Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(60 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(325 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(50 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(32 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3371 productos de "Endocrinología / Hormonas"
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Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFórmula:C46H66N10O12S2Pureza:98.93%Forma y color:SolidPeso molecular:1015.21Ref: TM-T20166L
1mg185,00€5mg415,00€10mg622,00€25mg1.119,00€50mg1.679,00€100mg2.520,00€200mg3.780,00€Leumorphin, human
CAS:Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-Fórmula:C150H224N42O46Pureza:98%Forma y color:SolidPeso molecular:3351.64AH 7563
CAS:AH 7563 is structurally classified as an opioid compound with analgesic properties. In mice, its ED50 for pain relief was 15.3 mg/kg when administered orally in the Phenylquinone test, and 15.5 mg/kg when injected subcutaneously in the Hot plate test.Fórmula:C16H24N2OForma y color:SolidPeso molecular:260.38U-48520
CAS:U-48520 is an agonist of the μ-opioid receptor (μ-opioid receptor) with an EC50 of 1561 nM.Fórmula:C16H23ClN2OForma y color:SolidPeso molecular:294.82(-)-9-Hydroxycorynantheidine
CAS:(-)-9-Hydroxycorynantheidine (9-O-Desmethyl mitragynine) is a demethylated analog of Mitragynine, functioning as a selective and partial agonist for the μ-opioid receptor (μ-opioid receptor). This compound inhibits electrically stimulated twitch contractions in the guinea pig ileum.Fórmula:C22H28N2O4Forma y color:SolidPeso molecular:384.47MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Fórmula:C37H47Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:680.71WAY-298630
CAS:Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.Fórmula:C17H15FN2O3SPureza:97.84%Forma y color:SolidPeso molecular:346.38Pro8-Oxytocin TFA
Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primate
Fórmula:C42H62N12O12S2·xC2HF3O2Pureza:98%Forma y color:SolidFluorphine
CAS:Fluorphine, an analog of Brorphine, binds to the μ-opioid receptor (MOR) with a Ki of 12.5 nM. It exhibits GTPγS binding activity with an EC50 of 75 nM and β-arrestin 2 recruitment activity with an EC50 of 377 nM, and it also has respiratory depressive effects.Fórmula:C20H22FN3OForma y color:SolidPeso molecular:339.41Orphine
CAS:Orphine is an opioid compound that can amplify the antinociceptive effects reduced by naloxone in mice.Fórmula:C20H23N3OForma y color:SolidPeso molecular:321.42PF-06478939 TFA
PF-06478939 TFA is a peptide that acts as a non-brain-penetrating agonist at the oxytocin (OT) and vasopressin receptors, exhibiting EC50 values of 0.01 nM andFórmula:C78H134N14O22S2·xC2HF3O2Pureza:98%Forma y color:Solid(Val3,Pro8)-Oxytocin
CAS:(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced efficacy agonist for β-arrestinFórmula:C41H60N12O12S2Pureza:98%Forma y color:SolidPeso molecular:977.12CSD-CH2(1,8)-NH2
CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM.Fórmula:C76H125N25O15S2Pureza:98%Forma y color:SolidPeso molecular:1693.09DALDA TFA
DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM.Fórmula:C30H45N9O5·xC2HF3O2Pureza:98%Forma y color:SolidPeso molecular:611.74 (free base)AH 8529
CAS:AH 8529 is an orally active opioid compound with analgesic properties.Fórmula:C16H23ClN2OForma y color:SolidPeso molecular:294.82N-Phenethylnoroxymorphone
CAS:N-Phenethylnoroxymorphone is an opioid compound that can enhance morphine-induced analgesia in rats. It is used in the research of neurological disorders.Fórmula:C24H25NO4Forma y color:SolidPeso molecular:391.46KOR agonist 3
KOR agonist 3 (Compound 5) is an agonist of the κ opioid receptor (κOR) with an EC50 of 0.88 nM. It also exhibits some activation of μOR, with an EC50 of 720 nM. However, KOR agonist 3 does not activate δOR at concentrations below 1 μM. Its ability to recruit β-Arrestin-2 is lower than that of U50488.Fórmula:C24H24N2O3Forma y color:SolidPeso molecular:388.46Pro8-Oxytocin
CAS:Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR and induces stronger behavioral effects comparedFórmula:C42H62N12O12S2Pureza:98%Forma y color:SolidPeso molecular:991.14Corynantheidine
CAS:Corynantheidine ((-)-Corynantheidine) is a partial agonist of the mu opioid receptor (MOR) and demonstrates MOR-dependent analgesic effects in mice.Fórmula:C22H28N2O3Forma y color:SolidPeso molecular:368.47AH 7959
CAS:AH 7959 is an orally active N-substituted cyclohexylmethylbenzamide compound that exhibits analgesic properties. In mice, the ED50 for oral and subcutaneous administration of AH 7959 exceeds 100 mg/kg.Fórmula:C19H26Cl2N2OForma y color:SolidPeso molecular:369.33
