Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"
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GABAA receptor agent 1
CAS:<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Fórmula:C13H8ClN3O2Pureza:99.31%Forma y color:SolidPeso molecular:273.675,5-Dimethyloxazolidine-2,4-dione
CAS:<p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>Fórmula:C5H7NO3Pureza:99.12%Forma y color:Drypowder PelletslargecrystalsPeso molecular:129.11Vinpocetine
CAS:<p>Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).</p>Fórmula:C22H26N2O2Pureza:99.85% - 99.98%Forma y color:White Crystalline SolidPeso molecular:350.45FG 7142
CAS:<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Fórmula:C13H11N3OPureza:98.75%Forma y color:SolidPeso molecular:225.25Torsemide
CAS:<p>Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.</p>Fórmula:C16H20N4O3SPureza:99.81%Forma y color:Crystalline SolidPeso molecular:348.42Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Fórmula:C14H18N2O2Pureza:97.37%Forma y color:White To Off-White Crystalline PowderPeso molecular:246.3FFN 206 dihydrochloride
CAS:<p>FFN 206 dihydrochloride: fluorescent VMAT2 marker, detects subcellular sites, non-inhibitory to DAT.</p>Fórmula:C12H15ClN2O2Pureza:98.96% - >99.99%Forma y color:SolidPeso molecular:254.71Piracetam
CAS:<p>Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.</p>Fórmula:C6H10N2O2Pureza:97.16%Forma y color:Crystals From Isopropanol SolidPeso molecular:142.16Afoxolaner
CAS:<p>Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.</p>Fórmula:C26H17ClF9N3O3Pureza:99.1% - 99.38%Forma y color:SolidPeso molecular:625.87Flufenamic acid
CAS:<p>Flufenamic acid (Arlef) is an anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties.</p>Fórmula:C14H10F3NO2Pureza:98.68%Forma y color:White To Light Yellow Crystalline PowderPeso molecular:281.23Halothane
CAS:<p>Halothane (Anestan) 可以减弱内皮依赖性舒张作用。</p>Fórmula:C2HBrClF3Pureza:98.50% - >99.99%Forma y color:Colorless Volatile Liquid Density 1 875 G / Cm3 Boiling Point 122 4°F (50 2°C) NoncombustiblePeso molecular:197.38Hydrochlorothiazide
CAS:<p>Hydrochlorothiazide (HCTZ) 是一种口服有效的噻嗪类的利尿药，可抑制转化 TGF-β/Smad 信号通路。它通过打开钙激活钾 (KCA) 通道发挥直接的血管松弛作用。它改善心脏功能，减少纤维化并具有降压作用。</p>Fórmula:C7H8ClN3O4S2Pureza:99.43% - 99.50%Forma y color:Crystals Physical Description Crystals Or White Powder (Ntp 1992)Peso molecular:297.74L-Cycloserine
CAS:<p>L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.</p>Fórmula:C3H6N2O2Pureza:99.45% - 99.92%Forma y color:Crystals White PowderPeso molecular:102.09Riparin III
CAS:<p>Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.</p>Fórmula:C16H17NO4Pureza:95.13%Forma y color:SolidPeso molecular:287.31BMS-394136
CAS:<p>BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as arrhythmias and atrial fibrillation.</p>Fórmula:C24H21Cl2FN4OPureza:98.19% - 98.67%Forma y color:SolidPeso molecular:471.35Phenazopyridine hydrochloride
CAS:<p>Phenazopyridine HCl, an oral urinary analgesic, may cause nausea, anemia, and liver/kidney toxicity. Possibly carcinogenic.</p>Fórmula:C11H12ClN5Pureza:99.27%Forma y color:Brownish-Yellow Crystals Aqueous Solutions Are Yellow To Brick-Red And Slightly Acidic; They May Be Stabilized By The AdditionPeso molecular:249.7RUVBL1/2 ATPase-IN-1
CAS:<p>RUVBL1/2 ATPase-IN-1 inhibits RUVBL1/2 ATPase (IC50: 6.0/7.7 μM); useful in cancer research.</p>Fórmula:C28H28F3N5OPureza:99.92%Forma y color:SolidPeso molecular:507.55Endovion
CAS:<p>Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.</p>Fórmula:C16H9BrF6N6OPureza:98.51%Forma y color:SolidPeso molecular:495.18NS8593 hydrochloride
CAS:<p>NS8593 hydrochloride (NS8593 HCl) is a potent and selective inhibitor of small conductance Ca2+-activated K+ channels (SK channels) .</p>Fórmula:C17H18ClN3Pureza:99.77%Forma y color:SolidPeso molecular:299.8Ropivacaine
CAS:<p>Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.</p>Fórmula:C17H26N2OPureza:97.75% - >99.99%Forma y color:SolidPeso molecular:274.40Dyclonine hydrochloride
CAS:<p>Dyclonine hydrochloride (Dyclonine HCl) , an over the counter throat lozenge, is found in Sucretswith local anesthetic effect .</p>Fórmula:C18H27NO2·HClPureza:99.35%Forma y color:White Crystalline SolidPeso molecular:325.87(Z)-Capsaicin
CAS:<p>(Z)-Capsaicin (Zucapsaicin) is a medication used to treat osteoarthritis of the knee and Others neuropathic pain.(Z)-Capsaicin is a synthetic cis isomer of</p>Fórmula:C18H27NO3Pureza:97.33% - 98.91%Forma y color:SolidPeso molecular:305.41Nicorandil
CAS:<p>Nicorandil (SG-75)(Ikorel) acts by relaxing the smooth muscle of the blood vessels, especially those of the venous system.</p>Fórmula:C8H9N3O4Pureza:98.14% - >99.99%Forma y color:White Or Off-White PowderPeso molecular:211.17Alinidine
CAS:<p>Alinidine is an HCN channel blocker with antiarrhythmic effects and can be used for the study of angina pectoris.</p>Fórmula:C12H13Cl2N3Pureza:98.91% - >99.99%Forma y color:SolidPeso molecular:270.16Tocainide hydrochloride
CAS:<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Fórmula:C11H17ClN2OPureza:97%Forma y color:SolidPeso molecular:228.72Flindokalner
CAS:<p>Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.</p>Fórmula:C16H10ClF4NO2Pureza:99.96%Forma y color:SolidPeso molecular:359.7URAT1 inhibitor 7
CAS:<p>URAT1 inhibitor 7, a uric acid transporter protein URAT1 inhibitor.URAT1 inhibitor 7 inhibits CYP2C9 and can be used in the study of hyperuricemia and gout.</p>Fórmula:C19H10ClFN4O3SPureza:97.65%Forma y color:SoildPeso molecular:428.82Glibenclamide
CAS:<p>Glibenclamide (Glyburide) is an antidiabetic sulfonylurea derivative with actions similar to those of chlorpropamide.</p>Fórmula:C23H28ClN3O5SPureza:99.05% - 99.75%Forma y color:SolidPeso molecular:494.00QX-314 chloride
CAS:<p>QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.</p>Fórmula:C16H27ClN2OPureza:99.73%Forma y color:SolidPeso molecular:298.85Gabapentin
CAS:<p>Gabapentin (Neurontin) is an Anti-epileptic Agent.</p>Fórmula:C9H17NO2Pureza:99.55% - 99.91%Forma y color:White To Off-White Crystalline Solid; Crystals From Ethanol/Ether SolidPeso molecular:171.24NBQX disodium
CAS:<p>NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity.</p>Fórmula:C12H6N4Na2O6SPureza:97.6% - 98.22%Forma y color:SolidPeso molecular:380.2415Clorsulon
CAS:<p>Clorsulon (L631529) is utilized for the treatment of Fasciola hepatica infections in calves and sheep.</p>Fórmula:C8H8Cl3N3O4S2Pureza:99.66% - 99.87%Forma y color:White To Off-White Crystalline PowderPeso molecular:380.66Miconazole
CAS:<p>Miconazole (R18134) is an imidazole antifungal agent that is used topically and by intravenous infusion.</p>Fórmula:C18H14Cl4N2OPureza:98% - >99.99%Forma y color:SolidPeso molecular:416.13Omeprazole
CAS:<p>Omeprazole (Losec) is a proton pump inhibitor (PPI), Omeprazole(Losec) is a potent brain penetrant neutral sphingomyelinase (N-SMase) inhibitor.</p>Fórmula:C17H19N3O3SPureza:98.43% - 98.48%Forma y color:White SolidPeso molecular:345.42Pivagabine
CAS:<p>Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.</p>Fórmula:C9H17NO3Pureza:99.87%Forma y color:SolidPeso molecular:187.24Phenelzine sulfate
CAS:<p>Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.</p>Fórmula:C8H14N2O4SPureza:98.38% - 99.83%Forma y color:SolidPeso molecular:234.27Ropivacaine hydrochloride
CAS:<p>Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activity</p>Fórmula:C17H26N2O·HClPureza:99.85% - 99.95%Forma y color:SolidPeso molecular:310.86Oxybutynin
CAS:<p>Oxybutynin (Ditropan) is a synthetic anticholinergic agent that is used for treatment of urinary incontinence and overactive bladder syndrome.</p>Fórmula:C22H31NO3Pureza:97.81% - 99.57%Forma y color:White To Off-White Crystalline PowderPeso molecular:357.49N-Acetylprocainamide
CAS:<p>N-Acetylprocainamide (NAPA), the N-acetylated metabolite of Procainamide, is a Class III antiarrhythmic agent, while procainamide is a Class Ia antiarrhythmic</p>Fórmula:C15H23N3O2Pureza:99.65% - 99.74%Forma y color:SolidPeso molecular:277.36VU591 hydrochloride
CAS:<p>VU591 hydrochloride is a selective Kir1.1 (ROMK) blocker with IC50 of 0.24 μM, not affecting Kir7.1, Kir2.1, Kir2.3, or Kir4.1, similar to VU 590.</p>Fórmula:C16H13ClN6O5Pureza:98.93% - 99.22%Forma y color:SolidPeso molecular:404.76Emamectin Benzoate
CAS:<p>Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods</p>Fórmula:C56H81NO15Pureza:98.68%Forma y color:SolidPeso molecular:1008.256Acetohexamide
CAS:<p>Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.</p>Fórmula:C15H20N2O4SPureza:99.19% - 99.85%Forma y color:Crystals From 90% Aq EthanolPeso molecular:324.40Hydroxyhexamide
CAS:<p>Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.</p>Fórmula:C15H22N2O4SPureza:98.91%Forma y color:SolidPeso molecular:326.41Gliclazide
CAS:<p>Gliclazide (SE1702), an oral antihyperglycemic agent, belongs to the sulfonylurea class of insulin secretagogues, which act by stimulating beta-cells of the</p>Fórmula:C15H21N3O3SPureza:99.58%Forma y color:SolidPeso molecular:323.41NS5806
CAS:<p>NS5806 activates K+ currents, slows KV4.2/4.3 decay with KChIP2, and boosts KV4.3/KChIP2 peaks (EC50=5.3μM).</p>Fórmula:C16H8Br2F6N6OPureza:97.95%Forma y color:SolidPeso molecular:574.07Meticrane
CAS:<p>Meticrane (Arresten) is a sulphonamide-derivative with thiazide-like diuretic activity.</p>Fórmula:C10H13NO4S2Pureza:99.16%Forma y color:SolidPeso molecular:275.34BIIB 722 Mesylate
CAS:<p>BIIB 722 Mesylate is a sodium-hydrogen exchange inhibitor with cardioprotective properties and can be used to study myocardial ischemia.</p>Fórmula:C19H23F3N6O5SPureza:99.57%Forma y color:SoildPeso molecular:504.483VU591
CAS:<p>VU591 is a selective extra-renal potassium channel inhibitor with an IC₅₀ of 0.24 μM.</p>Fórmula:C16H12N6O5Pureza:99.29% - 99.53%Forma y color:SolidPeso molecular:368.3Nav1.8-IN-4
CAS:<p>Nav1.8-IN-4 is a potent Nav1.8 channel inhibitor with potential analgesic activity.Nav1.8-IN-4 can be used for pain and neurological related disorders.</p>Fórmula:C20H14F4N2O3Pureza:99.83%Forma y color:SoildPeso molecular:406.33Tuvatexib
CAS:<p>Tuvatexib is a small molecule VDAC/HK2 dual modulator.</p>Fórmula:C21H23NO3Pureza:97.29% - 99.80%Forma y color:SolidPeso molecular:337.41E 0747 FA
<p>E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax in Purkinje fibers of porcine heart.E 0747 FA inhibits Na channels in cardiac cells.</p>Fórmula:C22H30ClN3O6Pureza:98.54%Forma y color:SolidPeso molecular:467.94Broflanilide
CAS:<p>Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.</p>Fórmula:C25H14BrF11N2O2Pureza:99.82%Forma y color:SolidPeso molecular:663.29Lansoprazole
CAS:<p>Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISON</p>Fórmula:C16H14F3N3O2SPureza:99.18% - 99.84%Forma y color:White Crystalline PowderPeso molecular:369.36NS1652
CAS:<p>NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.</p>Fórmula:C15H11F3N2O3Pureza:99.62%Forma y color:SolidPeso molecular:324.25VU6036720
<p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>Fórmula:C20H22ClFN4O2SPureza:98.1%Forma y color:SoildPeso molecular:436.93BI-749327
CAS:<p>BI-749327 is a high selectivity and orally bioavailable antagonist of TRPC6 (IC50s: 13 nM, 19 nM and 15 nM for mouse, human and guinea pig TRPC6).</p>Fórmula:C23H21F3N4O2Pureza:99.68%Forma y color:SolidPeso molecular:442.43NS13001
CAS:<p>NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).</p>Fórmula:C17H16ClN7Pureza:99.55%Forma y color:SolidPeso molecular:353.81Zamicastat
CAS:<p>Zamicastat (BIA 5-1058) inhibits DBH, P-gp (IC50=73.8μM), and BCRP (IC50=17.0μM).</p>Fórmula:C21H21F2N3OSPureza:99.58%Forma y color:SolidPeso molecular:401.47NMDA-IN-1
CAS:<p>NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).</p>Fórmula:C20H23ClFN3OPureza:99.57%Forma y color:SolidPeso molecular:375.87Pramocaine hydrochloride
CAS:<p>Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.</p>Fórmula:C17H27NO3·HClPureza:99.15% - 99.61%Forma y color:Crystals White Or Off White Crystalline PowderPeso molecular:329.86Cromolyn sodium
CAS:<p>Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.</p>Fórmula:C23H14Na2O11Pureza:99.4% - 99.95%Forma y color:Colorless Crystals From Ethanol + Ether White Crystalline PowderPeso molecular:512.33VU0134992 hydrochloride
CAS:<p>VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).</p>Fórmula:C20H32BrClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:447.841-EBIO
CAS:<p>1-EBIO (1-EBIO) is a calium channel agonist.</p>Fórmula:C9H10N2OPureza:98.75%Forma y color:SolidPeso molecular:162.19FFN 511
CAS:<p>Fluorescent false neurotransmitter (FFN)</p>Fórmula:C17H20N2O2Pureza:98%Forma y color:SolidPeso molecular:284.35Clomethiazole
CAS:<p>Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.</p>Fórmula:C6H8ClNSPureza:99.06%Forma y color:SolidPeso molecular:161.65TRPV4 agonist-1 free base
CAS:<p>TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).</p>Fórmula:C25H22F2N4O2Pureza:99.79%Forma y color:SolidPeso molecular:448.46Ethaverine hydrochloride
CAS:<p>Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.</p>Fórmula:C24H30ClNO4Pureza:99.66% - 99.90%Forma y color:SolidPeso molecular:431.96T16Ainh-A01
CAS:<p>T16Ainh-A01 is a potent TMEM16A chloride channel inhibitor with a 1 μM IC50, targeting CaCC.</p>Fórmula:C19H20N4O3S2Pureza:97.18% - 98.15%Forma y color:SolidPeso molecular:416.52Vocacapsaicin hydrochloride
CAS:<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Fórmula:C26H42ClN3O4Pureza:99.66% - 99.80%Forma y color:SolidPeso molecular:496.08ATP synthase inhibitor 1
CAS:<p>ATP synthase inhibitor 1 is an inhibitor of the c subunit of the F1/FO-ATP synthase complex.</p>Fórmula:C17H18ClN3O3S2Pureza:99.83%Forma y color:SolidPeso molecular:411.93GFB-8438
CAS:<p>GFB-8438 is a potent and subtype selective inhibitor of TRPC5(IC50s of 0.18 and 0.29 μM of hTRPC5 and hTRPC4, respectively).</p>Fórmula:C16H14ClF3N4O2Pureza:99.58%Forma y color:SolidPeso molecular:386.76Repaglinide
CAS:<p>Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.</p>Fórmula:C27H36N2O4Pureza:99.73% - >99.99%Forma y color:White To Off-White SolidPeso molecular:452.59Domperidone EP Impurity A
CAS:<p>Domperidone EP Impurity A is used as pharmaceutical intermediates.</p>Fórmula:C12H14ClN3OPureza:99.97%Forma y color:SolidPeso molecular:251.71Sulfacarbamide
CAS:<p>Sulfacarbamide (Sulfanilylurea) is a blood sugar-lowering agent.</p>Fórmula:C7H9N3O3SPureza:95.6% - 99.72%Forma y color:SolidPeso molecular:215.23Econazole
CAS:<p>Econazole ((±)-Econazol) is an imidazole derivative that is commonly used as a topical antifungal agent.</p>Fórmula:C18H15Cl3N2OPureza:98.11% - 99.97%Forma y color:SolidPeso molecular:381.68Ornidazole (Levo-)
CAS:<p>Ornidazole (Levo-) (Levornidazole) is the levo-isomer of Ornidazole.</p>Fórmula:C7H10ClN3O3Pureza:99.8%Forma y color:SolidPeso molecular:219.63Tertiapin-Q
CAS:<p>Tertiapin-Q is a bee toxin derivative that inhibits BK-type K(+) channels in a concentration-dependent manner, inhibiting efflux to K(+).</p>Fórmula:C106H175N35O24S4Pureza:98.06% - 98.09%Forma y color:SolidPeso molecular:2452CGP37157
CAS:<p>CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) is a Na+/Ca2+ exchanger inhibitor, inhibits Na+-induced Ca2+ release from</p>Fórmula:C15H11Cl2NOSPureza:99.92%Forma y color:SolidPeso molecular:324.22Manidipine dihydrochloride
CAS:<p>Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).</p>Fórmula:C35H40Cl2N4O6Pureza:99.76% - 99.86%Forma y color:SolidPeso molecular:683.62D-AP5
CAS:<p>D-AP5 (D-APV) is a NMDA receptor antagonist.</p>Fórmula:C5H12NO5PPureza:98.77% - >99.99%Forma y color:White Fine Crystalline PowderPeso molecular:197.13Etifoxine hydrochloride
CAS:<p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>Fórmula:C17H18Cl2N2OPureza:99.36%Forma y color:SolidPeso molecular:337.24CRAC intermediate 2
CAS:<p>CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.</p>Fórmula:C11H7F6N3Pureza:99.69%Forma y color:SolidPeso molecular:295.18PF-04885614
CAS:<p>PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.</p>Fórmula:C13H14F3N3OPureza:98.02%Forma y color:SolidPeso molecular:285.27Tolazamide
CAS:<p>Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.</p>Fórmula:C14H21N3O3SPureza:98% - >99.99%Forma y color:SolidPeso molecular:311.40Devapamil
CAS:<p>Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.</p>Fórmula:C26H36N2O3Pureza:99.63%Forma y color:SolidPeso molecular:424.58Vigabatrin
CAS:<p>Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-</p>Fórmula:C6H11NO2Pureza:99.47% - 99.88%Forma y color:SolidPeso molecular:129.16LAU159
CAS:<p>LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).</p>Fórmula:C17H12ClN3O2Pureza:98.7% - 99.38%Forma y color:SolidPeso molecular:325.75Oxiracetam
CAS:<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Fórmula:C6H10N2O3Pureza:99.67%Forma y color:White Crystalline PowderPeso molecular:158.16Permethrin
CAS:<p>Permethrin (NRDC-143) is a pyrethroid insecticide commonly used in the treatment of LICE INFESTATIONS and SCABIES.</p>Fórmula:C21H20Cl2O3Pureza:99.37% - 99.54%Forma y color:Colorless Crystals To A Viscous Liquid; Color White To Pale Yellow Permethrin Is A Pale Brown Liquid Relatively Water Insoluble Used As An InsecticidePeso molecular:391.29AR-C155858
CAS:<p>AR-C155858 is an inhibitor of monocarboxylate transporter MCT1 and MCT2 (Kis: 2.3 nM and 10 nM).</p>Fórmula:C21H27N5O5SPureza:98.96% - 99.42%Forma y color:SolidPeso molecular:461.53Oxybutynin chloride
CAS:<p>Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.</p>Fórmula:C22H32ClNO3Pureza:99.27% - >99.99%Forma y color:White PowderPeso molecular:393.96BMS-191095
CAS:<p>BMS-191095 is mitochondrial ATP-sensitive potassium (mitoKATP) channel activator.</p>Fórmula:C22H21ClN4O2Pureza:>99.99%Forma y color:SolidPeso molecular:408.88DCEBIO
CAS:<p>DCEBIO, a 1-EBIO derivative, enhances Cl- secretion via hIK1 K+ channel and apical conductance in T84 cells.</p>Fórmula:C9H8Cl2N2OPureza:99.89%Forma y color:SolidPeso molecular:231.08Chlormezanone
CAS:<p>Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.</p>Fórmula:C11H12ClNO3SPureza:99.89% - >99.99%Forma y color:Crystals SolidPeso molecular:273.74Isoguvacine hydrochloride
CAS:<p>Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.</p>Fórmula:C6H10ClNO2Pureza:99.59%Forma y color:SolidPeso molecular:163.6Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Fórmula:C12H21NO8SPureza:99.79% - 99.92%Forma y color:White To Off-White Crystalline PowderPeso molecular:339.36IA-Alkyne
CAS:<p>IA-Alkyne: TRPC agonist, cysteine-reactivity probe, potential in respiratory infection study.</p>Fórmula:C8H12INOPureza:99.76%Forma y color:SolidPeso molecular:265.09Eact
CAS:<p>Eact is a potent TMEM16A activator that also triggers TRPV1, causing itch, pain, and heat sensitivity.</p>Fórmula:C22H24N2O5SPureza:98.14%Forma y color:SolidPeso molecular:428.5Chlorpropamide
CAS:<p>Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary</p>Fórmula:C10H13ClN2O3SPureza:98.90%Forma y color:Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Peso molecular:276.74Gut restricted-7
CAS:<p>Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor.</p>Fórmula:C25H40FNaO6SPureza:98.81% - 99.27%Forma y color:SolidPeso molecular:510.64NaV1.7 inhibitor-1
CAS:<p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>Fórmula:C23H30FNO4SPureza:99.89%Forma y color:SolidPeso molecular:435.55Omeprazole metabolite Omeprazole sulfone
CAS:<p>Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.</p>Fórmula:C17H19N3O4SPureza:99.87%Forma y color:SolidPeso molecular:361.42Pentetrazol
CAS:<p>Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.</p>Fórmula:C6H10N4Pureza:99.7% - >99.99%Forma y color:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Peso molecular:138.17Nikethamide
CAS:<p>Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of end</p>Fórmula:C10H14N2OPureza:99.42%Forma y color:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Peso molecular:178.23Flumazenil
CAS:<p>Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous</p>Fórmula:C15H14FN3O3Pureza:99.72% - 99.98%Forma y color:Less Crystals Colourless CrystalsPeso molecular:303.29Eleclazine hydrochloride
CAS:<p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>Fórmula:C21H17ClF3N3O3Pureza:99.86%Forma y color:SolidPeso molecular:451.83Phenformin hydrochloride
CAS:<p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>Fórmula:C10H16ClN5Pureza:97.11% - 99.80%Forma y color:Lactic AcidosisPeso molecular:241.72ML418
CAS:<p>ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.</p>Fórmula:C19H24ClN3O3Pureza:99.3%Forma y color:SolidPeso molecular:377.874-Aminopyridine
CAS:<p>4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.</p>Fórmula:C5H6N2Pureza:91.61%Forma y color:SolidPeso molecular:94.11NS19504
CAS:<p>NS19504 is an activator of Ca2+-activated K+ channel with EC50 of 11.0 µM.</p>Fórmula:C10H9BrN2SPureza:99.87%Forma y color:SolidPeso molecular:269.16CIQ
CAS:<p>CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.</p>Fórmula:C26H26ClNO5Pureza:99.5%Forma y color:SolidPeso molecular:467.94Omeprazole sulfide
CAS:<p>Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.</p>Fórmula:C17H19N3O2SPureza:98.83%Forma y color:White To Slightly Collored Solid Solid CrystallinePeso molecular:329.42DSP-2230
CAS:<p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>Fórmula:C20H20F3N5O2Pureza:97.14%Forma y color:SolidPeso molecular:419.4ICA-27243
CAS:<p>ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.</p>Fórmula:C12H7ClF2N2OPureza:99.54%Forma y color:SolidPeso molecular:268.65Suloctidil
CAS:<p>Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.</p>Fórmula:C20H35NOSPureza:99.75% - >99.99%Forma y color:SolidPeso molecular:337.56Baclofen
CAS:<p>Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.</p>Fórmula:C10H12ClNO2Pureza:98% - >99.99%Forma y color:1992)Peso molecular:213.66Linopirdine
CAS:<p>Linopirdine (DuP 996) is a TRPV1 agonist.</p>Fórmula:C26H21N3OPureza:99.45% - 99.78%Forma y color:SolidPeso molecular:391.46Azosemide
CAS:<p>Azosemide is a potent NKCC1 inhibitor (IC50s: 0.246 µM and 0.197 µM for hNKCC1A and NKCC1B).</p>Fórmula:C12H11ClN6O2S2Pureza:99.84%Forma y color:SolidPeso molecular:370.84Methocarbamol
CAS:<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Fórmula:C11H15NO5Pureza:99.96%Forma y color:Crystals From Benzene SolidPeso molecular:241.24Trichlormethiazide
CAS:<p>Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.</p>Fórmula:C8H8Cl3N3O4S2Pureza:98.8% - 99.54%Forma y color:SolidPeso molecular:380.66Fluxametamide
CAS:<p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>Fórmula:C20H16Cl2F3N3O3Pureza:99.49%Forma y color:SolidPeso molecular:474.26γ-Aminobutyric acid
CAS:<p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>Fórmula:C4H9NO2Pureza:99.95%Forma y color:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderPeso molecular:103.12Cycloleucine
CAS:<p>Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.</p>Fórmula:C6H11NO2Pureza:99.90%Forma y color:SolidPeso molecular:129.16Linoleoyl glycine
CAS:<p>Linoleoyl glycine activates hKCNQ1/hKCNE1 channels, has analgesic properties, and is found in skin, spinal cord, and brain.</p>Fórmula:C20H35NO3Pureza:98.96%Forma y color:SolidPeso molecular:337.5Glipizide
CAS:<p>Glipizide (CP 28720) is a short-acting, second-generation sulfonylurea with hypoglycemic activity.</p>Fórmula:C21H27N5O4SPureza:99.67% - 99.75%Forma y color:SolidPeso molecular:445.54Diphenidol hydrochloride
CAS:<p>Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.</p>Fórmula:C21H28ClNOPureza:99.15% - 99.33%Forma y color:Crystals Soluble In Methanol WaterPeso molecular:345.91Ciclopirox olamine
CAS:<p>Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.</p>Fórmula:C14H24N2O3Pureza:99.16% - >99.99%Forma y color:White To Yellow Solid Solid Particulate/PowderPeso molecular:268.35Dooku1
CAS:<p>Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.</p>Fórmula:C13H9Cl2N3OSPureza:98.87% - 99.74%Forma y color:SolidPeso molecular:326.2Caloxin 2A1 TFA
<p>Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.</p>Fórmula:C66H92F3N19O24Pureza:99.89%Forma y color:SolidPeso molecular:1592.55BMS-195270
CAS:<p>BMS-195270 is a bio-active chemical.</p>Fórmula:C15H9ClF3N3O2Pureza:98.7%Forma y color:SolidPeso molecular:355.7Flavoxate hydrochloride
CAS:<p>Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.</p>Fórmula:C24H26ClNO4Pureza:99.78%Forma y color:White SolidPeso molecular:427.92Tocainide
CAS:<p>Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.</p>Fórmula:C11H16N2OPureza:99.84%Forma y color:SolidPeso molecular:192.26Celivarone
CAS:<p>Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and atrial fibrillation.</p>Fórmula:C34H47NO4Pureza:99.53%Forma y color:SolidPeso molecular:533.74MRZ 2-514
CAS:<p>MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with Ki</p>Fórmula:C11H6BrN3O3Pureza:98.459%Forma y color:SolidPeso molecular:308.09Prilocaine hydrochloride
CAS:<p>Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.</p>Fórmula:C13H21ClN2OPureza:99.97%Forma y color:Needles White Or Off White Crystalline PowderPeso molecular:256.77Z433927330
CAS:<p>Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).</p>Fórmula:C20H20N4O3Pureza:99.78%Forma y color:SolidPeso molecular:364.4Bupivacaine hydrochloride
CAS:<p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>Fórmula:C18H28N2O·HClPureza:99.9% - >99.99%Forma y color:SolidPeso molecular:324.89NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Fórmula:C20H24ClN3OPureza:99.56%Forma y color:SolidPeso molecular:357.88Bemegride
CAS:<p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>Fórmula:C8H13NO2Pureza:99.89%Forma y color:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Peso molecular:155.19IK1 inhibitor PA-6
CAS:<p>IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouse</p>Fórmula:C31H32N4O2Pureza:98.9%Forma y color:SolidPeso molecular:492.61Elexacaftor
CAS:<p>Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.</p>Fórmula:C26H34F3N7O4SPureza:98.87% - 99.87%Forma y color:SolidPeso molecular:597.65NS3623
CAS:<p>NS3623 is an activator of human ether-a-go-go-related gene potassium channels.</p>Fórmula:C15H10BrF3N6OPureza:97.06%Forma y color:SolidPeso molecular:427.18Lotilaner
CAS:<p>Lotilaner is a parasiticide.</p>Fórmula:C20H14Cl3F6N3O3SPureza:99.56%Forma y color:SolidPeso molecular:596.76EN6
CAS:<p>EN6, a small molecule, activates autophagy by modifying ATP6V1A, inhibiting mTORC1 and enhancing lysosomal function to clear TDP-43 aggregates.</p>Fórmula:C19H14F2N4O2Pureza:95.74% - 97.04%Forma y color:SolidPeso molecular:368.34Mebeverine hydrochloride
CAS:<p>Mebeverine hydrochloride (Colofac Hydrochloride), a β-phenylethylamine derivative, is a potent α1 repector inhibitor, relaxing the muscles in and around the gut</p>Fórmula:C25H35NO5Pureza:99.81% - 99.81%Forma y color:SolidPeso molecular:429.55Ethosuximide
CAS:<p>Ethosuximide (Zarontin) is an anticonvulsant, blocks the low voltage-activated T-type calcium channel used in the treatment of absence seizures unaccompanied by</p>Fórmula:C7H11NO2Pureza:98.87% - 99.72%Forma y color:Crystals From Acetone And Ether SolidPeso molecular:141.17MK-7622
CAS:<p>MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.</p>Fórmula:C25H25N3O2Pureza:99.77% - 99.8%Forma y color:SolidPeso molecular:399.48DMT1 blocker 2
CAS:<p>Compound 12f, a DMT1 blocker, inhibits DMT1 with a 0.83 IC50, potentially blocking intestinal iron absorption.</p>Fórmula:C16H13N3OPureza:99.68%Forma y color:SolidPeso molecular:263.29AZD 7009
CAS:<p>AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.</p>Fórmula:C23H34N4O5Pureza:98.42% - 98.51%Forma y color:SoildPeso molecular:446.54Moxidectin
CAS:<p>Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.</p>Fórmula:C37H53NO8Pureza:97.38%Forma y color:Appearance White Or Pale Yellow Amorphous PowderPeso molecular:639.82Phenibut
CAS:<p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>Fórmula:C10H13NO2Pureza:99.55%Forma y color:SolidPeso molecular:179.22γ-DGG acetate(6729-55-1 free base)
CAS:<p>gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.</p>Fórmula:C9H16N2O7Pureza:99.81%Forma y color:SolidPeso molecular:264.23GET73
CAS:<p>GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.</p>Fórmula:C13H16F3NO2Pureza:99.54%Forma y color:SolidPeso molecular:275.27Etimizol
CAS:<p>Etimizol improves memory by aiding the consolidation stage, effective against amnesia from hypoxia or brain injury.</p>Fórmula:C9H14N4O2Pureza:99%Forma y color:SolidPeso molecular:210.23Oxybuprocaine hydrochloride
CAS:<p>Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.</p>Fórmula:C17H29ClN2O3Pureza:>99.99%Forma y color:White Crystalline PowderPeso molecular:344.88DCPIB
CAS:<p>DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM</p>Fórmula:C22H28Cl2O4Pureza:99.79% - 99.87%Forma y color:SolidPeso molecular:427.36Doxapram hydrochloride hydrate
CAS:<p>Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.</p>Fórmula:C24H33ClN2O3C24H30N2O2·ClH·H2OPureza:99.64% - >99.99%Forma y color:SolidPeso molecular:432.99Glimepiride
CAS:<p>Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.</p>Fórmula:C24H34N4O5SPureza:97.84% - 98.87%Forma y color:White Cyrstalline SolidPeso molecular:490.62Disopyramide
CAS:<p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>Fórmula:C21H29N3OPureza:99.62%Forma y color:SolidPeso molecular:339.473,4,5-Trimethoxycinnamic acid
CAS:<p>3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the</p>Fórmula:C12H14O5Pureza:98.91%Forma y color:SolidPeso molecular:238.24Butamben
CAS:<p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>Fórmula:C11H15NO2Pureza:99.43%Forma y color:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Peso molecular:193.24Penicillin G sodium salt
CAS:<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Fórmula:C16H17N2NaO4SPureza:98.11%Forma y color:White To Off-White Crystalline PowderPeso molecular:356.37Leptomycin A
CAS:<p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>Fórmula:C32H46O6Pureza:98%Forma y color:SolidPeso molecular:526.7EVT-401
<p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>Fórmula:C22H20F4N2O3Forma y color:SolidPeso molecular:436.4Cavα2δ-IN-1
CAS:<p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>Fórmula:C18H27N5OForma y color:SolidPeso molecular:329.448Nitrazolam
CAS:<p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>Fórmula:C17H13N5O2Forma y color:SolidPeso molecular:319.32Elgodipine
CAS:<p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>Fórmula:C29H33FN2O6Pureza:98.95% - 99.50%Forma y color:SolidPeso molecular:524.58GS-9191 PM
<p>GS-9191 PM: novel antitumorviral bis-amide prodrug, inhibits MDR1/BCRP, has antiproliferative activity.</p>Fórmula:C11H16N6OPureza:99.79%Forma y color:SoildPeso molecular:248.28TRPA1 Antagonist 3
CAS:<p>TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.</p>Fórmula:C11H8ClN3Forma y color:SolidPeso molecular:217.66(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Fórmula:C6H11NO2Forma y color:SolidPeso molecular:129.16GsMTx4
CAS:<p>GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).</p>Fórmula:C185H273N49O45S6Pureza:98%Forma y color:SolidPeso molecular:4095.84BeKm-1
CAS:<p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>Fórmula:C174H261N51O52S6Pureza:98%Forma y color:SolidPeso molecular:4091.65GeX-2
CAS:<p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>Fórmula:C103H169N43O27Forma y color:SolidPeso molecular:2441.72α,β-Methylene-ATP dilithium
CAS:<p>α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.</p>Fórmula:C11H16Li2N5O12P3Forma y color:SolidPeso molecular:517.07GpTx-1 TFA
<p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with >20-fold and >950-fold selectivity, respectively.</p>Forma y color:Odour SolidWAY-326766
CAS:<p>WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).</p>Fórmula:C21H23N3O5Pureza:98.76%Forma y color:SolidPeso molecular:397.42AChE/Aβ-IN-1
<p>AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting the</p>Fórmula:C20H25BrN4Forma y color:SolidPeso molecular:401.34Anisatin
<p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>Fórmula:C15H20O8Forma y color:SolidPeso molecular:328.317Trans (2,3)-Dihydrotetrabenazine
CAS:<p>Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).</p>Fórmula:C19H29NO3Pureza:98%Forma y color:SolidPeso molecular:319.44LRRK2-IN-15
<p>LRRK2-IN-15 is an inhibitor of LRRK2. It exhibits an IC50 value of 5 nM in PBMC cells and 1.5 μM for BCRP. This compound is utilized in the research of Parkinson's disease.</p>Forma y color:Odour SolidTP-050
CAS:<p>TP-050: potent, selective NMDAR agonist, EC50 0.51 µM (GluN2A), 9.6 µM (GluN2D), BBB permeable, boosts hippocampal LTP.</p>Fórmula:C16H15ClF2N6OForma y color:SolidPeso molecular:380.78Albanin A
<p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>Fórmula:C20H18O6Forma y color:SolidPeso molecular:354.358Jingzhaotoxin-XII TFA
<p>Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.</p>Forma y color:Odour Solid3-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Fórmula:C3H10NO2PForma y color:SolidPeso molecular:123.092Huwentoxin I
CAS:<p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>Fórmula:C161H246N48O44S6Pureza:98%Forma y color:SolidPeso molecular:3750.36LY-466195
CAS:<p>LY-466195 is a competitive antagonist of GLUK5 receptor.</p>Fórmula:C16H24F2N2O4Forma y color:SolidPeso molecular:346.37Hyp9
CAS:<p>Hyp9, a specific agonist for the transient receptor potential canonical 6 (TRPC6) channel, is utilized in spinal cord injury (SCI) research [1].</p>Fórmula:C18H26O5Forma y color:SolidPeso molecular:322.40AChE/Aβ-IN-2
<p>AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.</p>Fórmula:C20H25ClN4Forma y color:SolidPeso molecular:356.89Chlorotoxin TFA
<p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>Fórmula:C160H250F3N53O49S11Forma y color:SolidPeso molecular:4109.74JAMI1001A
CAS:<p>JAMI1001A enhances AMPA receptor signaling, slows deactivation/desensitization for flip/flop isoforms.</p>Fórmula:C16H17F3N4O3SForma y color:SolidPeso molecular:402.39SLC26A3-IN-2
CAS:<p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>Fórmula:C19H13ClN2O2SPureza:99.86%Forma y color:SolidPeso molecular:368.84Homocarnosine
CAS:<p>Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.</p>Fórmula:C10H16N4O3Forma y color:SolidPeso molecular:240.26Idactamab
CAS:<p>Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.</p>Pureza:> 95%Forma y color:LiquidPeso molecular:146.2 kDaAnticonvulsant agent 9
<p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>Fórmula:C22H24N4O2Forma y color:SolidPeso molecular:376.45Crofelemer
CAS:<p>Crofelemer (Provir) is an orally active antidiarrheal agent. It targets the cystic fibrosis transmembrane conductance regulator (CFTR) and calcium-activated chloride channels (CACC), which are responsible for chloride and fluid secretion in the gastrointestinal tract. Crofelemer is applicable for research in diarrhea-related conditions.</p>Forma y color:Solid2,4,6-Tri-tert-butylphenol
CAS:<p>2,4,6-Tri-tert-butylphenol inhibits the Ca2+ ATPase activity of human red blood cell membranes and can be used in related research in the field of life sciences.</p>Fórmula:C18H30OPureza:99.55%Forma y color:SolidPeso molecular:262.43Bendroflumethiazide
CAS:<p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>Fórmula:C15H14F3N3O4S2Pureza:98% - >99.99%Forma y color:Crystals From Dioxane SolidPeso molecular:421.41Levamlodipine besylate Hemipentahydrate
CAS:<p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>Fórmula:C20H25ClN2O5·C6H6O3SH2OForma y color:SolidPeso molecular:1224.18Analgesic/antidepressant agent-1
<p>Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.</p>Fórmula:C22H25ClN2O2Forma y color:SolidPeso molecular:384.9Resolvin D2 methyl ester
CAS:<p>RvD2 is an anti-inflammatory lipid made from docosahexaenoic acid by 15- and 5-lipoxygenase. Its methyl ester may serve as a prodrug.</p>Fórmula:C23H34O5Forma y color:SolidPeso molecular:390.52
