Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(56 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(166 productos)
- LHRH(1 productos)
- Receptor de opioides(326 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(90 productos)
- Reductasa(50 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(32 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3371 productos de "Endocrinología / Hormonas"
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DPP-4/GPR119 modulator 1
CAS:Orally active DPP-4 inhibitor/GPR119 agonist, Compound 22 lowers glucose, moderate hERG inhibition, IC50 4.9 µM, for diabetes research.Fórmula:C30H39ClN10O3Forma y color:SolidPeso molecular:623.15(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
CAS:(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].Fórmula:C48H74N12O12S2Pureza:98%Forma y color:SolidPeso molecular:1075.3Bexirestrant
CAS:Bexirestrant is an orally active ER-α degrader commonly employed in the research of antiestrogen and antineoplastic therapies.Fórmula:C29H26F3NO2Forma y color:SolidPeso molecular:477.527Ganoderic acid Df
CAS:<p>Ganoderic acid Df, a lanostane triterpenoid from Ganoderma lucidum, inhibits aldose reductase with IC50 of 22.8 μM.</p>Fórmula:C30H44O7Forma y color:SolidPeso molecular:516.67Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFórmula:C46H66N10O12S2Pureza:98.93%Forma y color:SolidPeso molecular:1015.21Ref: TM-T20166L
1mg185,00€5mg415,00€10mg622,00€25mg1.119,00€50mg1.679,00€100mg2.520,00€200mg3.780,00€Inocoterone acetate
CAS:Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.Fórmula:C18H26O3Forma y color:SolidPeso molecular:290.40NH-3
CAS:NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding and cofactor recruitment.Fórmula:C28H27NO6Pureza:97.79% - 99.40%Forma y color:SolidPeso molecular:473.52Ref: TM-T40548
1mg217,00€5mg550,00€10mg792,00€25mg1.206,00€50mg1.605,00€100mg2.175,00€500mg4.389,00€1mL*10mM (DMSO)492,00€AM-5262
CAS:AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.Fórmula:C33H35FO4Forma y color:SolidPeso molecular:514.63ER degrader 4
CAS:ER degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1].Fórmula:C26H19FO4SForma y color:SolidPeso molecular:446.49Leumorphin, human
CAS:Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-Fórmula:C150H224N42O46Pureza:98%Forma y color:SolidPeso molecular:3351.64Saprisartan
CAS:Saprisartan (GR-138950, GR-138950X) is an AT1 receptor antagonist used for the treatment of heart failure and blood pressure.Fórmula:C25H22BrF3N4O4SForma y color:SolidPeso molecular:611.43AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Fórmula:C16H24N2OForma y color:SolidPeso molecular:260.38U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Fórmula:C16H23ClN2OForma y color:SolidPeso molecular:294.82(-)-9-Hydroxycorynantheidine
CAS:(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.Fórmula:C22H28N2O4Forma y color:SolidPeso molecular:384.47Antidiabetic agent 15
<p>Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.</p>Fórmula:C26H23NO5Forma y color:SolidPeso molecular:429.15762Nurr1 agonist 12
Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.Fórmula:C18H12ClN3OForma y color:SolidPeso molecular:321.76MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Fórmula:C37H47Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:680.71WAY-298630
CAS:Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.Fórmula:C17H15FN2O3SPureza:97.84%Forma y color:SolidPeso molecular:346.38Pro8-Oxytocin TFA
<p>Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primate</p>Fórmula:C42H62N12O12S2·xC2HF3O2Pureza:98%Forma y color:SolidMyrciacetin
CAS:Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.Fórmula:C17H16O6Forma y color:SolidPeso molecular:316.309
