N7O2
    Pureza:98% - 99.95%
    Forma y color:Solid
    Peso molecular:525.53
  • BAY 61-3606

    CAS:
    <p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>
    Fórmula:C20H18N6O3
    Pureza:98.72%
    Forma y color:Solid
    Peso molecular:390.4
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Fórmula:C30H18O10
    Pureza:98.21% - 99.22%
    Forma y color:Odourless Whitish Solid
    Peso molecular:538.46
  • WYC-209

    CAS:
    <p>WYC-209 inhibits proliferation of malignant murine melanoma tumor-repopulating cells (TRCs, IC50: 0.19 uM). It targets the retinoic acid receptor (RAR).</p>
    Fórmula:C20H20N2O3S
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:368.45
  • KW-2449

    CAS:
    <p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>
    Fórmula:C20H20N4O
    Pureza:98.43% - 99.69%
    Forma y color:Solid
    Peso molecular:332.4
  • Nafamostat mesylate

    CAS:
    <p>Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis</p>
    Fórmula:C19H17N5O2·2CH4O3S
    Pureza:97.36% - 99.76%
    Forma y color:Tan To Pale Orange Solid
    Peso molecular:539.58
  • Etidronic acid

    CAS:
    <p>Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.</p>
    Fórmula:C2H8O7P2
    Pureza:99.93% - ≥95%
    Forma y color:Liquid Syrup
    Peso molecular:206.03
  • Dinaciclib

    CAS:
    <p>Dinaciclib (SCH 727965) is a CDK inhibitor that selectively inhibits CDK1, CDK2, CDK5, and CDK9 (IC50 = 3/1/1/4 nM).</p>
    Fórmula:C21H28N6O2
    Pureza:98.21% - 99.75%
    Forma y color:Solid
    Peso molecular:396.49
  • Astragalin

    CAS:
    <p>Astragalin (Kaempferol 3-O-glucoside) is a biologically active natural flavonoid.</p>
    Fórmula:C21H20O11
    Pureza:98.8% - ≥95%
    Forma y color:Solid
    Peso molecular:448.38
  • Phellamurin

    CAS:
    <p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>
    Fórmula:C26H30O11
    Pureza:97.91%
    Forma y color:Solid
    Peso molecular:518.51
  • Pracinostat

    CAS:
    <p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>
    Fórmula:C20H30N4O2
    Pureza:99.15% - 99.67%
    Forma y color:Solid
    Peso molecular:358.48
  • 2-Hydroxychalcone

    CAS:
    <p>2-Hydroxychalcone (2-(2-Hydroxybenzal)Acetophenone) can be used as antiparasitic hit compounds when Methoxylated. It inhibits invasion of breast cancer cells.</p>
    Fórmula:C15H12O2
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:224.25
  • GMB-475

    CAS:
    <p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>
    Fórmula:C43H46F3N7O7S
    Pureza:98.78% - >99.99%
    Forma y color:Solid
    Peso molecular:861.93
  • Citric acid monohydrate

    CAS:
    <p>Citric Acid Monohydrate: tricarboxylic, from citrus, antioxidant, stabilizes drugs, preservative.</p>
    Fórmula:C6H10O8
    Pureza:99.87%
    Forma y color:White Solid Crystalline
    Peso molecular:210.14
  • Protosappanin B

    CAS:
    <p>Protosappanin B enhances cell survival, growth protein 43; degrades p53 via MDM2 ubiquitination.</p>
    Fórmula:C16H16O6
    Pureza:98% - 98.86%
    Forma y color:Solid
    Peso molecular:304.29
  • GSK1059615

    CAS:
    <p>GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.</p>
    Fórmula:C18H11N3O2S
    Pureza:99.3% - ≥95%
    Forma y color:Solid
    Peso molecular:333.36
  • STF-118804

    CAS:
    <p>STF-118804 is a highly specific NAMPT inhibitor; reduces the viability of most B-ALL cell lines with IC50 &lt;10 nM.</p>
    Fórmula:C25H23N3O4S
    Pureza:98.66%
    Forma y color:Solid
    Peso molecular:461.53
  • [6]-Gingerol

    CAS:
    <p>[6]-Gingerol ((S)-(+)-[6]Gingerol), an antioxidant, protects HL-60 cells from oxidative stress. It has protective effects for tumors.</p>
    Fórmula:C17H26O4
    Pureza:98% - 99.66%
    Forma y color:Light Yellow Oiliness
    Peso molecular:294.39
  • SKI II

    CAS:
    SKI II is a selective non-ATP S1P receptor inhibitor with an IC50 of 0.5 μM; it doesn't inhibit PKCα, PI3K, or ERK2.
    Fórmula:C15H11ClN2OS
    Pureza:99.34% - 99.93%
    Forma y color:Solid
    Peso molecular:302.78
  • Diffractaic Acid

    CAS:
    <p>Diffractaic Acid (NSC 685595) can inhibit LTB4 biosynthesis in A-23187-stimulated bovine PMNL cells with activity value of 8 μM.</p>
    Fórmula:C20H22O7
    Pureza:99.81% - 99.87%
    Forma y color:Solid
    Peso molecular:374.38
  • NSC 95397

    CAS:
    <p>NSC 95397 is a potent inhibitor of Cdc25 dual specificity phosphatase(Ki of 32, 96, and 40 nM for Cdc25A, Cdc25B, and Cdc25C, respectively).</p>
    Fórmula:C14H14O4S2
    Pureza:98.66%
    Forma y color:Solid
    Peso molecular:310.39
  • S-trityl-L-Cysteine

    CAS:
    <p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>
    Fórmula:C22H21NO2S
    Pureza:97.02%
    Forma y color:Almost White To Light Yellow Granular Powder
    Peso molecular:363.47
  • Pioglitazone potassium

    CAS:
    <p>Pioglitazone potassium is an oral PPARγ agonist with EC50 of 0.93 μM (human) and 0.99 μM (mouse), used in diabetes research.</p>
    Fórmula:C19H19KN2O3S
    Forma y color:Solid
    Peso molecular:394.53
  • Daphnetin

    CAS:
    <p>Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR (IC50: 7.67 μM), PKA (IC50: 9.33 μM),</p>
    Fórmula:C9H6O4
    Pureza:97.47% - 99.8%
    Forma y color:Solid
    Peso molecular:178.14
  • kauran-16,17-diol

    CAS:
    <p>Kauran-16,17-diol, a natural diterpenoid product, exhibits anti-tumoral and apoptosis-inducing activities by inhibiting NO production in LPS-induced RAW 264.7</p>
    Fórmula:C20H34O2
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:306.48
  • Mocetinostat

    CAS:
    <p>Mocetinostat (MG0103) is an orally available HDAC inhibitor with most potency for HDAC1 (IC50: 0.15 μM), 2- to 10- fold selectivity against HDAC2/3/11.</p>
    Fórmula:C23H20N6O
    Pureza:99% - 99.21%
    Forma y color:Solid
    Peso molecular:396.44
  • LRRK2-IN-1

    CAS:
    LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.
    Fórmula:C31H38N8O3
    Pureza:98% - 98.82%
    Forma y color:Solid
    Peso molecular:570.69
  • Atezolizumab

    CAS:
    <p>Atezolizumab is an antibody inhibitor, a humanized monoclonal antibody, IgG1, which targets PD-L1. Atezolizumab has antitumor effect. Cost-effective and quality-assured.</p>
    Pureza:95.10% - 99.3% (SEC-HPLC)
    Forma y color:Liquid
    Peso molecular:145 kDa
  • HO-3867

    CAS:
    HO-3867, an analog of curcumin, is a sspecific STAT3 inhibitor.
    Fórmula:C28H30F2N2O2
    Pureza:91.18% - 99.21%
    Forma y color:Solid
    Peso molecular:464.55
  • LCL161

    CAS:
    LCL161 is a SMAC mimetic, an IAP antagonist with oral activity that inhibits XIAP and cIAP1. LCL161 has potential antitumor activity. Cost-effective and quality-assured.
    Fórmula:C26H33FN4O3S
    Pureza:99.13% - 99.87%
    Forma y color:Solid
    Peso molecular:500.63
  • Rilmenidine Phosphate

    CAS:
    <p>Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.</p>
    Fórmula:C10H19N2O5P
    Pureza:99.87% - ≥95%
    Forma y color:Solid
    Peso molecular:278.24
  • Elesclomol

    CAS:
    <p>Elesclomol (STA-4783) is an oxidative stress inducer and a highly lipophilic copper ion carrier.</p>
    Fórmula:C19H20N4O2S2
    Pureza:97.17% - 99.51%
    Forma y color:Solid
    Peso molecular:400.52
  • SGI-1776

    CAS:
    <p>SGI-1776 (Pim-Kinase Inhibitor IX) has been used in trials studying the treatment of Prostate Cancer, Non-Hodgkins Lymphoma, and Relapsed/Refractory Leukemias.</p>
    Fórmula:C20H22F3N5O
    Pureza:99.3% - >99.99%
    Forma y color:Solid
    Peso molecular:405.42
  • L-Asparaginase

    CAS:
    <p>L-Asparaginase, an enzyme for acute lymphoblastic leukemia treatment, is administered via injection.</p>
    Fórmula:NA
    Pureza:97%
    Forma y color:Solid
    Peso molecular:N/A
  • Lobaplatin

    CAS:
    Lobaplatin (D-19466) (D-19466) is a diastereometric mixture of platinum(II) complexe.
    Fórmula:C9H18N2O3Pt
    Pureza:98.00%
    Forma y color:Solid
    Peso molecular:397.33
  • CCT128930 hydrochloride

    CAS:
    <p>CCT128930 hydrochloride: Potent AKT inhibitor (IC50=6 nM), 28x selective over PKA, 20x over p70S6K, induces cell cycle arrest &amp; DNA damage.</p>
    Fórmula:C18H21Cl2N5
    Pureza:98.55%
    Forma y color:Solid
    Peso molecular:378.3
  • Bufotalin

    CAS:
    <p>1. Bufotalin (Bufotaline)e is a kind of poisonous secretions of toads.</p>
    Fórmula:C26H36O6
    Pureza:99.45% - 99.91%
    Forma y color:White To Off-White Solid
    Peso molecular:444.56
  • GDC-0152

    CAS:
    <p>GDC-0152 is a potent inhibitor of IAPs.</p>
    Fórmula:C25H34N6O3S
    Pureza:97.18% - 99.32%
    Forma y color:Solid
    Peso molecular:498.64
  • Supinoxin

    CAS:
    <p>Supinoxin (RX-5902) is an oral anti-cancer drug targeting p68 RNA helicase, inducing apoptosis in TNBC cells (IC50: 10-20nM).</p>
    Fórmula:C22H24FN5O4
    Pureza:99.83% - 99.95%
    Forma y color:Solid
    Peso molecular:441.46
  • BX-912

    CAS:
    <p>BX-912 inhibits PDK1 with IC50 of 12 nM; over 10x more selective versus C-Kit, EGFR, PKA, PKC.</p>
    Fórmula:C20H23BrN8O
    Pureza:98.29% - 99.34%
    Forma y color:Solid
    Peso molecular:471.35
  • 8-​Prenylnaringenin

    CAS:
    <p>8-Prenylnaringenin is a phytoestrogen with high estrogenic activity,</p>
    Fórmula:C20H20O5
    Pureza:98.26% - 99.46%
    Forma y color:Solid
    Peso molecular:340.37