Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(33 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3420 productos de "Endocrinología / Hormonas"
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Human PTH-(1-31) amide
CAS:Human PTH-(1-31) amide, an analog of PTH, effectively stimulates phosphatidylcholine hydrolysis and promotes the release of adenylyl cyclase [1].Fórmula:C162H270N50O46S2Forma y color:SolidPeso molecular:3718.31MOR agonist-4
MOR agonist-4 (2d), having an EC50 of 11 nM, is a G protein-biased agonist of the Kappa opioid receptor (KOR). This compound features a triazole-based, electron-withdrawing CF3 group and a bias factor of 38. MOR agonist-4 is utilized for antipruritic and analgesic applications.Forma y color:Odour SolidArg-Glu(edans)-Ile-His-Pro-Phe-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(dabcyl)-Arg
Arg-Glu(edans)-Ile-His-Pro-Phe-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys(dabcyl)-Arg is a fluorescent renin substrate based on the N-terminal tetrapeptide sequence of human angiotensinogen (hTDP).Fórmula:C129H179N37O24SPeso molecular:2662.36444Osteostatin (1-5) amide (human, bovine, dog, horse, mouse, rabbit, rat)
CAS:Osteostatin (1-5) amide (human, bovine, dog, horse, mouse, rabbit, rat), also known as Human PTHrP (107-111) amide, is a C-terminal fragment of parathyroidFórmula:C27H42N10O7Peso molecular:618.69Kisspeptin-14 human
CAS:Kisspeptin-14 human is an active fragment peptide of Kisspeptin encoded by the KiSS-1 gene. Kisspeptin-14 human is a GPR54 agonist for human and rat.Fórmula:C82H112N22O21Forma y color:SolidPeso molecular:1741.9Acetalin-2
CAS:Acetalin-2, an opioid peptide with the sequence Ac-Arg-Phe-Met-Trp-Met-Arg-NH2, selectively binds to [3 H]DAMGO with a Ki value of 93.3 nM [1].Fórmula:C44H66N14O7S2Peso molecular:967.21Antiproliferative agent-51
Antiproliferative agent-51 (Compound 18h) inhibits estrogen receptor α (ERα)-mediated transcription with an IC50 of 1.6 nM. It also suppresses the proliferation of cancer cells ZR-75, with an IC50 of 0.031 μM, and exhibits antitumor activity in mouse models.Fórmula:C43H50N4O9Peso molecular:766.35778Chymase
CAS:Chymase is a proteolytic enzyme predominantly found in mast cells (MC), fibroblasts, and vascular endothelial cells. It is released into the extracellular matrix in response to inflammatory signals, tissue damage, and cellular stress. Chymase also plays a role in the generation of angiotensin II (Ang II), making it significant for cardiovascular disease research.Termitomycamide B
CAS:Termitomycamide B, a fatty acid from T. titanicus, protects Neuro2a cells from ER stress-induced death at 0.1 μg/ml.Fórmula:C28H40N2O2Forma y color:SolidPeso molecular:436.63β-Chlornaltrexamine dihydrochloride
CAS:β-Chlornaltrexamine dihydrochloride (β-CNA dihydrochloride) is an effective long-term antagonist of opioid receptors. It efficiently blocks the inhibition of dopamine release mediated by κ opioid receptor agonists. This compound is useful in the research of pain perception mechanisms.Fórmula:C24H34Cl4N2O3Forma y color:SolidPeso molecular:540.35Ota-vasotocin
CAS:Ota-vasotocin is a ligand utilized in quantitative receptor autoradiography for oxytocin receptors.Fórmula:C54H79N11O13S2Peso molecular:1154.41TRV055
CAS:TRV055: Gq-biased AT1R ligand, stimulates Gq signaling, aids Gq-biased agonist development.Fórmula:C42H57N9O9Forma y color:SolidPeso molecular:831.972[Asp5]-Oxytocin
CAS:[Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity.Fórmula:C43H65N11O13S2Peso molecular:1008.18Morphiceptin
CAS:Morphiceptin is a synthetic tetrapeptide with morphinelike activities, highly specific for morphine receptors, but not for enkephalin receptors.Fórmula:C28H35N5O5Peso molecular:521.61Detrothyronine
CAS:Detrothyronine is a biochemical.Fórmula:C15H12I3NO4Forma y color:SolidPeso molecular:650.97Biotin-Oxytocin
Biotin-Oxytocin (Biotin-α-Hypophamine; Biotin-Oxytocic hormone) is a biologically active peptide. It is oxytocin labeled with biotin at the N-terminus.Fórmula:C53H80N14O14S3Peso molecular:1232.51406[Asp5]-Oxytocin acetate
[Asp5]-Oxytocin acetate: a biologically active neurohypophyseal hormone analogue, inducing uterine contractions, effects magnified by Mg2+.Fórmula:C45H69N11O15S2Peso molecular:1068.22BPRMU191
CAS:BPRMU191 is a distinct mu-opioid receptor (MOR) modulator with an EC50 of 2.17 μM in FLIPR Ca2+ assays conducted on CHO-K1/MOR/Gα15 cells. Additionally, BPRMU191 interacts with MOR in the presence of naloxone.Fórmula:C17H14FNO3SForma y color:SolidPeso molecular:331.36Saprisartan
CAS:Saprisartan (GR-138950, GR-138950X) is an AT1 receptor antagonist used for the treatment of heart failure and blood pressure.Fórmula:C25H22BrF3N4O4SForma y color:SolidPeso molecular:611.43Keap1-IN-1
Keap1-IN-1 (Compound 27) is an inhibitor of Keap1, functioning by covalently modifying the Cys151 residue on the BTB domain of KEAP1, thereby disrupting the interaction between Keap and Nrf. It enhances the mRNA expression of the antioxidant response element (ARE) dependent gene NQO1, with an EC50 of 160 nM, and exhibits cytotoxicity in U2OS cells, with an EC50 of 527 nM.Fórmula:C17H21Cl2N2O5PS3Forma y color:SolidPeso molecular:531.434
