Apoptosis
Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.
Subcategorías de "Apoptosis"
- ASK(6 productos)
- BCL(11 productos)
- Caspasa(127 productos)
- FOXO1(3 productos)
- IAP(65 productos)
- Mdm2(12 productos)
- PD-1 / PD-L1(126 productos)
- PDK(9 productos)
- PERK(24 productos)
- Serina / treonina quinasa(15 productos)
- Survivin(13 productos)
- TNF(91 productos)
- c-RET(51 productos)
- p53(62 productos)
Mostrar 6 subcategorías más
Se han encontrado 5622 productos de "Apoptosis"
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Nodinitib-1
CAS:Nodinitib-1 (CID-1088438) is a potent and selective NOD1 inhibitor with an IC50 of 0.56 μM.Fórmula:C14H13N3O2SPureza:99.97% - >99.99%Forma y color:SolidPeso molecular:287.34Zinc Protoporphyrin
CAS:<p>Zinc Protoporphyrin is an oral HO-1 inhibitor that reduces PG's protection against H2O2 and has anti-cancer properties.</p>Fórmula:C34H32N4O4ZnPureza:95.43% - 99.27%Forma y color:SolidPeso molecular:626.02JQ-1 (carboxylic acid)
CAS:<p>JQ-1 (carboxylic acid) is a cell-permeable BRD4 inhibitor with IC50s of 77 nM for BRD4(1) and 33 nM for BRD4(2)</p>Fórmula:C19H17ClN4O2SPureza:99.14% - 99.9%Forma y color:SolidPeso molecular:400.88PCI-34051
CAS:<p>PCI-34051 is an effective and selective HDAC8 inhibitor (IC50: 10 nM).</p>Fórmula:C17H16N2O3Pureza:97.219% - 98.29%Forma y color:SolidPeso molecular:296.32GW 5074
CAS:<p>GW 5074 (Raf1 Kinase Inhibitor I)(IC50=9 nM) is an effective and specific c-Raf inhibitor.</p>Fórmula:C15H8Br2INO2Pureza:99.32%Forma y color:SolidPeso molecular:520.94ML311
CAS:<p>ML311 is a selective inhibitor of the Mcl-1/Bim interaction.</p>Fórmula:C23H24F3N3OPureza:99.75%Forma y color:SolidPeso molecular:415.45A-1155463
CAS:<p>A-1155463, a highly potent and selective BCL-XL inhibitor, shows picomolar binding affinity to BCL-XL, and >1000-fold weaker binding to BCL-2, BCL-W and MCL-1.</p>Fórmula:C35H32FN5O4S2Pureza:96.1% - 99%Forma y color:SolidPeso molecular:669.79PI-1840
CAS:<p>PI-1840 is a reversible and selective chymotrypsin-like (CT-L) inhibitor, with little proteasome proteolytic effects on trypsin-like (T-L) and PGPH-L.</p>Fórmula:C22H26N4O3Pureza:98.82%Forma y color:SolidPeso molecular:394.47(E)-Flavokawain A
CAS:(E)-Flavokawain A, a novel chalcone from kava extract, induces apoptosis by involvement of Bax protein-dependent and mitochondria-dependent apoptotic pathway.Fórmula:C18H18O5Pureza:98% - 99.75%Forma y color:SolidPeso molecular:314.33Lenalidomide hemihydrate
CAS:<p>Lenalidomide hemihydrate inhibits TNF-α (IC50=13nM) and binds CRBN/DDB1 complexes.</p>Fórmula:C13H13N3O3H2OPureza:96.22%Forma y color:SolidPeso molecular:268.28ERK1/2 inhibitor 2
CAS:<p>ERK1/2 inhibitor 2 (ASTX029) is a selective and orally bioavailable ERK 1/2 inhibitor, with potential antineoplastic activity.</p>Fórmula:C29H31ClFN5O5Pureza:98.99%Forma y color:SolidPeso molecular:584.04Isolongifolene
CAS:<p>Isolongifolene ((-)-Isolongifolene), a tricyclic sesquiterpene isolated from Murraya koenigii, exhibits antioxidant, anti-inflammatory, anticancer, and</p>Fórmula:C15H24Pureza:90.13% - 99.46%Forma y color:Colorless Or Light Yellow LiquidPeso molecular:204.35Quinocetone
CAS:<p>Quinocetone is an animal growth promoter and potential anti-tumor activity.</p>Fórmula:C18H14N2O3Pureza:98.06%Forma y color:SolidPeso molecular:306.32CM-272
CAS:CM-272 is a dual G9a/DNA methyltransferases (DNMTs) inhibitor.Fórmula:C28H38N4O3Pureza:97.83%Forma y color:SolidPeso molecular:478.63Cynaroside
CAS:<p>Cynaroside (Luteolin 7-O-Glucoside) is a flavone, a flavonoid-like chemical compound. It has an anti-oxidant effect, inhibiting lipid and protein oxidation.</p>Fórmula:C21H20O11Pureza:98% - >99.99%Forma y color:SolidPeso molecular:448.38PF-4989216
CAS:PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.Fórmula:C18H13FN6OSPureza:99.85%Forma y color:SolidPeso molecular:380.4Clodronate disodium tetrahydrate
CAS:<p>Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.</p>Fórmula:CH10Cl2Na2O10P2Pureza:98%Forma y color:SolidPeso molecular:360.92MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Forma y color:SolidPeso molecular:470.512'-OMe-Guanosine
CAS:<p>2'-OMe-Guanosine is a modified nucleoside produced by the action of tRNA guanosine-2'-o-methyltransferase. 2'-OMe-Guanosine has a certain pro-apoptotic effect.</p>Fórmula:C11H15N5O5Pureza:99.93%Forma y color:White SolidPeso molecular:297.27Isoliensinine
CAS:<p>Isoliensinine (Isoliensinin) is a natural product, a bisbenzylisoquinoline alkaloid. Isoliensinine has antitumor and antioxidant effects. Cost effective and quality assured.</p>Fórmula:C37H42N2O6Pureza:98.53% - 99.79%Forma y color:SolidPeso molecular:610.74PI-103
CAS:<p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>Fórmula:C19H16N4O3Pureza:97.79% - 99.3%Forma y color:SolidPeso molecular:348.36OSI-930
CAS:<p>OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.</p>Fórmula:C22H16F3N3O2SPureza:99.67%Forma y color:SolidPeso molecular:443.44Tauroursodeoxycholate
CAS:<p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>Fórmula:C26H45NO6SPureza:98.77% - 99.93%Forma y color:White SolidPeso molecular:499.7Larotrectinib sulfate
CAS:<p>Larotrectinib sulfate (LOXO-101 sulfate) is an oral active and specific ATP-competitive inhibitor of tropomyosin receptor kinases (TRK).</p>Fórmula:C21H22F2N6O2·H2O4SPureza:98.62% - 99.76%Forma y color:SolidPeso molecular:526.51Psoralen
CAS:<p>Psoralen (Ficusin) is a furocoumarin that intercalates with DNA, inhibiting DNA synthesis and cell division.</p>Fórmula:C11H6O3Pureza:99.3% - 99.87%Forma y color:Crystals From Ether Crystalline SolidPeso molecular:186.16BI-6C9
CAS:<p>BI-6C9 is an inhibitor of tBid (Kd = 20 μM).BI-6c9 prevented MOMP and mitochondrial fission, and protected the cells from cell death.</p>Fórmula:C23H25N3O4S2Pureza:98.39%Forma y color:SolidPeso molecular:471.59TVB-3166
CAS:<p>TVB-3166: reversible, selective FASN inhibitor, induces apoptosis, hinders xenograft growth (IC50: 42 nM FASN, 81 nM palmitate synthesis).</p>Fórmula:C24H24N4OPureza:99.53% - 99.57%Forma y color:SolidPeso molecular:384.47A-1331852
CAS:<p>A-1331852 is a potent and selectiveBCL-XL inhibitor and may be useful in the treatment of cancer, immune and autoimmune diseases.</p>Fórmula:C38H38N6O3SPureza:98.15% - >99.99%Forma y color:SolidPeso molecular:658.81Alogliptin Benzoate
CAS:<p>Alogliptin Benzoate, a potent DPP-4 inhibitor with >10,000-fold selectivity over DPP-8/9, may also curb TLR-4-induced inflammation.</p>Fórmula:C25H27N5O4Pureza:99.94% - >99.99%Forma y color:White PowderPeso molecular:461.51HA14-1
CAS:<p>HA14-1, a Bcl-2/Bcl-XL antagonist, is a non-peptidic ligand of a Bcl-2 surface pocket (IC50: ~9 μM).</p>Fórmula:C17H17BrN2O5Pureza:95.07% - 98%Forma y color:SolidPeso molecular:409.23Isobutylparaben
CAS:<p>Isobutylparaben is a preservative and preservative insecticide.</p>Fórmula:C11H14O3Pureza:99.36%Forma y color:White CreamPeso molecular:194.233-hydroxy-3-phenylpentanamide
CAS:<p>Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.</p>Fórmula:C11H15NO2Pureza:98.42%Forma y color:SolidPeso molecular:193.24Sepantronium bromide
CAS:<p>Sepantronium bromide (YM155) is a small-molecule proapoptotic agent with potential antineoplastic activity.</p>Fórmula:C20H19BrN4O3Pureza:99.68% - 99.85%Forma y color:SolidPeso molecular:443.26Sirtinol
CAS:Sirtinol is a selective SIRT1/2 inhibitor (IC50: 131/38 μM).Fórmula:C26H22N2O2Pureza:97.12% - 99.96%Forma y color:SolidPeso molecular:394.47Etretinate
CAS:<p>Etretinate (Ro 10-9359), an oral retinoid, treats psoriasis by promoting cell differentiation and reducing cell growth and inflammation.</p>Fórmula:C23H30O3Pureza:97.89%Forma y color:Crystals Crystalline SolidPeso molecular:354.48Afatinib Dimaleate
CAS:<p>Afatinib Dimaleate (BIBW 2992MA2) is an orally bioavailable anilino-quinazoline derivative and inhibitor of the EGFR family, with antineoplastic activity.</p>Fórmula:C32H33ClFN5O11Pureza:98.11% - 99.87%Forma y color:SolidPeso molecular:718.08Prosapogenin A
CAS:<p>Prosapogenin A (Progenin III) has anticancer activity.</p>Fórmula:C39H62O12Pureza:99.60% - 99.75%Forma y color:SolidPeso molecular:722.9SKI-178
CAS:<p>SKI-178 is a sphingosine kinase 1 (SphK1) inhibitor with IC50 of 0.1-1.8 μM.</p>Fórmula:C21H22N4O4Pureza:97.09%Forma y color:SolidPeso molecular:394.42Embelin
CAS:<p>Embelin (Embelic acid), isolated from the Japanese Ardisia herb, is an inhibitor of the X-linked inhibitor of apoptosis (IC50: 4.1 uM).</p>Fórmula:C17H26O4Pureza:97.07% - 99.88%Forma y color:SolidPeso molecular:294.39GW779439X
CAS:GW779439X is an inhibitor of CDK.Fórmula:C22H21F3N8Pureza:97.87%Forma y color:SolidPeso molecular:454.45Sacubitril/Valsartan
CAS:<p>Sacubitril/Valsartan (LCZ696) is an orally bioavailable, dual angiotensin II receptor and neprilysin inhibitor for treatment of hypertension and heart failure.</p>Fórmula:C48H55N6O8Na3·5H2OPureza:99.75% - >99.99%Forma y color:SolidPeso molecular:957.99HX 531
CAS:<p>HX 531 is a RXR antagonist (IC50 of 18 nM).Cost-effective and quality-assured.</p>Fórmula:C29H29N3O4Pureza:98.59% - 99.86%Forma y color:SolidPeso molecular:483.56PP121
CAS:<p>PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.</p>Fórmula:C17H17N7Pureza:98.45% - 99.67%Forma y color:SolidPeso molecular:319.36GSK 3 Inhibitor IX
CAS:<p>GSK 3 Inhibitor IX (6-BIO) is a selective reversible, ATP-competitive inhibitor of GSK-3α/β and CDK1-cyclinB complex.</p>Fórmula:C16H10BrN3O2Pureza:98% - 99.72%Forma y color:SolidPeso molecular:356.17SZL P1-41
CAS:<p>SZL P1-41 inhibits Skp2, blocks complex formation, and halts ubiquitination, promoting cell senescence, reducing glycolysis, and exhibiting antitumor effects.</p>Fórmula:C24H24N2O3SPureza:99.60% - 99.87%Forma y color:SolidPeso molecular:420.52Niraparib tosylate monohyrate
CAS:Niraparib (MK-4827), a PARP inhibitor, boosts DNA breaks to trigger genomic instability and apoptosis, offering anti-cancer effects.Fórmula:C26H30N4O5SPureza:97.7% - 99.99%Forma y color:SolidPeso molecular:510.61Fimasartan
CAS:<p>Fimasartan (BR-A-657), an ARB, treats hypertension and heart failure; safe with hydrochlorothiazide.</p>Fórmula:C27H31N7OSPureza:98.96%Forma y color:SolidPeso molecular:501.65DC661
CAS:<p>DC661 is a palmitoyl-protein thioesterase 1 (PPT1) inhibitor that acts as an anti-lysosomal agent by inhibiting autophagy, demonstrating anti-cancer activity.</p>Fórmula:C31H39Cl2N5Pureza:99.07%Forma y color:SolidPeso molecular:552.58MG 149
CAS:<p>MG 149 (Tip60 HAT inhibitor) is a selective and potent Tip60 inhibitor with IC50 of 74 uM, similar potentcy for MOF(IC50= 47 uM).</p>Fórmula:C22H28O3Pureza:98.69% - 99.86%Forma y color:SolidPeso molecular:340.46MSC 2032964A
CAS:<p>MSC 2032964A: Potent, selective ASK1 inhibitor, IC50=93 nM, oral, brain-permeable, curbs neuroinflammation, blocks LPS-induced ASK1/p38 activation.</p>Fórmula:C16H13F3N6OPureza:99.76%Forma y color:SolidPeso molecular:362.31CHS-828
CAS:<p>CHS-828 (GMX1778), a pyridyl cyanoguanidine, is an effective inhibitor of NAD+ biosynthesis enzyme NAMPT (IC50 <25 nM).</p>Fórmula:C19H22ClN5OPureza:98% - 99.9%Forma y color:SolidPeso molecular:371.86Rigosertib
CAS:<p>Rigosertib, a multi-kinase inhibitor targeting PLK1 (IC50: 9 nM), induces apoptosis and G2/M arrest by disrupting PI3K/Akt.</p>Fórmula:C21H25NO8SPureza:99.53%Forma y color:SolidPeso molecular:451.49ABT-737
CAS:<p>ABT-737 is a BH3 mimetic and an inhibitor of Bcl-2, Bcl-xL, and Bcl-w. ABT-737 exhibits antitumor activity and anti-aging activity. Cost-effective and quality-assured.</p>Fórmula:C42H45ClN6O5S2Pureza:98.15% - >99.99%Forma y color:SolidPeso molecular:813.43BAY 87-2243
CAS:BAY 87-2243 is a potent and selective inhibitor of hypoxia-inducible factor-1 (HIF-1).Fórmula:C26H26F3N7O2Pureza:98% - 99.95%Forma y color:SolidPeso molecular:525.53Sodium benzoate
CAS:<p>Sodium benzoate (Benzoic acid sodium salt) is a D-Amino Acid Oxidase Inhibitor.Sodium Benzoate is a Food Preservative.</p>Fórmula:C7H5NaO2Pureza:99.72%Forma y color:White Solid CrystallinePeso molecular:144.10LW6
CAS:LW6 (HIF-1α inhibitor) is a novel HIF-1 inhibitor.Fórmula:C26H29NO5Pureza:98.1% - 98.22%Forma y color:SolidPeso molecular:435.51Clodronic acid disodium salt
CAS:<p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>Fórmula:CH4Cl2O6P0·2NaPureza:>99.99% - ≥98%Forma y color:White SolidPeso molecular:288.86BAY 61-3606
CAS:<p>BAY 61-3606 (Syk inhibitor IV) is a potent, ATP-competitive, reversible, and highly selective inhibitor of Syk tyrosine kinase activity (Ki= 7.5 nM), exhibiting</p>Fórmula:C20H18N6O3Pureza:98.72%Forma y color:SolidPeso molecular:390.4Atractylenolide III
CAS:<p>Atractylenolide III could treat cognitive issues and lung cancer by modulating apoptosis factors.</p>Fórmula:C15H20O3Pureza:99.53% - 99.82%Forma y color:SolidPeso molecular:248.32Amentoflavone
CAS:<p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>Fórmula:C30H18O10Pureza:98.21% - 99.22%Forma y color:Odourless Whitish SolidPeso molecular:538.46Wogonin
CAS:<p>Wogonin (Vogonin) is a cell-permeable and orally available flavonoid that displays anti-inflammatory and anticancer properties.</p>Fórmula:C16H12O5Pureza:98% - 99.8%Forma y color:Yellow CrystalPeso molecular:284.26Formosanin C
CAS:<p>Formosanin C (Polyphyllin B) is a compound isolated from Rhizoma Paridis, showed pro-apoptosis and immunoregulation with antitumor activity.</p>Fórmula:C51H82O20Pureza:99.75% - >99.99%Forma y color:SolidPeso molecular:1015.18WYC-209
CAS:<p>WYC-209 inhibits proliferation of malignant murine melanoma tumor-repopulating cells (TRCs, IC50: 0.19 uM). It targets the retinoic acid receptor (RAR).</p>Fórmula:C20H20N2O3SPureza:99.77%Forma y color:SolidPeso molecular:368.45Cyasterone
CAS:<p>Cyasterone (Cyasteron), a natural EGFR inhibitor, can inhibit the growth of A549 and MGC823 cells, via regulating EGFR signaling pathway, it may be a promising</p>Fórmula:C29H44O8Pureza:99.32% - 99.70%Forma y color:SolidPeso molecular:520.65Garcinol
CAS:<p>Garcinol: inhibits HATs/PCAF (IC50=7/5 μM), anti-inflammatory, anti-cancer, anti-cholinesterase (AChE IC50=0.66 μM, BChE IC50=7.39 μM).</p>Fórmula:C38H50O6Pureza:98.59%Forma y color:SolidPeso molecular:602.8Temsirolimus
CAS:<p>Temsirolimus (CCI-779) is a specific mTOR inhibitor ( IC50: 1.76 μM), used in the treatment of advanced renal cell cancer.</p>Fórmula:C56H87NO16Pureza:97.76% - >99.99%Forma y color:White Crystalline PowderPeso molecular:1030.29Calcimycin
CAS:<p>Calcimycin (A-23187) is a polyether antibiotic that transports Ca²⁺, uncouples phosphorylation, and inhibits ATPase in mitochondria.</p>Fórmula:C29H37N3O6Pureza:98%Forma y color:SolidPeso molecular:523.62Licochalcone D
CAS:<p>Licochalcone D may treat melanoma and heart injury, halt cell spread, and reduce inflammation and allergies.</p>Fórmula:C21H22O5Pureza:99.03% - 99.9%Forma y color:SolidPeso molecular:354.4Nitidine chloride
CAS:1.Fórmula:C21H18ClNO4Pureza:96.59% - 99.55%Forma y color:SolidPeso molecular:383.82MAZ51
CAS:MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.Fórmula:C21H18N2OPureza:98.53%Forma y color:SolidPeso molecular:314.38MPI-0479605
CAS:<p>MPI-0479605 is an ATP competitive and selective inhibitor.</p>Fórmula:C22H29N7OPureza:97.59% - >99.99%Forma y color:SolidPeso molecular:407.51(-)-Alkannin
CAS:<p>(-)-Alkannin (Shikonin) is a natural red naphthoquinone pigment, has antimicrobial, anti-tumor, and anti-inflammatory effects.</p>Fórmula:C16H16O5Pureza:98.18% - 98.8%Forma y color:White Or Slightly Yellow Crystalline Powder SolidPeso molecular:288.3TCS-PIM-1-4a
CAS:<p>SMI-4a, a Pim inhibitor, activates AMPK, halts mTORC1, and kills various myeloid/lymphoid cells (IC50=0.8-40μM).</p>Fórmula:C11H6F3NO2SPureza:99.89%Forma y color:SolidPeso molecular:273.23Dihydrorotenone
CAS:Dihydrorotenone is a potent mitochondrial inhibitor and probably induces Parkinsonian syndrome.Fórmula:C23H24O6Pureza:98.98% - 99.58%Forma y color:SolidPeso molecular:396.43C646
CAS:<p>C646, a histone acetyltransferase inhibitor, inhibits p300 (Ki: 400 nM, in a cell-free assay).</p>Fórmula:C24H19N3O6Pureza:98% - 99.21%Forma y color:SolidPeso molecular:445.42KW-2449
CAS:<p>KW-2449 is a multiple-targeted inhibitor, mostly for Flt3, modestly effective to Bcr-Abl, FGFR1, and Aurora A; little inhibitory on PDGFRβ, IGF-1R, EGFR.</p>Fórmula:C20H20N4OPureza:98.43% - 99.69%Forma y color:SolidPeso molecular:332.4Quisinostat
CAS:Quisinostat (JNJ-26481585), a second-gen HDAC inhibitor, is most potent for HDAC1 (IC50 0.11 nM) and selectively affects HDACs 2, 4, 10, and 11.Fórmula:C21H26N6O2Pureza:96.01% - ≥98%Forma y color:SolidPeso molecular:394.47α-Hederin
CAS:<p>Alpha-Hederin (Tauroside E) is a water-soluble pentacyclic triterpenoid saponin found in the seeds of Nigella sativa, with hemolytic and apoptotic properties.</p>Fórmula:C41H66O12Pureza:99.44% - 99.89%Forma y color:SolidPeso molecular:750.96Nafamostat mesylate
CAS:<p>Nafamostat mesylate (FUT-175), a synthetic serine protease inhibitor, has been used for the treatment of allergic disorders such as asthma, allergic rhinitis</p>Fórmula:C19H17N5O2·2CH4O3SPureza:97.36% - 99.76%Forma y color:Tan To Pale Orange SolidPeso molecular:539.58AKT inhibitor VIII
CAS:<p>AKT inhibitor VIII (AKTi-1/2) is a highly specific Akt1/2 inhibitor (IC50: 58/210 nM). The selectivity for Akt1 is higher about 36-fold than Akt3.</p>Fórmula:C34H29N7OPureza:98.31% - 98.65%Forma y color:Pale Yellow SolidPeso molecular:551.64BMS-536924
CAS:<p>BMS-536924 (BMS 536924) is an ATP-competitive IGF-1R/IR inhibitor with IC50 of 100 nM/73 nM, modest activity for Mek, Fak, and Lck with very little activity for</p>Fórmula:C25H26ClN5O3Pureza:99.02%Forma y color:SolidPeso molecular:479.96Teneligliptin hydrobromide
CAS:<p>Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.</p>Fórmula:C22H30N6OSBrHPureza:97.83% - 99.92%Forma y color:SolidPeso molecular:628.86Flurbiprofen Axetil
CAS:<p>Flurbiprofen Axetil (Lipfen) is an anti-inflammatory used as an analgesic.</p>Fórmula:C19H19FO4Pureza:97.58% - 98%Forma y color:SolidPeso molecular:330.359-Methoxycamptothecin
CAS:9-Methoxycamptothecin (MCPT) has antitumour activities through topoisomerase inhibition.Fórmula:C21H18N2O5Pureza:98.49% - 99.56%Forma y color:SolidPeso molecular:378.38Sodium taurodeoxycholate hydrate
CAS:<p>Sodium taurodeoxycholate hydrate (Taurodeoxycholic acid sodium salt monohydrate) has been used in a study to assess the effect of submicellar concentrations of</p>Fórmula:C26H44NO6S·Na·H2OPureza:99.78%Forma y color:SolidPeso molecular:539.7NSC 73150
CAS:<p>6-Methyl-1H-pyrimidin-4-one (NSC 73150) shows antitumor effects, impeding growth in breast, lung, liver cancer, and inducing apoptosis.</p>Fórmula:C12H12N4O2Pureza:99.84%Forma y color:SolidPeso molecular:244.25Etidronic acid
CAS:<p>Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.</p>Fórmula:C2H8O7P2Pureza:99.93% - ≥95%Forma y color:Liquid SyrupPeso molecular:206.03RH01687
CAS:<p>RH01687 is a potent β-cell protector , exhibits β-cell-protective activities against endoplasmic reticulum (ER) stress.</p>Fórmula:C12H9ClN6O2SPureza:97.93%Forma y color:SolidPeso molecular:336.76Ispinesib
CAS:<p>Ispinesib (SB-715992), a selective, effectvie and reversible inhibitor of kinesin spindle protein (KSP), is derived from quinazolinone, with antineoplastic</p>Fórmula:C30H33ClN4O2Pureza:98% - 99.09%Forma y color:SolidPeso molecular:517.06BMS-833923
CAS:<p>BMS-833923 (XL-139), an orally bioavailable Smoothened antagonist, inhibits BODIPY cyclopamine binding to SMO in a dose-dependent manner (IC50: 21 nM).</p>Fórmula:C30H27N5OPureza:99.47% - 99.76%Forma y color:SolidPeso molecular:473.574E1rcat
CAS:<p>4E1RCat is a dual inhibitor of eIF4E:eIF4 g and eIF4E:4E-BP1 interaction. And it inhibits the binding of eIF4 g to eIF4E with IC50 of 3.2 μM.</p>Fórmula:C28H18N2O6Pureza:99.47%Forma y color:SolidPeso molecular:478.454-MMPB
CAS:<p>15-Lipoxygenase Inhibitor 1 is a selective inhibitor of 15-lipoxygenase, with an IC50 of 18 μM.</p>Fórmula:C16H19N5SPureza:97.18%Forma y color:SolidPeso molecular:313.42β-Lapachone
CAS:<p>β-Lapachone (ARQ-501) is a specific DNA topoisomerase I inhibitor, and no inhibitory activities against DNA topoisomerase II or ligase.</p>Fórmula:C15H14O3Pureza:99.76% - 99.88%Forma y color:SolidPeso molecular:242.27MX69
CAS:<p>MX69 is the MDM2/XIAP inhibitor, blocking the MDM2 protein-XIAP RNA interaction, leading to MDM2 degradation.</p>Fórmula:C27H26N2O4SPureza:97.27% - 99.57%Forma y color:SolidPeso molecular:474.57Macitentan
CAS:<p>Macitentan (ACT-064992) is an endothelin receptor antagonist that is used in the therapy of pulmonary arterial hypertension (PAH).</p>Fórmula:C19H20Br2N6O4SPureza:98% - >99.99%Forma y color:SolidPeso molecular:588.27Bay 11-7085
CAS:<p>Bay 11-7085 can irreversibly inhibit the IκBα phosphorylation induced by TNFα (IC50: 10 μM).</p>Fórmula:C13H15NO2SPureza:99.76% - 99.94%Forma y color:White SolidPeso molecular:249.33Lubiprostone
CAS:<p>Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.</p>Fórmula:C20H32F2O5Pureza:97.31% - 98.54%Forma y color:White Odorless Crystals Or Crystalline PowderPeso molecular:390.46Dinaciclib
CAS:<p>Dinaciclib (SCH 727965) is a CDK inhibitor that selectively inhibits CDK1, CDK2, CDK5, and CDK9 (IC50 = 3/1/1/4 nM).</p>Fórmula:C21H28N6O2Pureza:98.21% - 99.75%Forma y color:SolidPeso molecular:396.49Genistein
CAS:<p>Genistein (NPI 031L) is a natural soy isoflavone, a multi-targeted tyrosine kinase inhibitor. Genistein has antitumor effects. Cost effective and quality assured.</p>Fórmula:C15H10O5Pureza:98.22% - 99.64%Forma y color:Rectangular Or Six-Sided Rods From 60% Alcohol Dendritic Needles From Ether SolidPeso molecular:270.24(1E,6E)-Bis(demethoxy)curcumin
CAS:<p>(1E,6E)-Bis(demethoxy)curcumin (Curcumin III) is a natural demethoxy derivative of curcumin,with anti-inflammatory and anti-cancer activities.</p>Fórmula:C19H16O4Pureza:97.45%Forma y color:SolidPeso molecular:308.33UNC1215
CAS:<p>UNC1215, a potent MBT antagonist, targets L3MBTL3 with high selectivity (IC50: 40 nM, Kd: 120 nM, 50x versus MBT family).</p>Fórmula:C32H43N5O2Pureza:98% - 99.04%Forma y color:SolidPeso molecular:529.72H-Gly-Arg-Gly-Asp-Asn-Pro-OH
CAS:<p>RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.</p>Fórmula:C23H38N10O10Pureza:>99.99%Forma y color:SolidPeso molecular:614.61Astragalin
CAS:<p>Astragalin (Kaempferol 3-O-glucoside) is a biologically active natural flavonoid.</p>Fórmula:C21H20O11Pureza:98.8% - ≥95%Forma y color:SolidPeso molecular:448.38Spautin-1
CAS:Spautin-1 is an autophagy inhibitor that can suppress the deubiquitination activity of ubiquitin-specific peptidase USP10 and USP13. Cost-effective and quality-assured.Fórmula:C15H11F2N3Pureza:97.69% - 98.99%Forma y color:SolidPeso molecular:271.26AES-350
CAS:<p>AES-350, an HDAC6 inhibitor (IC50: 0.0244 μM), also targets HDAC-3, -8, -11, induces AML cell apoptosis, and aids AML research.</p>Fórmula:C18H20N2O3Pureza:98.82%Forma y color:SolidPeso molecular:312.36Tyrphostin AG 879
CAS:<p>Tyrphostin AG 879 (AG 879) effectively inhibits HER2/ErbB2 (IC50: 1 μM), 100- and 500-fold higher selective to ErbB2 than EGFR and PDGFR.</p>Fórmula:C18H24N2OSPureza:99.05%Forma y color:SolidPeso molecular:316.46BML-210
CAS:<p>BML-210 (CAY10433) is a new-type HDAC inhibitor.</p>Fórmula:C20H25N3O2Pureza:96.37% - 98.12%Forma y color:SolidPeso molecular:339.43Medicarpin
CAS:<p>Medicarpin, an ER agonist, stimulates osteoblasts, enhances peak bone mass, has no uterine effects, and is orally bioavailable.</p>Fórmula:C16H14O4Pureza:99.32% - 99.86%Forma y color:SolidPeso molecular:270.28Oleuropein
CAS:Oleuropein is an antioxidant polyphenol isolated from olive leaf.Fórmula:C25H32O13Pureza:98% - 99.95%Forma y color:Brown PowderPeso molecular:540.51Isobavachalcone
CAS:<p>Isobavachalcone (Corylifolinin) is a chalcone constituent of Angelica keiskei, has potent anti-inflammatory activity, possible can ameliorate neuronal injury in</p>Fórmula:C20H20O4Pureza:98% - 99.76%Forma y color:SolidPeso molecular:324.37Phellamurin
CAS:<p>Phellamurin blocks intestinal P-glycoprotein dose-dependently and it seriously interacts with cyclosporin; coadministration should be avoided.</p>Fórmula:C26H30O11Pureza:97.91%Forma y color:SolidPeso molecular:518.51AZ 628
CAS:<p>AZ628 is a new pan-Raf inhibitor for BRAF, BRAFV600E, and c-Raf-1 with IC50 of 105 nM, 34 nM and 29 nM, also inhibits VEGFR2, DDR2, Lyn, Flt1, FMS, etc.</p>Fórmula:C27H25N5O2Pureza:99.50%Forma y color:SolidPeso molecular:451.52Pracinostat
CAS:<p>Pracinostat (SB939) is a novel HDAC inhibitor with improved in vivo properties compared to other HDAC inhibitors currently in Clinicalal trials, allowing oral</p>Fórmula:C20H30N4O2Pureza:99.15% - 99.67%Forma y color:SolidPeso molecular:358.48Apremilast
CAS:Apremilast (CC-10004) (CC-10004) is a potent and orally active PDE4 (IC50=74 nM) with anti-inflammation activities.Fórmula:C22H24N2O7SPureza:98.13% - 99.95%Forma y color:SolidPeso molecular:460.50FLLL32
CAS:<p>FLLL32 is an effective JAK2/STAT3 inhibitor (IC50 of <5 μM).</p>Fórmula:C28H32O6Pureza:97% - 97.90%Forma y color:SolidPeso molecular:464.55Palmatine chloride
CAS:<p>Palmatine chloride an isoquinoline alkaloid, is an important medicinal herbal extract with diverse pharmacological and biological properties.</p>Fórmula:C21H22ClNO4Pureza:97.9% - 99.47%Forma y color:SolidPeso molecular:387.8572-Hydroxychalcone
CAS:<p>2-Hydroxychalcone (2-(2-Hydroxybenzal)Acetophenone) can be used as antiparasitic hit compounds when Methoxylated. It inhibits invasion of breast cancer cells.</p>Fórmula:C15H12O2Pureza:99.6%Forma y color:SolidPeso molecular:224.25RITA
CAS:<p>RITA (NSC-652287) forms DNA-DNA/protein cross-links without DNA breaks; disrupts p53/Mdm2 like nutlin-3.</p>Fórmula:C14H12O3S2Pureza:98.49% - 99.55%Forma y color:SolidPeso molecular:292.37Bortezomib
CAS:<p>Bortezomib (LDP 341) is a 20S proteasome inhibitor (Ki=0.6 nM) that is reversible and selective.</p>Fórmula:C19H25BN4O4Pureza:97.79% - >99.99%Forma y color:Yellow SolidPeso molecular:384.24Danshensu
CAS:<p>Danshensu (Dan shen suan A) is an active ingredient of Salvia miltiorrhiza with wide cardiovascular benefit.</p>Fórmula:C9H10O5Pureza:98.4% - 99.74%Forma y color:SolidPeso molecular:198.17Ketorolac
CAS:<p>Ketorolac (Acuvail) is an NSAID that blocks prostaglandin synthesis, related to heterocyclic acetic acids.</p>Fórmula:C15H13NO3Pureza:99.68%Forma y color:White Crystalline Or White PowderPeso molecular:255.27TPCA-1
CAS:<p>TPCA-1 (TPCA1) is an effective and specific IKK-2 inhibitor (IC50: 17.9 nM); shows >22-fold selectivity over IKK-1 and >550-fold selectivity over others kinases</p>Fórmula:C12H10FN3O2SPureza:95.03% - 97.86%Forma y color:SolidPeso molecular:279.29ML162
CAS:ML162 is a covalent glutathione peroxidase 4 (GPX4) inhibitor that induces ferroptosis. ML162 has antitumor activity. Cost-effective and quality-assured.Fórmula:C23H22Cl2N2O3SPureza:98.42% - 99.55%Forma y color:SolidPeso molecular:477.4Poziotinib
CAS:<p>Poziotinib (NOV120101)(NOV120101; HM781-36B) is an irreversible HER1/2/4 inhibitor (IC50s: 3/5/23 nM).</p>Fórmula:C23H21Cl2FN4O3Pureza:98.69% - 99.78%Forma y color:SolidPeso molecular:491.34Kumatakenin
CAS:<p>Kumatakenin can suppress >80% of the SOS-inducing activity of Trp-P-1 at <0.06 micromol/mL.</p>Fórmula:C17H14O6Pureza:97.44% - 98.29%Forma y color:SolidPeso molecular:314.29BG45
CAS:<p>BG45 is an HDAC I type inhibitor with IC50 of 289 nM, 2.0 μM, 2.2 μM and >20 μM for HDAC3/1/2/6 in cell-free assays, respectively.</p>Fórmula:C11H10N4OPureza:99.77%Forma y color:SolidPeso molecular:214.22SGI-1027
CAS:<p>SGI-1027 (DNA Methyltransferase Inhibitor II) is an effective and selective inhibitor of DNA methyltransferase (DNMT).</p>Fórmula:C27H23N7OPureza:99.45% - 99.78%Forma y color:SolidPeso molecular:461.52GMB-475
CAS:<p>GMB-475, a PROTAC-based BCR-ABL1 inhibitor, tackles drug resistance by promoting VHL-mediated degradation.</p>Fórmula:C43H46F3N7O7SPureza:98.78% - >99.99%Forma y color:SolidPeso molecular:861.93Benidipine hydrochloride
CAS:<p>Benidipine hydrochloride (Coniel) , a hydrochloride salt form of benidipine, is used as a blocker of dihydropyridine calcium channel.</p>Fórmula:C28H32ClN3O6Pureza:99.80%Forma y color:SolidPeso molecular:542.03AZD-8055
CAS:<p>AZD8055 is an ATP-competitive mTOR inhibitor (IC50: 0.8 nM in MDA-MB-468 cells). It is ~1,000-fold selective for mTOR over all PI3K isoforms.</p>Fórmula:C25H31N5O4Pureza:98% - 99.69%Forma y color:SolidPeso molecular:465.54NADPH tetracyclohexanamine
CAS:<p>NADPH tetracyclohexanamine (NADPH (tetracyclohexanamine)) is a cofactor and biological reducing agent.</p>Fórmula:C45H82N11O17P3Pureza:98.73% - 99.05%Forma y color:SolidPeso molecular:1142.12GSK3326595
CAS:<p>GSK3326595 (EPZ015938) is an inhibitor of protein arginine methyltransferase 5 (PRMT5)(IC50:6.2 nM.).</p>Fórmula:C24H32N6O3Pureza:97.7% - 99.63%Forma y color:SolidPeso molecular:452.55KY-05009
CAS:<p>KY-05009 blocks TGF-β1 EMT in lung cancer cells, inhibits TNIK, Wnt genes, induces apoptosis, and is an ATP-competitive TNIK inhibitor (Ki = 100 nM).</p>Fórmula:C18H16N4O2SPureza:99.89%Forma y color:SolidPeso molecular:352.41Arctigenin
CAS:<p>(-)-Arctigenin ((-)-Arctigenin) is found in burdock.</p>Fórmula:C21H24O6Pureza:98% - 99.51%Forma y color:SolidPeso molecular:372.41Onvansertib
CAS:Onvansertib (NMS-1286937) is a PLK1 inhibitor with high selectivity and oral activity. Onvansertib has antitumor activity. Cost-effective and quality-assured.Fórmula:C24H27F3N8O3Pureza:98.3% - 99.88%Forma y color:SolidPeso molecular:532.52Tofacitinib
CAS:<p>Tofacitinib (Tasocitinib) is an orally Janus kinase inhibitor. Tofacitinib is used for the treatment of rheumatoid arthritis. Cost effective and quality assured.</p>Fórmula:C16H20N6OPureza:99% - >99.99%Forma y color:SolidPeso molecular:312.37Ginsenoside Rh2
CAS:<p>Ginsenoside Rh2 (20(S)-Ginsenoside Rh2), an extract of red Panax ginseng, is a potent anti-inflammatory and anticancer drug.</p>Fórmula:C36H62O8Pureza:99.20% - 99.76%Forma y color:White PowderPeso molecular:622.87MPP dihydrochloride (289726-02-9 Free base)
CAS:<p>MPP dihydrochloride is a highly selective antagonist of estrogen receptor alpha (ERα).</p>Fórmula:C29H33Cl2N3O3Forma y color:SolidPeso molecular:542.5Siramesine hydrochloride
CAS:<p>Siramesine hydrochloride (Lu 28-179 hydrochloride) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of Y cells and to exhibit</p>Fórmula:C30H32ClFN2OPureza:99.72% - >99.99%Forma y color:SolidPeso molecular:491.04Piclidenoson
CAS:<p>Piclidenoson (CF-101), a selective agonist of adenosine A3 receptor(EC50 values of 0.11 μM), induces robust anti-inflammatory effect in psoriasis patients.</p>Fórmula:C18H19IN6O4Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:510.29CIL56
CAS:<p>CIL56 (CA3) is a small molecule that induces cellular ferroptosis through the production of iron-dependent reactive oxygen species (ROS).</p>Fórmula:C23H27N3O5S2Pureza:99.46% - 99.91%Forma y color:SolidPeso molecular:489.61SBI-0640756
CAS:SBI-0640756 (SBI-756) (SBI-756) is a first-in-class inhibitor that targets eIF4G1 and disrupts the eIF4F complex.Fórmula:C23H14ClFN2O2Pureza:99.75%Forma y color:SolidPeso molecular:404.82Oxychlororaphine
CAS:<p>Oxychlororaphine (phenazine-1-carboxamide) inhibits strongly the growth of Streptomyces sp. 441.</p>Fórmula:C13H9N3OPureza:98.3%Forma y color:Green-Yellow SolidPeso molecular:223.23Pitavastatin sodium
CAS:<p>Pitavastatin sodium inhibits HMG-CoA reductase, enhances LDL-C receptors, and has various protective effects.</p>Fórmula:C25H23FNNaO4Forma y color:SolidPeso molecular:443.45Avadomide
CAS:<p>Avadomide (CC 122) is an orally available pleiotropic pathway modulator with potential antineoplastic activity.</p>Fórmula:C14H14N4O3Pureza:99.56%Forma y color:SolidPeso molecular:286.29PHA-793887
CAS:<p>PHA-793887 has been used in trials studying the treatment of Advanced/Metastatic Solid Tumors.</p>Fórmula:C19H31N5O2Pureza:98.02% - >99.99%Forma y color:SolidPeso molecular:361.48L67
CAS:<p>L67 (DNA Ligase Inhibitor) is a competitive human DNA ligase inhibitor, inhibits DNA ligases I and III (IC50: 10 μM).</p>Fórmula:C16H14Br2N4O4Pureza:98.34% - 99.56%Forma y color:SolidPeso molecular:486.11ALSTERPAULLONE
CAS:Alsterpaullone is a Cyclin-Dependent Kinase Inhibitor, Mediated Toxicity in HeLa Cells Through Apoptosis-Inducing EffecFórmula:C16H11N3O3Pureza:99.8%Forma y color:SolidPeso molecular:293.28ENMD-1068 hydrochloride
CAS:<p>ENMD-1068 hydrochloride: selective PAR2 antagonist, counters liver fibrosis, hinders endometrial cell growth, and induces apoptosis in studies.</p>Fórmula:C15H30ClN3O2Forma y color:SolidPeso molecular:319.87D-Pantothenic acid sodium
CAS:D-Pantothenic acid sodium, a sodium salt of D-pantothenate, is a vital B5 derivative, aiding fat, carb, and amino acid oxidation.Fórmula:C9H16NNaO5Pureza:97.98%Forma y color:White PowderPeso molecular:241.22β-mangostin
CAS:β-Mangostin: a xanthone in Cratoxylum arborescens, fights bacteria, malaria, tuberculosis (MIC 6.25μg/mL), and cancer.Fórmula:C25H28O6Pureza:98.01% - 99.97%Forma y color:Faintly Yellow PowderPeso molecular:424.49Rhosin hydrochloride
CAS:<p>Rhosin hydrochloride is a specific inhibitor of the RhoA subfamily Rho GTPases.Cost-effective and quality-assured.</p>Fórmula:C20H20Cl2N6OPureza:97.33% - 98.92%Forma y color:SolidPeso molecular:431.318VR23
CAS:<p>VR23: Potent proteasome inhibitor; IC50: 1 nM trypsin, 50-100 nM chymotrypsin, 3 μM caspase-like.</p>Fórmula:C19H16ClN5O6SPureza:98.99% - 99.22%Forma y color:SolidPeso molecular:477.88EPI-001
CAS:<p>EPI-001 is an androgen receptor N-terminal domain antagonist with IC50 of ～6 μM and a selective PPAR-gamma modulator.</p>Fórmula:C21H27ClO5Pureza:99% - 99.67%Forma y color:SolidPeso molecular:394.897,8-Dihydroxyflavone
CAS:<p>7,8-Dihydroxyflavone (7,8-DHF) is a naturally-occurring flavone and exist in Tridax procumbens, Godmania aesculifolia, and primula tree leaves.</p>Fórmula:C15H10O4Pureza:98.48% - 99.81%Forma y color:SolidPeso molecular:254.241A-116
CAS:<p>1A-116 is a specific Rac1 inhibitor.</p>Fórmula:C16H16F3N3Pureza:99.71%Forma y color:SolidPeso molecular:307.31Capmatinib 2HCl
CAS:<p>Capmatinib 2HCl (INC-280 2HCl), a c-MET inhibitor, is potent (IC50 = 0.13 nM), highly specific, and induces apoptosis in tumor cells.</p>Fórmula:C23H19Cl2FN6OPureza:98.80%Forma y color:SolidPeso molecular:485.34INH6
CAS:<p>INH6, an effective Hec1 inhibitor, selectively disrupts the Hec1/Nek2 interaction and induces chromosome mis-alignment.</p>Fórmula:C19H18N2OSPureza:98.81%Forma y color:SolidPeso molecular:322.42Urolithin A
CAS:<p>Urolithin A is a metabolite of ellagic acid, which inhibits DNA synthesis and induces apoptosis and autophagy. Cost-effective and quality-assured.</p>Fórmula:C13H8O4Pureza:99.14% - 99.67%Forma y color:SolidPeso molecular:228.2Cannabigerol
CAS:Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; alsoFórmula:C21H32O2Pureza:99.59% - 99.92%Forma y color:SolidPeso molecular:316.48Trigonelline
CAS:<p>Trigonelline (Trigenolline), an alkaloid with potential antidiabetic activity, is present in considerable amounts in coffee.</p>Fórmula:C7H7NO2Pureza:97.585% - 99.49%Forma y color:Prisms Aqueous From Alcohol + Water SolidPeso molecular:137.14TT-232 TFA(147159-51-1 free base)
CAS:<p>TT2-32 TFA induces a biphasic activation of phosphotyrosine phosphatase activity in human colon tumor cell line, SW620</p>Fórmula:C47H59F3N10O11S2Pureza:99.27% - 99.8%Forma y color:SolidPeso molecular:1061.16(Z)-Mirin
CAS:<p>(Z)-Mirin is a potent Mre11–Rad50–Nbs1 (MRN) complex inhibitor, and inhibits Mre11-associated exonuclease activity.</p>Fórmula:C10H8N2O2SPureza:99.67% - 99.76%Forma y color:SolidPeso molecular:220.25Cidofovir dihydrate
CAS:<p>Cidofovir dihydrate: Injectable anti-CMV; suppresses CMV by inhibiting viral DNA polymerase; treats CMV retinitis in AIDS.</p>Fórmula:C8H18N3O8PPureza:99.44%Forma y color:SolidPeso molecular:315.22Phenazine methylsulfate
CAS:<p>Phenazine methylsulfate is anti-bacterial agents.</p>Fórmula:C14H14N2O4SPureza:97.67% - >99.99%Forma y color:Yellow CrystallinePeso molecular:306.34Tetramethylcurcumin
CAS:<p>Tetramethylcurcumin is a novel curcumin analog, is an effective inhibitors of STAT3 phosphorylation, DNA binding activity, and transactivation in vitro.it also</p>Fórmula:C25H28O6Pureza:97.69% - 99.94%Forma y color:SolidPeso molecular:424.49Dantrolene
CAS:Dantrolene is a postsynaptic muscle relaxant by inhibiting Ca2+ ions release from sarcoplasmic reticulum stores by antagonizing ryanodine receptors.Fórmula:C14H10N4O5Pureza:99.97%Forma y color:Crystals From Aq DimethylformamidePeso molecular:314.25Tauroursodeoxycholate sodium
CAS:<p>Tauroursodeoxycholate sodium (TUDC) is an endoplasmic reticulum (ER) stress inhibitor, used for the treatment of gallstones and liver cirrhosis.</p>Fórmula:C26H44NNaO6SPureza:97.90%Forma y color:SolidPeso molecular:521.69CRT0066101 dihydrochloride
CAS:<p>CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).</p>Fórmula:C18H22N6O·2HClPureza:99.85%Forma y color:SolidPeso molecular:411.33Cinobufagin
CAS:<p>Cinobufagin (Cinobufagine) is a selective Na+/K+-ATPase inhibitor. The activity of Cinobufagin is same as ouabain.</p>Fórmula:C26H34O6Pureza:97.77% - 99.97%Forma y color:SolidPeso molecular:442.54Onatasertib
CAS:<p>Onatasertib (CC223) is an orally available mTOR inhibitor with potential antitumor activity.</p>Fórmula:C21H27N5O3Pureza:99.14% - 99.97%Forma y color:SolidPeso molecular:397.47Euphorbia Factor L2
CAS:<p>Euphorbia Factor L2 alleviates lipopolysaccharide-induced acute lung injury and inflammation through inhibits NF-κB activation.</p>Fórmula:C38H42O9Pureza:99.53% - 99.96%Forma y color:SolidPeso molecular:642.73Talampanel
CAS:<p>Talampanel (LY-300164), an oral selective AMPA receptor antagonist, exhibits anti-seizure and neuroprotective properties.</p>Fórmula:C19H19N3O3Pureza:98.3%Forma y color:SolidPeso molecular:337.37NADPH tetrasodium salt
CAS:<p>NADPH tetrasodium salt is the reduced form of the electron acceptor nicotinamide adenine dinucleotide phosphate, which acts as an electron donor in a variety of</p>Fórmula:C21H26N7Na4O17P3Pureza:97.15% - >99.99%Forma y color:SolidPeso molecular:833.35Liproxstatin-1 hydrochloride
CAS:<p>Liproxstatin-1 hydrochloride is a high-potency ferroptosis inhibitor capable of effectively preventing ferroptotic cell death, with an IC50 value of 22 nM [1].</p>Fórmula:C19H22Cl2N4Forma y color:SolidPeso molecular:377.31Thalidomide-O-C6-NH2 hydrochloride
CAS:<p>Thalidomide-O-C6-NH2 hydrochloride (4-((6-aminohexyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione hydrochloride) is a synthesized E3 ligase ligand-</p>Fórmula:C19H24ClN3O5Pureza:97.45%Forma y color:SolidPeso molecular:409.86Omaveloxolone
CAS:<p>Omaveloxolone (RTA-408) (RTA-408) is a synthetic triterpenoid that activates the cytoprotective transcription factor Nrf2 and inhibits NF-κB signaling. Phase 2.</p>Fórmula:C33H44F2N2O3Pureza:98.7% - 99.92%Forma y color:SolidPeso molecular:554.71Cladribine
CAS:<p>Cladribine (2CdA), an adenosine deaminase inhibitor, is utilized in the treatment of lymphoproliferative diseases.</p>Fórmula:C10H12ClN5O3Pureza:99.58% - >99.99%Forma y color:White Crystalline SolidPeso molecular:285.69(ZE)-SU9516
CAS:<p>(ZE)-SU9516 is a selectively potent ATP-competitive inhibitor of CDKs.</p>Fórmula:C13H11N3O2Pureza:99.59%Forma y color:SolidPeso molecular:241.25Pyraclostrobin
CAS:Pyraclostrobin is one of the most heavily used fungicides that inhibits mitochondrial complex III of fungal and mammalian cells.Fórmula:C19H18ClN3O4Pureza:99.89%Forma y color:SolidPeso molecular:387.82TCS PrP Inhibitor 13
CAS:<p>TCS PrP Inhibitor 13 (5-(4-Nitrophenyl)-2-Phenyl-4H-Pyrazol-3-One) is an antiprion agent inhibiting protease-resistant prion protein (PrP-res) accumulation.</p>Fórmula:C15H11N3O3Pureza:99.7%Forma y color:SolidPeso molecular:281.27Azathioprine Sodium
CAS:<p>Azathioprine Sodium is a pro-drug converted to 6-MP, inhibiting DNA/RNA synthesis, curbing cell proliferation, especially in lymphocytes.</p>Fórmula:C9H6N7NaO2SForma y color:SolidPeso molecular:299.24β-Elemonic Acid
CAS:<p>β-Elemonic Acid (3-Oxotirucallenoic Acid) exhibits anti-inflammatory effects, which inhibits proliferation by inducing hypoploid cells and cell apoptosis.</p>Fórmula:C30H46O3Pureza:99.61% - 99.8%Forma y color:SolidPeso molecular:454.68PF-3758309
CAS:<p>PF-3758309 (PF-03758309) (IC50=1.3 nM), a pyrrolopyrazole inhibitor of PAK4, has effective ATP-competition.</p>Fórmula:C25H30N8OSPureza:97.70%Forma y color:SolidPeso molecular:490.62Imipramine hydrochloride
CAS:<p>Imipramine HCl: 1st-gen tricyclic antidepressant, inhibits serotonin and norepinephrine uptake, blocks aSMase, reduces MV/exosome secretion.</p>Fórmula:C19H25ClN2Pureza:99.65% - 99.98%Forma y color:White To Off-White /Hydrochloride/ Un 1230 3/Pg 2Peso molecular:316.87Vatalanib dihydrochloride
CAS:<p>Vatalanib dihydrochloride (PTK787 dihydrochloride)(IC50=37 nM) is an inhibitor of VEGFR2/KDR.</p>Fórmula:C20H15ClN4·2HClPureza:99.16%Forma y color:White To Off-White Crystalline PowderPeso molecular:419.73AZD5582 acetate (1258392-53-8 free base)
<p>AZD5582 acetate is an inhibitor of IAPs, which binds to the BIR3 domains cIAP1, cIAP2, and XIAP with IC50s of 15, 21, and 15 nM, respectively.</p>Fórmula:C60H82N8O10Pureza:97.76%Forma y color:SolidPeso molecular:1075.36Thalidomide-O-amido-C4-NH2 TFA
CAS:<p>Thalidomide-O-amido-C4-NH2 TFA (E3 ligase Ligand-Linker Conjugates 19 TFA) is a synthesized E3 ligase ligand-linker conjugate.</p>Fórmula:C21H23F3N4O8Pureza:95%Forma y color:SolidPeso molecular:516.42Maduramicin ammonium
CAS:<p>Maduramicin ammonium (Maduramycin Ammonium) is an anticoccidial agent for the the treatment of Eimeria spp., E.</p>Fórmula:C47H83NO17Pureza:99.83%Forma y color:White Crystalline PowderPeso molecular:934.20Morroniside
CAS:<p>Morroniside regulates liver inflammation, lipid metabolism, protects against diabetic kidney damage, and guards the brain from ischemic injury.</p>Fórmula:C17H26O11Pureza:99.70% - 99.84%Forma y color:SolidPeso molecular:406.38Diclofenac Potassium
CAS:<p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>Fórmula:C14H10Cl2KNO2Pureza:99.51%Forma y color:White To Yellowish Crystalline PowderPeso molecular:334.24C188-9
CAS:<p>C188-9 (TTI-101) is a Stat3 inhibitor with an IC50 of 4-7 μM.</p>Fórmula:C27H21NO5SPureza:98.07% - >99.99%Forma y color:SolidPeso molecular:471.52Thalidomide-O-amido-PEG2-C2-NH2 TFA
CAS:<p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>Fórmula:C23H27F3N4O10Pureza:95.74% - 99%Forma y color:SolidPeso molecular:576.48BAY 11-7082
CAS:BAY 11-7082 (BAY 11-7821) is an NF-κB inhibitor that inhibits TNFα-induced IκBα phosphorylation (IC50=10 μM).Fórmula:C10H9NO2SPureza:98% - 99.92%Forma y color:SolidPeso molecular:207.25OSU-T315
CAS:<p>OSU-T315 (OSU-T315 (1,5-regioisomer)) (1,5-regioisomer) is a ILK inhibitor.</p>Fórmula:C30H30F3N5OPureza:98.69%Forma y color:SolidPeso molecular:533.59Ganetespib
CAS:<p>Ganetespib (STA-9090) is a synthetic small-molecule inhibitor of heat shock protein 90 (Hsp90) with potential antineoplastic activity.</p>Fórmula:C20H20N4O3Pureza:98% - 99.95%Forma y color:SolidPeso molecular:364.4Trametinib (DMSO solvate)
CAS:<p>Trametinib (DMSO solvate) (GSK-1120212 (DMSO solvate)) is a Highly Potent and Selective MEK Inhibitor that specifically inhibits MEK1/2(IC50 :2 nM)</p>Fórmula:C28H29FIN5O5SPureza:98.82% - 99.92%Forma y color:SolidPeso molecular:693.53Notopterol
CAS:1. Notopterol induces apoptosis and inhibits cell cycle-specific.Fórmula:C21H22O5Pureza:97.57% - 99.82%Forma y color:SolidPeso molecular:354.40Terrestrosin D
CAS:<p>Terrestrosin D triggers apoptosis, halts cell cycles, and blocks angiogenesis in tumor cells, displaying anti-cancer effects.</p>Fórmula:C50H80O23Pureza:99.92% - 99.96%Forma y color:SolidPeso molecular:1049.16
